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Таблетки Zoetis Апоквел, 16 мг
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Таблетки Zoetis Апоквел, 16 мг, 100 мл, 100 г, 100шт. в уп., 1уп., 16 мг

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Артикул Маркета
103714816877
Вид животного
Назначение средства
Форма выпуска
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Оклацитиниба малеат, входящий в состав препарата, в терапевтической дозе угнетает функции провоспалительных, проаллергических и пруритогенных (зудогенных) цитокинов, зависимых от ферментативной активности янус-киназы JAK1 или JAK3, целенаправленное воздействие на которые позволяет ингибировать ключевые механизмы возникновения зуда, ассоциированного с аллергией, и способствует устранению симптомов местного воспаления; на цитокины, участвующие в кроветворении и зависимые от JAK2, существенно не влияет. После перорального введения препарата оклацитиниба малеат быстро всасывается в желудочно-кишечном тракте (биодоступность составляет 89%), поступает в системный кровоток, достигая максимальной концентрации в плазме менее чем через 1 час, проникает в большинство органов и тканей, практически не метаболизируется, выводится из организма в неизмененной форме, преимущественно с мочой, период полувыведения составляет 3-4 часа. Апоквел по степени воздействия на организм относится к веществам умеренно опасным (3 класс опасности по ГОСТ 12.1.007) со слабо выраженными кумулятивными свойствами, в рекомендуемой дозе не обладает мутагенной, канцерогенной, эмбриотоксической и тератогенной активностью."},{"name":"Состав","value":"оклацитиниба малеат (в пересчете на оклацитиниб) 16 мг, а также вспомогательные вещества: микрокристаллическая целлюлоза, лактоза моногидрат, карбоксиметил-крахмал натрия, магния стеарат, плёнкообразователь «Opadry II White» и вода очищенная"},{"name":"Показания к применению","value":"для лечения зуда, вызванного аллергическим дерматитом и профилактики атопического дерматита у собак"},{"name":"Противопоказания","value":"Противопоказанием к применению Апоквела является индивидуальная непереносимость животным его компонентов. Не допускается применение препарата собакам с признаками иммуносупрессии, такими как гиперадренокортицизм, а также собакам с прогрессирующими злокачественными новообразованиями."},{"name":"Побочные действия","value":"Побочные явления и осложнения при кратковременном применении Апоквела могут проявляться угнетенным состоянием, расстройством функции желудочно-кишечного тракта, циститом; у животных, получающих Апоквел более 16 дней, приблизительно в 1% случаев может наблюдаться повышение аппетита и агрессия, кожные и подкожные новообразования, инфекции кожи, вызванные дрожжевыми грибками, увеличением лимфатических узлов, обострением демодекоза и онкологических заболеваний."},{"name":"Передозировка","value":"При передозировке лекарственного препарата у животного могут наблюдаться следующие симптомы: угнетенное состояние, рвота, диарея, локальные алопеции, утолщение кожной складки, образование струпьев и корочек, межпальцевые кисты, отек конечностей. Специфические антидоты отсутствуют, животному применяют симптоматическое лечение."},{"name":"Взаимодействие","value":"При совместном применении Апоквела с противомикробными, противовоспалительными и противопаразитарными препаратами фармакологического взаимодействия не выявлено. Не следует применять Апоквел совместно с иммунодепрессантами и противосудорожными препаратами."},{"name":"Особые указания","value":"Пустые флаконы из-под лекарственного препарата запрещается использовать для бытовых целей, они подлежат утилизации с бытовыми отходами. Особенности действия при первом применении препарата и при его отмене не выявлены. Следует избегать пропусков при введении очередной дозы препарата, так как это может привести к снижению эффективности. В случае пропуска очередной дозы, применение Апоквела возобновляют в соответствии с настоящей инструкцией. Апоквел не предназначен для применения продуктивным животным."},{"name":"Применение у беременных и кормящих животных","value":"не следует применять Апоквел сукам в период беременности и лактации"},{"name":"Способ применения и дозы","value":"применяют собакам перорально индивидуально с руки, или в смеси с кормом, или вводят принудительно в пасть в разовой дозе 0,4-0,6 мг оклацитиниба на 1 кг массы животного два раза в день, не более 14 суток; в качестве поддерживающей терапии при атопическом дерматите — один раз в сутки в той же дозе, но не более 14 недель"},{"name":"Фармакокинетика","value":"после перорального введения препарата оклацитиниба малеат быстро всасывается в желудочно-кишечном тракте (биодоступность составляет 89 %), поступает в системный кровоток, достигая максимальной концентрации в плазме менее чем через 1 час, проникает в большинство органов и тканей, практически не метаболизируется, выводится из организма в неизмененной форме, преимущественно с мочой, период полувыведения составляет 3-4 часа"},{"name":"Условия отпуска","value":"без рецепта"},{"name":"Условия хранения","value":"Хранят препарат в закрытой упаковке производителя, в сухом, защищенном от света месте, отдельно от продуктов питания и кормов при температуре от 0 °С до 25 °С."},{"name":"Регистрационный номер","value":"№ПВИ-3-1.16/04707"},{"name":"Дата государственной регистрации","value":"20.02.2021"},{"name":"Дополнительная информация","value":"При переводе на корм Alleva Equilibrium рекомендуется постепенно в течение 1-2 недель замещать предыдущий корм на новый."}]}},"fullSpecsGrouped":{"6336985730195497350":{"groups":[{"name":"Общие сведения","items":[{"value":"Zoetis","transition":{"params":{"glfilters":["7893318:13582700"]},"type":"catalog"},"name":"Бренд"},{"value":"лекарственный препарат","transition":{"params":{"glfilters":["34324371:35649313"]},"type":"catalog"},"name":"Тип препарата"},{"name":"Действующее вещество","value":"оклацитиниб"},{"name":"Форма выпуска","value":"таблетки для перорального применения"},{"value":"100 шт.","transition":{"params":{"glfilters":["14805583:100~100"]},"type":"catalog"},"name":"Количество в упаковке"},{"value":"100 мл","transition":{"params":{"glfilters":["24139073:100~100"]},"type":"catalog"},"name":"Объем"},{"name":"Вес","value":"100 г"},{"name":"Упаковка","value":"банка"},{"value":"при аллергии","transition":{"params":{"glfilters":["27143691:37167814"]},"type":"catalog"},"name":"Назначение средства"},{"value":"собаки","transition":{"params":{"glfilters":["43903290:44628264"]},"type":"catalog"},"name":"Вид животного"},{"value":"взрослые, молодые, пожилые","transition":{"params":{"glfilters":["34074939:35635216,35635215,35635213"]},"type":"catalog"},"name":"Возраст животного"},{"name":"Минимальный возраст применения","value":"12 мес"},{"name":"Размер животного","value":"крупные породы, крупный, маленький"},{"name":"Минимальный вес животного","value":"13.5 кг"},{"name":"Максимальный вес животного","value":"80 кг"},{"name":"Страна производства","value":"Италия"}]},{"name":"Фармакологические свойства","items":[{"name":"Описание средства","value":"овальные таблетки белого или почти белого цвета, покрытые пленочной оболочкой, с разделительной бороздкой посередине и c надписью на обеих сторонах таблетки: L"},{"name":"Фармакологическая группа","value":"относится к лекарственным препаратам группы селективных ингибиторов янус-киназы (JAK)"},{"name":"Фармакологическое действие","value":"Апоквел относится к лекарственным препаратам группы селективных ингибиторов янус-киназы (JAK). 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Пэй
64 999
–42%
без карты
 
38 000
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Таблетки Zoetis Апоквел, 16 мг
Таблетки Zoetis Апоквел, 16 мг, 100 мл, 100 г, 100шт. в уп., 1уп., 16 мг
Цена с картой Яндекс Пэй:37 620
Скидка: 42%
–42 %
Вместо:
38 00064 999
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Войдите, и станет дешевлеВ аккаунте больше скидок
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Ветеринарная аптека "Здоровые Лапы"
Ветеринарная аптека "Здоровые Лапы"
Магазин4 26 оценок
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Доставка Маркета
11 июня, по клику  0
Москва
11 июня, пункт выдачи  0
Москва
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    Рейтинг товара: 4.8 из 5на основе 4 оценки
      
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    Рейтинг товара: 4.7 из 5на основе 12 оценок
      
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    Рейтинг товара: 4.3 из 5на основе 24 оценки
      
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    Рейтинг товара: 5.0 из 5на основе 49 оценок
      
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    Рейтинг товара: 4.6 из 5на основе 573 оценки
      
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    Рейтинг товара: 4.4 из 5на основе 5 оценок
      
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О товаре

Zoetis Апоквел 16 мг, 100 таб – единственный препарат, разрывающий цикл зуда и воспаления при дерматите у собак.
Селективный ингибитор янус-киназы (JAK) для снятия зуда у собак.
Действие в течение 4 часов после введения.
Хорошо переносится животными.
Подходит для купирования острых и хронических состояний.
Апоквел назначают собакам при дерматите, вызванным аллергией (блошиной, контактной, пищевой, паразитарной), и при атопическом дерматите для устранения зуда и уменьшения воспаления. Не допускается применение препарата собакам, с признаками иммуносупрессии, такими как гиперадренокортицизм, а также собакам, с прогрессирующими злокачественными новообразованиями.
Бренд
Zoetis
Тип препарата
лекарственный препарат
Действующее вещество
оклацитиниб
Форма выпуска
таблетки для перорального применения
Количество в упаковке
100 шт.
Объем
100 мл
Вес
100 г
Упаковка
банка
Назначение средства
при аллергии
Вид животного
собаки
Возраст животного
взрослые, молодые, пожилые
Минимальный возраст применения
12 мес
Размер животного
крупные породы, крупный, маленький
Минимальный вес животного
13.5 кг
Максимальный вес животного
80 кг
Страна производства
Италия
Описание средства
овальные таблетки белого или почти белого цвета, покрытые пленочной оболочкой, с разделительной бороздкой посередине и c надписью на обеих сторонах таблетки: L
Фармакологическая группа
относится к лекарственным препаратам группы селективных ингибиторов янус-киназы (JAK)
Фармакологическое действие
Апоквел относится к лекарственным препаратам группы селективных ингибиторов янус-киназы (JAK). Оклацитиниба малеат, входящий в состав препарата, в терапевтической дозе угнетает функции провоспалительных, проаллергических и пруритогенных (зудогенных) цитокинов, зависимых от ферментативной активности янус-киназы JAK1 или JAK3, целенаправленное воздействие на которые позволяет ингибировать ключевые механизмы возникновения зуда, ассоциированного с аллергией, и способствует устранению симптомов местного воспаления; на цитокины, участвующие в кроветворении и зависимые от JAK2, существенно не влияет. После перорального введения препарата оклацитиниба малеат быстро всасывается в желудочно-кишечном тракте (биодоступность составляет 89%), поступает в системный кровоток, достигая максимальной концентрации в плазме менее чем через 1 час, проникает в большинство органов и тканей, практически не метаболизируется, выводится из организма в неизмененной форме, преимущественно с мочой, период полувыведения составляет 3-4 часа. Апоквел по степени воздействия на организм относится к веществам умеренно опасным (3 класс опасности по ГОСТ 12.1.007) со слабо выраженными кумулятивными свойствами, в рекомендуемой дозе не обладает мутагенной, канцерогенной, эмбриотоксической и тератогенной активностью.
Состав
оклацитиниба малеат (в пересчете на оклацитиниб) 16 мг, а также вспомогательные вещества: микрокристаллическая целлюлоза, лактоза моногидрат, карбоксиметил-крахмал натрия, магния стеарат, плёнкообразователь «Opadry II White» и вода очищенная
Показания к применению
для лечения зуда, вызванного аллергическим дерматитом и профилактики атопического дерматита у собак
Противопоказания
Противопоказанием к применению Апоквела является индивидуальная непереносимость животным его компонентов. Не допускается применение препарата собакам с признаками иммуносупрессии, такими как гиперадренокортицизм, а также собакам с прогрессирующими злокачественными новообразованиями.
Побочные действия
Побочные явления и осложнения при кратковременном применении Апоквела могут проявляться угнетенным состоянием, расстройством функции желудочно-кишечного тракта, циститом; у животных, получающих Апоквел более 16 дней, приблизительно в 1% случаев может наблюдаться повышение аппетита и агрессия, кожные и подкожные новообразования, инфекции кожи, вызванные дрожжевыми грибками, увеличением лимфатических узлов, обострением демодекоза и онкологических заболеваний.
Передозировка
При передозировке лекарственного препарата у животного могут наблюдаться следующие симптомы: угнетенное состояние, рвота, диарея, локальные алопеции, утолщение кожной складки, образование струпьев и корочек, межпальцевые кисты, отек конечностей. Специфические антидоты отсутствуют, животному применяют симптоматическое лечение.
Взаимодействие
При совместном применении Апоквела с противомикробными, противовоспалительными и противопаразитарными препаратами фармакологического взаимодействия не выявлено. Не следует применять Апоквел совместно с иммунодепрессантами и противосудорожными препаратами.
Особые указания
Пустые флаконы из-под лекарственного препарата запрещается использовать для бытовых целей, они подлежат утилизации с бытовыми отходами. Особенности действия при первом применении препарата и при его отмене не выявлены. Следует избегать пропусков при введении очередной дозы препарата, так как это может привести к снижению эффективности. В случае пропуска очередной дозы, применение Апоквела возобновляют в соответствии с настоящей инструкцией. Апоквел не предназначен для применения продуктивным животным.
Применение у беременных и кормящих животных
не следует применять Апоквел сукам в период беременности и лактации
Способ применения и дозы
применяют собакам перорально индивидуально с руки, или в смеси с кормом, или вводят принудительно в пасть в разовой дозе 0,4-0,6 мг оклацитиниба на 1 кг массы животного два раза в день, не более 14 суток; в качестве поддерживающей терапии при атопическом дерматите — один раз в сутки в той же дозе, но не более 14 недель
Фармакокинетика
после перорального введения препарата оклацитиниба малеат быстро всасывается в желудочно-кишечном тракте (биодоступность составляет 89 %), поступает в системный кровоток, достигая максимальной концентрации в плазме менее чем через 1 час, проникает в большинство органов и тканей, практически не метаболизируется, выводится из организма в неизмененной форме, преимущественно с мочой, период полувыведения составляет 3-4 часа
Условия отпуска
без рецепта
Условия хранения
Хранят препарат в закрытой упаковке производителя, в сухом, защищенном от света месте, отдельно от продуктов питания и кормов при температуре от 0 °С до 25 °С.
Регистрационный номер
№ПВИ-3-1.16/04707
Дата государственной регистрации
20.02.2021
Дополнительная информация
При переводе на корм Alleva Equilibrium рекомендуется постепенно в течение 1-2 недель замещать предыдущий корм на новый.
Перед покупкой уточняйте характеристики и комплектацию у продавца.
Есть противопоказания, посоветуйтесь с врачом.
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
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Вопросы о товаре
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Войдите в аккаунт

И тогда откроется корзина, а цены на Маркете могут стать ниже
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