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Таблетки Zoetis Апоквел, 5.4 мг
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Описание
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Таблетки Zoetis Апоквел, 5.4 мг, 26 г, 20шт. в уп., 1уп.

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Артикул Маркета
103542541590
Вид животного
Назначение средства
Форма выпуска
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Вместо:
4 1824 403
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Таблетки Zoetis Апоквел, 5.4 мг
Таблетки Zoetis Апоквел, 5.4 мг, 26 г, 20шт. в уп., 1уп.
Цена с картой Яндекс Пэй:4 098
Скидка: 7%
–7 %
Вместо:
4 1824 403
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Войдите, и станет дешевлеВ аккаунте больше скидок
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Доставка Маркета
12 июня, курьер  0 ₽
Москва
12 июня, по клику  0 ₽
15-30 мин. курьером в удобный момент
12 июня, пункт выдачи  0 ₽
Москва
Animal City
Магазин4.7 1.5K оценок
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Ещё может подойти
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    Рейтинг товара: 4.9 из 5на основе 122 оценки
      
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    Рейтинг товара: 4.6 из 5на основе 12 оценок
      
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    Рейтинг товара: 4.8 из 5на основе 146 оценок
      
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    Рейтинг товара: 4.8 из 5на основе 4 оценки
      
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    Рейтинг товара: 4.7 из 5на основе 12 оценок
      
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    Рейтинг товара: 4.6 из 5на основе 573 оценки
      
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Инструкция
Бренд
Zoetis
Тип препарата
лекарственный препарат
Действующее вещество
оклацитиниб
Форма выпуска
таблетки для перорального применения
Количество в упаковке
20 шт.
Вес
26 г
Упаковка
банка
Назначение средства
для кожи
Вид животного
кошки, собаки
Возраст животного
взрослые
Размер животного
крупный, маленький, средние породы, средний
Страна производства
Италия
Описание средства
овальные таблетки белого или почти белого цвета, покрытые пленочной оболочкой, с разделительной бороздкой посередине и c надписью на обеих сторонах таблетки: L
Фармакологическая группа
относится к лекарственным препаратам группы селективных ингибиторов янус-киназы (JAK)
Фармакологическое действие
оклацитиниба малеат, входящий в состав препарата, в терапевтической дозе угнетает функции провоспалительных, проаллергических и пруритогенных (зудогенных) цитокинов, зависимых от ферментативной активности янус-киназы JAK1 или JAK3, целенаправленное воздействие на которые позволяет ингибировать ключевые механизмы возникновения зуда, ассоциированного с аллергией, и способствует устранению симптомов местного воспаления; на цитокины, участвующие в кроветворении и зависимые от JAK2, существенно не влияет
Состав
Оклацитиниба малеат (в пересчете на оклацитиниб) 16 мг, а также вспомогательные вещества: микрокристаллическая целлюлоза, лактоза моногидрат, карбоксиметил-крахмал натрия, магния стеарат, плёнкообразователь «Opadry II White» и вода очищенная.
Показания к применению
Апоквел назначают собакам при дерматите, ассоциированном с аллергией (контактный, пищевой, паразитарный) в целях устранения зуда и уменьшения очаговых изменений кожи, а также для профилактики рецидивов атопического дерматита.
Противопоказания
противопоказанием к применению Апоквела является индивидуальная непереносимость животным его компонентов; не допускается применение препарата собакам, с признаками иммуносупрессии, такими как гиперадренокортицизм, а также собакам, с прогрессирующими злокачественными новообразованиями; не следует применять препарат кобелям в период вязки, собакам моложе 12-месячного возраста и/или массой менее 3 кг, а также щенным и кормящим сукам
Побочные действия
заключаются в угнетенном состоянии, расстройстве функции желудочно-кишечного тракта, циститом; у животных, получающих Апоквел более 16 дней, приблизительно в 1 % случаев может наблюдаться повышение аппетита и агрессия, кожные и подкожные образования
Передозировка
при передозировке лекарственного препарата у животного могут наблюдаться следующие симптомы: угнетенное состояние, рвота, диарея, локальные алопеции, утолщение кожной складки, образование струпьев и корочек, межпальцевые кисты, отек конечностей. Специфические антидоты отсутствуют, животному применяют симптоматическое лечение
Взаимодействие
При совместном применении Апоквела с противомикробными, противовоспалительными и противопаразитарными препаратами фармакологического взаимодействия не выявлено. Не следует применять Апоквел совместно с иммунодепрессантами и противосудорожными препаратами.
Особые указания
пустые флаконы из-под лекарственного препарата запрещается использовать для бытовых целей, они подлежат утилизации с бытовыми отходами; следует избегать пропусков при введении очередной дозы препарата, так как это может привести к снижению эффективности; в случае пропуска очередной дозы, применение Апоквела возобновляют в соответствии с настоящей инструкцией
Применение у беременных и кормящих животных
запрещается применять Апоквел сукам в период беременности и лактации
Способ применения и дозы
Апоквел применяют собакам перорально индивидуально с руки, или в смеси с кормом, или вводят принудительно в пасть в разовой дозе 0,4-0,6 мг оклацитиниба на 1 кг массы животного два раза в день, не более 14 суток; в качестве поддерживающей терапии при атопическом дерматите – один раз в сутки в той же дозе, но не более 14 недель. Схема и длительность курса применения препарата зависят от этиологии и патогенеза дерматита, клинического состояния животного и определяются лечащим ветеринарным врачом.
Фармакокинетика
после перорального введения препарата оклацитиниба малеат быстро всасывается в желудочно-кишечном тракте (биодоступность составляет 89 %), поступает в системный кровоток, достигая максимальной концентрации в плазме менее чем через 1 час, проникает в большинство органов и тканей, практически не метаболизируется, выводится из организма в неизмененной форме, преимущественно с мочой, период полувыведения составляет 3-4 часа
Условия отпуска
без рецепта
Условия хранения
Хранят препарат в закрытой упаковке производителя, в сухом, защищенном от света месте, отдельно от продуктов питания и кормов при температуре от 0 °С до 25 °С.
Регистрационный номер
№ПВИ-3-1.16/04707
Дата государственной регистрации
20.02.2021
Дополнительная информация
Схема и длительность курса применения препарата зависят от этиологии и патогенеза дерматита, клинического состояния животного и определяются лечащим ветеринарным врачом.
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Войдите в аккаунт

И тогда откроется корзина, а цены на Маркете могут стать ниже
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