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Описание

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Аллафорте таб. пролонг. действ., 25 мг, 20 шт.

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Дозировка: 25 мг

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Количество штук в упаковке, шт.: 20

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0,025 г.\u003Cbr\u003EВспомогательные вещества: крахмал прежелатинизированный, лактоза моногидрат, гипромеллоза, кальция стеарат, кремния диоксид коллоидный (аэросил А-380) - 0,230 г.\u003Cbr\u003EСостав на одну таблетку 50 мг:\u003Cbr\u003EДействующее вещество: Лаппаконитина гидробромид (Аллапинин) (в пересчете на 100 % вещества) - 0,050 г.\u003Cbr\u003EВспомогательные вещества: крахмал прежелатинизированный, лактоза моногидрат, гипромеллоза, кальция стеарат, кремния диоксид коллоидный (аэросил А-380) - 0,350 г."},{"name":"Действующее вещество","value":"Лаппаконитина гидробромид","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28710831"]}}},{"name":"Способ применения и дозы","value":"Прием препарата следует начинать под наблюдением врача.\u003Cbr\u003EВнутрь, после приема пищи, проглатывая таблетку целиком и запивая небольшим количеством воды комнатной температуры.\u003Cbr\u003EТаблетки категорически запрещается разламывать, измельчать или разжевывать!\u003Cbr\u003EДоза препарата Аллафорте подбирается индивидуально. Лечение следует начинать с назначения таблеток по 25 мг каждые 8 часов. При отсутствии или недостаточности терапевтического эффекта дозу следует увеличить - таблетки по 25 мг через каждые 6 часов или таблетки по 50 мг через каждые 12 часов. Судить о терапевтическом действии препарата при его первом применении или при увеличении его дозы следует не ранее, чем через 2-3 суток регулярного применения препарата.\u003Cbr\u003EДля предупреждения нежелательных влияний препарата на проводящую систему сердца его применение и увеличение дозы следует контролировать с помощью ЭКГ. Регистрировать ЭКГ целесообразно через 1-2 часа после приема очередной разовой дозы препарата. При удлинении интервала PQ до 300 мс или развитии предсердно-желудочковых блокад более высокой степени дозу следует уменьшить, при необходимости временно прекратив лечение. Безопасным является удлинение комплекса QRS на величину до 25 % от исходной, но при этом длительность QRS не должна превышать 140 мс. Недопустимо удлинение комплекса QRS свыше 50 % от исходного или более 160 мс!\u003Cbr\u003EМаксимальная суточная доза препарата составляет 100 мг (25 мг 4 раза в сутки или 50 мг 2 раза в сутки). В дозе более 100 мг в сутки препарат принимать не рекомендуется ввиду отсутствия контролируемых клинических исследований. Перевод пациентов, принимающих препарат Аллапинин, на лечение препаратом Аллафорте осуществляется путем простой замены, начиная с момента очередного приема одного препарата на другой с применением одинаковых доз и интервалов между приемами.\u003Cbr\u003EПродолжительность лечения и коррекция режима дозирования (увеличение дозы) определяется врачом."},{"name":"Побочные действия","value":"Оценка частоты возникновения побочных реакций произведена на основании следующих критериев: очень частые (≥ 1/10), частые (от ≥ 1/100 до \u003C 1/10), нечастые (от ≥ 1/1000 до \u003C 1/100), редкие (от ≥ 1/10 000 до \u003C 1/1000), очень редкие (\u003C 1/10 000), частота неизвестна (данные по оценке частоты отсутствуют).\u003Cbr\u003EНарушения со стороны центральной нервной системы\u003Cbr\u003Eочень часто: головокружение, головная боль, ощущение тяжести в голове, атаксия;\u003Cbr\u003EНарушения со стороны органа зрения\u003Cbr\u003Eочень часто: диплопия;\u003Cbr\u003EНарушения со стороны сердца\u003Cbr\u003Eочень часто: нарушения внутрижелудочковой и AV проводимости; изменения на ЭКГ: удлинение интервала PQ, расширение комплекса QRS;\u003Cbr\u003Eчасто: синусовая тахикардия (при длительном применении), повышение АД; нечасто: аритмогенное действие;\u003Cbr\u003EНарушения со стороны кожи и подкожных тканей\u003Cbr\u003Eчасто: аллергические реакции, гиперемия кожных покровов;\u003Cbr\u003EЛабораторные и инструментальные данные\u003Cbr\u003EОчень часто: изменения на ЭКГ: удлинение интервала PQ, расширение комплекса QRS."},{"name":"Фармакологическое действие","value":"Антиаритмический препарат IC класса. Действующее вещество препарата представляет собой бромистоводородную соль алкалоида лаппаконитина с сопутствующими алкалоидами, получаемую из травы борца белоустого или из корневищ и корней борца белоустого - Aconitum leucostomum Worosch., или из корневищ с корнями борца северного (борца высокого) - Aconitum septentrionale Koelle (A. excelsum Reichenb.), семейства лютиковые - Ranunculaceae, или из технической суммы алкалоидов семейства лютиковых.\u003Cbr\u003EФармакодинамика\u003Cbr\u003EВ основе механизма антиаритмического действия лежит блокировка «быстрых» натриевых каналов мембран кардиомиоцитов. Лаппаконитина гидробромид вызывает замедление атриовентрикулярной (AV) и внутрижелудочковой проводимости, угнетает проведение по дополнительным путям при синдроме Вольфа-Паркинсона-Уайта, укорачивает эффективный и функциональный рефрактерные периоды предсердий, AV узла, пучка Гиса и волокон Пуркинье. Не влияет на продолжительность интервала QT, проводимость по AV узлу в антероградном направлении, частоту сердечных сокращений (ЧСС) и артериальное давление (АД), сократимость миокарда (при исходном отсутствии явлений сердечной недостаточности). Не угнетает автоматизм синусового узла, не оказывает отрицательного инотропного действия, не обладает антигипертензивным и м-холинолитическим действием. Лаппаконитина гидробромид оказывает умеренное спазмолитическое, коронарорасширяющее, местноанестезирующее и седативное действие.\u003Cbr\u003EПри приеме внутрь эффект развивается через 40-60 минут, сохраняется на достигнутом уровне 4-5 часов и постепенно снижается. В целом действие препарата после однократного приема внутрь сохраняется не менее 12 часов."},{"name":"Фармакологическая группа","value":"антиаритмические средства"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"В защищенном от света месте, при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Сравнительно небольшая терапевтическая широта препарата может способствовать интоксикации, особенно при сочетании с другими антиаритмическими средствами.\u003Cbr\u003EСимптомы: удлинение интервала PQ и QT, расширение комплекса QRS, увеличение амплитуды зубца Т, брадикардия, синоатриальная и атриовентрикулярная блокада, асистолия, пароксизмы полиморфной желудочковой тахикардии, снижение сократимости миокарда, выраженное снижение АД, головокружение, затуманенность зрения, головная боль, желудочно-кишечные расстройства.\u003Cbr\u003EЛечение: симптоматическое, промывание желудка, дефибрилляция, введение добутамина, диазепама; при необходимости - искусственная вентиляция легких и непрямой массаж сердца.\u003Cbr\u003EДля лечения желудочковой тахикардии не применять антиаритмические средства IA и IC класса."},{"name":"Применение при беременности и кормлении грудью","value":"Беременность\u003Cbr\u003EПрименение препарата при беременности не рекомендуется ввиду отсутствия контролируемых исследований.\u003Cbr\u003EПо данным доклинических исследований лаппаконитина гидробромид в дозах 1 -5 мг/кг не обладает тератогенным и эмбриотоксическим действием.\u003Cbr\u003EПрименение препарата при беременности возможно только по жизненным показаниям, если предполагаемая польза для матери превышает потенциальный риск развития побочных эффектов у плода/ребенка.\u003Cbr\u003EПериод грудного вскармливания\u003Cbr\u003EДанные о выделении лаппаконитина гидробромида в грудное молоко отсутствуют. Применение препарата не рекомендуется в период грудного вскармливания.\u003Cbr\u003EЕсли применение препарата Аллафорте в период лактации необходимо, грудное вскармливание следует прекратить."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"При применении препарата необходимо соблюдать осторожность при управлении транспортными средствами и занятии другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций в связи с риском развития головокружения."},{"name":"Особые указания","value":"С осторожностью:\u003Cbr\u003E\nПрименять пациентам с электрокардиостимулятором, при AV блокаде I степени, хронической сердечной недостаточности I-II функционального класса по классификации NYHA, нарушении внутрижелудочковой проводимости, синдроме слабости синусового узла (СССУ), брадикардии, тяжелых нарушениях периферического кровообращения, закрытоугольной глаукоме, доброкачественной гипертрофии предстательной железы, нарушении проводимости по волокнам Пуркинье, блокаде одной из ножек пучка Гиса, нарушении водно-электролитного обмена (гипокалиемия, гиперкалиемия, гипомагниемия), при одновременном приеме других антиаритмических средств.\u003Cbr\u003EОсобые указания:\u003Cbr\u003EПрепарат применяют по назначению врача.\u003Cbr\u003EПеред началом применения препарата необходимо устранить нарушения водно-электролитного обмена, в период терапии необходим контроль водно¬электролитного баланса крови.\u003Cbr\u003EКаждый пациент, который принимает препарат, должен проходить электрокардиографическое и клиническое обследование до начала терапии и в период ее проведения для раннего выявления побочного действия, оценки эффективности препарата и необходимости продолжения терапии.\u003Cbr\u003EУ пациентов с установленным электрокардиостимулятором может повышаться порог стимуляции. Электрокардиостимуляторы необходимо проверять и при необходимости перепрограммировать.\u003Cbr\u003EПри развитии головной боли, головокружения, диплопии следует уменьшить дозу препарата.\u003Cbr\u003EПри появлении синусовой тахикардии на фоне длительного применения препарата показано применение бета-адреноблокаторов (в индивидуально подобранных дозах).\u003Cbr\u003EПри применении антиаритмических средств IC класса у пациентов с тяжелыми органическими изменениями миокарда могут возникать серьезные нежелательные реакции. Применение препарата у таких пациентов возможно только после тщательной оценки ожидаемой пользы и возможного риска для пациентов, и должно осуществляться под наблюдением врача-кардиолога, имеющего опыт лечения соответствующих нарушений сердечного ритма.\u003Cbr\u003EС особой осторожностью следует применять препарат у пациентов с ишемической болезнью сердца и стабильной стенокардией напряжения, поскольку одним из предрасполагающих факторов аритмогенного действия антиаритмических препаратов IC класса является преходящая ишемия миокарда и высокая ЧСС. Препарат следует с осторожностью применять совместно с другими антиаритмическими препаратами в связи с повышенным риском аритмогенного действия.\u003Cbr\u003EУстановлено неблагоприятное влияние других антиаритмических препаратов IC класса на электрофизиологические показатели и клинические проявления при синдроме Бругада. Опыт применения лаппаконитина гидробромида при синдроме Бругада отсутствует, в связи с чем применение препарата у пациентов с синдромом Бругада противопоказано.\u003Cbr\u003EПрепарат предназначен для длительной профилактической антиаритмической терапии. Имеющийся ограниченный клинический опыт не позволяет рекомендовать применение препарата внутрь для купирования пароксизмов наджелудочковой и желудочковой тахикардии.\u003Cbr\u003EВлияние терапии лаппаконитина гидробромидом на выживаемость или частоту внезапной смерти пациентов с желудочковыми нарушениями сердечного ритма не изучалось в клинических исследованиях.\u003Cbr\u003EВспомогательные вещества\u003Cbr\u003EПрепарат Аллафорте содержит лактозы моногидрат. Пациентам с редко встречающимися наследственными заболеваниями, такими как непереносимость галактозы, непереносимость лактозы вследствие дефицита лактазы или синдром галактозной мальабсорбции, не следует принимать данный лекарственный препарат."},{"name":"Взаимодействие","value":"-при одновременном применении лаппаконитина гидробромида с другими антиаритмическими средствами повышается риск развития аритмогенного действия;\u003Cbr\u003E-лаппаконитина гидробромид усиливает эффект недеполяризующих миорелаксантов;\u003Cbr\u003E-при одновременном применении лаппаконитина гидробромида с другими антиаритмическими средствами повышается риск развития побочных эффектов, связанных с влиянием на функцию синусового узла и предсердно-желудочковую проводимость; требуется индивидуальный подбор доз каждого из этих препаратов;\u003Cbr\u003E-в клиническом исследовании при применении лаппаконитина гидробромида на фоне стандартной гипотензивной терапии ингибиторами ангиотензинпреврагцающего фермента, антагонистами рецепторов к ангиотензину ii, блокаторами «медленных» кальциевых каналов производных дигидропиридина, бета-адреноблокаторами не наблюдалось усиления или ослабления антигипертензивного действия;\u003Cbr\u003E-индукторы микросомальных ферментов печени не влияют на эффективность лаппаконитина гидробромида;\u003Cbr\u003E-не имеется данных о неблагоприятном влиянии лаппаконитина гидробромида на эффективность и безопасность непрямых антикоагулянтов."},{"name":"Регистрационный номер","value":"ЛП-004040"},{"name":"Дата государственной регистрации","value":"26.09.2022"},{"name":"Владелец регистрационного удостоверения","value":"Фармцентр Вилар","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313","7893318:16003015"]}}},{"name":"Изготовитель","value":"Фармцентр Вилар"},{"name":"Фасовщик","value":"Фармцентр Вилар"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Аллафорте","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["17796364:18007780"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"13435693244782992754":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"сердце"},{"name":"Назначение","value":"аритмия, наджелудочковая тахикардия, нарушение ритма сердца, пароксизмальная наджелудочковая тахикардия, синдром Вольфа-Паркинсона-Уайта, трепетание предсердий, фибрилляция предсердий, экстрасистолия"},{"name":"Показания к применению","value":"-наджелудочковая и желудочковая экстрасистолия;\u003Cbr\u003E-пароксизмальная форма фибрилляции и трепетания предсердий;\u003Cbr\u003E-пароксизмальная наджелудочковая тахикардия, в том числе и при синдроме Вольфа-Паркинсона-Уайта (WPW);\u003Cbr\u003E-пароксизмальная желудочковая тахикардия (при отсутствии органических изменений миокарда)."},{"name":"Противопоказания","value":"-повышенная чувствительность к лаппаконитина гидробромиду или к любому другому компоненту препарата;\u003Cbr\u003E-синоатриальная блокада;\u003Cbr\u003E-AV блокада II и III степени (без электрокардиостимулятора);\u003Cbr\u003E-кардиогенный шок;\u003Cbr\u003E-блокада правой ножки пучка Гиса, сочетающаяся с блокадой одной из ветвей левой ножки;\u003Cbr\u003E-тяжелая артериальная гипотензия (систолическое АД менее 90 мм рт;ст;);\u003Cbr\u003E-хроническая сердечная недостаточность III-IV функционального класса по классификации NYHA;\u003Cbr\u003E-выраженная гипертрофия миокарда левого желудочка (≥1,4 см);\u003Cbr\u003E-постинфарктный кардиосклероз;\u003Cbr\u003E-синдром Бругада;\u003Cbr\u003E-острый инфаркт миокарда;\u003Cbr\u003E-тяжелые нарушения функции печени и/или почек;\u003Cbr\u003E-непереносимость лактозы;\u003Cbr\u003E-беременность и период грудного вскармливания;"},{"name":"Состав","value":"1 таблетка препарата Аллафорте содержит в качестве действующего вещества Лаппаконитина гидробромид 25 мг или 50 мг.\u003Cbr\u003EСостав на одну таблетку 25 мг:\u003Cbr\u003EДействующее вещество: Лаппаконитина гидробромид (Аллапинин) (в пересчете на 100 % вещества) - 0,025 г.\u003Cbr\u003EВспомогательные вещества: крахмал прежелатинизированный, лактоза моногидрат, гипромеллоза, кальция стеарат, кремния диоксид коллоидный (аэросил А-380) - 0,230 г.\u003Cbr\u003EСостав на одну таблетку 50 мг:\u003Cbr\u003EДействующее вещество: Лаппаконитина гидробромид (Аллапинин) (в пересчете на 100 % вещества) - 0,050 г.\u003Cbr\u003EВспомогательные вещества: крахмал прежелатинизированный, лактоза моногидрат, гипромеллоза, кальция стеарат, кремния диоксид коллоидный (аэросил А-380) - 0,350 г."},{"name":"Действующее вещество","value":"Лаппаконитина гидробромид"},{"name":"Способ применения и дозы","value":"Прием препарата следует начинать под наблюдением врача.\u003Cbr\u003EВнутрь, после приема пищи, проглатывая таблетку целиком и запивая небольшим количеством воды комнатной температуры.\u003Cbr\u003EТаблетки категорически запрещается разламывать, измельчать или разжевывать!\u003Cbr\u003EДоза препарата Аллафорте подбирается индивидуально. Лечение следует начинать с назначения таблеток по 25 мг каждые 8 часов. При отсутствии или недостаточности терапевтического эффекта дозу следует увеличить - таблетки по 25 мг через каждые 6 часов или таблетки по 50 мг через каждые 12 часов. Судить о терапевтическом действии препарата при его первом применении или при увеличении его дозы следует не ранее, чем через 2-3 суток регулярного применения препарата.\u003Cbr\u003EДля предупреждения нежелательных влияний препарата на проводящую систему сердца его применение и увеличение дозы следует контролировать с помощью ЭКГ. Регистрировать ЭКГ целесообразно через 1-2 часа после приема очередной разовой дозы препарата. При удлинении интервала PQ до 300 мс или развитии предсердно-желудочковых блокад более высокой степени дозу следует уменьшить, при необходимости временно прекратив лечение. Безопасным является удлинение комплекса QRS на величину до 25 % от исходной, но при этом длительность QRS не должна превышать 140 мс. Недопустимо удлинение комплекса QRS свыше 50 % от исходного или более 160 мс!\u003Cbr\u003EМаксимальная суточная доза препарата составляет 100 мг (25 мг 4 раза в сутки или 50 мг 2 раза в сутки). В дозе более 100 мг в сутки препарат принимать не рекомендуется ввиду отсутствия контролируемых клинических исследований. Перевод пациентов, принимающих препарат Аллапинин, на лечение препаратом Аллафорте осуществляется путем простой замены, начиная с момента очередного приема одного препарата на другой с применением одинаковых доз и интервалов между приемами.\u003Cbr\u003EПродолжительность лечения и коррекция режима дозирования (увеличение дозы) определяется врачом."},{"name":"Побочные действия","value":"Оценка частоты возникновения побочных реакций произведена на основании следующих критериев: очень частые (≥ 1/10), частые (от ≥ 1/100 до \u003C 1/10), нечастые (от ≥ 1/1000 до \u003C 1/100), редкие (от ≥ 1/10 000 до \u003C 1/1000), очень редкие (\u003C 1/10 000), частота неизвестна (данные по оценке частоты отсутствуют).\u003Cbr\u003EНарушения со стороны центральной нервной системы\u003Cbr\u003Eочень часто: головокружение, головная боль, ощущение тяжести в голове, атаксия;\u003Cbr\u003EНарушения со стороны органа зрения\u003Cbr\u003Eочень часто: диплопия;\u003Cbr\u003EНарушения со стороны сердца\u003Cbr\u003Eочень часто: нарушения внутрижелудочковой и AV проводимости; изменения на ЭКГ: удлинение интервала PQ, расширение комплекса QRS;\u003Cbr\u003Eчасто: синусовая тахикардия (при длительном применении), повышение АД; нечасто: аритмогенное действие;\u003Cbr\u003EНарушения со стороны кожи и подкожных тканей\u003Cbr\u003Eчасто: аллергические реакции, гиперемия кожных покровов;\u003Cbr\u003EЛабораторные и инструментальные данные\u003Cbr\u003EОчень часто: изменения на ЭКГ: удлинение интервала PQ, расширение комплекса QRS."},{"name":"Фармакологическое действие","value":"Антиаритмический препарат IC класса. Действующее вещество препарата представляет собой бромистоводородную соль алкалоида лаппаконитина с сопутствующими алкалоидами, получаемую из травы борца белоустого или из корневищ и корней борца белоустого - Aconitum leucostomum Worosch., или из корневищ с корнями борца северного (борца высокого) - Aconitum septentrionale Koelle (A. excelsum Reichenb.), семейства лютиковые - Ranunculaceae, или из технической суммы алкалоидов семейства лютиковых.\u003Cbr\u003EФармакодинамика\u003Cbr\u003EВ основе механизма антиаритмического действия лежит блокировка «быстрых» натриевых каналов мембран кардиомиоцитов. Лаппаконитина гидробромид вызывает замедление атриовентрикулярной (AV) и внутрижелудочковой проводимости, угнетает проведение по дополнительным путям при синдроме Вольфа-Паркинсона-Уайта, укорачивает эффективный и функциональный рефрактерные периоды предсердий, AV узла, пучка Гиса и волокон Пуркинье. Не влияет на продолжительность интервала QT, проводимость по AV узлу в антероградном направлении, частоту сердечных сокращений (ЧСС) и артериальное давление (АД), сократимость миокарда (при исходном отсутствии явлений сердечной недостаточности). Не угнетает автоматизм синусового узла, не оказывает отрицательного инотропного действия, не обладает антигипертензивным и м-холинолитическим действием. Лаппаконитина гидробромид оказывает умеренное спазмолитическое, коронарорасширяющее, местноанестезирующее и седативное действие.\u003Cbr\u003EПри приеме внутрь эффект развивается через 40-60 минут, сохраняется на достигнутом уровне 4-5 часов и постепенно снижается. В целом действие препарата после однократного приема внутрь сохраняется не менее 12 часов."},{"name":"Фармакологическая группа","value":"антиаритмические средства"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В защищенном от света месте, при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Сравнительно небольшая терапевтическая широта препарата может способствовать интоксикации, особенно при сочетании с другими антиаритмическими средствами.\u003Cbr\u003EСимптомы: удлинение интервала PQ и QT, расширение комплекса QRS, увеличение амплитуды зубца Т, брадикардия, синоатриальная и атриовентрикулярная блокада, асистолия, пароксизмы полиморфной желудочковой тахикардии, снижение сократимости миокарда, выраженное снижение АД, головокружение, затуманенность зрения, головная боль, желудочно-кишечные расстройства.\u003Cbr\u003EЛечение: симптоматическое, промывание желудка, дефибрилляция, введение добутамина, диазепама; при необходимости - искусственная вентиляция легких и непрямой массаж сердца.\u003Cbr\u003EДля лечения желудочковой тахикардии не применять антиаритмические средства IA и IC класса."},{"name":"Применение при беременности и кормлении грудью","value":"Беременность\u003Cbr\u003EПрименение препарата при беременности не рекомендуется ввиду отсутствия контролируемых исследований.\u003Cbr\u003EПо данным доклинических исследований лаппаконитина гидробромид в дозах 1 -5 мг/кг не обладает тератогенным и эмбриотоксическим действием.\u003Cbr\u003EПрименение препарата при беременности возможно только по жизненным показаниям, если предполагаемая польза для матери превышает потенциальный риск развития побочных эффектов у плода/ребенка.\u003Cbr\u003EПериод грудного вскармливания\u003Cbr\u003EДанные о выделении лаппаконитина гидробромида в грудное молоко отсутствуют. Применение препарата не рекомендуется в период грудного вскармливания.\u003Cbr\u003EЕсли применение препарата Аллафорте в период лактации необходимо, грудное вскармливание следует прекратить."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"При применении препарата необходимо соблюдать осторожность при управлении транспортными средствами и занятии другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций в связи с риском развития головокружения."},{"name":"Особые указания","value":"С осторожностью:\u003Cbr\u003E\nПрименять пациентам с электрокардиостимулятором, при AV блокаде I степени, хронической сердечной недостаточности I-II функционального класса по классификации NYHA, нарушении внутрижелудочковой проводимости, синдроме слабости синусового узла (СССУ), брадикардии, тяжелых нарушениях периферического кровообращения, закрытоугольной глаукоме, доброкачественной гипертрофии предстательной железы, нарушении проводимости по волокнам Пуркинье, блокаде одной из ножек пучка Гиса, нарушении водно-электролитного обмена (гипокалиемия, гиперкалиемия, гипомагниемия), при одновременном приеме других антиаритмических средств.\u003Cbr\u003EОсобые указания:\u003Cbr\u003EПрепарат применяют по назначению врача.\u003Cbr\u003EПеред началом применения препарата необходимо устранить нарушения водно-электролитного обмена, в период терапии необходим контроль водно¬электролитного баланса крови.\u003Cbr\u003EКаждый пациент, который принимает препарат, должен проходить электрокардиографическое и клиническое обследование до начала терапии и в период ее проведения для раннего выявления побочного действия, оценки эффективности препарата и необходимости продолжения терапии.\u003Cbr\u003EУ пациентов с установленным электрокардиостимулятором может повышаться порог стимуляции. Электрокардиостимуляторы необходимо проверять и при необходимости перепрограммировать.\u003Cbr\u003EПри развитии головной боли, головокружения, диплопии следует уменьшить дозу препарата.\u003Cbr\u003EПри появлении синусовой тахикардии на фоне длительного применения препарата показано применение бета-адреноблокаторов (в индивидуально подобранных дозах).\u003Cbr\u003EПри применении антиаритмических средств IC класса у пациентов с тяжелыми органическими изменениями миокарда могут возникать серьезные нежелательные реакции. Применение препарата у таких пациентов возможно только после тщательной оценки ожидаемой пользы и возможного риска для пациентов, и должно осуществляться под наблюдением врача-кардиолога, имеющего опыт лечения соответствующих нарушений сердечного ритма.\u003Cbr\u003EС особой осторожностью следует применять препарат у пациентов с ишемической болезнью сердца и стабильной стенокардией напряжения, поскольку одним из предрасполагающих факторов аритмогенного действия антиаритмических препаратов IC класса является преходящая ишемия миокарда и высокая ЧСС. Препарат следует с осторожностью применять совместно с другими антиаритмическими препаратами в связи с повышенным риском аритмогенного действия.\u003Cbr\u003EУстановлено неблагоприятное влияние других антиаритмических препаратов IC класса на электрофизиологические показатели и клинические проявления при синдроме Бругада. Опыт применения лаппаконитина гидробромида при синдроме Бругада отсутствует, в связи с чем применение препарата у пациентов с синдромом Бругада противопоказано.\u003Cbr\u003EПрепарат предназначен для длительной профилактической антиаритмической терапии. Имеющийся ограниченный клинический опыт не позволяет рекомендовать применение препарата внутрь для купирования пароксизмов наджелудочковой и желудочковой тахикардии.\u003Cbr\u003EВлияние терапии лаппаконитина гидробромидом на выживаемость или частоту внезапной смерти пациентов с желудочковыми нарушениями сердечного ритма не изучалось в клинических исследованиях.\u003Cbr\u003EВспомогательные вещества\u003Cbr\u003EПрепарат Аллафорте содержит лактозы моногидрат. Пациентам с редко встречающимися наследственными заболеваниями, такими как непереносимость галактозы, непереносимость лактозы вследствие дефицита лактазы или синдром галактозной мальабсорбции, не следует принимать данный лекарственный препарат."},{"name":"Взаимодействие","value":"-при одновременном применении лаппаконитина гидробромида с другими антиаритмическими средствами повышается риск развития аритмогенного действия;\u003Cbr\u003E-лаппаконитина гидробромид усиливает эффект недеполяризующих миорелаксантов;\u003Cbr\u003E-при одновременном применении лаппаконитина гидробромида с другими антиаритмическими средствами повышается риск развития побочных эффектов, связанных с влиянием на функцию синусового узла и предсердно-желудочковую проводимость; требуется индивидуальный подбор доз каждого из этих препаратов;\u003Cbr\u003E-в клиническом исследовании при применении лаппаконитина гидробромида на фоне стандартной гипотензивной терапии ингибиторами ангиотензинпреврагцающего фермента, антагонистами рецепторов к ангиотензину ii, блокаторами «медленных» кальциевых каналов производных дигидропиридина, бета-адреноблокаторами не наблюдалось усиления или ослабления антигипертензивного действия;\u003Cbr\u003E-индукторы микросомальных ферментов печени не влияют на эффективность лаппаконитина гидробромида;\u003Cbr\u003E-не имеется данных о неблагоприятном влиянии лаппаконитина гидробромида на эффективность и безопасность непрямых антикоагулянтов."},{"name":"Регистрационный номер","value":"ЛП-004040"},{"name":"Дата государственной регистрации","value":"26.09.2022"},{"name":"Владелец регистрационного удостоверения","value":"Фармцентр Вилар"},{"name":"Изготовитель","value":"Фармцентр Вилар"},{"name":"Фасовщик","value":"Фармцентр Вилар"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Аллафорте"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_14916588632605838069"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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562 ₽

Скидка: 15%
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Вместо:663 ₽
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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
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  • Рейтинг товара: 4.9 из 5
    на основе 174 оценки
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  • Рейтинг товара: 4.5 из 5
    на основе 8 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 43 оценки
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-yqtz316zrn/addToCartButton":{"offerId":"g676gn9fZPrM0qt0OrFDeg","skuId":"186530622","pendingCartItem":{"productId":1401075876,"offerId":"g676gn9fZPrM0qt0OrFDeg","showPlaceId":"OTNDnItfwRMjN9MRHuEMMnA_dhOybheybDZX1vfuIh9JLvJ0wS9aMXmmwFuq92Jyx_nHADk8vvmzgDhr8g85VRsgX9zAwHU7W6XYahdmdJ-BDDrQSHYUL7Mhk4sYpvEKsQ7r_7eAvvK08wD0t3O5DnG6plolbBA-05jlmyeiuCXb-HJ9aeZBAAotnQ2QFFF_7h775Xf_8xVZ0l1E9T79BQ,,","feeShow":"OTNDnItfwRMjN9MRHuEMMnA_dhOybheybDZX1vfuIh9JLvJ0wS9aMXmmwFuq92Jyx_nHADk8vvmzgDhr8g85VRsgX9zAwHU7W6XYahdmdJ-BDDrQSHYUL7Mhk4sYpvEKsQ7r_7eAvvK08wD0t3O5DnG6plolbBA-05jlmyeiuCXb-HJ9aeZBAAotnQ2QFFF_7h775Xf_8xVZ0l1E9T79BQ,,","skuId":"186530622","shopId":55106433,"price":{"applicablePriceDiscounts":[],"discount":{"oldMin":"181","percent":12},"value":"159","currency":"RUR"},"hid":"15756887","name":"Беталок Зок таб. с замедл. высвоб. п/о, 25 мг, 14 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  • Рейтинг товара: 4.9 из 5
    на основе 12 оценок
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  • Рейтинг товара: 5 из 5
    на основе 6 оценок
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-pco7potb43c/addToCartButton":{"offerId":"82VwWWQcFaPK7O7D__NvBA","skuId":"228042234","pendingCartItem":{"productId":1401075599,"offerId":"82VwWWQcFaPK7O7D__NvBA","showPlaceId":"OTNDnItfwRMjN9MRHuEMMnA_dhOybheyRz0cx3O5-MMyyb_mRewUU6kBcto3ZeRlMXzNHSNCPbHc7fYGZ8XCoLpbjF5Dq4tR2Uskz45uik2AuSVyOBlD-FdjDsCkdJJL21hreePJWYp8busTuFWsrYgRwvF-Dfr6FnESMjOxS-SQ-QWcZzF248RCR4ronR8B62OaDftGEz3ZGSPgo8Frug,,","feeShow":"OTNDnItfwRMjN9MRHuEMMnA_dhOybheyRz0cx3O5-MMyyb_mRewUU6kBcto3ZeRlMXzNHSNCPbHc7fYGZ8XCoLpbjF5Dq4tR2Uskz45uik2AuSVyOBlD-FdjDsCkdJJL21hreePJWYp8busTuFWsrYgRwvF-Dfr6FnESMjOxS-SQ-QWcZzF248RCR4ronR8B62OaDftGEz3ZGSPgo8Frug,,","skuId":"228042234","shopId":55106433,"price":{"applicablePriceDiscounts":[],"value":"55","currency":"RUR"},"hid":"15756887","name":"Верапамил таб. п/о плен., 40 мг, 30 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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-9t5sp83ezd/addToCartButton":{"offerId":"ZlskALOwnoYz8rGfq5Alag","skuId":"186481406","pendingCartItem":{"productId":1778173749,"offerId":"ZlskALOwnoYz8rGfq5Alag","showPlaceId":"OTNDnItfwRMjN9MRHuEMMnA_dhOybheyk--Y27pUzQDbDX8ShoCTTr9hXEceuxSXBxRSD6pVsi8N5pbSyg_iMqSNyod_uPgGVN8Ca_NCigV2jtAk2MH2aiPK_WGGaXiFkz-aueNfEjYLt54GyDy6eQbg6px5LqqX4j3NaO9Sb1rN6IPTprZzIx6Jej6NvYd8ud-ZfcR8vKzKzr7E_FhghQ,,","feeShow":"OTNDnItfwRMjN9MRHuEMMnA_dhOybheyk--Y27pUzQDbDX8ShoCTTr9hXEceuxSXBxRSD6pVsi8N5pbSyg_iMqSNyod_uPgGVN8Ca_NCigV2jtAk2MH2aiPK_WGGaXiFkz-aueNfEjYLt54GyDy6eQbg6px5LqqX4j3NaO9Sb1rN6IPTprZzIx6Jej6NvYd8ud-ZfcR8vKzKzr7E_FhghQ,,","skuId":"186481406","shopId":55106433,"price":{"applicablePriceDiscounts":[],"value":"783","currency":"RUR"},"hid":"15756887","name":"Предизин таб. таб. пролонг. действ., 35 мг, 60 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  • Рейтинг товара: 5 из 5
    на основе 10 оценок
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Инструкция

Показания к применению

-наджелудочковая и желудочковая экстрасистолия;
-пароксизмальная форма фибрилляции и трепетания предсердий;
-пароксизмальная наджелудочковая тахикардия, в том числе и при синдроме Вольфа-Паркинсона-Уайта (WPW);
-пароксизмальная желудочковая тахикардия (при отсутствии органических изменений миокарда).

Противопоказания

-повышенная чувствительность к лаппаконитина гидробромиду или к любому другому компоненту препарата;
-синоатриальная блокада;
-AV блокада II и III степени (без электрокардиостимулятора);
-кардиогенный шок;
-блокада правой ножки пучка Гиса, сочетающаяся с блокадой одной из ветвей левой ножки;
-тяжелая артериальная гипотензия (систолическое АД менее 90 мм рт;ст;);
-хроническая сердечная недостаточность III-IV функционального класса по классификации NYHA;
-выраженная гипертрофия миокарда левого желудочка (≥1,4 см);
-постинфарктный кардиосклероз;
-синдром Бругада;
-острый инфаркт миокарда;
-тяжелые нарушения функции печени и/или почек;
-непереносимость лактозы;
-беременность и период грудного вскармливания;

Способ применения и дозы

Прием препарата следует начинать под наблюдением врача.
Внутрь, после приема пищи, проглатывая таблетку целиком и запивая небольшим количеством воды комнатной температуры.
Таблетки категорически запрещается разламывать, измельчать или разжевывать!
Доза препарата Аллафорте подбирается индивидуально. Лечение следует начинать с назначения таблеток по 25 мг каждые 8 часов. При отсутствии или недостаточности терапевтического эффекта дозу следует увеличить - таблетки по 25 мг через каждые 6 часов или таблетки по 50 мг через каждые 12 часов. Судить о терапевтическом действии препарата при его первом применении или при увеличении его дозы следует не ранее, чем через 2-3 суток регулярного применения препарата.
Для предупреждения нежелательных влияний препарата на проводящую систему сердца его применение и увеличение дозы следует контролировать с помощью ЭКГ. Регистрировать ЭКГ целесообразно через 1-2 часа после приема очередной разовой дозы препарата. При удлинении интервала PQ до 300 мс или развитии предсердно-желудочковых блокад более высокой степени дозу следует уменьшить, при необходимости временно прекратив лечение. Безопасным является удлинение комплекса QRS на величину до 25 % от исходной, но при этом длительность QRS не должна превышать 140 мс. Недопустимо удлинение комплекса QRS свыше 50 % от исходного или более 160 мс!
Максимальная суточная доза препарата составляет 100 мг (25 мг 4 раза в сутки или 50 мг 2 раза в сутки). В дозе более 100 мг в сутки препарат принимать не рекомендуется ввиду отсутствия контролируемых клинических исследований. Перевод пациентов, принимающих препарат Аллапинин, на лечение препаратом Аллафорте осуществляется путем простой замены, начиная с момента очередного приема одного препарата на другой с применением одинаковых доз и интервалов между приемами.
Продолжительность лечения и коррекция режима дозирования (увеличение дозы) определяется врачом.
Полная инструкция
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Аллафорте таб. пролонг. действ.
Аллафорте таб. пролонг. действ., 25 мг, 20 шт.
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Инструкция

562 ₽

Скидка: 15%
–15 %
Вместо:663 ₽
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5.0
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