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Описание

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Кофеин-бензоат натрия р-р для п/к введ. амп., 200 мг/мл, 1 мл, 10 шт.

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Коротко о товаре

Артикул Маркета
4453167417
Действующее вещество
Возраст
от 18 лет
Инструкция
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Высшая разовая доза - 0,4 г, высшая суточная доза - 1 г."},{"name":"Побочные действия","value":"Со стороны нервной системы: возбуждение, тревожность, тремор, беспокойство, головная боль, головокружение, эпилептические припадки, усиление рефлексов, тахипноэ, бессонница; при внезапной отмене - усиление торможения центральной нервной системы, повышенная утомляемость, сонливость, мышечное напряжение.\u003Cbr\u003EСо стороны сердечно-сосудистой системы: сердцебиение, тахикардия, аритмия, повышение артериального давления.\u003Cbr\u003EСо стороны пищеварительной системы: тошнота, рвота, обострение язвенной болезни. \u003Cbr\u003EПрочие: заложенность носа, при длительном применении - привыкание, лекарственная зависимость."},{"name":"Фармакологическое действие","value":"Кофеин - метилксантин. оказывающий психостимулирующий и аналептический эффект. Конкурентно блокирует центральные и периферические А1 и А2 аденозиновые рецепторы. Тормозит активность фосфодиэстеразы в центральной нервной системе, сердце, гладкомышечных органах, скелетных мышцах, жировой ткани, способствует накоплению в них циклического аденозинмонофосфата и циклического гуанозинмонофосфата (данный эффект наблюдается при применении только высоких доз кофеина). Стимулирует центры продолговатого мозга (дыхательный и сосудодвигательный), а также центр n.vagus, оказывает прямое возбуждающее влияние на кору головною мозга. В высоких дозах облегчает межнейрональную проводимость в спинном мозге, усиливая спинномозговые рефлексы. Повышает умственную и физическую работоспособность, стимулирует психическую деятельность, двигательную активность, укорачивает время реакций, временно уменьшает утомление и сонливость. В мачых дозах преобладает эффект стимуляции, а в больших -эффект угнетения нервной системы. Учащает и углубляет дыхание, обычно оказывает положительный ино-, хроно-, батмо- и дромотропный эффект (поскольку влияние на сердечно-сосудистую систему складывается из прямого стимулирующего действия на миокард и одновременного возбуждающего влияния на центры п. vagus, результирующий эффект зависит от преобладания того или иного действия). Стимулирует сосудодвигательный центр и оказывает непосредственное релаксирующее действие на сосудистую стенку, что приводит к расширению сосудов сердца, скелетных мышц и ночек, при этом тонус церебральных артерий повышается (вызывает сужение сосудов головного мозга, что сопровождается снижением мозгового кровотока и давления кислорода в головном мозге). Артериальное давление изменяется под действием сосудистых и сердечных механизмов влияния кофеина: при нормальном исходном артериальном давлении кофеин не изменяет или слегка повышает его, при артериальной гипотензии нормализует его.\u003Cbr\u003EОказывает спазмолитическое действие на гладкую мускулатуру (в т.ч. бронходилатирующий эффект), на поперечнополосатую - стимулирующее. Повышает секреторную активность желудка и диурез (снижение реабсорбции ионов натрия и воды в проксимальных и дистальных почечных канальцах, а также расширение сосудов почек и увеличение фильтрации в почечных клубочках).\u003Cbr\u003EСнижает агрегацию тромбоцитов и высвобождение гистамина из тучных клеток.\u003Cbr\u003EПовышает основной обмен: увеличивает гликогенолиз, повышает липолиз."},{"name":"Фармакологическая группа","value":"психостимуляторы"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-nervnoi-sistemy","categoryId":"15756525","navnodeId":"72478","glfilters":["35947170:36763748"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"При температуре не выше 25 °C.Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: гастралгия, ажитация, тревожность, возбуждение, двигательное беспокойство, спутанность сознания, делирий, обезвоживание, тахикардия, аритмия, гипертермия, учащенное мочеиспускание, головная боль, повышенная тактильная или болевая чувствительность, тремор или мышечные подергивания; тошнота и рвота, иногда с кровыо; звон в ушах, эпилептические припадки (при острой передозировке - тонико-клонические). Кофеин в дозах более 300 мг/сут (в т.ч. на фоне злоупотребления кофе - более 4 чашек натурального кофе по 150 мл) может вызывать состояние тревоги, тремор, головную боль, спутанность сознания, экстрасистолию.\u003Cbr\u003EЛечение: симптоматическая терапия, поддержание вентиляции легких и оксигенации, при эпилептических припадках - внутривенно диазепам, фенобарбитал или фенитоин, поддержание баланса жидкости и солей, гемодиализ."},{"name":"Применение при беременности и кормлении грудью","value":"Применение во время беременности противопоказано. При необходимости применения препарата в период лактации на время лечения следует прекратить грудное вскармливание."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Препарат не следует применять во время работы водителям транспортных средств и людям, профессия которых требует повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"С осторожностью: Глаукома, повышенная возбудимость, пожилой возраст, эпилепсия и склонность к судорожным припадкам.\u003Cbr\u003EСледует иметь в виду, что внезапное прекращение приема может приводить к усилению торможения центральной нервной системы (сонливость, депрессия).\u003Cbr\u003EВлияние на центральную нервную систему зависит от типа нервной системы и может проявляться как возбуждением, так и торможением высшей нервной деятельности. В связи с тем, что действие кофеина на артериальное давление складывается из сосудистого и кардиального компонентов, в результате может развиваться как эффект стимуляции сердца, так и угнетение (слабое) его деятельности."},{"name":"Взаимодействие","value":"Кофеин является антагонистом аденозина (могут потребоваться большие дозы аденозина). При совместном применении кофеина и барбитуратов, примидона, противосудорожных лекарственных средств (производные гидантоина, особенно фенитоин) возможно усиление метаболизма и увеличение клиренса кофеина; циметидина, пероральных контрацептивных лекарственных средств, дисульфирама, ципрофлоксацина, норфлоксацина - снижение метаболизма кофеина в печени (замедление его выведения и увеличение концентрации в крови).\u003Cbr\u003EКофеинсодержащие напитки и др. лекарственные средства, стимулирующие центральную нервную систему - возможна чрезмерная стимуляция центральной нервной системы.\u003Cbr\u003EМексилетин - снижает выведение кофеина до 50 %; никотин - увеличивает скорость выведения кофеина.\u003Cbr\u003EИнгибиторы моноаминоксидазы, фуразолидон, прокарбазин и селегилин - большие дозы кофеина могут вызывать развитие опасных аритмий сердца или выраженного повышения артериального давления.\u003Cbr\u003EКофеин снижает всасывание препаратов кальция в желудочно-кишечном тракте.\u003Cbr\u003EСнижает эффект наркотических и снотворных лекарственных средств. Увеличивает выведение препаратов лития с мочой.\u003Cbr\u003EУскоряет всасывание и усиливает действие сердечных гликозидов, повышает их токсичность.\u003Cbr\u003EСовместное применение кофеина с бета-адреноблокаторами может приводить к взаимному подавлению терапевтических эффектов; с адренергическими бронхорасширяющими лекарственными средствами - к дополнительной стимуляции центральной нервной системы и др. аддитивным токсическим эффектам.\u003Cbr\u003EКофеин может снижать клиренс теофиллина и. возможно, др. ксантинов, увеличивая возможность аддитивных фармакодинамических и токсических эффектов."},{"name":"Регистрационный номер","value":"П N010971"},{"name":"Дата государственной регистрации","value":"29.03.2019"},{"name":"Владелец регистрационного удостоверения","value":"Борисовский завод медицинских препаратов","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-nervnoi-sistemy","categoryId":"15756525","navnodeId":"72478","glfilters":["34324371:35649313","7893318:14945147"]}}},{"name":"Изготовитель","value":"Борисовский завод медицинских препаратов"},{"name":"Фасовщик","value":"Борисовский завод медицинских препаратов"},{"name":"Страна бренда","value":"Беларусь"},{"name":"Страна-производитель","value":"Беларусь"},{"name":"Название препарата","value":"Кофеин-бензоат натрия","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-nervnoi-sistemy","categoryId":"15756525","navnodeId":"72478","glfilters":["17796364:18028590"]}}},{"name":"Срок годности","value":"60 мес."}]}},"fullSpecsGrouped":{"16636777798738980134":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"нервная система"},{"name":"Назначение","value":"артериальная гипертензия, повышение работоспособности, угнетение дыхания"},{"name":"Показания к применению","value":"Снижение умственной и физической работоспособности, сонливость, головная боль сосудистого генеза (в т.ч. мигрень), умеренная артериальная гипотензия, угнетение дыхания (в т.ч. при легких отравлениях наркотическими анальгетиками и снотворными лекарственными препаратами, оксидом углерода), восстановление легочной вентиляции после использования общей анестезии."},{"name":"Противопоказания","value":"Гиперчувствительность (в т.ч. к др. ксантинам), тревожные расстройства (агорафобия, панические расстройства), органические заболевания сердечно-сосудистой системы (в т.ч. острый инфаркт миокарда, атеросклероз), пароксизмальная тахикардия, частая желудочковая экстрасистолия, артериальная гипертензия, нарушения сна, детский возраст до 18 лет, беременность и период лактации."},{"name":"Состав","value":"Одна ампула содержит: действующие вещества: кофеин - 80 мг, натрия бензоат -120 мг; вспомогательные вещества: 0,1 М раствор натрия гидроксида, вода для инъекций."},{"name":"Действующее вещество","value":"Кофеин"},{"name":"Способ применения и дозы","value":"Подкожно взрослым по 1 мл раствора (100-200 мг). Высшая разовая доза - 0,4 г, высшая суточная доза - 1 г."},{"name":"Побочные действия","value":"Со стороны нервной системы: возбуждение, тревожность, тремор, беспокойство, головная боль, головокружение, эпилептические припадки, усиление рефлексов, тахипноэ, бессонница; при внезапной отмене - усиление торможения центральной нервной системы, повышенная утомляемость, сонливость, мышечное напряжение.\u003Cbr\u003EСо стороны сердечно-сосудистой системы: сердцебиение, тахикардия, аритмия, повышение артериального давления.\u003Cbr\u003EСо стороны пищеварительной системы: тошнота, рвота, обострение язвенной болезни. \u003Cbr\u003EПрочие: заложенность носа, при длительном применении - привыкание, лекарственная зависимость."},{"name":"Фармакологическое действие","value":"Кофеин - метилксантин. оказывающий психостимулирующий и аналептический эффект. Конкурентно блокирует центральные и периферические А1 и А2 аденозиновые рецепторы. Тормозит активность фосфодиэстеразы в центральной нервной системе, сердце, гладкомышечных органах, скелетных мышцах, жировой ткани, способствует накоплению в них циклического аденозинмонофосфата и циклического гуанозинмонофосфата (данный эффект наблюдается при применении только высоких доз кофеина). Стимулирует центры продолговатого мозга (дыхательный и сосудодвигательный), а также центр n.vagus, оказывает прямое возбуждающее влияние на кору головною мозга. В высоких дозах облегчает межнейрональную проводимость в спинном мозге, усиливая спинномозговые рефлексы. Повышает умственную и физическую работоспособность, стимулирует психическую деятельность, двигательную активность, укорачивает время реакций, временно уменьшает утомление и сонливость. В мачых дозах преобладает эффект стимуляции, а в больших -эффект угнетения нервной системы. Учащает и углубляет дыхание, обычно оказывает положительный ино-, хроно-, батмо- и дромотропный эффект (поскольку влияние на сердечно-сосудистую систему складывается из прямого стимулирующего действия на миокард и одновременного возбуждающего влияния на центры п. vagus, результирующий эффект зависит от преобладания того или иного действия). Стимулирует сосудодвигательный центр и оказывает непосредственное релаксирующее действие на сосудистую стенку, что приводит к расширению сосудов сердца, скелетных мышц и ночек, при этом тонус церебральных артерий повышается (вызывает сужение сосудов головного мозга, что сопровождается снижением мозгового кровотока и давления кислорода в головном мозге). Артериальное давление изменяется под действием сосудистых и сердечных механизмов влияния кофеина: при нормальном исходном артериальном давлении кофеин не изменяет или слегка повышает его, при артериальной гипотензии нормализует его.\u003Cbr\u003EОказывает спазмолитическое действие на гладкую мускулатуру (в т.ч. бронходилатирующий эффект), на поперечнополосатую - стимулирующее. Повышает секреторную активность желудка и диурез (снижение реабсорбции ионов натрия и воды в проксимальных и дистальных почечных канальцах, а также расширение сосудов почек и увеличение фильтрации в почечных клубочках).\u003Cbr\u003EСнижает агрегацию тромбоцитов и высвобождение гистамина из тучных клеток.\u003Cbr\u003EПовышает основной обмен: увеличивает гликогенолиз, повышает липолиз."},{"name":"Фармакологическая группа","value":"психостимуляторы"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"При температуре не выше 25 °C.Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: гастралгия, ажитация, тревожность, возбуждение, двигательное беспокойство, спутанность сознания, делирий, обезвоживание, тахикардия, аритмия, гипертермия, учащенное мочеиспускание, головная боль, повышенная тактильная или болевая чувствительность, тремор или мышечные подергивания; тошнота и рвота, иногда с кровыо; звон в ушах, эпилептические припадки (при острой передозировке - тонико-клонические). Кофеин в дозах более 300 мг/сут (в т.ч. на фоне злоупотребления кофе - более 4 чашек натурального кофе по 150 мл) может вызывать состояние тревоги, тремор, головную боль, спутанность сознания, экстрасистолию.\u003Cbr\u003EЛечение: симптоматическая терапия, поддержание вентиляции легких и оксигенации, при эпилептических припадках - внутривенно диазепам, фенобарбитал или фенитоин, поддержание баланса жидкости и солей, гемодиализ."},{"name":"Применение при беременности и кормлении грудью","value":"Применение во время беременности противопоказано. При необходимости применения препарата в период лактации на время лечения следует прекратить грудное вскармливание."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Препарат не следует применять во время работы водителям транспортных средств и людям, профессия которых требует повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"С осторожностью: Глаукома, повышенная возбудимость, пожилой возраст, эпилепсия и склонность к судорожным припадкам.\u003Cbr\u003EСледует иметь в виду, что внезапное прекращение приема может приводить к усилению торможения центральной нервной системы (сонливость, депрессия).\u003Cbr\u003EВлияние на центральную нервную систему зависит от типа нервной системы и может проявляться как возбуждением, так и торможением высшей нервной деятельности. В связи с тем, что действие кофеина на артериальное давление складывается из сосудистого и кардиального компонентов, в результате может развиваться как эффект стимуляции сердца, так и угнетение (слабое) его деятельности."},{"name":"Взаимодействие","value":"Кофеин является антагонистом аденозина (могут потребоваться большие дозы аденозина). При совместном применении кофеина и барбитуратов, примидона, противосудорожных лекарственных средств (производные гидантоина, особенно фенитоин) возможно усиление метаболизма и увеличение клиренса кофеина; циметидина, пероральных контрацептивных лекарственных средств, дисульфирама, ципрофлоксацина, норфлоксацина - снижение метаболизма кофеина в печени (замедление его выведения и увеличение концентрации в крови).\u003Cbr\u003EКофеинсодержащие напитки и др. лекарственные средства, стимулирующие центральную нервную систему - возможна чрезмерная стимуляция центральной нервной системы.\u003Cbr\u003EМексилетин - снижает выведение кофеина до 50 %; никотин - увеличивает скорость выведения кофеина.\u003Cbr\u003EИнгибиторы моноаминоксидазы, фуразолидон, прокарбазин и селегилин - большие дозы кофеина могут вызывать развитие опасных аритмий сердца или выраженного повышения артериального давления.\u003Cbr\u003EКофеин снижает всасывание препаратов кальция в желудочно-кишечном тракте.\u003Cbr\u003EСнижает эффект наркотических и снотворных лекарственных средств. Увеличивает выведение препаратов лития с мочой.\u003Cbr\u003EУскоряет всасывание и усиливает действие сердечных гликозидов, повышает их токсичность.\u003Cbr\u003EСовместное применение кофеина с бета-адреноблокаторами может приводить к взаимному подавлению терапевтических эффектов; с адренергическими бронхорасширяющими лекарственными средствами - к дополнительной стимуляции центральной нервной системы и др. аддитивным токсическим эффектам.\u003Cbr\u003EКофеин может снижать клиренс теофиллина и. возможно, др. ксантинов, увеличивая возможность аддитивных фармакодинамических и токсических эффектов."},{"name":"Регистрационный номер","value":"П N010971"},{"name":"Дата государственной регистрации","value":"29.03.2019"},{"name":"Владелец регистрационного удостоверения","value":"Борисовский завод медицинских препаратов"},{"name":"Изготовитель","value":"Борисовский завод медицинских препаратов"},{"name":"Фасовщик","value":"Борисовский завод медицинских препаратов"},{"name":"Страна бренда","value":"Беларусь"},{"name":"Страна-производитель","value":"Беларусь"},{"name":"Название препарата","value":"Кофеин-бензоат натрия"},{"name":"Срок годности","value":"60 мес."}]}],"transitionId":"tr_9170507888457463148"}}}}
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Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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Инструкция

Показания к применению

Снижение умственной и физической работоспособности, сонливость, головная боль сосудистого генеза (в т.ч. мигрень), умеренная артериальная гипотензия, угнетение дыхания (в т.ч. при легких отравлениях наркотическими анальгетиками и снотворными лекарственными препаратами, оксидом углерода), восстановление легочной вентиляции после использования общей анестезии.

Противопоказания

Гиперчувствительность (в т.ч. к др. ксантинам), тревожные расстройства (агорафобия, панические расстройства), органические заболевания сердечно-сосудистой системы (в т.ч. острый инфаркт миокарда, атеросклероз), пароксизмальная тахикардия, частая желудочковая экстрасистолия, артериальная гипертензия, нарушения сна, детский возраст до 18 лет, беременность и период лактации.

Способ применения и дозы

Подкожно взрослым по 1 мл раствора (100-200 мг). Высшая разовая доза - 0,4 г, высшая суточная доза - 1 г.
Полная инструкция
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Кофеин-бензоат натрия р-р для п/к введ. амп.
Кофеин-бензоат натрия р-р для п/к введ. амп., 200 мг/мл, 1 мл, 10 шт.
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Инструкция

49 ₽

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5.0
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У продавца:11 оценок·3 отзыва
У всех продавцов:25 оценок·9 отзывов
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3 месяца назад • ВИКТОР ИЩЕНКО • Куплен на Маркете
Достоинства: отличное лекарство для поднятия давления!
Недостатки: нет
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5 месяцев назад • Юлия Кухарчук • Куплен на Маркете
Достоинства: Отлично
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7 месяцев назад • Алексей П. • Куплен на Маркете
Достоинства: эффективность
Недостатки: нет
Посмотреть все отзывы на Маркете
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