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Описание

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Гептор таб. п/о кш/раств., 400 мг, 20 шт.

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Количество штук в упаковке, шт.: 20

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системы","value":"желчный пузырь и желчевыводящие пути, печень","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-pishchevareniia","categoryId":"15756506","navnodeId":"72470","glfilters":["34045610:34516032,34516029"]}}},{"name":"Назначение","value":"внутрипеченочный холестаз, нарушение функции печени, острые гепатиты, печеночная энцефалопатия, синдром алкогольной абстиненции, токсические поражения печени, холангит, холецистит, хронические гепатиты, хронический алкогольный гепатит, цирроз печени","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-pishchevareniia","categoryId":"15756506","navnodeId":"72470","glfilters":["36476390:36618841,36618605,36618595,36618554,36618493,36618449,36617929,36617671,36617579,36617299,36617278"]}}},{"name":"Показания к применению","value":"Внутрипеченочный холестаз при прецирротических и цирротических состояниях, который может наблюдаться при следующих заболеваниях:\u003Cbr\u003E- жировая дистрофия печени;\u003Cbr\u003E- хронический гепатит;\u003Cbr\u003E- токсические поражения печени различной этиологии, включая алкогольные, вирусные, лекарственные (антибиотики, противоопухолевые, противотуберкулезные и противовирусные препараты, трициклические антидепрессанты, пероральные контрацептивы);\u003Cbr\u003E\n- хронический некалькулезный (бескаменный) холецистит;\u003Cbr\u003E- холангит;\u003Cbr\u003E- цирроз печени;\u003Cbr\u003E- энцефалопатия, в т.ч. ассоциированная с печеночной недостаточностью (алкогольная и др.);\u003Cbr\u003E- внутрипеченочный холестаз у беременных;\u003Cbr\u003E- симптомы депрессии."},{"name":"Противопоказания","value":"- Генетические нарушения, влияющие на метиониновый цикл и/или вызывающие гомоцистинурию и/или гипергомоцистеинемию (дефицит цистатион-бета-синтазы, нарушение метаболизма витамина В 12 (цианокобаламин));\u003Cbr\u003E- гиперчувствительность к любому из компонентов препарата;\u003Cbr\u003E- возраст до 18 лет (опыт медицинского применения у детей ограничен);\u003Cbr\u003E- биполярные расстройства.\u003Cbr\u003E"},{"name":"Состав","value":"Состав на одну таблетку\u003Cbr\u003E\nДействующее вещество: Адеметионина тозилата дисульфат в пересчет на адеметионин-ион - 400 мг.\u003Cbr\u003EВспомогательные вещества: Полипласдон Икс Эл-10 (кросповидон) - 19 мг, целлюлоза микрокристаллическая - 53 мг, маннитол (маннит) - 53 мг, магния стеарат - 15 мг, масса таблетки без оболочки - 950 мг.\u003Cbr\u003E\nСостав оболочки: Акрил-из желтый - 61.3 мг, [метакриловой кислоты и этилакрилата сополимер ( 1:1 ) - 24.52 мг, тальк - 22.83 мг, титана диоксид - 5.52 мг, кремния диоксид коллоидный (аэросил) - 0.77 мг, триэтилцитрат - 2.94 мг, натрия гидрокарбонат - 0.73 мг, натрия лаурилсульфат - 0.31 мг, железа оксид желтый - 1.84 мг, хинолиновый желтый алюминиевый лак] - 1.84 мг, гипромеллоза (Оксипропилметилцеллюлоза) - 21.0 мг, пласдон ЭС-630 (коповидон) - 9.0 мг, макрогол 6000 (Полиэтиленгликоль 6000) - 3.7 мг, масса таблетки с оболочкой - 1045 мг."},{"name":"Действующее вещество","value":"Адеметионин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-pishchevareniia","categoryId":"15756506","navnodeId":"72470","glfilters":["27144131:28710768"]}}},{"name":"Способ применения и дозы","value":"Способ применения и дозы:\u003Cbr\u003EВнутрь.\u003Cbr\u003EТаблетки следует принимать целиком, не разжевывая, желательно в первой половине дня между приемами пищи.\u003Cbr\u003EТаблетки препарата Гептор следует вынимать из блистера непосредственно перед приемом внутрь.\u003Cbr\u003EНачальная терапия:\u003Cbr\u003EРекомендуемая доза составляет 10-25 мг/кг/сут.\u003Cbr\u003EВнутрипеченочный холестаз\u003Cbr\u003EДоза составляет от 800 мг/сут до 1600 мг/сут.\u003Cbr\u003EДепрессия\u003Cbr\u003EДоза составляет от 800 мг/сут до 1600 мг/сут.\u003Cbr\u003EДлительность терапии определяется врачом.\u003Cbr\u003E\nТерапия препаратом Гептор может быть начата с внутривенного или внутримышечного введения с последующим применением препарата Гептор в виде таблеток или сразу с применения препарата Гептор в виде таблеток.\u003Cbr\u003EПациенты пожилого возраста\u003Cbr\u003EКлинический опыт применения препарата Гептор не выявил каких-либо различий в его эффективности у пациентов пожилого возраста и пациентов более молодого возраста. Однако, учитывая высокую вероятность имеющихся нарушений функции печени, почек или сердца, другой сопутствующей патологии или одновременной терапии с другими лекарственными средствами, дозу препарата Гептор пожилым пациентам следует подбирать с осторожностью, начиная применение препарата с нижнего предела диапазона доз.\u003Cbr\u003EПочечная недостаточность\u003Cbr\u003EИмеются ограниченные клинические данные о применении препарата Гептор у пациентов с почечной недостаточностью, в связи с этим рекомендуется соблюдать осторожность при применении препарата Гептор утаких пациентов.\u003Cbr\u003EПеченочная недостаточность\u003Cbr\u003EПараметры фармакокинетики адеметионина сходны у здоровых добровольцев и у пациентов с хроническими заболеваниями печени.\u003Cbr\u003EДети\u003Cbr\u003EПрименение препарата Гептор у детей противопоказано (эффективность и безопасность не установлены)."},{"name":"Побочные действия","value":"Побочное действие:\u003Cbr\u003EСо стороны пищеварительной системы: часто - тошнота, боли в животе, диарея; редко - рвота, сухость во рту, эзофагит, диспепсия, метеоризм, желудочно-кишечная боль, желудочно-кишечное кровотечение, печеночная колика.\u003Cbr\u003EСо стороны нервной системы: редко - спутанность сознания, бессонница, головокружение, головная боль, парестезии.\u003Cbr\u003EСо стороны костно-мышечной системы: редко - артралгии, мышечные судороги\u003Cbr\u003EСо стороны мочевыделительной системы: редко - инфекции мочевыводящих путей.\u003Cbr\u003EСо стороны кожных покровов: редко - гипергидроз, зуд, кожная сыпь.\u003Cbr\u003EМестные реакции: редко - реакции в месте введения; очень редко - реакции в месте введения, некроз кожи в месте введения.\u003Cbr\u003EАллергические реакции: редко - анафилактические реакции; очень редко - отек Квинке, отек гортани.\u003Cbr\u003EПрочие: редко - приливы, поверхностный флебит, астения, озноб, гриппоподобные симптомы, слабость, периферические отеки, гипертермия."},{"name":"Фармакологическое действие","value":"Гептор относится к группе гепатопротекторов с антидепрессивной активностью. Оказывает холеретическое и холекинетическое действие. Обладает дезинтоксикационным, регенерирующим, антиоксидантным, антифиброзирующим и нейропротективным действием.\u003Cbr\u003EВосполняет дефицит S-аденозил-L-метионина (адеметионина) и стимулирует его выработку в организме, содержится во всех средах организма. Наибольшая концентрация адеметионина отмечена в печени и мозге. Выполняет ключевую роль в метаболических процессах организма, принимает участие в важных биохимических реакциях: трансметилировании, транссульфурировании, трансаминировании. В реакциях трансметилирования адеметионин донирует метильную группу для синтеза фосфолипидов клеточных мембран, нейротрансмитгеров, нуклеиновых кислот, белков, гормонов и др. В реакциях транссульфурирования адеметионин является предшественником цистеина, таурина, глютатиона (обеспечивая окислительно-восстановительный механизм клеточной детоксикации), коэнзима А (включается в биохимические реакции цикла трикарбоновых кислот и восполняет энергетический потенциал клетки). Повышает содержание глутамина в печени, цистеина и таурина в плазме; снижает содержание метионина в сыворотке, нормализуя метаболические реакции в печени. После декарбоксилирования участвует в реакциях аминопропилирования, как предшественник полиаминов путресцина (стимулятор регенерации клеток и пролиферации гепатоцитов), спермидина и спермина, входящих в структуру рибосом, что уменьшает риск фиброзирования. Оказывает холеретическое действие. Адеметионин нормализует синтез эндогенного фосфатидилхолина в гепатоцитах, что повышает текучесть и поляризацию мембран. Это улучшает функцию ассоциированных с мембранами гепатоцитов транспортных систем желчных кислот и способствует пассажу желчных кислот в желчевыводящие пути. Эффективен при внутридольковом варианте холестаза (нарушение синтеза и тока желчи). Адеметионин снижает токсичность желчных кислот в гепатоците, осуществляя их конъюгирование и сульфатирование. Конъюгация с таурином повышает растворимость желчных кислот и выведение их из гепатоцита. Процесс сульфатирования желчных кислот способствует возможности их элиминации почками, облегчает прохождение через мембрану гепатоцита и выведение с желчью. Кроме этого, сами сульфатированные желчные кислоты дополнительно защищают мембраны клеток печени от токсического действия несульфатированных желчных кислот (в высоких концентрациях присутствующих в гепатоцитах при внутрипеченочном холестазе). У пациентов с диффузными заболеваниями печени (цирроз, гепатит) с синдромом внутрипеченочного холестаза адеметионин снижает выраженность кожного зуда и изменений биохимических показателей, в т.ч. концентрации прямого билирубина, активности щелочной фосфатазы, аминотрансфераз и др. Холеретический и гепатопротективный эффект сохраняется до З месяцев после прекращения лечения. Показана эффективность при гепатопатиях, обусловленных различными гепатотоксическими препаратами. Антидепрессивная активность проявляется постепенно, начиная с конца 1 недели лечения, и стабилизируется в течение 2 недель лечения."},{"name":"Фармакологическая группа","value":"прочие препараты для желудочно-кишечного тракта и обмена веществ, аминокислоты и их производные"},{"name":"Форма выпуска","value":"таблетки, покрытые кишечнорастворимой оболочкой"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-pishchevareniia","categoryId":"15756506","navnodeId":"72470","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"В сухом, защищенном от света месте, при температуре не выше 25°С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Передозировка препарата Гептор маловероятна. В случае передозировки рекомендуется наблюдение за пациентом и проведение симптоматической терапии."},{"name":"Применение при беременности и кормлении грудью","value":"В клинических исследованиях было показано, что применение адеметионина в III триместре беременности не вызывало никаких нежелательных эффектов. Применение препарата Гептор у беременных в I триместре и в период грудного вскармливания возможно, только если потенциальная польза для матери превышает возможный риск для плода или ребенка."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"У некоторых пациентов при приеме препарата Гептор может возникнуть головокружение. Не рекомендуется водить автомобиль и работать с механизмами во время приема препарата до тех пор, пока у пациента не возникнет уверенность, что терапия не влияет на способность заниматься подобного вида деятельностью."},{"name":"Особые указания","value":"Меры предосторожности при применении\u003Cbr\u003EУчитывая тонизирующий эффект препарата, не рекомендуется принимать перед сном. Пероральное применение препарата пациентами с циррозом печени, ассоциированным с гиперазотемией, должно проводиться под наблюдением врача с контролем уровня азота. Таблетки препарата покрыты специальной оболочкой, растворяющейся только в кишечнике, благодаря чему адеметионин высвобождается в 12-перстной кишке. У пациентов с биполярным аффективным расстройством приём адеметионина может индуцировать инверсию аффекта (развитие гипомании или мании)."},{"name":"Взаимодействие","value":"Известных взаимодействий с другими лекарственными средствами не наблюдалось.\u003Cbr\u003EЕсть сообщение о синдроме избытка серотонина у пациента, принимавшего адеметионин и кломипрамин. Считается, что такое взаимодействие возможно, и следует с осторожностью назначать адеметионин вместе с селективными ингибиторами обратного захвата серотонина, трициклическими антидепрессантами (такими как кломипрамин), а также травами и препаратами, содержащими триптофан."},{"name":"Регистрационный номер","value":"ЛС-001820"},{"name":"Дата государственной регистрации","value":"31.03.2022"},{"name":"Владелец регистрационного удостоверения","value":"ВЕРОФАРМ","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-pishchevareniia","categoryId":"15756506","navnodeId":"72470","glfilters":["34324371:35649313","7893318:11037274"]}}},{"name":"Изготовитель","value":"ВЕРОФАРМ"},{"name":"Фасовщик","value":"ВЕРОФАРМ"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Гептор","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-pishchevareniia","categoryId":"15756506","navnodeId":"72470","glfilters":["17796364:18020099"]}}},{"name":"Срок годности","value":"24 мес."}]}},"fullSpecsGrouped":{"88121564196921442":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"желчный пузырь и желчевыводящие пути, печень"},{"name":"Назначение","value":"внутрипеченочный холестаз, нарушение функции печени, острые гепатиты, печеночная энцефалопатия, синдром алкогольной абстиненции, токсические поражения печени, холангит, холецистит, хронические гепатиты, хронический алкогольный гепатит, цирроз печени"},{"name":"Показания к применению","value":"Внутрипеченочный холестаз при прецирротических и цирротических состояниях, который может наблюдаться при следующих заболеваниях:\u003Cbr\u003E- жировая дистрофия печени;\u003Cbr\u003E- хронический гепатит;\u003Cbr\u003E- токсические поражения печени различной этиологии, включая алкогольные, вирусные, лекарственные (антибиотики, противоопухолевые, противотуберкулезные и противовирусные препараты, трициклические антидепрессанты, пероральные контрацептивы);\u003Cbr\u003E\n- хронический некалькулезный (бескаменный) холецистит;\u003Cbr\u003E- холангит;\u003Cbr\u003E- цирроз печени;\u003Cbr\u003E- энцефалопатия, в т.ч. ассоциированная с печеночной недостаточностью (алкогольная и др.);\u003Cbr\u003E- внутрипеченочный холестаз у беременных;\u003Cbr\u003E- симптомы депрессии."},{"name":"Противопоказания","value":"- Генетические нарушения, влияющие на метиониновый цикл и/или вызывающие гомоцистинурию и/или гипергомоцистеинемию (дефицит цистатион-бета-синтазы, нарушение метаболизма витамина В 12 (цианокобаламин));\u003Cbr\u003E- гиперчувствительность к любому из компонентов препарата;\u003Cbr\u003E- возраст до 18 лет (опыт медицинского применения у детей ограничен);\u003Cbr\u003E- биполярные расстройства.\u003Cbr\u003E"},{"name":"Состав","value":"Состав на одну таблетку\u003Cbr\u003E\nДействующее вещество: Адеметионина тозилата дисульфат в пересчет на адеметионин-ион - 400 мг.\u003Cbr\u003EВспомогательные вещества: Полипласдон Икс Эл-10 (кросповидон) - 19 мг, целлюлоза микрокристаллическая - 53 мг, маннитол (маннит) - 53 мг, магния стеарат - 15 мг, масса таблетки без оболочки - 950 мг.\u003Cbr\u003E\nСостав оболочки: Акрил-из желтый - 61.3 мг, [метакриловой кислоты и этилакрилата сополимер ( 1:1 ) - 24.52 мг, тальк - 22.83 мг, титана диоксид - 5.52 мг, кремния диоксид коллоидный (аэросил) - 0.77 мг, триэтилцитрат - 2.94 мг, натрия гидрокарбонат - 0.73 мг, натрия лаурилсульфат - 0.31 мг, железа оксид желтый - 1.84 мг, хинолиновый желтый алюминиевый лак] - 1.84 мг, гипромеллоза (Оксипропилметилцеллюлоза) - 21.0 мг, пласдон ЭС-630 (коповидон) - 9.0 мг, макрогол 6000 (Полиэтиленгликоль 6000) - 3.7 мг, масса таблетки с оболочкой - 1045 мг."},{"name":"Действующее вещество","value":"Адеметионин"},{"name":"Способ применения и дозы","value":"Способ применения и дозы:\u003Cbr\u003EВнутрь.\u003Cbr\u003EТаблетки следует принимать целиком, не разжевывая, желательно в первой половине дня между приемами пищи.\u003Cbr\u003EТаблетки препарата Гептор следует вынимать из блистера непосредственно перед приемом внутрь.\u003Cbr\u003EНачальная терапия:\u003Cbr\u003EРекомендуемая доза составляет 10-25 мг/кг/сут.\u003Cbr\u003EВнутрипеченочный холестаз\u003Cbr\u003EДоза составляет от 800 мг/сут до 1600 мг/сут.\u003Cbr\u003EДепрессия\u003Cbr\u003EДоза составляет от 800 мг/сут до 1600 мг/сут.\u003Cbr\u003EДлительность терапии определяется врачом.\u003Cbr\u003E\nТерапия препаратом Гептор может быть начата с внутривенного или внутримышечного введения с последующим применением препарата Гептор в виде таблеток или сразу с применения препарата Гептор в виде таблеток.\u003Cbr\u003EПациенты пожилого возраста\u003Cbr\u003EКлинический опыт применения препарата Гептор не выявил каких-либо различий в его эффективности у пациентов пожилого возраста и пациентов более молодого возраста. Однако, учитывая высокую вероятность имеющихся нарушений функции печени, почек или сердца, другой сопутствующей патологии или одновременной терапии с другими лекарственными средствами, дозу препарата Гептор пожилым пациентам следует подбирать с осторожностью, начиная применение препарата с нижнего предела диапазона доз.\u003Cbr\u003EПочечная недостаточность\u003Cbr\u003EИмеются ограниченные клинические данные о применении препарата Гептор у пациентов с почечной недостаточностью, в связи с этим рекомендуется соблюдать осторожность при применении препарата Гептор утаких пациентов.\u003Cbr\u003EПеченочная недостаточность\u003Cbr\u003EПараметры фармакокинетики адеметионина сходны у здоровых добровольцев и у пациентов с хроническими заболеваниями печени.\u003Cbr\u003EДети\u003Cbr\u003EПрименение препарата Гептор у детей противопоказано (эффективность и безопасность не установлены)."},{"name":"Побочные действия","value":"Побочное действие:\u003Cbr\u003EСо стороны пищеварительной системы: часто - тошнота, боли в животе, диарея; редко - рвота, сухость во рту, эзофагит, диспепсия, метеоризм, желудочно-кишечная боль, желудочно-кишечное кровотечение, печеночная колика.\u003Cbr\u003EСо стороны нервной системы: редко - спутанность сознания, бессонница, головокружение, головная боль, парестезии.\u003Cbr\u003EСо стороны костно-мышечной системы: редко - артралгии, мышечные судороги\u003Cbr\u003EСо стороны мочевыделительной системы: редко - инфекции мочевыводящих путей.\u003Cbr\u003EСо стороны кожных покровов: редко - гипергидроз, зуд, кожная сыпь.\u003Cbr\u003EМестные реакции: редко - реакции в месте введения; очень редко - реакции в месте введения, некроз кожи в месте введения.\u003Cbr\u003EАллергические реакции: редко - анафилактические реакции; очень редко - отек Квинке, отек гортани.\u003Cbr\u003EПрочие: редко - приливы, поверхностный флебит, астения, озноб, гриппоподобные симптомы, слабость, периферические отеки, гипертермия."},{"name":"Фармакологическое действие","value":"Гептор относится к группе гепатопротекторов с антидепрессивной активностью. Оказывает холеретическое и холекинетическое действие. Обладает дезинтоксикационным, регенерирующим, антиоксидантным, антифиброзирующим и нейропротективным действием.\u003Cbr\u003EВосполняет дефицит S-аденозил-L-метионина (адеметионина) и стимулирует его выработку в организме, содержится во всех средах организма. Наибольшая концентрация адеметионина отмечена в печени и мозге. Выполняет ключевую роль в метаболических процессах организма, принимает участие в важных биохимических реакциях: трансметилировании, транссульфурировании, трансаминировании. В реакциях трансметилирования адеметионин донирует метильную группу для синтеза фосфолипидов клеточных мембран, нейротрансмитгеров, нуклеиновых кислот, белков, гормонов и др. В реакциях транссульфурирования адеметионин является предшественником цистеина, таурина, глютатиона (обеспечивая окислительно-восстановительный механизм клеточной детоксикации), коэнзима А (включается в биохимические реакции цикла трикарбоновых кислот и восполняет энергетический потенциал клетки). Повышает содержание глутамина в печени, цистеина и таурина в плазме; снижает содержание метионина в сыворотке, нормализуя метаболические реакции в печени. После декарбоксилирования участвует в реакциях аминопропилирования, как предшественник полиаминов путресцина (стимулятор регенерации клеток и пролиферации гепатоцитов), спермидина и спермина, входящих в структуру рибосом, что уменьшает риск фиброзирования. Оказывает холеретическое действие. Адеметионин нормализует синтез эндогенного фосфатидилхолина в гепатоцитах, что повышает текучесть и поляризацию мембран. Это улучшает функцию ассоциированных с мембранами гепатоцитов транспортных систем желчных кислот и способствует пассажу желчных кислот в желчевыводящие пути. Эффективен при внутридольковом варианте холестаза (нарушение синтеза и тока желчи). Адеметионин снижает токсичность желчных кислот в гепатоците, осуществляя их конъюгирование и сульфатирование. Конъюгация с таурином повышает растворимость желчных кислот и выведение их из гепатоцита. Процесс сульфатирования желчных кислот способствует возможности их элиминации почками, облегчает прохождение через мембрану гепатоцита и выведение с желчью. Кроме этого, сами сульфатированные желчные кислоты дополнительно защищают мембраны клеток печени от токсического действия несульфатированных желчных кислот (в высоких концентрациях присутствующих в гепатоцитах при внутрипеченочном холестазе). У пациентов с диффузными заболеваниями печени (цирроз, гепатит) с синдромом внутрипеченочного холестаза адеметионин снижает выраженность кожного зуда и изменений биохимических показателей, в т.ч. концентрации прямого билирубина, активности щелочной фосфатазы, аминотрансфераз и др. Холеретический и гепатопротективный эффект сохраняется до З месяцев после прекращения лечения. Показана эффективность при гепатопатиях, обусловленных различными гепатотоксическими препаратами. Антидепрессивная активность проявляется постепенно, начиная с конца 1 недели лечения, и стабилизируется в течение 2 недель лечения."},{"name":"Фармакологическая группа","value":"прочие препараты для желудочно-кишечного тракта и обмена веществ, аминокислоты и их производные"},{"name":"Форма выпуска","value":"таблетки, покрытые кишечнорастворимой оболочкой"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В сухом, защищенном от света месте, при температуре не выше 25°С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Передозировка препарата Гептор маловероятна. В случае передозировки рекомендуется наблюдение за пациентом и проведение симптоматической терапии."},{"name":"Применение при беременности и кормлении грудью","value":"В клинических исследованиях было показано, что применение адеметионина в III триместре беременности не вызывало никаких нежелательных эффектов. Применение препарата Гептор у беременных в I триместре и в период грудного вскармливания возможно, только если потенциальная польза для матери превышает возможный риск для плода или ребенка."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"У некоторых пациентов при приеме препарата Гептор может возникнуть головокружение. Не рекомендуется водить автомобиль и работать с механизмами во время приема препарата до тех пор, пока у пациента не возникнет уверенность, что терапия не влияет на способность заниматься подобного вида деятельностью."},{"name":"Особые указания","value":"Меры предосторожности при применении\u003Cbr\u003EУчитывая тонизирующий эффект препарата, не рекомендуется принимать перед сном. Пероральное применение препарата пациентами с циррозом печени, ассоциированным с гиперазотемией, должно проводиться под наблюдением врача с контролем уровня азота. Таблетки препарата покрыты специальной оболочкой, растворяющейся только в кишечнике, благодаря чему адеметионин высвобождается в 12-перстной кишке. У пациентов с биполярным аффективным расстройством приём адеметионина может индуцировать инверсию аффекта (развитие гипомании или мании)."},{"name":"Взаимодействие","value":"Известных взаимодействий с другими лекарственными средствами не наблюдалось.\u003Cbr\u003EЕсть сообщение о синдроме избытка серотонина у пациента, принимавшего адеметионин и кломипрамин. Считается, что такое взаимодействие возможно, и следует с осторожностью назначать адеметионин вместе с селективными ингибиторами обратного захвата серотонина, трициклическими антидепрессантами (такими как кломипрамин), а также травами и препаратами, содержащими триптофан."},{"name":"Регистрационный номер","value":"ЛС-001820"},{"name":"Дата государственной регистрации","value":"31.03.2022"},{"name":"Владелец регистрационного удостоверения","value":"ВЕРОФАРМ"},{"name":"Изготовитель","value":"ВЕРОФАРМ"},{"name":"Фасовщик","value":"ВЕРОФАРМ"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Гептор"},{"name":"Срок годности","value":"24 мес."}]}],"transitionId":"tr_2246038013891411137"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

Где купить

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1 234 ₽

  • Сегодня, самовывоз  0 ₽
Рейтинг 5 из 5
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Ещё может подойти

  • Рейтинг товара: 4.8 из 5
    на основе 870 оценок
    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  • Рейтинг товара: 4.4 из 5
    на основе 8 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 251 оценка
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  • Рейтинг товара: 5 из 5
    на основе 3 оценки
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  • Рейтинг товара: 5 из 5
    на основе 52 оценки
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  • Рейтинг товара: 4.9 из 5
    на основе 247 оценок
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  • Рейтинг товара: 5 из 5
    на основе 8 оценок
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  • Рейтинг товара: 5 из 5
    на основе 19 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 55 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 16 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 10 оценок
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-c5gdnn0dce6/addToCartButton":{"offerId":"9qRzH24hw192SQvE0VCC7g","skuId":"835237084","pendingCartItem":{"productId":1778171608,"offerId":"9qRzH24hw192SQvE0VCC7g","showPlaceId":"OTNDnItfwRMjN9MRHuEMMq_ESgpxF-mXJkgNsOF8_mrAzM5GqtrcDro0FXDGzjKY6foJz6XaQkm4nq2_IkvkPxZiBZKgx1OzB2zmBlcxx9FOJjNPTlD7IXJczAuFORvFq_n7JK_vUfPcWyqtErz0gOe_OwLzS2nXb7lNd5OV0yWKvONvxp-3yrC6fQy9gOPkIwIJ0fM-l0MqlEYiv4OQDQ,,","feeShow":"OTNDnItfwRMjN9MRHuEMMq_ESgpxF-mXJkgNsOF8_mrAzM5GqtrcDro0FXDGzjKY6foJz6XaQkm4nq2_IkvkPxZiBZKgx1OzB2zmBlcxx9FOJjNPTlD7IXJczAuFORvFq_n7JK_vUfPcWyqtErz0gOe_OwLzS2nXb7lNd5OV0yWKvONvxp-3yrC6fQy9gOPkIwIJ0fM-l0MqlEYiv4OQDQ,,","skuId":"835237084","shopId":77075781,"price":{"applicablePriceDiscounts":[],"value":"1058","currency":"RUR"},"hid":"15756506","name":"Гептразан таб. кш/раств., 400 мг, 20 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{"widgets":{"@light/ScrollBoxControls":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/controls":{"parentId":"wti8lnxsoam","itemsCount":12,"ratio":[2,13],"withScrollBoxGap":false,"gapWidth":4,"rightButtonOffset":0,"leftButtonOffset":0}}},"meta":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/controls":{"name":"@light/ScrollBoxControls"}}}

Инструкция

Показания к применению

Внутрипеченочный холестаз при прецирротических и цирротических состояниях, который может наблюдаться при следующих заболеваниях:
- жировая дистрофия печени;
- хронический гепатит;
- токсические поражения печени различной этиологии, включая алкогольные, вирусные, лекарственные (антибиотики, противоопухолевые, противотуберкулезные и противовирусные препараты, трициклические антидепрессанты, пероральные контрацептивы);
- хронический некалькулезный (бескаменный) холецистит;
- холангит;
- цирроз печени;
- энцефалопатия, в т.ч. ассоциированная с печеночной недостаточностью (алкогольная и др.);
- внутрипеченочный холестаз у беременных;
- симптомы депрессии.

Противопоказания

- Генетические нарушения, влияющие на метиониновый цикл и/или вызывающие гомоцистинурию и/или гипергомоцистеинемию (дефицит цистатион-бета-синтазы, нарушение метаболизма витамина В 12 (цианокобаламин));
- гиперчувствительность к любому из компонентов препарата;
- возраст до 18 лет (опыт медицинского применения у детей ограничен);
- биполярные расстройства.

Способ применения и дозы

Способ применения и дозы:
Внутрь.
Таблетки следует принимать целиком, не разжевывая, желательно в первой половине дня между приемами пищи.
Таблетки препарата Гептор следует вынимать из блистера непосредственно перед приемом внутрь.
Начальная терапия:
Рекомендуемая доза составляет 10-25 мг/кг/сут.
Внутрипеченочный холестаз
Доза составляет от 800 мг/сут до 1600 мг/сут.
Депрессия
Доза составляет от 800 мг/сут до 1600 мг/сут.
Длительность терапии определяется врачом.
Терапия препаратом Гептор может быть начата с внутривенного или внутримышечного введения с последующим применением препарата Гептор в виде таблеток или сразу с применения препарата Гептор в виде таблеток.
Пациенты пожилого возраста
Клинический опыт применения препарата Гептор не выявил каких-либо различий в его эффективности у пациентов пожилого возраста и пациентов более молодого возраста. Однако, учитывая высокую вероятность имеющихся нарушений функции печени, почек или сердца, другой сопутствующей патологии или одновременной терапии с другими лекарственными средствами, дозу препарата Гептор пожилым пациентам следует подбирать с осторожностью, начиная применение препарата с нижнего предела диапазона доз.
Почечная недостаточность
Имеются ограниченные клинические данные о применении препарата Гептор у пациентов с почечной недостаточностью, в связи с этим рекомендуется соблюдать осторожность при применении препарата Гептор утаких пациентов.
Печеночная недостаточность
Параметры фармакокинетики адеметионина сходны у здоровых добровольцев и у пациентов с хроническими заболеваниями печени.
Дети
Применение препарата Гептор у детей противопоказано (эффективность и безопасность не установлены).
Полная инструкция
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Гептор таб. п/о кш/раств.
Гептор таб. п/о кш/раств., 400 мг, 20 шт.
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Инструкция

1 234 ₽

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5.0
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У продавца:45 оценок·7 отзывов
У всех продавцов:316 оценок·81 отзыв
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user avatar
4 месяца назад • Марина К. • Куплен на Маркете
Достоинства: полный аналог Гептрала
Недостатки: нет
Комментарий: принимаю профилактически ,отметила положительные изменения в самочувствии и анализах
user avatar
5 месяцев назад • Евгений П. • Куплен на Маркете
Достоинства: Очень эффективный препарат, нет побочных эффектов. Хорошо переносится.
Недостатки: нет,
Комментарий: рекомендую!
user avatar
Неделю назад • Kristibog • Куплен на Маркете
Достоинства: за две недели, билирубин пришёл в норму
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Заказывайте в новом приложении
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