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Новокаин р-р д/ин., 0.5%, 5 мл, 10 шт.

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Объем, мл: 5

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Коротко о товаре

Артикул Маркета
3123167417
Действующее вещество
Возраст
от 12 лет
Инструкция
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Для уменьшения всасывания и удлинения действия при местной анестезии дополнительно вводят 0,1% раствор эпинефрина - по 1 капле на 2-5-10 мл раствора прокаты.\u003Cbr\u003EПри паранефральной блокаде (по Л. В. Вишневскому) в околопочечную клетчатку вводят 50-80 мл 0,5% раствора или 100-150 мл 0,25%, а при вагосимпатической блокаде - 30-100 мл 0,25% раствора.\u003Cbr\u003EДля циркуляторной или паравертебральной блокад внутрикожно вводят 0,25% или 0,5% раствор.\u003Cbr\u003EВысшие дозы для инфильтрационной анестезии для взрослых: первая разовая доза в начале операции - не более 500 мл 0,25% раствора и 150 мл 0,5% раствора. Максимальная доза для применения у детей старше 12 лет - 15 мг/кг.\u003Cbr\u003EПорядок работы с полимерной ампулой:\u003Cbr\u003E1. Взять ампулу и встряхнуть ее, удерживая за горлышко.\u003Cbr\u003E2. Сдавить ампулу рукой, при этом не должно происходить выделение препарата, и вращающими движениями повернуть и отделить клапан.\u003Cbr\u003E3. Через образовавшееся отверстие немедленно соединить шприц с ампулой.\u003Cbr\u003E4. Перевернуть ампулу и медленно набрать в шприц ее содержимое.\u003Cbr\u003E5. Надеть иглу на шприц."},{"name":"Побочные действия","value":"Со стороны центральной и периферической системы: головная боль, головокружение, сонливость, слабость, тризм, тремор, нистагм, стойкая анестезия, двигательное беспокойство, потеря сознания, судороги, зрительные и слуховые нарушения.\u003Cbr\u003EСо стороны сердечно-сосудистой системы: повышение или снижение артериального давления, коллапс, периферическая вазодилатация, брадикардия, аритмия, боль в грудной клетке, изменения распространения возбуждения в сердце, которые проявляются на ЭКГ в виде плоского зубца Т или укорочения сегмента ST.\u003Cbr\u003EСо стороны дыхательной системы: спазмы дыхательных путей или затруднение дыхания.\u003Cbr\u003EСо стороны мочевыделительной системы: непроизвольное мочеиспускание.\u003Cbr\u003EСо стороны пищеварительной системы: тошнота, рвота.\u003Cbr\u003EСо стороны крови: метгемоглобинемия.\u003Cbr\u003EАллергические реакции: аллергические реакции, вплоть до анафилактического шока.\u003Cbr\u003EПрочие: возвращение боли, стойкая анестезия, гипотермия, дрожь, отек губ, лица, рта, языка и горла."},{"name":"Фармакологическое действие","value":"Местноанестезирующее средство с умеренной анестезирующей активностью и большой широтой терапевтического действия. Являясь слабым основанием, блокирует натриевые каналы, препятствует генерации импульсов в окончаниях чувствительных нервов и проведению импульсов по нервным волокнам. Изменяет потенциал действия в мембранах нервных клеток без выраженного влияния на потенциал покоя. Подавляет проведение не только болевых, но и импульсов другой модальности.\u003Cbr\u003EПри всасывании и непосредственном сосудистом введении в ток крови снижает возбудимость периферических холинергических систем, уменьшает образование и высвобождение ацетилхолина из преганглионарных окончаний (обладает некоторым ганглиоблокирующим действием), устраняет спазм гладкой мускулатуры, уменьшает возбудимость миокарда и моторных зон коры головного мозга. Устраняет нисходящие тормозные влияния ретикулярной формации ствола мозга. Угнетает полисинаптические рефлексы. В больших дозах может вызывать судороги. Обладает короткой анестезирующей активностью (продолжительность инфильтрационной анестезии составляет 0,5-1 ч)."},{"name":"Фармакологическая группа","value":"местноанестезирующее средство"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный","transition":{"type":"catalog","params":{"categorySlug":"anesteziia-rastvoriteli-i-kontrastnye-veshchestva","categoryId":"15758037","navnodeId":"72693","glfilters":["35947170:36763748"]}}},{"name":"Минимальный возраст применения","value":"от 12 лет"},{"name":"Условия хранения","value":"Хранить при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"При использовании в высоких дозах возможно избыточное всасывание.\u003Cbr\u003EСимптомы: бледность кожных покровов и слизистых оболочек, головокружение, тошнота, рвота, \"холодный\" пот, учащение дыхания, тахикардия, снижение артериального давления вплоть до коллапса, апноэ, метгемоглобинемия. Действие на центральную нервную систему проявляется чувством страха, галлюцинациями, судорогами, двигательным возбуждением.\u003Cbr\u003EЛечение: поддержание адекватной легочной вентиляции, дезинтоксикационная симптоматическая терапия."},{"name":"Применение при беременности и кормлении грудью","value":"При беременности и в период грудного вскармливания безопасность и эффективность препарата не установлена.\u003Cbr\u003EПрименение препарата при беременности и в период грудного вскармливания возможно только по назначению врача, если предполагаемая польза для матери превышает потенциальный риск для плода или ребенка."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо воздерживаться от вождения автотранспорта и занятий потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"С осторожностью:\u003Cbr\u003E- Экстренные операции, сопровождающиеся острой кровопотерей;\u003Cbr\u003E- состояния, сопровождающиеся снижением печеночного кровотока (например, при хронической сердечной недостаточности, заболеваниях печени);\u003Cbr\u003E- прогрессирование сердечно-сосудистой недостаточности (обычно вследствие развития блокад сердца и шока);\u003Cbr\u003E- воспалительные заболевания или инфицирование места инъекции;\u003Cbr\u003E- дефицит псевдохолинэстеразы;\u003Cbr\u003E- почечная недостаточность;\u003Cbr\u003E- детский возраст (от 12 до 18 лег);\u003Cbr\u003E- пожилые пациенты (старше 65 лет);\u003Cbr\u003E- ослабленные больные."},{"name":"Взаимодействие","value":"Усиливает угнетающее действие на центральную нервную систему средств для общей анестезии, снотворных и седативных препаратов, наркотических анальгетиков и транквилизаторов.\u003Cbr\u003EАнтикоагулянты (ардепарин натрия, далтепарин натрия, данапароид натрия, эноксапарин натрия, гепарин, варфарин) повышают риск развития кровотечений.\u003Cbr\u003EПри обработке 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йодид, тиотепа) снижают метаболизм прокаина.\u003Cbr\u003EМетаболит прокаина (пара-аминобензойная кислота) является антагонистом сульфаниламидов.\u003Cbr\u003EПри применении местноанестезирующих средств для эпидуральной анестезии с гуанадрелом, с гуанетидином, мекамиламином, триметафана камзилатом повышается риск развития резкого снижения артериального давления и брадикардии."},{"name":"Регистрационный номер","value":"ЛП-003091"},{"name":"Дата государственной регистрации","value":"19.03.2021"},{"name":"Владелец регистрационного удостоверения","value":"Гротекс","transition":{"type":"catalog","params":{"categorySlug":"anesteziia-rastvoriteli-i-kontrastnye-veshchestva","categoryId":"15758037","navnodeId":"72693","glfilters":["34324371:35649313","7893318:16002823"]}}},{"name":"Изготовитель","value":"Гротекс"},{"name":"Фасовщик","value":"Гротекс"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название 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тканях (для анестезии методом ползучего инфильтрата)."},{"name":"Состав","value":"1 мл препарата содержит:\u003Cbr\u003E0,25% раствор\u003Cbr\u003Eактивное вещество: прокаина гидрохлорид - 2,5 мг;\u003Cbr\u003Eвспомогательные вещества: 0,1М раствор хлористоводородной кислоты - до pH 3,8-4,5; вода для инъекций - до 1 мл,\u003Cbr\u003E0,5% раствор\u003Cbr\u003Eактивное вещество: прокаина гидрохлорид - 5 мг;\u003Cbr\u003Eвспомогательные вещества: 0,1 М раствор хлористоводородной кислоты - до pH 3,8-4,5; вода для инъекций - до 1 мл."},{"name":"Действующее вещество","value":"Прокаин"},{"name":"Способ применения и дозы","value":"Для инфильтрационной анестезии применяют 0,25% и 0,5% растворы; для анестезии по методу Вишневского (тугая ползучая инфильтрация) - 0,125% и 0,25% растворы. Для уменьшения всасывания и удлинения действия при местной анестезии дополнительно вводят 0,1% раствор эпинефрина - по 1 капле на 2-5-10 мл раствора прокаты.\u003Cbr\u003EПри паранефральной блокаде (по Л. В. Вишневскому) в околопочечную клетчатку вводят 50-80 мл 0,5% раствора или 100-150 мл 0,25%, а при вагосимпатической блокаде - 30-100 мл 0,25% раствора.\u003Cbr\u003EДля циркуляторной или паравертебральной блокад внутрикожно вводят 0,25% или 0,5% раствор.\u003Cbr\u003EВысшие дозы для инфильтрационной анестезии для взрослых: первая разовая доза в начале операции - не более 500 мл 0,25% раствора и 150 мл 0,5% раствора. Максимальная доза для применения у детей старше 12 лет - 15 мг/кг.\u003Cbr\u003EПорядок работы с полимерной ампулой:\u003Cbr\u003E1. Взять ампулу и встряхнуть ее, удерживая за горлышко.\u003Cbr\u003E2. Сдавить ампулу рукой, при этом не должно происходить выделение препарата, и вращающими движениями повернуть и отделить клапан.\u003Cbr\u003E3. Через образовавшееся отверстие немедленно соединить шприц с ампулой.\u003Cbr\u003E4. Перевернуть ампулу и медленно набрать в шприц ее содержимое.\u003Cbr\u003E5. Надеть иглу на шприц."},{"name":"Побочные действия","value":"Со стороны центральной и периферической системы: головная боль, головокружение, сонливость, слабость, тризм, тремор, нистагм, стойкая анестезия, двигательное беспокойство, потеря сознания, судороги, зрительные и слуховые нарушения.\u003Cbr\u003EСо стороны сердечно-сосудистой системы: повышение или снижение артериального давления, коллапс, периферическая вазодилатация, брадикардия, аритмия, боль в грудной клетке, изменения распространения возбуждения в сердце, которые проявляются на ЭКГ в виде плоского зубца Т или укорочения сегмента ST.\u003Cbr\u003EСо стороны дыхательной системы: спазмы дыхательных путей или затруднение дыхания.\u003Cbr\u003EСо стороны мочевыделительной системы: непроизвольное мочеиспускание.\u003Cbr\u003EСо стороны пищеварительной системы: тошнота, рвота.\u003Cbr\u003EСо стороны крови: метгемоглобинемия.\u003Cbr\u003EАллергические реакции: аллергические реакции, вплоть до анафилактического шока.\u003Cbr\u003EПрочие: возвращение боли, стойкая анестезия, гипотермия, дрожь, отек губ, лица, рта, языка и горла."},{"name":"Фармакологическое действие","value":"Местноанестезирующее средство с умеренной анестезирующей активностью и большой широтой терапевтического действия. Являясь слабым основанием, блокирует натриевые каналы, препятствует генерации импульсов в окончаниях чувствительных нервов и проведению импульсов по нервным волокнам. Изменяет потенциал действия в мембранах нервных клеток без выраженного влияния на потенциал покоя. Подавляет проведение не только болевых, но и импульсов другой модальности.\u003Cbr\u003EПри всасывании и непосредственном сосудистом введении в ток крови снижает возбудимость периферических холинергических систем, уменьшает образование и высвобождение ацетилхолина из преганглионарных окончаний (обладает некоторым ганглиоблокирующим действием), устраняет спазм гладкой мускулатуры, уменьшает возбудимость миокарда и моторных зон коры головного мозга. Устраняет нисходящие тормозные влияния ретикулярной формации ствола мозга. Угнетает полисинаптические рефлексы. В больших дозах может вызывать судороги. Обладает короткой анестезирующей активностью (продолжительность инфильтрационной анестезии составляет 0,5-1 ч)."},{"name":"Фармакологическая группа","value":"местноанестезирующее средство"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный"},{"name":"Минимальный возраст применения","value":"от 12 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"Хранить при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"При использовании в высоких дозах возможно избыточное всасывание.\u003Cbr\u003EСимптомы: бледность кожных покровов и слизистых оболочек, головокружение, тошнота, рвота, \"холодный\" пот, учащение дыхания, тахикардия, снижение артериального давления вплоть до коллапса, апноэ, метгемоглобинемия. Действие на центральную нервную систему проявляется чувством страха, галлюцинациями, судорогами, двигательным возбуждением.\u003Cbr\u003EЛечение: поддержание адекватной легочной вентиляции, дезинтоксикационная симптоматическая терапия."},{"name":"Применение при беременности и кормлении грудью","value":"При беременности и в период грудного вскармливания безопасность и эффективность препарата не установлена.\u003Cbr\u003EПрименение препарата при беременности и в период грудного вскармливания возможно только по назначению врача, если предполагаемая польза для матери превышает потенциальный риск для плода или ребенка."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо воздерживаться от вождения автотранспорта и занятий потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"С осторожностью:\u003Cbr\u003E- Экстренные операции, сопровождающиеся острой кровопотерей;\u003Cbr\u003E- состояния, сопровождающиеся снижением печеночного кровотока (например, при хронической сердечной недостаточности, заболеваниях печени);\u003Cbr\u003E- прогрессирование сердечно-сосудистой недостаточности (обычно вследствие развития блокад сердца и шока);\u003Cbr\u003E- воспалительные заболевания или инфицирование места инъекции;\u003Cbr\u003E- дефицит псевдохолинэстеразы;\u003Cbr\u003E- почечная недостаточность;\u003Cbr\u003E- детский возраст (от 12 до 18 лег);\u003Cbr\u003E- пожилые пациенты (старше 65 лет);\u003Cbr\u003E- ослабленные больные."},{"name":"Взаимодействие","value":"Усиливает угнетающее действие на центральную нервную систему средств для общей анестезии, снотворных и седативных препаратов, наркотических анальгетиков и транквилизаторов.\u003Cbr\u003EАнтикоагулянты (ардепарин натрия, далтепарин натрия, данапароид натрия, эноксапарин натрия, гепарин, варфарин) повышают риск развития кровотечений.\u003Cbr\u003EПри обработке места инъекции местного анестетика дезинфицирующими растворами, содержащими тяжелые металлы, повышается риск развития местной реакции в виде болезненности и отека.\u003Cbr\u003EОдновременное применение с ингибиторами моноаминоксидазы (фуразолидон, прокарбазин, селегилин) повышает риск развития гипотонии.\u003Cbr\u003EУсиливают и удлиняют действие миорелаксантов.\u003Cbr\u003EПри применении прокаина совместно с наркотическими анальгетиками отмечается аддитивный эффект, что используется при проведении спинальной и эпидуральной анестезии, при этом усиливается угнетение дыхания.\u003Cbr\u003EВазоконстрикторы (эпинефрин, метоксамин, фенилэфрин) удлиняют местно-анестезирующее действие.\u003Cbr\u003EПрокаин снижает антимиастеническое действие лекарственных средств, особенно при применении его в высоких дозах, что требует дополнительной коррекции лечения миастении.\u003Cbr\u003EИнгибиторы холинэстеразы (антимиастенические лекарственные средства, циклофосфамид, демекария бромид, экотиопата йодид, тиотепа) снижают метаболизм прокаина.\u003Cbr\u003EМетаболит прокаина (пара-аминобензойная кислота) является антагонистом сульфаниламидов.\u003Cbr\u003EПри применении местноанестезирующих средств для эпидуральной анестезии с гуанадрелом, с гуанетидином, мекамиламином, триметафана камзилатом повышается риск развития резкого снижения артериального давления и брадикардии."},{"name":"Регистрационный номер","value":"ЛП-003091"},{"name":"Дата государственной регистрации","value":"19.03.2021"},{"name":"Владелец регистрационного удостоверения","value":"Гротекс"},{"name":"Изготовитель","value":"Гротекс"},{"name":"Фасовщик","value":"Гротекс"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Новокаин"},{"name":"Срок годности","value":"24 мес."}]}],"transitionId":"tr_16352333257925465733"}}}}
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    на основе 15 оценок
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  • Рейтинг товара: 5 из 5
    на основе 3 оценки
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-59wfhujdfcg/addToCartButton":{"offerId":"1insO6i_CkqBUBKcJCSqWw","skuId":"228060826","pendingCartItem":{"productId":1404816472,"offerId":"1insO6i_CkqBUBKcJCSqWw","showPlaceId":"OTNDnItfwRMjN9MRHuEMMvnGlta_LWTI7ZKt0B772j2NnuVRlmXgs9NqRxp_vFKZ6w4F3G0v0gRiwAzOrmZhsCZYtMscMB26d7MnoJqRoJQPCJda5pR7Ef8i3NetW0Lo1IwrG7JDJqZ8f31a5C2IZKxT3CbOBIuBLc1tJaGb3aV54MGsM4eJ4twV6vkkaJP3x4-OAbSo7pdr6XVKbsiUFw,,","feeShow":"OTNDnItfwRMjN9MRHuEMMvnGlta_LWTI7ZKt0B772j2NnuVRlmXgs9NqRxp_vFKZ6w4F3G0v0gRiwAzOrmZhsCZYtMscMB26d7MnoJqRoJQPCJda5pR7Ef8i3NetW0Lo1IwrG7JDJqZ8f31a5C2IZKxT3CbOBIuBLc1tJaGb3aV54MGsM4eJ4twV6vkkaJP3x4-OAbSo7pdr6XVKbsiUFw,,","skuId":"228060826","shopId":55106433,"price":{"applicablePriceDiscounts":[],"value":"157","currency":"RUR"},"hid":"15758037","name":"Новокаин буфус р-р д/ин., 5 мг/мл, 5 мл, 10 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  • Рейтинг товара: 5 из 5
    на основе 10 оценок
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  • Рейтинг товара: 5 из 5
    на основе 3 оценки
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  • {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-nr2ggvofpv/addToCartButton":{"offerId":"v7U5k1fQaHXX4yiqvASjDA","skuId":"228007906","pendingCartItem":{"productId":1404816426,"offerId":"v7U5k1fQaHXX4yiqvASjDA","showPlaceId":"OTNDnItfwRMjN9MRHuEMMvnGlta_LWTI6cfRyAvSbDJ2oHo2jSYPhZSi2_yrGKk-mQsjNGgOFVzW0AcOIaNSIELV-Xk3TTLLV3QgQ67VcsWmLCppQWBoezv8M-qf33fvD17Kr27JOxLNHxL63Zcz663npUPXNCos8bvJfU62-_m4W5vwlkgJrUzbm1KyS4bhDJmTA6nwPQMyLoVnMIBtzw,,","feeShow":"OTNDnItfwRMjN9MRHuEMMvnGlta_LWTI6cfRyAvSbDJ2oHo2jSYPhZSi2_yrGKk-mQsjNGgOFVzW0AcOIaNSIELV-Xk3TTLLV3QgQ67VcsWmLCppQWBoezv8M-qf33fvD17Kr27JOxLNHxL63Zcz663npUPXNCos8bvJfU62-_m4W5vwlkgJrUzbm1KyS4bhDJmTA6nwPQMyLoVnMIBtzw,,","skuId":"228007906","shopId":4035369,"price":{"applicablePriceDiscounts":[],"value":"48","currency":"RUR"},"hid":"15758037","name":"Новокаин р-р д/ин., 5 мг/мл, 5 мл, 10 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  • Рейтинг товара: 4.7 из 5
    на основе 13 оценок
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  • Рейтинг товара: 5 из 5
    на основе 4 оценки
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  • Рейтинг товара: 5 из 5
    на основе 4 оценки
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  • Рейтинг товара: 5 из 5
    на основе 7 оценок
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  • Рейтинг товара: 5 из 5
    на основе 32 оценки
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Инструкция

Показания к применению

- Инфильтрационная (в том числе внутрикостная) анестезия;
- вагосимпатическая шейная, паранефральная, циркулярная и паравертебральная блокады.

Противопоказания

- Гиперчувствительность (в том числе к парааминобензойной кислоте и другим местным анестетикам);
- детский возраст до 12 лет:
- выраженные фиброзные изменения в тканях (для анестезии методом ползучего инфильтрата).

Способ применения и дозы

Для инфильтрационной анестезии применяют 0,25% и 0,5% растворы; для анестезии по методу Вишневского (тугая ползучая инфильтрация) - 0,125% и 0,25% растворы. Для уменьшения всасывания и удлинения действия при местной анестезии дополнительно вводят 0,1% раствор эпинефрина - по 1 капле на 2-5-10 мл раствора прокаты.
При паранефральной блокаде (по Л. В. Вишневскому) в околопочечную клетчатку вводят 50-80 мл 0,5% раствора или 100-150 мл 0,25%, а при вагосимпатической блокаде - 30-100 мл 0,25% раствора.
Для циркуляторной или паравертебральной блокад внутрикожно вводят 0,25% или 0,5% раствор.
Высшие дозы для инфильтрационной анестезии для взрослых: первая разовая доза в начале операции - не более 500 мл 0,25% раствора и 150 мл 0,5% раствора. Максимальная доза для применения у детей старше 12 лет - 15 мг/кг.
Порядок работы с полимерной ампулой:
1. Взять ампулу и встряхнуть ее, удерживая за горлышко.
2. Сдавить ампулу рукой, при этом не должно происходить выделение препарата, и вращающими движениями повернуть и отделить клапан.
3. Через образовавшееся отверстие немедленно соединить шприц с ампулой.
4. Перевернуть ампулу и медленно набрать в шприц ее содержимое.
5. Надеть иглу на шприц.
Полная инструкция
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Новокаин р-р д/ин.
Новокаин р-р д/ин., 0.5%, 5 мл, 10 шт.
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Инструкция

99 ₽

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5.0
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