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Описание

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Ацекардол таб. п/о плен. кш/раств., 100 мг, 30 шт.

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Дозировка: 100 мг

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50 мг, 100 мг, 300 мг;\u003Cbr\u003EВспомогательные вещества: повидон низкомолекулярный (поливинилпирролидон низкомолекулярный медицинский 12600 + 2700), крахмал кукурузный, целлюлоза микрокристаллическая, магния стеарат, тальк, лактозы моногидрат (сахар молочный).\u003Cbr\u003EВспомогательные вещества для получения покрытия: целлацефат (ацетилфталил- целлюлоза), титана диоксид, касторовое масло."},{"name":"Действующее вещество","value":"Ацетилсалициловая кислота","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28709804"]}}},{"name":"Способ применения и дозы","value":"Таблетки препарата Ацекардол следует принимать перед едой, запивая большим количеством жидкости, 1 раз в сутки. Ацекардол предназначен для длительного применения. Длительность терапии определяется врачом.\u003Cbr\u003EПрофилактика при подозрении острого инфаркта миокарда: 100 мг в сутки или 300 мг через день (первую таблетку необходимо разжевать для более быстрого всасывания).\u003Cbr\u003EПрофилактика впервые возникшего острого инфаркта миокарда при наличии факторов риска: 100 мг в сутки или 300 мг через день.\u003Cbr\u003EПрофилактика повторного инфаркта миокарда и нестабильная стенокардия: 100 - 300 мг в сутки.\u003Cbr\u003EПрофилактика ишемического инсульта и преходящего нарушения мозгового кровообращения: 100 - 300 мг в сутки.\u003Cbr\u003EПрофилактика тромбоэмболии после операций и инвазивных вмешательств на сосудах: 100 - 300 мг в сутки.\u003Cbr\u003EПрофилактика тромбоза глубоких вен и тромбоэмболии легочной артерии и ее ветвей: 100 мг в сутки или 300 мг через день."},{"name":"Побочные действия","value":"Со стороны пищеварительной системы: тошнота, изжога, рвота, боли в животе; язвы слизистой оболочки желудка и двенадцатиперстной кишки; перфоративные яз¬вы желудка и двенадцатиперстной кишки, желудочно-кишечные кровотечения, пре¬ходящие нарушения функции печени с повышением активности \"печеночных\" трансаминаз.\u003Cbr\u003EСо стороны системы кроветворения: назначение АСК сопровождается повы¬шенным риском кровотечений вследствие ингибирующего действия АСК на агрега¬цию тромбоцитов, анемия.\u003Cbr\u003EАллергические реакции: кожная сыпь, кожный зуд, крапивница, отек Квинке, ри¬нит, отек слизистой оболочки носа, кардиореспираторный дистресс-синдром, а так¬же тяжелые реакции, включая анафилактический шок.\u003Cbr\u003EСо стороны дыхательной системы: бронхоспазм.\u003Cbr\u003EСо стороны центральной нервной системы: головокружение, снижение слуха, головная боль, шум в ушах.\u003Cbr\u003EЕсли любые из указанных побочных эффектов усугубляются, или Вы заметили любые другие побочные эффекты не указанные в инструкции, сообщите об этом врачу."},{"name":"Фармакологическое действие","value":"В основе механизма антиагрегантного действия ацетилсалициловой кислоты (АСК) лежит необратимое ингибирование циклооксигеназы (ЦОГ-1), в результате чего блокируется синтез тромбоксана А2 и подавляется агрегация тромбоцитов. Антиагрегантный эффект развивается даже после применения малых доз препарата и сохраняется в течение 7 суток после однократного приема. Считается, что АСК име¬ет и другие механизмы подавления агрегации тромбоцитов.\u003Cbr\u003EВ высоких дозах АСК (свыше 300 мг/сутки) также оказывает противовоспали¬тельное, жаропонижающее и анальгезирующее действие."},{"name":"Фармакологическая группа","value":"антиагреганты"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"При температуре не выше 25 °С. Хранить в местах, недоступных для детей."},{"name":"Передозировка","value":"Передозировка маловероятна вследствие низкого содержания АСК в препарате.\u003Cbr\u003EПревышение дозы АСК сопряжено с риском желудочно-кишечного кровотечения.\u003Cbr\u003EПередозировка особенно опасна у пациентов пожилого возраста.\u003Cbr\u003EСимптомы передозировки от легкой до средней степени тяжести: головокружении, шум в ушах, ухудшение слуха, повышенное потоотделение (в том числе профузное), тошнота, рвота, головная боль, спутанность сознания, тахипноэ, гипервентиляция, респираторный алкалоз.\u003Cbr\u003EЛечение: желудочный лаваж, многократный прием активированного угля, форсированный щелочной диурез, восстановление водно-электролитного баланса и кислотно-основного состояния.\u003Cbr\u003EСимптомы передозировки от средней до тяжелой степени:\u003Cbr\u003E- респираторный алкалоз с компенсаторным метаболическим ацидозом;\u003Cbr\u003E- гиперпирексия (крайне высокая температура тела);\u003Cbr\u003E- нарушения дыхания: гипервентиляция, некардиогенный отек легких, угнетение дыхания, асфиксия;\u003Cbr\u003E- нарушения со стороны сердечно-сосудистой системы: нарушения ритма сердца, снижение артериального давления, угнетение сердечной деятельности;\u003Cbr\u003E- нарушения водно-электролитного баланса: дегидратация, нарушение функции по¬чек от олигурии вплоть до развития почечной недостаточности, характеризующееся гипокалиемией, гипернатриемией, гипонатриемией;\u003Cbr\u003E- нарушение метаболизма глюкозы: гипергликемия, гипогликемия (особенно у детей), кетоацидоз;\u003Cbr\u003E- шум в ушах, глухота;\u003Cbr\u003E- желудочно-кишечные кровотечения;\u003Cbr\u003E- гематологические нарушения: от ингибирования агрегации тромбоцитов до коагулопатии, удлинение протромбинового времени, гипопротромбинемия;\u003Cbr\u003E- неврологические нарушения: токсическая энцефалопатия и угнетение функции центральной нервной системы (сонливость, спутанность сознания, кома, судороги).\u003Cbr\u003EЛечение: немедленная госпитализация в специализированные отделения для проведения экстренной терапии - желудочный лаваж, многократный прием активированного угля, форсированный щелочной диурез, гемодиализ, восстановление водно-электролитного баланса и кислотно-основного состояния, симптоматическая тера¬пия. При проведении щелочного диуреза необходимо добиться значений pH между 7,5 и 8. Форсированный щелочной диурез следует проводить, когда концентрация салицилатов в плазме составляет более 500 мг/л (3,6 ммоль/л) у взрослых и 300 мг/л (2, 2 ммоль/л) у детей.\u003Cbr\u003E\u003Cbr\u003E"},{"name":"Применение при беременности и кормлении грудью","value":"Применение больших доз салицилатов в первые 3 месяца беременности ассоции¬руется с повышенной частотой дефектов развития плода (расщепленное небо, пороки сердца). Назначение салицилатов в I триместре беременности противопоказано. Во II триместре беременности салицилаты можно назначать только с учетом строгой оценки риска для плода и пользы для матери, предпочтительно в дозах не выше 150 мг/сутки и непродолжительно.\u003Cbr\u003EВ последнем триместре беременности салицилаты в высокой дозе (более 300 мг/сутки) вызывают ослабление родовой деятельности, преждевременное за¬крытие артериального протока у плода, повышенную кровоточивость у матери и плода, а назначение непосредственно перед родами может вызвать внутричерепные кровоизлияния, особенно у недоношенных детей. Назначение салицилатов в последнем триместре беременности противопоказано.\u003Cbr\u003EСалицилаты и их метаболиты в небольших количествах проникают в грудное молоко, поэтому в период лактации следует отменить грудное вскармливание."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Во время приема препарата Ацекардол следует соблюдать осторожность при управлении транспортными средствами, механизмами и при выполнении других потенциально опасных видов деятельности, требующих повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"С осторожностью:\u003Cbr\u003EПри подагре, гиперурикемии, т.к. АСК в низких дозах снижает экскрецию моче¬вой кислоты; следует иметь в виду, что АСК в низких дозах может спровоцировать развитие подагры у предрасположенных пациентов (имеющих сниженную экскре¬цию мочевой кислоты); язвенной болезни желудка и двенадцатиперстной кишки или желудочно-кишечных кровотечениях (в анамнезе); нарушении функции печени (класс А по шкале Чайлд-Пью); нарушении функции почек (КК более 30 мл/мин); бронхиальной астме, хронических заболеваниях органов дыхания, сенной лихорадке, полипозе носа, лекарственной аллергии, одновременном приеме метотрексата в дозе менее 15 мг/нед; сопутствующей терапии антикоагулянтами, беременности (II триместр); при предполагаемом хирургическом вмешательстве (включая незначи¬тельные, например, экстракция зуба), так как АСК может вызывать склонность к развитию кровотечений в течение нескольких дней после приема препарата.\u003Cbr\u003EЕсли у Вас одно из перечисленных заболевания, перед приемом препарата обяза-тельно проконсультируйтесь с врачом.\u003Cbr\u003EАСК может провоцировать бронхоспазм, а также вызывать приступы бронхиаль¬ной астмы и другие реакции повышенной чувствительности. Факторами риска яв¬ляются наличие бронхиальной астмы в анамнезе, сенной лихорадки, полипоза носа, хронических заболеваний дыхательной системы, а также аллергических реакций на другие препараты (например, кожные реакции, зуд, крапивница).\u003Cbr\u003EИнгибирующее действие АСК на агрегацию тромбоцитов сохраняется в течение нескольких дней после приема, в связи с чем, возможно повышение риска кровотечений в ходе оперативного вмешательства или в послеоперационном периоде. При необходимости абсолютного исключения кровоточивости в ходе оперативного вме¬шательства необходимо по возможности полностью отказаться от применения АСК в предоперационном периоде.\u003Cbr\u003EАцетилсалициловая кислота в низких дозах может спровоцировать развитие по¬дагры у предрасположенных лиц (имеющих сниженную экскрецию мочевой кисло¬ты).\u003Cbr\u003EПри сочетанном применении ГКС и салицилатов следует помнить, что во Время лечения концентрация салицилатов в крови снижена, а после отмены ГКС возможна передозировка салицилатов.\u003Cbr\u003EПревышение дозы ацетилсалициловой кислоты сопряжено с риском желудочно-кишечного кровотечения."},{"name":"Взаимодействие","value":"АСК при одновременном применении усиливает действие следующих лекарст-венных средств:\u003Cbr\u003E- метотрексата за счет снижения почечного клиренса и вытеснения его из связи с белками плазмы, также сочетание ацетилсалициловой кислоты с метотрексатом сопровождается повышенной частотой развития побочных эффектов со стороны органов кроветворения;\u003Cbr\u003E- гепарина и непрямых антикоагулянтов за счет нарушения функции тромбоцитов и вытеснения непрямых антикоагулянтов из связи с белками плазмы;\u003Cbr\u003E- тромболитических средств и антиагрегантов;\u003Cbr\u003E- дигоксина вследствие снижения его почечной экскреции;\u003Cbr\u003E- гипогликемических средств (инсулина и производных сульфонилмочевины) за счет гипогликемических свойств самой ацетилсалициловой кислоты в высоких до¬зах и вытеснения производных сульфонилмочевины из связи с белками плазмы;\u003Cbr\u003E- вальпроевой кислоты за счет вытеснения ее из связи с белками плазмы.\u003Cbr\u003EСочетание ацетилсалициловой кислоты с антикоагулянтами, тромболитиками и антиагрегантами сопровождается повышенным риском развития кровотечения.\u003Cbr\u003EПри одновременном приеме ацетилсалициловой кислоты с алкоголем наблюдает¬ся усиление токсического действия алкоголя на центральную нервную систему, повышается риск повреждения слизистой оболочки желудочно-кишечного тракта и удлинения времени кровотечения.\u003Cbr\u003EАСК ослабляет действие урикозурических препаратов - бензбромарона (снижение урикозурического эффекта вследствие конкурентного подавления почечной канальцевой экскреции мочевой кислоты), ингибиторов ангиотензинпревращающего фер¬мента (АПФ) (отмечается дозозависимое снижение скорости клубочковой фильтрации в результате ингибирования простагландинов, обладающих сосудорасширяю-щим действием, соответственно ослабление гипотензивного действия), диуретиков (при совместном применении с АСК в высоких дозах отмечается снижение скорости клубочковой фильтрации в результате снижения синтеза простагландинов в почках).\u003Cbr\u003EУсиливая элиминацию салицилатов, системные глюкокортикостероиды(ГКС) ослабляют их действие."},{"name":"Регистрационный номер","value":"ЛС-000680"},{"name":"Дата государственной регистрации","value":"04.06.2013"},{"name":"Владелец регистрационного удостоверения","value":"Синтез","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313","7893318:10970801"]}}},{"name":"Изготовитель","value":"Синтез"},{"name":"Фасовщик","value":"Синтез"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Ацекардол","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["17796364:18007807"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"4179599423635485372":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Органы и системы","value":"кровеносные сосуды, сердце"},{"name":"Назначение","value":"профилактика венозной тромбоэмболии, профилактика инсульта, профилактика инфаркта миокарда, профилактика тромбоза глубоких вен и тромбоэмболии легочной артерии и ее ветвей, профилактика тромбоэмболии, стенокардия"},{"name":"Показания к применению","value":"- профилактика острого инфаркта миокарда при наличии факторов риска (например, сахарный диабет, гиперлипидемия, артериальная гипертензия, ожирение, курение, пожилой возраст) и повторного инфаркта миокарда;\u003Cbr\u003E- нестабильная стенокардия;\u003Cbr\u003E- профилактика ишемического инсульта (в том числе у пациентов с преходящим нарушением мозгового кровообращения);\u003Cbr\u003E- профилактика тромбоэмболии после операций и инвазивных вмешательств на сосудах (например, аортокоронарное шунтирование, эндартерэктомия сонных арте¬рий, артериовенозное шунтирование, ангиопластика и стентирование коронарных артерий, ангиопластика сонных артерий);\u003Cbr\u003E- профилактика тромбоза глубоких вен и тромбоэмболии легочной артерии и ее ветвей (в том числе, при длительной иммобилизации в результате обширного хирургического вмешательства)."},{"name":"Противопоказания","value":"Гиперчувствительность к АСК, эрозивно-язвенные поражения ЖКТ (в фазе обострения), желудочно-кишечное кровотечение, геморрагический диатез, бронхиальная астма, индуцированная приемом салицилатов, полное или неполное сочетание бронхиальной астмы, рецидивирующего полипоза носа и околоносовых пазух и непереносимости АСК, выраженная почечная недостаточность (клиренс креатинина (КК) менее 30 мл/мин), выраженная печеночная недостаточность (класс В и С по шкале Чайлд-Пью), хроническая сердечная недостаточность (III-IV функционального класса по классификации NYHA), одновременный прием метотрексата в дозе 15 мг/нед и более, беременность (I и III триместр), период лактации, детский возраст до 18 лет, дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция."},{"name":"Состав","value":"Состав на одну таблетку:\u003Cbr\u003EАктивное вещество: ацетилсалициловая кислота - 50 мг, 100 мг, 300 мг;\u003Cbr\u003EВспомогательные вещества: повидон низкомолекулярный (поливинилпирролидон низкомолекулярный медицинский 12600 + 2700), крахмал кукурузный, целлюлоза микрокристаллическая, магния стеарат, тальк, лактозы моногидрат (сахар молочный).\u003Cbr\u003EВспомогательные вещества для получения покрытия: целлацефат (ацетилфталил- целлюлоза), титана диоксид, касторовое масло."},{"name":"Действующее вещество","value":"Ацетилсалициловая кислота"},{"name":"Способ применения и дозы","value":"Таблетки препарата Ацекардол следует принимать перед едой, запивая большим количеством жидкости, 1 раз в сутки. Ацекардол предназначен для длительного применения. Длительность терапии определяется врачом.\u003Cbr\u003EПрофилактика при подозрении острого инфаркта миокарда: 100 мг в сутки или 300 мг через день (первую таблетку необходимо разжевать для более быстрого всасывания).\u003Cbr\u003EПрофилактика впервые возникшего острого инфаркта миокарда при наличии факторов риска: 100 мг в сутки или 300 мг через день.\u003Cbr\u003EПрофилактика повторного инфаркта миокарда и нестабильная стенокардия: 100 - 300 мг в сутки.\u003Cbr\u003EПрофилактика ишемического инсульта и преходящего нарушения мозгового кровообращения: 100 - 300 мг в сутки.\u003Cbr\u003EПрофилактика тромбоэмболии после операций и инвазивных вмешательств на сосудах: 100 - 300 мг в сутки.\u003Cbr\u003EПрофилактика тромбоза глубоких вен и тромбоэмболии легочной артерии и ее ветвей: 100 мг в сутки или 300 мг через день."},{"name":"Побочные действия","value":"Со стороны пищеварительной системы: тошнота, изжога, рвота, боли в животе; язвы слизистой оболочки желудка и двенадцатиперстной кишки; перфоративные яз¬вы желудка и двенадцатиперстной кишки, желудочно-кишечные кровотечения, пре¬ходящие нарушения функции печени с повышением активности \"печеночных\" трансаминаз.\u003Cbr\u003EСо стороны системы кроветворения: назначение АСК сопровождается повы¬шенным риском кровотечений вследствие ингибирующего действия АСК на агрега¬цию тромбоцитов, анемия.\u003Cbr\u003EАллергические реакции: кожная сыпь, кожный зуд, крапивница, отек Квинке, ри¬нит, отек слизистой оболочки носа, кардиореспираторный дистресс-синдром, а так¬же тяжелые реакции, включая анафилактический шок.\u003Cbr\u003EСо стороны дыхательной системы: бронхоспазм.\u003Cbr\u003EСо стороны центральной нервной системы: головокружение, снижение слуха, головная боль, шум в ушах.\u003Cbr\u003EЕсли любые из указанных побочных эффектов усугубляются, или Вы заметили любые другие побочные эффекты не указанные в инструкции, сообщите об этом врачу."},{"name":"Фармакологическое действие","value":"В основе механизма антиагрегантного действия ацетилсалициловой кислоты (АСК) лежит необратимое ингибирование циклооксигеназы (ЦОГ-1), в результате чего блокируется синтез тромбоксана А2 и подавляется агрегация тромбоцитов. Антиагрегантный эффект развивается даже после применения малых доз препарата и сохраняется в течение 7 суток после однократного приема. Считается, что АСК име¬ет и другие механизмы подавления агрегации тромбоцитов.\u003Cbr\u003EВ высоких дозах АСК (свыше 300 мг/сутки) также оказывает противовоспали¬тельное, жаропонижающее и анальгезирующее действие."},{"name":"Фармакологическая группа","value":"антиагреганты"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"При температуре не выше 25 °С. Хранить в местах, недоступных для детей."},{"name":"Передозировка","value":"Передозировка маловероятна вследствие низкого содержания АСК в препарате.\u003Cbr\u003EПревышение дозы АСК сопряжено с риском желудочно-кишечного кровотечения.\u003Cbr\u003EПередозировка особенно опасна у пациентов пожилого возраста.\u003Cbr\u003EСимптомы передозировки от легкой до средней степени тяжести: головокружении, шум в ушах, ухудшение слуха, повышенное потоотделение (в том числе профузное), тошнота, рвота, головная боль, спутанность сознания, тахипноэ, гипервентиляция, респираторный алкалоз.\u003Cbr\u003EЛечение: желудочный лаваж, многократный прием активированного угля, форсированный щелочной диурез, восстановление водно-электролитного баланса и кислотно-основного состояния.\u003Cbr\u003EСимптомы передозировки от средней до тяжелой степени:\u003Cbr\u003E- респираторный алкалоз с компенсаторным метаболическим ацидозом;\u003Cbr\u003E- гиперпирексия (крайне высокая температура тела);\u003Cbr\u003E- нарушения дыхания: гипервентиляция, некардиогенный отек легких, угнетение дыхания, асфиксия;\u003Cbr\u003E- нарушения со стороны сердечно-сосудистой системы: нарушения ритма сердца, снижение артериального давления, угнетение сердечной деятельности;\u003Cbr\u003E- нарушения водно-электролитного баланса: дегидратация, нарушение функции по¬чек от олигурии вплоть до развития почечной недостаточности, характеризующееся гипокалиемией, гипернатриемией, гипонатриемией;\u003Cbr\u003E- нарушение метаболизма глюкозы: гипергликемия, гипогликемия (особенно у детей), кетоацидоз;\u003Cbr\u003E- шум в ушах, глухота;\u003Cbr\u003E- желудочно-кишечные кровотечения;\u003Cbr\u003E- гематологические нарушения: от ингибирования агрегации тромбоцитов до коагулопатии, удлинение протромбинового времени, гипопротромбинемия;\u003Cbr\u003E- неврологические нарушения: токсическая энцефалопатия и угнетение функции центральной нервной системы (сонливость, спутанность сознания, кома, судороги).\u003Cbr\u003EЛечение: немедленная госпитализация в специализированные отделения для проведения экстренной терапии - желудочный лаваж, многократный прием активированного угля, форсированный щелочной диурез, гемодиализ, восстановление водно-электролитного баланса и кислотно-основного состояния, симптоматическая тера¬пия. При проведении щелочного диуреза необходимо добиться значений pH между 7,5 и 8. Форсированный щелочной диурез следует проводить, когда концентрация салицилатов в плазме составляет более 500 мг/л (3,6 ммоль/л) у взрослых и 300 мг/л (2, 2 ммоль/л) у детей.\u003Cbr\u003E\u003Cbr\u003E"},{"name":"Применение при беременности и кормлении грудью","value":"Применение больших доз салицилатов в первые 3 месяца беременности ассоции¬руется с повышенной частотой дефектов развития плода (расщепленное небо, пороки сердца). Назначение салицилатов в I триместре беременности противопоказано. Во II триместре беременности салицилаты можно назначать только с учетом строгой оценки риска для плода и пользы для матери, предпочтительно в дозах не выше 150 мг/сутки и непродолжительно.\u003Cbr\u003EВ последнем триместре беременности салицилаты в высокой дозе (более 300 мг/сутки) вызывают ослабление родовой деятельности, преждевременное за¬крытие артериального протока у плода, повышенную кровоточивость у матери и плода, а назначение непосредственно перед родами может вызвать внутричерепные кровоизлияния, особенно у недоношенных детей. Назначение салицилатов в последнем триместре беременности противопоказано.\u003Cbr\u003EСалицилаты и их метаболиты в небольших количествах проникают в грудное молоко, поэтому в период лактации следует отменить грудное вскармливание."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Во время приема препарата Ацекардол следует соблюдать осторожность при управлении транспортными средствами, механизмами и при выполнении других потенциально опасных видов деятельности, требующих повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"С осторожностью:\u003Cbr\u003EПри подагре, гиперурикемии, т.к. АСК в низких дозах снижает экскрецию моче¬вой кислоты; следует иметь в виду, что АСК в низких дозах может спровоцировать развитие подагры у предрасположенных пациентов (имеющих сниженную экскре¬цию мочевой кислоты); язвенной болезни желудка и двенадцатиперстной кишки или желудочно-кишечных кровотечениях (в анамнезе); нарушении функции печени (класс А по шкале Чайлд-Пью); нарушении функции почек (КК более 30 мл/мин); бронхиальной астме, хронических заболеваниях органов дыхания, сенной лихорадке, полипозе носа, лекарственной аллергии, одновременном приеме метотрексата в дозе менее 15 мг/нед; сопутствующей терапии антикоагулянтами, беременности (II триместр); при предполагаемом хирургическом вмешательстве (включая незначи¬тельные, например, экстракция зуба), так как АСК может вызывать склонность к развитию кровотечений в течение нескольких дней после приема препарата.\u003Cbr\u003EЕсли у Вас одно из перечисленных заболевания, перед приемом препарата обяза-тельно проконсультируйтесь с врачом.\u003Cbr\u003EАСК может провоцировать бронхоспазм, а также вызывать приступы бронхиаль¬ной астмы и другие реакции повышенной чувствительности. Факторами риска яв¬ляются наличие бронхиальной астмы в анамнезе, сенной лихорадки, полипоза носа, хронических заболеваний дыхательной системы, а также аллергических реакций на другие препараты (например, кожные реакции, зуд, крапивница).\u003Cbr\u003EИнгибирующее действие АСК на агрегацию тромбоцитов сохраняется в течение нескольких дней после приема, в связи с чем, возможно повышение риска кровотечений в ходе оперативного вмешательства или в послеоперационном периоде. При необходимости абсолютного исключения кровоточивости в ходе оперативного вме¬шательства необходимо по возможности полностью отказаться от применения АСК в предоперационном периоде.\u003Cbr\u003EАцетилсалициловая кислота в низких дозах может спровоцировать развитие по¬дагры у предрасположенных лиц (имеющих сниженную экскрецию мочевой кисло¬ты).\u003Cbr\u003EПри сочетанном применении ГКС и салицилатов следует помнить, что во Время лечения концентрация салицилатов в крови снижена, а после отмены ГКС возможна передозировка салицилатов.\u003Cbr\u003EПревышение дозы ацетилсалициловой кислоты сопряжено с риском желудочно-кишечного кровотечения."},{"name":"Взаимодействие","value":"АСК при одновременном применении усиливает действие следующих лекарст-венных средств:\u003Cbr\u003E- метотрексата за счет снижения почечного клиренса и вытеснения его из связи с белками плазмы, также сочетание ацетилсалициловой кислоты с метотрексатом сопровождается повышенной частотой развития побочных эффектов со стороны органов кроветворения;\u003Cbr\u003E- гепарина и непрямых антикоагулянтов за счет нарушения функции тромбоцитов и вытеснения непрямых антикоагулянтов из связи с белками плазмы;\u003Cbr\u003E- тромболитических средств и антиагрегантов;\u003Cbr\u003E- дигоксина вследствие снижения его почечной экскреции;\u003Cbr\u003E- гипогликемических средств (инсулина и производных сульфонилмочевины) за счет гипогликемических свойств самой ацетилсалициловой кислоты в высоких до¬зах и вытеснения производных сульфонилмочевины из связи с белками плазмы;\u003Cbr\u003E- вальпроевой кислоты за счет вытеснения ее из связи с белками плазмы.\u003Cbr\u003EСочетание ацетилсалициловой кислоты с антикоагулянтами, тромболитиками и антиагрегантами сопровождается повышенным риском развития кровотечения.\u003Cbr\u003EПри одновременном приеме ацетилсалициловой кислоты с алкоголем наблюдает¬ся усиление токсического действия алкоголя на центральную нервную систему, повышается риск повреждения слизистой оболочки желудочно-кишечного тракта и удлинения времени кровотечения.\u003Cbr\u003EАСК ослабляет действие урикозурических препаратов - бензбромарона (снижение урикозурического эффекта вследствие конкурентного подавления почечной канальцевой экскреции мочевой кислоты), ингибиторов ангиотензинпревращающего фер¬мента (АПФ) (отмечается дозозависимое снижение скорости клубочковой фильтрации в результате ингибирования простагландинов, обладающих сосудорасширяю-щим действием, соответственно ослабление гипотензивного действия), диуретиков (при совместном применении с АСК в высоких дозах отмечается снижение скорости клубочковой фильтрации в результате снижения синтеза простагландинов в почках).\u003Cbr\u003EУсиливая элиминацию салицилатов, системные глюкокортикостероиды(ГКС) ослабляют их действие."},{"name":"Регистрационный номер","value":"ЛС-000680"},{"name":"Дата государственной регистрации","value":"04.06.2013"},{"name":"Владелец регистрационного удостоверения","value":"Синтез"},{"name":"Изготовитель","value":"Синтез"},{"name":"Фасовщик","value":"Синтез"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Ацекардол"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_14210066621057973629"}}}}
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32 ₽

  • Сегодня, курьер магазина  249 ₽
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  • Рейтинг товара: 4.9 из 5
    на основе 142 оценки
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-qzvnhbdzc9q/addToCartButton":{"offerId":"_A74cT-lOG9oQEnGg1vKzw","skuId":"228089895","pendingCartItem":{"productId":1401075797,"offerId":"_A74cT-lOG9oQEnGg1vKzw","showPlaceId":"OTNDnItfwRMjN9MRHuEMMq1uNlkSxp0i7kzxAEdAVPkwlo__zEikJiQOAxwynrIhxBB7Qv77IKsZmAEcIEZzibexC-Ct9XiOVdJW7HzDaQVfHuoYWL-P2INuL1dAMQZK1kY-7HXfHaDP8NAqBAHlobrbpt_w_YdRm5epmRTngn8-Q2_8UD9v6CZDoguWxJVyeWwr33NOynxI5UkZ-vcY3g,,","feeShow":"OTNDnItfwRMjN9MRHuEMMq1uNlkSxp0i7kzxAEdAVPkwlo__zEikJiQOAxwynrIhxBB7Qv77IKsZmAEcIEZzibexC-Ct9XiOVdJW7HzDaQVfHuoYWL-P2INuL1dAMQZK1kY-7HXfHaDP8NAqBAHlobrbpt_w_YdRm5epmRTngn8-Q2_8UD9v6CZDoguWxJVyeWwr33NOynxI5UkZ-vcY3g,,","skuId":"228089895","shopId":11693184,"price":{"applicablePriceDiscounts":[{"priceWithDiscount":"149","type":"ya-card","totalPercentWithDiscount":1}],"value":"150","currency":"RUR"},"hid":"15756887","name":"Тромбо АСС таб. п/о плен. кш/раств., 100 мг, 100 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  • Рейтинг товара: 5 из 5
    на основе 23 оценки
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  • Рейтинг товара: 4.9 из 5
    на основе 28 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 62 оценки
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  • Рейтинг товара: 5 из 5
    на основе 20 оценок
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-fl5d4gtpqqn/addToCartButton":{"offerId":"Va7IZFLPuJAcDG0WThZf6Q","skuId":"228093566","pendingCartItem":{"productId":1401075806,"offerId":"Va7IZFLPuJAcDG0WThZf6Q","showPlaceId":"OTNDnItfwRMjN9MRHuEMMq1uNlkSxp0iKt-pIsqmHYNVqI12pf5ZJ68Vy6tdM90mjnagYLIYKLxxhelK5b5AvbIBH2Xw21sP60D8QYsbFpps3Mivr8QM2F22yIJ_7BlkrwZCfPsbE2mu2DCkFaYFSzMK4zzpRIgCiPypETww7FPOZHGag5pyx9lJ2QDfQG3bVAMBkRKS2xpQEAQgtX2H8Q,,","feeShow":"OTNDnItfwRMjN9MRHuEMMq1uNlkSxp0iKt-pIsqmHYNVqI12pf5ZJ68Vy6tdM90mjnagYLIYKLxxhelK5b5AvbIBH2Xw21sP60D8QYsbFpps3Mivr8QM2F22yIJ_7BlkrwZCfPsbE2mu2DCkFaYFSzMK4zzpRIgCiPypETww7FPOZHGag5pyx9lJ2QDfQG3bVAMBkRKS2xpQEAQgtX2H8Q,,","skuId":"228093566","shopId":11693184,"price":{"applicablePriceDiscounts":[{"priceWithDiscount":"213","type":"ya-card","totalPercentWithDiscount":1}],"value":"215","currency":"RUR"},"hid":"15756887","name":"Фазостабил таб. п/о плен., 75 мг+15.2 мг, 100 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  • Рейтинг товара: 5 из 5
    на основе 4 оценки
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  • Рейтинг товара: 4.3 из 5
    на основе 7 оценок
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  • Рейтинг товара: 4.8 из 5
    на основе 25 оценок
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  • Рейтинг товара: 4.8 из 5
    на основе 130 оценок
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Инструкция

Показания к применению

- профилактика острого инфаркта миокарда при наличии факторов риска (например, сахарный диабет, гиперлипидемия, артериальная гипертензия, ожирение, курение, пожилой возраст) и повторного инфаркта миокарда;
- нестабильная стенокардия;
- профилактика ишемического инсульта (в том числе у пациентов с преходящим нарушением мозгового кровообращения);
- профилактика тромбоэмболии после операций и инвазивных вмешательств на сосудах (например, аортокоронарное шунтирование, эндартерэктомия сонных арте¬рий, артериовенозное шунтирование, ангиопластика и стентирование коронарных артерий, ангиопластика сонных артерий);
- профилактика тромбоза глубоких вен и тромбоэмболии легочной артерии и ее ветвей (в том числе, при длительной иммобилизации в результате обширного хирургического вмешательства).

Противопоказания

Гиперчувствительность к АСК, эрозивно-язвенные поражения ЖКТ (в фазе обострения), желудочно-кишечное кровотечение, геморрагический диатез, бронхиальная астма, индуцированная приемом салицилатов, полное или неполное сочетание бронхиальной астмы, рецидивирующего полипоза носа и околоносовых пазух и непереносимости АСК, выраженная почечная недостаточность (клиренс креатинина (КК) менее 30 мл/мин), выраженная печеночная недостаточность (класс В и С по шкале Чайлд-Пью), хроническая сердечная недостаточность (III-IV функционального класса по классификации NYHA), одновременный прием метотрексата в дозе 15 мг/нед и более, беременность (I и III триместр), период лактации, детский возраст до 18 лет, дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция.

Способ применения и дозы

Таблетки препарата Ацекардол следует принимать перед едой, запивая большим количеством жидкости, 1 раз в сутки. Ацекардол предназначен для длительного применения. Длительность терапии определяется врачом.
Профилактика при подозрении острого инфаркта миокарда: 100 мг в сутки или 300 мг через день (первую таблетку необходимо разжевать для более быстрого всасывания).
Профилактика впервые возникшего острого инфаркта миокарда при наличии факторов риска: 100 мг в сутки или 300 мг через день.
Профилактика повторного инфаркта миокарда и нестабильная стенокардия: 100 - 300 мг в сутки.
Профилактика ишемического инсульта и преходящего нарушения мозгового кровообращения: 100 - 300 мг в сутки.
Профилактика тромбоэмболии после операций и инвазивных вмешательств на сосудах: 100 - 300 мг в сутки.
Профилактика тромбоза глубоких вен и тромбоэмболии легочной артерии и ее ветвей: 100 мг в сутки или 300 мг через день.
Полная инструкция
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Ацекардол таб. п/о плен. кш/раств.
Ацекардол таб. п/о плен. кш/раств., 100 мг, 30 шт.
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Инструкция

32 ₽

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