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Описание

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Эуфиллин таб., 150 мг, 30 шт.

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Детям внутрь следует назначать из расчета 7-10 мг/кг в сут в 4 приема. Длительность курса лечения - от нескольких дней до нескольких месяцев, в зависимости от течения заболевания и переносимости препарата. Высшие дозы эуфиллина для взрослых внутрь: разовая - 0,5 г, суточная - 1,5 г. Высшие дозы для детей внутрь: разовая - 7 мг/кг, суточная - 15 мг/кг."},{"name":"Побочные действия","value":"Со стороны нервной системы: головокружение, головная боль, бессонница, возбуждение, тревожность, раздражительность, тремор.\u003Cbr\u003E\nСо стороны сердечно-сосудистой системы: сердцебиение, тахикардия (в том числе у плода при приеме беременной в III триместре), аритмии, кардиалгия, снижение артериального давления, увеличение частоты приступов стенокардии.\u003Cbr\u003EСо стороны пищеварительной системы: гастралгия, тошнота, рвота, гастроэзофагеальный рефлюкс, изжога, обострение язвенной болезни, диарея, при длительном приеме - снижение аппетита.\u003Cbr\u003EАллергические реакции: кожная сыпь, зуд, лихорадка.\u003Cbr\u003EПрочие: боль в груди, тахипноэ, ощущение приливов к лицу, альбуминурия, гематурия, гипогликемия, усиление диуреза, повышенное потоотделение."},{"name":"Фармакологическое действие","value":"Эуфиллин - бронхолитическое средство, производное ксантина; ингибирует фосфодиэстеразу, увеличивает накопление в тканях циклического аденозинмонофосфата, блокирует аденозиновые (пуриновые) рецепторы; снижает поступление ионов кальция через каналы клеточных мембран, уменьшает сократительную активность гладкой мускулатуры.\u003Cbr\u003E\nРасслабляет мускулатуру бронхов, увеличивает мукоцилиарный клиренс, стимулирует сокращение диафрагмы, улучшает функцию дыхательных и межреберных мышц, стимулирует дыхательный центр, повышает его чувствительность к углекислому газу и улучшает альвеолярную вентиляцию, что в конечном итоге приводит к снижению тяжести и частоты эпизодов апноэ. Нормализуя дыхательную функцию, способствует насыщению крови кислородом и снижению концентрации углекислоты.\u003Cbr\u003EОказывает стимулирующее влияние на деятельность сердца, увеличивает силу и число сердечных сокращений, повышает коронарный кровоток и потребность миокарда в кислороде. Снижает тонус кровеносных сосудов (главным образом, сосудов мозга, кожи и почек).\u003Cbr\u003EОказывает периферическое венодилатирующее действие, уменьшает легочное сосудистое сопротивление, снижает давление в \"малом\" круге кровообращения.\u003Cbr\u003EУвеличивает почечный кровоток, оказывает умеренный диуретический эффект.\u003Cbr\u003EРасширяет внепеченочные желчные пути.\u003Cbr\u003EТормозит агрегацию тромбоцитов (подавляет фактор активации тромбоцитов и PgE2 альфа), повышает устойчивость эритроцитов к деформации (улучшает реологические свойства крови), уменьшает тромбообразование и нормализует микроциркуляцию.\u003Cbr\u003EОбладает токолитическим действием, повышает кислотность желудочного сока.\u003Cbr\u003EПри использовании в больших дозах обладает энилептогенным действием."},{"name":"Фармакологическая группа","value":"бронходилатирующее средство - фосфодиэстеразы ингибитор"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-astmy","categoryId":"15756897","navnodeId":"72498","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 3 лет"},{"name":"Условия хранения","value":"В защищенном от света месте, при температуре не выше 25°С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: снижение аппетита, гастралгия, диарея, тошнота, рвота (в том числе с кровью), желудочно-кишечное кровотечение, тахипноэ, гиперемия кожи лица, тахикардия, желудочковые аритмии, бессонница, двигательное возбуждение, тревожность, светобоязнь, тремор, судороги. При тяжелом отравлении могут развиться эпилептоидные припадки (особенно у детей без возникновения каких-либо предвестников), гипоксия, метаболический ацидоз, гипергликемия, гипокалиемия, снижение артериального давления, некроз скелетных мышц, спутанность сознания, почечная недостаточность с миоглобинурией.\u003Cbr\u003EЛечение: отмена препарата, промывание желудка, применение активированного угля, слабительных лекарственных средств, промывание кишечника комбинацией полиэтиленгликоля и электролитов, форсированный диурез, гемосорбция, плазмосорбция, гемодиализ (эффективность не высока, перитонеальный диализ не эффективен), симптоматическая терапия (в том числе метоклопрамид и ондансетрон - при рвоте). При возникновении судорог поддерживать проходимость дыхательных путей и проводить оксигенотерапию. Для купирования припадка - в/в диазепам 0,1-0,3 мг/кг (но не более 10 мг). При сильной тошноте и рвоте - метоклопрамид или ондансетрон (в/в)."},{"name":"Применение при беременности и кормлении грудью","value":"С осторожностью беременность, период лактации."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо воздерживаться от вождения транспорта и занятий другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Соблюдать осторожность при употреблении больших количеств кофеинсодержащих продуктов или напитков."},{"name":"Взаимодействие","value":"Повышает вероятность развития побочных эффектов глюкокортикостероидов, минералокортикостероидов (гипернатриемия), средств для общей анестезии (возрастает риск возникновения желудочковых аритмий), ксантинов и средств, возбуждающих центральную нервную систему (увеличивает нейротоксичность), бета-адреностимуляторов.\u003Cbr\u003E\nПротиводиарейные препараты и энтеросорбенты снижают всасывание аминофиллина.\u003Cbr\u003E\nРифампицин, фенобарбитал, фенитоин, изониазид, карбамазепин, сульфинпиразон, аминоглутетимид, пероральные эстрогенсодержащие контрацептивы и морацизин, являясь индукторами микросомальных ферментов печени, повышают клиренс аминофиллина, что может потребовать увеличения его дозы.\u003Cbr\u003EПри одновременном применении с антибиотиками группы макролидов, линкомицином, аллопуринолом, циметидином, изопреналином, эноксацином, небольшими дозами этанола, дисульфирамом, фторхинолонами, рекомбинантным интерфероном-альфа, метотрексатом, мексилетином, пропафеноном, тиабендазолом, тиклопидином, верапамилом и при вакцинации против гриппа интенсивность действия аминофиллина может увеличиваться, что может потребовать снижения его дозы.\u003Cbr\u003EУсиливает действие бета-адреностимуляторов и диуретиков (в том числе за счет увеличения клубочковой фильтрации), снижает эффективность препаратов лития и бета-адреноблокаторов.\u003Cbr\u003EСовместим со спазмолитиками, не применяют совместно с другими производными ксантина."},{"name":"Регистрационный номер","value":"ЛП-003432"},{"name":"Дата государственной регистрации","value":"09.02.2021"},{"name":"Владелец регистрационного удостоверения","value":"Усолье-Сибирский химфармзавод","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-astmy","categoryId":"15756897","navnodeId":"72498","glfilters":["34324371:35649313","7893318:16003123"]}}},{"name":"Изготовитель","value":"Усолье-Сибирский химфармзавод"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Эуфиллин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-astmy","categoryId":"15756897","navnodeId":"72498","glfilters":["17796364:18053304"]}}},{"name":"Срок годности","value":"61 мес."}]}},"fullSpecsGrouped":{"7305927362138408868":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"дыхательная система"},{"name":"Назначение","value":"\"легочное\" сердце, бронхиальная астма, бронхит, ночное апноэ, хроническая обструктивная болезнь легких, эмфизема легких"},{"name":"Показания к применению","value":"Бронхообструктивный синдром любого генеза: бронхиальная астма (препарат выбора у больных с астмой физического напряжения и как дополнительное средство при др. формах), хроническая обструктивная болезнь легких, эмфизема легких, хронический обструктивный бронхит, легочная гипертензия, \"легочное\" сердце, ночное апноэ."},{"name":"Противопоказания","value":"Гиперчувствительность (в том числе к другим производным ксантина: кофеин, пентоксифиллин, теобромин), эпилепсия, язвенная болезнь желудка и двенадцатиперстной кишки (в стадии обострения), гастрит с повышенной кислотностью, артериальная гипер- или гипотензия тяжелого течения, тахиаритмии, геморрагический инсульт, кровоизлияние в сетчатку глаза, детский возраст (до 3 лет)."},{"name":"Состав","value":"Активные вещества: аминофиллин 150 мг;\u003Cbr\u003Eвспомогательные вещества: крахмал картофельный - 48,0 мг, кальция стеарат - 2,0 мг."},{"name":"Действующее вещество","value":"Аминофиллин"},{"name":"Способ применения и дозы","value":"Внутрь, взрослым Эуфиллин следует назначать по 150 мг на прием 1-3 раза в день после еды. Детям внутрь следует назначать из расчета 7-10 мг/кг в сут в 4 приема. Длительность курса лечения - от нескольких дней до нескольких месяцев, в зависимости от течения заболевания и переносимости препарата. Высшие дозы эуфиллина для взрослых внутрь: разовая - 0,5 г, суточная - 1,5 г. Высшие дозы для детей внутрь: разовая - 7 мг/кг, суточная - 15 мг/кг."},{"name":"Побочные действия","value":"Со стороны нервной системы: головокружение, головная боль, бессонница, возбуждение, тревожность, раздражительность, тремор.\u003Cbr\u003E\nСо стороны сердечно-сосудистой системы: сердцебиение, тахикардия (в том числе у плода при приеме беременной в III триместре), аритмии, кардиалгия, снижение артериального давления, увеличение частоты приступов стенокардии.\u003Cbr\u003EСо стороны пищеварительной системы: гастралгия, тошнота, рвота, гастроэзофагеальный рефлюкс, изжога, обострение язвенной болезни, диарея, при длительном приеме - снижение аппетита.\u003Cbr\u003EАллергические реакции: кожная сыпь, зуд, лихорадка.\u003Cbr\u003EПрочие: боль в груди, тахипноэ, ощущение приливов к лицу, альбуминурия, гематурия, гипогликемия, усиление диуреза, повышенное потоотделение."},{"name":"Фармакологическое действие","value":"Эуфиллин - бронхолитическое средство, производное ксантина; ингибирует фосфодиэстеразу, увеличивает накопление в тканях циклического аденозинмонофосфата, блокирует аденозиновые (пуриновые) рецепторы; снижает поступление ионов кальция через каналы клеточных мембран, уменьшает сократительную активность гладкой мускулатуры.\u003Cbr\u003E\nРасслабляет мускулатуру бронхов, увеличивает мукоцилиарный клиренс, стимулирует сокращение диафрагмы, улучшает функцию дыхательных и межреберных мышц, стимулирует дыхательный центр, повышает его чувствительность к углекислому газу и улучшает альвеолярную вентиляцию, что в конечном итоге приводит к снижению тяжести и частоты эпизодов апноэ. Нормализуя дыхательную функцию, способствует насыщению крови кислородом и снижению концентрации углекислоты.\u003Cbr\u003EОказывает стимулирующее влияние на деятельность сердца, увеличивает силу и число сердечных сокращений, повышает коронарный кровоток и потребность миокарда в кислороде. Снижает тонус кровеносных сосудов (главным образом, сосудов мозга, кожи и почек).\u003Cbr\u003EОказывает периферическое венодилатирующее действие, уменьшает легочное сосудистое сопротивление, снижает давление в \"малом\" круге кровообращения.\u003Cbr\u003EУвеличивает почечный кровоток, оказывает умеренный диуретический эффект.\u003Cbr\u003EРасширяет внепеченочные желчные пути.\u003Cbr\u003EТормозит агрегацию тромбоцитов (подавляет фактор активации тромбоцитов и PgE2 альфа), повышает устойчивость эритроцитов к деформации (улучшает реологические свойства крови), уменьшает тромбообразование и нормализует микроциркуляцию.\u003Cbr\u003EОбладает токолитическим действием, повышает кислотность желудочного сока.\u003Cbr\u003EПри использовании в больших дозах обладает энилептогенным действием."},{"name":"Фармакологическая группа","value":"бронходилатирующее средство - фосфодиэстеразы ингибитор"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 3 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В защищенном от света месте, при температуре не выше 25°С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: снижение аппетита, гастралгия, диарея, тошнота, рвота (в том числе с кровью), желудочно-кишечное кровотечение, тахипноэ, гиперемия кожи лица, тахикардия, желудочковые аритмии, бессонница, двигательное возбуждение, тревожность, светобоязнь, тремор, судороги. При тяжелом отравлении могут развиться эпилептоидные припадки (особенно у детей без возникновения каких-либо предвестников), гипоксия, метаболический ацидоз, гипергликемия, гипокалиемия, снижение артериального давления, некроз скелетных мышц, спутанность сознания, почечная недостаточность с миоглобинурией.\u003Cbr\u003EЛечение: отмена препарата, промывание желудка, применение активированного угля, слабительных лекарственных средств, промывание кишечника комбинацией полиэтиленгликоля и электролитов, форсированный диурез, гемосорбция, плазмосорбция, гемодиализ (эффективность не высока, перитонеальный диализ не эффективен), симптоматическая терапия (в том числе метоклопрамид и ондансетрон - при рвоте). При возникновении судорог поддерживать проходимость дыхательных путей и проводить оксигенотерапию. Для купирования припадка - в/в диазепам 0,1-0,3 мг/кг (но не более 10 мг). При сильной тошноте и рвоте - метоклопрамид или ондансетрон (в/в)."},{"name":"Применение при беременности и кормлении грудью","value":"С осторожностью беременность, период лактации."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо воздерживаться от вождения транспорта и занятий другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Соблюдать осторожность при употреблении больших количеств кофеинсодержащих продуктов или напитков."},{"name":"Взаимодействие","value":"Повышает вероятность развития побочных эффектов глюкокортикостероидов, минералокортикостероидов (гипернатриемия), средств для общей анестезии (возрастает риск возникновения желудочковых аритмий), ксантинов и средств, возбуждающих центральную нервную систему (увеличивает нейротоксичность), бета-адреностимуляторов.\u003Cbr\u003E\nПротиводиарейные препараты и энтеросорбенты снижают всасывание аминофиллина.\u003Cbr\u003E\nРифампицин, фенобарбитал, фенитоин, изониазид, карбамазепин, сульфинпиразон, аминоглутетимид, пероральные эстрогенсодержащие контрацептивы и морацизин, являясь индукторами микросомальных ферментов печени, повышают клиренс аминофиллина, что может потребовать увеличения его дозы.\u003Cbr\u003EПри одновременном применении с антибиотиками группы макролидов, линкомицином, аллопуринолом, циметидином, изопреналином, эноксацином, небольшими дозами этанола, дисульфирамом, фторхинолонами, рекомбинантным интерфероном-альфа, метотрексатом, мексилетином, пропафеноном, тиабендазолом, тиклопидином, верапамилом и при вакцинации против гриппа интенсивность действия аминофиллина может увеличиваться, что может потребовать снижения его дозы.\u003Cbr\u003EУсиливает действие бета-адреностимуляторов и диуретиков (в том числе за счет увеличения клубочковой фильтрации), снижает эффективность препаратов лития и бета-адреноблокаторов.\u003Cbr\u003EСовместим со спазмолитиками, не применяют совместно с другими производными ксантина."},{"name":"Регистрационный номер","value":"ЛП-003432"},{"name":"Дата государственной регистрации","value":"09.02.2021"},{"name":"Владелец регистрационного удостоверения","value":"Усолье-Сибирский химфармзавод"},{"name":"Изготовитель","value":"Усолье-Сибирский химфармзавод"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Эуфиллин"},{"name":"Срок годности","value":"61 мес."}]}],"transitionId":"tr_11572573475447121411"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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Ещё может подойти

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Инструкция

Показания к применению

Бронхообструктивный синдром любого генеза: бронхиальная астма (препарат выбора у больных с астмой физического напряжения и как дополнительное средство при др. формах), хроническая обструктивная болезнь легких, эмфизема легких, хронический обструктивный бронхит, легочная гипертензия, "легочное" сердце, ночное апноэ.

Противопоказания

Гиперчувствительность (в том числе к другим производным ксантина: кофеин, пентоксифиллин, теобромин), эпилепсия, язвенная болезнь желудка и двенадцатиперстной кишки (в стадии обострения), гастрит с повышенной кислотностью, артериальная гипер- или гипотензия тяжелого течения, тахиаритмии, геморрагический инсульт, кровоизлияние в сетчатку глаза, детский возраст (до 3 лет).

Способ применения и дозы

Внутрь, взрослым Эуфиллин следует назначать по 150 мг на прием 1-3 раза в день после еды. Детям внутрь следует назначать из расчета 7-10 мг/кг в сут в 4 приема. Длительность курса лечения - от нескольких дней до нескольких месяцев, в зависимости от течения заболевания и переносимости препарата. Высшие дозы эуфиллина для взрослых внутрь: разовая - 0,5 г, суточная - 1,5 г. Высшие дозы для детей внутрь: разовая - 7 мг/кг, суточная - 15 мг/кг.
Полная инструкция
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Эуфиллин таб.
Эуфиллин таб., 150 мг, 30 шт.
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Инструкция

29 ₽

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1.0
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