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Амлодипин-Прана таб., 10 мг, 90 шт.

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Количество штук в упаковке, шт.: 90

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Коротко о товаре

Инструкция
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гипертензия","transition":{"type":"list","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["36476390:36619024,36618715,36618511,36618237,36617589"]}}},{"name":"действующее вещество","value":"Амлодипин","transition":{"type":"list","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28709386"]}}},{"name":"возраст","value":"от 18 лет"},{"name":"форма выпуска","value":"таблетки"},{"name":"страна-производитель","value":"Россия"}]}},"compactSpecs":{"16872425295943092503":{"specItems":[{"name":"Артикул Маркета","value":"3288356885","withCopyValueButton":true},{"name":"Тип препарата","value":"Рецептурный лекарственный препарат","transition":{"type":"list","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27272850:1,0","34324371:35649313"]}}},{"name":"Действующее вещество","value":"Амлодипин","transition":{"type":"list","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28709386"]}}},{"name":"Возраст","value":"От 18 лет"},{"name":"Форма выпуска","value":"Таблетки"}]}},"fullSpecs":{"16872425295943092503":{"specItems":[{"name":"Тип препарата","value":"лекарственный препарат","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313"]}}},{"name":"Рецептурный препарат","value":"да","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27272850:1,0"]}}},{"name":"Органы и системы","value":"кровеносная система, кровеносные сосуды, сердце"},{"name":"Назначение","value":"артериальная гипертензия, гипертония, стенокардия, стенокардия Принцметала, эссенциальная гипертензия","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["36476390:36619024,36618715,36618511,36618237,36617589"]}}},{"name":"Показания к применению","value":"Артериальная гипертензия (монотерапия или в комбинации с другими антигипертензивными средствами).\u003Cbr\u003EСтабильная стенокардия напряжения и вазоспастическая стенокардия (стенокардия Принцметала) (монотерапия или в комбинации с другими антиангинальными средствами)."},{"name":"Противопоказания","value":"Повышенная чувствительность к амлодипину, производным дигидропиридина и другим компонентам препарата;\u003Cbr\u003Eвыраженная артериальная гипотензия (систолическое АД менее 90 мм рт.ст.);\u003Cbr\u003Eколлапс, кардиогенный шок;\u003Cbr\u003Eнестабильная стенокардия (за исключением стенокардии Принцметала);\u003Cbr\u003Eклинически значимый стеноз аорты;\u003Cbr\u003Eбеременность и период лактации;\u003Cbr\u003Eвозраст до 18 лет (эффективность и безопасность не изучены);\u003Cbr\u003Eнепереносимость лактозы, дефицит лактазы или глюкозо-галактозная мальабсорбция.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EНарушениях функции печени, синдроме слабости синусового узла (выраженная брадикардия, тахикардия), хронической сердечной недостаточности неишемической этиологии III-1V функционального класса по классификации NYHA, артериальной гипотензии, аортальном стенозе, митральном стенозе, гипертрофической обструктивной кардиомиопатии (ГОКМП), остром инфаркте миокарда (и в течение 1 месяца после инфаркта миокарда), в пожилом возрасте."},{"name":"Состав","value":"Каждая таблетка содержит:\u003Cbr /\u003Eв качестве активного компонента: амлодипина безилата 6,93 мг и 13,86 мг, что соответствует 5 мг и 10 мг амлодипина.\u003Cbr /\u003Eвспомогательные вещества: крахмал кукурузный, лактоза, целлюлоза микрокристаллическая, магния стеарат"},{"name":"Действующее вещество","value":"Амлодипин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28709386"]}}},{"name":"Способ применения и дозы","value":"Внутрь, начальная доза для лечения артериальной гипертензии и стенокардии составляет 5 мг препарата 1 раз в сутки. Доза максимально может быть увеличена до 10 мг 1 раз в сутки. При артериальной гипертензии поддерживающая доза может быть 2,5 - 5 мг (1/2 таблетки по 5 мг - 1 таблетка по 5 мг) в сутки.\u003Cbr\u003EУ пациентов пожилого возраста может увеличиваться Т1/2 амлодипина и снижаться клиренс креатинина (КК). Изменения доз не требуется, но необходимо более тщательное наблюдение за пациентами.\u003Cbr\u003EНе требуется изменения дозы при одновременном назначении с тиазидными диуретиками, бета-адреноблокаторам и ингибиторами ангиотензинпревращающего фермента (АГ1Ф).\u003Cbr\u003EНe требуется изменения дозы у пациентов с почечной недостаточностью."},{"name":"Побочные действия","value":"Со стороны сердечно-сосудистой системы: часто - сердцебиение, периферические отеки (отечность лодыжек и стоп), \"приливы\" крови к коже лица: иногда - чрезмерное снижение АД; очень редко - обморок, одышка, васкулит, ортостатическая гипотензия, развитие или усугубление течения сердечной недостаточности, нарушения ритма сердца (включая брадикардию, желудочковую тахикардию и мерцание предсердии), инфаркт миокарда, боли в грудной клетке.\u003Cbr\u003EСо стороны центральной и периферической нервной системы: часто - головная боль, головокружение, повышенная утомляемость, сонливость; иногда - астения, общее недомогание, гипестезии, парестезии, периферическая нейропатия, тремор, бессонница, лабильность настроения, необычные сновидения, повышенная возбудимость, депрессия, тревожность, очей редко - мигрень, повышенное потоотделение, апатия.\u003Cbr\u003EСо стороны пищеварительной системы: часто - тошнота, боли в животе; иногда - рвота, запор или диарея, метеоризм, диспепсия, анорексия, сухость слизистой оболочки полости рта, жажда; редко - гиперплазия десен, повышение аппетита; очень редко - панкреатит, гастрит, желтуха (обусловленные холестазом), гипербилирубинемия, повышение активности \"печеночных\" трансаминаз, гепатит.\u003Cbr\u003EСо стороны органов кроветворения: очень редко - тромбоцитопеническая пурпура, лейкопения, тромбоцитопения.\u003Cbr\u003EСо стороны мочеполовой системы: иногда - учащенное мочеиспускание, болезненное мочеиспускание, никтурия, импотенция, очень редко - дизурия, полиурия.\u003Cbr\u003EСо стороны дыхательном системы: иногда - одышка, ринит, очень редко - кашель.\u003Cbr\u003EСо стороны кожных покровов: редко - дерматит, очень редко - алопеция, ксеродермия, холодный пот, нарушение пигментации кожи.\u003Cbr\u003EАллергические реакции: кожный зуд, сыпь (в том числе эритематозная, макулопапулезная сыпь, крапивница), ангионевротический отек, мультиформная эритема.\u003Cbr\u003EСо стороны опорно-двигательного аппарата: иногда - мышечные судороги, миалгия, артралгия, боль в спине, артроз, редко - миастения.\u003Cbr\u003EПрочие: иногда - звон в ушах, диплопия, нарушение аккомодации, ксерофтальмия, конъюнктивит, боль в глазах, озноб, носовое кровотечение, гинекомастия, очень редко - паросмия, гипергликемия."},{"name":"Фармакологическое действие","value":"Производное дигидропиридина - блокатор \"медленных\" кальциевых каналов (БМКК) II поколения, оказывает антиангинальное и гипотензивное действие. Связываясь с дигидропиридиновыми рецепторами, блокирует кальциевые каналы, снижает трансмембранный переход ионов кальция в клетку (в большей степени в гладкомышечные клетки сосудов, чем в кардиомиоциты).\u003Cbr\u003EАнтиангинальное действие обусловлено расширением коронарных и периферических артерий и артериол: при стенокардии уменьшает выраженность ишемии миокарда; расширяя периферические артериолы, снижает общее периферическое сосудистое сопротивление (ОПСС), уменьшает пред нагрузку на сердце, снижает потребность миокарда в кислороде. Расширяет главные коронарные артерии и артериолы в неизмененных и ишемизированных зонах миокарда, увеличивает поступление кислорода в миокард (особенно при вазоспастической стенокардии); предотвращает развитие спазма коронарных артерий (в т.ч. вызванного курением). У больных стабильной стенокардией разовая суточная доза увеличивает толерантность к физической нагрузке, замедляет развитие стенокардии и \"ишемической\" депрессии сегмента ST, снижает частоту приступов стенокардии и потребления нитроглицерина и других нитратов. \u003Cbr\u003EОказывает длительный дозозависимый гипотензивный эффект. Гипотензивное действие обусловлено прямым вазодилатирующим влиянием на гладкие мышцы сосудов. При артериальной гипертензии разовая доза обеспечивает клинически значимое снижение артериального давления (АД) на протяжении 24 ч (в положении больного \"лежа\" и \"стоя\"). Ортостатическая гипотензия при назначении амлодипина встречается достаточно редко. Не вызывает снижения толерантности к физической нагрузке, фракции выброса левого желудочка. Уменьшает степень гипертрофии миокарда левого желудочка. Не оказывает влияния на сократимость и проводимость миокарда, нс вызывает рефлекторного увеличения частоты сердечных сокращений (ЧСС), тормозит агрегацию тромбоцитов, повышает скорость клубочковой фильтрации, обладает слабым натрийуретическим действием. При диабетической нефропатии не увеличивает выраженность микроальбуминурии. Не оказывает какого-либо неблагоприятного влияния на обмен веществ и концентрацию липидов плазмы крови и может применяться при лечении больных бронхиальной астмой, сахарным диабетом и подагрой. Значимое снижение АД наблюдается через 6-10 часов, длительность эффекта 24 часа."},{"name":"Фармакологическая группа","value":"блокатор \"медленных\" кальциевых каналов"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"В сухом, защищенном от света месте, при температуре не выше 25°С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: чрезмерная периферическая вазодилатация с выраженным и возможно длительным снижением АД, коллапс, шок.\u003Cbr\u003EЛечение: промывание желудка, назначение активированного угля, поддержание функции сердечно-сосудистой системы, контроль показателей функции сердца и легких, приподнятое, выше уровня головы, положение нижних конечностей, контроль объема циркулирующей крови и диуреза. Для восстановления тонуса сосудов - применение сосудосуживающих средств (при отсутствии противопоказаний к их применению); с целью устранения последствий блокады кальциевых каналов - внутривенное введение кальция глюконата. Гемодиализ неэффективен."},{"name":"Применение при беременности и кормлении грудью","value":"Безопасность применения амлодипина при беременности и в период кормления грудью не установлена, поэтому препарат амлодипин не следует назначать беременным и в период лактации."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения следует соблюдать осторожность при вождении автотранспорта и занятии потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"В период лечения препаратом необходимо контролировать массу тела и потребление натрия, назначение соответствующей диеты. Необходимо поддержание гигиены зубов и наблюдение у стоматолога (для предотвращения болезненности, кровоточивости и гиперплазии десен).\u003Cbr\u003EПациентам с малой массой тела, пациентам невысокого роста и больным с выраженным нарушением функции печени может потребоваться меньшая доза.\u003Cbr\u003EУ пожилых пациентов может удлиняться T1/2 и клиренс препарата. Изменения доз для пожилых пациентов нс требуется; при увеличении дозы необходимо более тщательное наблюдение за пациентами.\u003Cbr\u003EПри нарушении функции печени также может удлиняться Т1/2 препарата. Поэтому таким пациентам препарат необходимо назначать с осторожностью. Несмотря на то, что прекращение приема препарата не сопровождается развитием синдрома \"отмены\", прекращение лечения желательно проводить, постепенно уменьшая дозу препарата. Эффективность и безопасность препарата при гипертензивном кризе не установлена."},{"name":"Взаимодействие","value":"Амлодипин может безопасно применяться для лечения артериальной гипертензии вместе с тиазидными диуретиками, альфа-адреноблокаторами, бета-адреноблокаторами или ингибиторами АПФ. У пациентов со стабильной стенокардией препарат можно комбинировать с другими антиангинальными средствами, например, с нитратами пролонгированного или короткого действия, бета-адреноблокаторами.\u003Cbr\u003EАмлодипин можно одновременно применять с нестероидными противовоспалительными препаратами (НПВП) (особенно индометацином), антибактериальными средствами и гипогликемическими средствами для приема внутрь. \u003Cbr\u003EВозможно усиление антиангинального и гипотензивного действия БМКК при совместном применении с тиазидными и \"петлевыми\" диуретиками, верапамилом, ингибиторами АПФ, бета-адреноблокаторами и нитратами, а так же усиление их гипотензивного действия при совместном применении с альфа 1 -адреноблокаторами, нейролептиками. \u003Cbr\u003EХотя при изучении амлодипина отрицательного инотропного действия обычно не наблюдали, тем не менее, некоторые БМКК могут усиливать выраженность отрицательного инотропного действия антиаритмических средств и вызывающих удлинение интервала QT (например, амиодарон и хинидин). \u003Cbr\u003EОднократный прием 100 мг силденафила у больных эссенциальной гипертензией не оказывает влияния на параметры фармакокинетики амлодипина. \u003Cbr\u003EПовторное применение амлодипина в дозе 10 мг и аторвастатина в дозе 80 мг не сопровождается значительными изменениями показателей фармакокинетики аторвастатина. \u003Cbr\u003EЭтанол (напитки, содержащие алкоголь): амлодипин при однократном и повторном применении в дозе 10 мг не влияет на фармакокинетику этанола. Противовирусные средства (ритонавир) увеличивает плазменные концентрации БМКК, в т.ч. амлодипина. \u003Cbr\u003EНейролептики и изофлуран - усиление гипотензивного действия производных дигидропиридина. \u003Cbr\u003EПрепараты кальция могут уменьшать эффект БМКК. \u003Cbr\u003EПри совместном применении амлодипина с препаратами лития возможно усиление проявления нейротоксичности (тошнота, рвота, диарея, атаксия, тремор, шум в ушах). \u003Cbr\u003EАмлодипин не изменяет фармакокинетику циклоспорина. \u003Cbr\u003EНе оказывает влияние на концентрацию в сыворотке крови дигоксина и его почечный клиренс. \u003Cbr\u003EНе оказывает существенного влияние на действие варфарина (протромбиновое время). \u003Cbr\u003EЦиметидин не влияет на фармакокинетику амлодипина. \u003Cbr\u003EВ исследованиях in vitro амлодипин не влияет на связывание с белками крови дигоксина, фенитоина, варфарина и индометацина. \u003Cbr\u003EГрейпфрутовый сок: одновременный однократный прием 240 мг грейпфрутового сока и 10 мг амлодипина внутрь не сопровождается существенным изменением фармакокинетики амлодипина."},{"name":"Регистрационный номер","value":"ЛСР-000849/10"},{"name":"Дата государственной регистрации","value":"16.05.2017"},{"name":"Владелец регистрационного удостоверения","value":"ПРАНАФАРМ","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313","7893318:12507927"]}}},{"name":"Изготовитель","value":"ПРАНАФАРМ"},{"name":"Фасовщик","value":"ПРАНАФАРМ"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Амлодипин-Прана","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["17796364:18020738"]}}},{"name":"Срок годности","value":"507 дн."}]}},"fullSpecsGrouped":{"16872425295943092503":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"кровеносная система, кровеносные сосуды, сердце"},{"name":"Назначение","value":"артериальная гипертензия, гипертония, стенокардия, стенокардия Принцметала, эссенциальная гипертензия"},{"name":"Показания к применению","value":"Артериальная гипертензия (монотерапия или в комбинации с другими антигипертензивными средствами).\u003Cbr\u003EСтабильная стенокардия напряжения и вазоспастическая стенокардия (стенокардия Принцметала) (монотерапия или в комбинации с другими антиангинальными средствами)."},{"name":"Противопоказания","value":"Повышенная чувствительность к амлодипину, производным дигидропиридина и другим компонентам препарата;\u003Cbr\u003Eвыраженная артериальная гипотензия (систолическое АД менее 90 мм рт.ст.);\u003Cbr\u003Eколлапс, кардиогенный шок;\u003Cbr\u003Eнестабильная стенокардия (за исключением стенокардии Принцметала);\u003Cbr\u003Eклинически значимый стеноз аорты;\u003Cbr\u003Eбеременность и период лактации;\u003Cbr\u003Eвозраст до 18 лет (эффективность и безопасность не изучены);\u003Cbr\u003Eнепереносимость лактозы, дефицит лактазы или глюкозо-галактозная мальабсорбция.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EНарушениях функции печени, синдроме слабости синусового узла (выраженная брадикардия, тахикардия), хронической сердечной недостаточности неишемической этиологии III-1V функционального класса по классификации NYHA, артериальной гипотензии, аортальном стенозе, митральном стенозе, гипертрофической обструктивной кардиомиопатии (ГОКМП), остром инфаркте миокарда (и в течение 1 месяца после инфаркта миокарда), в пожилом возрасте."},{"name":"Состав","value":"Каждая таблетка содержит:\u003Cbr /\u003Eв качестве активного компонента: амлодипина безилата 6,93 мг и 13,86 мг, что соответствует 5 мг и 10 мг амлодипина.\u003Cbr /\u003Eвспомогательные вещества: крахмал кукурузный, лактоза, целлюлоза микрокристаллическая, магния стеарат"},{"name":"Действующее вещество","value":"Амлодипин"},{"name":"Способ применения и дозы","value":"Внутрь, начальная доза для лечения артериальной гипертензии и стенокардии составляет 5 мг препарата 1 раз в сутки. Доза максимально может быть увеличена до 10 мг 1 раз в сутки. При артериальной гипертензии поддерживающая доза может быть 2,5 - 5 мг (1/2 таблетки по 5 мг - 1 таблетка по 5 мг) в сутки.\u003Cbr\u003EУ пациентов пожилого возраста может увеличиваться Т1/2 амлодипина и снижаться клиренс креатинина (КК). Изменения доз не требуется, но необходимо более тщательное наблюдение за пациентами.\u003Cbr\u003EНе требуется изменения дозы при одновременном назначении с тиазидными диуретиками, бета-адреноблокаторам и ингибиторами ангиотензинпревращающего фермента (АГ1Ф).\u003Cbr\u003EНe требуется изменения дозы у пациентов с почечной недостаточностью."},{"name":"Побочные действия","value":"Со стороны сердечно-сосудистой системы: часто - сердцебиение, периферические отеки (отечность лодыжек и стоп), \"приливы\" крови к коже лица: иногда - чрезмерное снижение АД; очень редко - обморок, одышка, васкулит, ортостатическая гипотензия, развитие или усугубление течения сердечной недостаточности, нарушения ритма сердца (включая брадикардию, желудочковую тахикардию и мерцание предсердии), инфаркт миокарда, боли в грудной клетке.\u003Cbr\u003EСо стороны центральной и периферической нервной системы: часто - головная боль, головокружение, повышенная утомляемость, сонливость; иногда - астения, общее недомогание, гипестезии, парестезии, периферическая нейропатия, тремор, бессонница, лабильность настроения, необычные сновидения, повышенная возбудимость, депрессия, тревожность, очей редко - мигрень, повышенное потоотделение, апатия.\u003Cbr\u003EСо стороны пищеварительной системы: часто - тошнота, боли в животе; иногда - рвота, запор или диарея, метеоризм, диспепсия, анорексия, сухость слизистой оболочки полости рта, жажда; редко - гиперплазия десен, повышение аппетита; очень редко - панкреатит, гастрит, желтуха (обусловленные холестазом), гипербилирубинемия, повышение активности \"печеночных\" трансаминаз, гепатит.\u003Cbr\u003EСо стороны органов кроветворения: очень редко - тромбоцитопеническая пурпура, лейкопения, тромбоцитопения.\u003Cbr\u003EСо стороны мочеполовой системы: иногда - учащенное мочеиспускание, болезненное мочеиспускание, никтурия, импотенция, очень редко - дизурия, полиурия.\u003Cbr\u003EСо стороны дыхательном системы: иногда - одышка, ринит, очень редко - кашель.\u003Cbr\u003EСо стороны кожных покровов: редко - дерматит, очень редко - алопеция, ксеродермия, холодный пот, нарушение пигментации кожи.\u003Cbr\u003EАллергические реакции: кожный зуд, сыпь (в том числе эритематозная, макулопапулезная сыпь, крапивница), ангионевротический отек, мультиформная эритема.\u003Cbr\u003EСо стороны опорно-двигательного аппарата: иногда - мышечные судороги, миалгия, артралгия, боль в спине, артроз, редко - миастения.\u003Cbr\u003EПрочие: иногда - звон в ушах, диплопия, нарушение аккомодации, ксерофтальмия, конъюнктивит, боль в глазах, озноб, носовое кровотечение, гинекомастия, очень редко - паросмия, гипергликемия."},{"name":"Фармакологическое действие","value":"Производное дигидропиридина - блокатор \"медленных\" кальциевых каналов (БМКК) II поколения, оказывает антиангинальное и гипотензивное действие. Связываясь с дигидропиридиновыми рецепторами, блокирует кальциевые каналы, снижает трансмембранный переход ионов кальция в клетку (в большей степени в гладкомышечные клетки сосудов, чем в кардиомиоциты).\u003Cbr\u003EАнтиангинальное действие обусловлено расширением коронарных и периферических артерий и артериол: при стенокардии уменьшает выраженность ишемии миокарда; расширяя периферические артериолы, снижает общее периферическое сосудистое сопротивление (ОПСС), уменьшает пред нагрузку на сердце, снижает потребность миокарда в кислороде. Расширяет главные коронарные артерии и артериолы в неизмененных и ишемизированных зонах миокарда, увеличивает поступление кислорода в миокард (особенно при вазоспастической стенокардии); предотвращает развитие спазма коронарных артерий (в т.ч. вызванного курением). У больных стабильной стенокардией разовая суточная доза увеличивает толерантность к физической нагрузке, замедляет развитие стенокардии и \"ишемической\" депрессии сегмента ST, снижает частоту приступов стенокардии и потребления нитроглицерина и других нитратов. \u003Cbr\u003EОказывает длительный дозозависимый гипотензивный эффект. Гипотензивное действие обусловлено прямым вазодилатирующим влиянием на гладкие мышцы сосудов. При артериальной гипертензии разовая доза обеспечивает клинически значимое снижение артериального давления (АД) на протяжении 24 ч (в положении больного \"лежа\" и \"стоя\"). Ортостатическая гипотензия при назначении амлодипина встречается достаточно редко. Не вызывает снижения толерантности к физической нагрузке, фракции выброса левого желудочка. Уменьшает степень гипертрофии миокарда левого желудочка. Не оказывает влияния на сократимость и проводимость миокарда, нс вызывает рефлекторного увеличения частоты сердечных сокращений (ЧСС), тормозит агрегацию тромбоцитов, повышает скорость клубочковой фильтрации, обладает слабым натрийуретическим действием. При диабетической нефропатии не увеличивает выраженность микроальбуминурии. Не оказывает какого-либо неблагоприятного влияния на обмен веществ и концентрацию липидов плазмы крови и может применяться при лечении больных бронхиальной астмой, сахарным диабетом и подагрой. Значимое снижение АД наблюдается через 6-10 часов, длительность эффекта 24 часа."},{"name":"Фармакологическая группа","value":"блокатор \"медленных\" кальциевых каналов"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В сухом, защищенном от света месте, при температуре не выше 25°С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: чрезмерная периферическая вазодилатация с выраженным и возможно длительным снижением АД, коллапс, шок.\u003Cbr\u003EЛечение: промывание желудка, назначение активированного угля, поддержание функции сердечно-сосудистой системы, контроль показателей функции сердца и легких, приподнятое, выше уровня головы, положение нижних конечностей, контроль объема циркулирующей крови и диуреза. Для восстановления тонуса сосудов - применение сосудосуживающих средств (при отсутствии противопоказаний к их применению); с целью устранения последствий блокады кальциевых каналов - внутривенное введение кальция глюконата. Гемодиализ неэффективен."},{"name":"Применение при беременности и кормлении грудью","value":"Безопасность применения амлодипина при беременности и в период кормления грудью не установлена, поэтому препарат амлодипин не следует назначать беременным и в период лактации."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения следует соблюдать осторожность при вождении автотранспорта и занятии потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"В период лечения препаратом необходимо контролировать массу тела и потребление натрия, назначение соответствующей диеты. Необходимо поддержание гигиены зубов и наблюдение у стоматолога (для предотвращения болезненности, кровоточивости и гиперплазии десен).\u003Cbr\u003EПациентам с малой массой тела, пациентам невысокого роста и больным с выраженным нарушением функции печени может потребоваться меньшая доза.\u003Cbr\u003EУ пожилых пациентов может удлиняться T1/2 и клиренс препарата. Изменения доз для пожилых пациентов нс требуется; при увеличении дозы необходимо более тщательное наблюдение за пациентами.\u003Cbr\u003EПри нарушении функции печени также может удлиняться Т1/2 препарата. Поэтому таким пациентам препарат необходимо назначать с осторожностью. Несмотря на то, что прекращение приема препарата не сопровождается развитием синдрома \"отмены\", прекращение лечения желательно проводить, постепенно уменьшая дозу препарата. Эффективность и безопасность препарата при гипертензивном кризе не установлена."},{"name":"Взаимодействие","value":"Амлодипин может безопасно применяться для лечения артериальной гипертензии вместе с тиазидными диуретиками, альфа-адреноблокаторами, бета-адреноблокаторами или ингибиторами АПФ. У пациентов со стабильной стенокардией препарат можно комбинировать с другими антиангинальными средствами, например, с нитратами пролонгированного или короткого действия, бета-адреноблокаторами.\u003Cbr\u003EАмлодипин можно одновременно применять с нестероидными противовоспалительными препаратами (НПВП) (особенно индометацином), антибактериальными средствами и гипогликемическими средствами для приема внутрь. \u003Cbr\u003EВозможно усиление антиангинального и гипотензивного действия БМКК при совместном применении с тиазидными и \"петлевыми\" диуретиками, верапамилом, ингибиторами АПФ, бета-адреноблокаторами и нитратами, а так же усиление их гипотензивного действия при совместном применении с альфа 1 -адреноблокаторами, нейролептиками. \u003Cbr\u003EХотя при изучении амлодипина отрицательного инотропного действия обычно не наблюдали, тем не менее, некоторые БМКК могут усиливать выраженность отрицательного инотропного действия антиаритмических средств и вызывающих удлинение интервала QT (например, амиодарон и хинидин). \u003Cbr\u003EОднократный прием 100 мг силденафила у больных эссенциальной гипертензией не оказывает влияния на параметры фармакокинетики амлодипина. \u003Cbr\u003EПовторное применение амлодипина в дозе 10 мг и аторвастатина в дозе 80 мг не сопровождается значительными изменениями показателей фармакокинетики аторвастатина. \u003Cbr\u003EЭтанол (напитки, содержащие алкоголь): амлодипин при однократном и повторном применении в дозе 10 мг не влияет на фармакокинетику этанола. Противовирусные средства (ритонавир) увеличивает плазменные концентрации БМКК, в т.ч. амлодипина. \u003Cbr\u003EНейролептики и изофлуран - усиление гипотензивного действия производных дигидропиридина. \u003Cbr\u003EПрепараты кальция могут уменьшать эффект БМКК. \u003Cbr\u003EПри совместном применении амлодипина с препаратами лития возможно усиление проявления нейротоксичности (тошнота, рвота, диарея, атаксия, тремор, шум в ушах). \u003Cbr\u003EАмлодипин не изменяет фармакокинетику циклоспорина. \u003Cbr\u003EНе оказывает влияние на концентрацию в сыворотке крови дигоксина и его почечный клиренс. \u003Cbr\u003EНе оказывает существенного влияние на действие варфарина (протромбиновое время). \u003Cbr\u003EЦиметидин не влияет на фармакокинетику амлодипина. \u003Cbr\u003EВ исследованиях in vitro амлодипин не влияет на связывание с белками крови дигоксина, фенитоина, варфарина и индометацина. \u003Cbr\u003EГрейпфрутовый сок: одновременный однократный прием 240 мг грейпфрутового сока и 10 мг амлодипина внутрь не сопровождается существенным изменением фармакокинетики амлодипина."},{"name":"Регистрационный номер","value":"ЛСР-000849/10"},{"name":"Дата государственной регистрации","value":"16.05.2017"},{"name":"Владелец регистрационного удостоверения","value":"ПРАНАФАРМ"},{"name":"Изготовитель","value":"ПРАНАФАРМ"},{"name":"Фасовщик","value":"ПРАНАФАРМ"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Амлодипин-Прана"},{"name":"Срок годности","value":"507 дн."}]}],"transitionId":"tr_16126422868032808310"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

Где купить

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198 ₽

Скидка: 20%
–20 %
Вместо:248 ₽
  • 11-13 июня, самовывоз  0 ₽
Рейтинг 4.9 из 5
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  • Рейтинг товара: 4.7 из 5
    на основе 34 оценки
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-rew7fcwkmkb/addToCartButton":{"offerId":"-BW8eyNmLdewcuve-R_xPA","skuId":"227933878","pendingCartItem":{"productId":1401075437,"offerId":"-BW8eyNmLdewcuve-R_xPA","showPlaceId":"OTNDnItfwRMjN9MRHuEMMhi59sH_lB2ZtNH5zNE5kGLvoKdvZEkum9rh5uGD43hid5elOb0OT-R05crk8fkEL-pao9XO0C5ELsf1wI6cqEoANvoG4a3Mg6gid9XT1hlwKGPPCZTXY-XoSWxiS0U3qtcReRgTVPuUdLE5kHvSC3DvWm4MyDdg4UXvsMATbdt6UIx2718BJVDmWM6RUCTXuw,,","feeShow":"OTNDnItfwRMjN9MRHuEMMhi59sH_lB2ZtNH5zNE5kGLvoKdvZEkum9rh5uGD43hid5elOb0OT-R05crk8fkEL-pao9XO0C5ELsf1wI6cqEoANvoG4a3Mg6gid9XT1hlwKGPPCZTXY-XoSWxiS0U3qtcReRgTVPuUdLE5kHvSC3DvWm4MyDdg4UXvsMATbdt6UIx2718BJVDmWM6RUCTXuw,,","skuId":"227933878","shopId":77075781,"price":{"applicablePriceDiscounts":[],"value":"135","currency":"RUR"},"hid":"15756887","name":"Амлодипин таб., 10 мг, 30 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  • Рейтинг товара: 4.7 из 5
    на основе 69 оценок
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  • Рейтинг товара: 5 из 5
    на основе 19 оценок
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-79fo9qbxhh4/addToCartButton":{"offerId":"E2yTJId5EreSACR60yB7SA","skuId":"101465762432","pendingCartItem":{"productId":1451489305,"offerId":"E2yTJId5EreSACR60yB7SA","showPlaceId":"OTNDnItfwRMjN9MRHuEMMhi59sH_lB2ZxL5tuvW88vMT0OA97O5zqYfriik2jKHFkHGA_n5ry72OKmcnrULXcpV5_m349ymwU9B2gCarPsv0qqj_JvrG9btN_5zsG2511ry5i3gAjPYHL8vgr3po_3izN6BYxC86uY5oTkzpgq6-vyXWJjFb16FuYWnPBukIsG2U83mZ9jrtfR-3OlOfzw,,","feeShow":"OTNDnItfwRMjN9MRHuEMMhi59sH_lB2ZxL5tuvW88vMT0OA97O5zqYfriik2jKHFkHGA_n5ry72OKmcnrULXcpV5_m349ymwU9B2gCarPsv0qqj_JvrG9btN_5zsG2511ry5i3gAjPYHL8vgr3po_3izN6BYxC86uY5oTkzpgq6-vyXWJjFb16FuYWnPBukIsG2U83mZ9jrtfR-3OlOfzw,,","skuId":"101465762432","shopId":4035369,"price":{"applicablePriceDiscounts":[],"value":"58","currency":"RUR"},"hid":"15756887","name":"Амлодипин Реневал таб., 5 мг, 30 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  • Рейтинг товара: 4.8 из 5
    на основе 72 оценки
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  • {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-8oor0xzma7f/addToCartButton":{"offerId":"97V1cetJRUAyHpWt3KWluQ","skuId":"227830013","pendingCartItem":{"productId":1778173627,"offerId":"97V1cetJRUAyHpWt3KWluQ","showPlaceId":"OTNDnItfwRMjN9MRHuEMMhi59sH_lB2ZTpRyKV4mOE7RJ_tqRBuiP1a7REe1NMqHI9NLAEXu0WMcLzouZnVFj3WqiTvuR8NtdwAOgttpvdEvUEJNuhgyyO5_HssFdXU1zcIDIuVMaaRyghM9JBBYlSvNqaQaI09O_THHz_E45ORFKV4vJ-oBAp4-ykW0JHSfc2bbD5SXgiJ5SHDEXdcGgg,,","feeShow":"OTNDnItfwRMjN9MRHuEMMhi59sH_lB2ZTpRyKV4mOE7RJ_tqRBuiP1a7REe1NMqHI9NLAEXu0WMcLzouZnVFj3WqiTvuR8NtdwAOgttpvdEvUEJNuhgyyO5_HssFdXU1zcIDIuVMaaRyghM9JBBYlSvNqaQaI09O_THHz_E45ORFKV4vJ-oBAp4-ykW0JHSfc2bbD5SXgiJ5SHDEXdcGgg,,","skuId":"227830013","shopId":55106433,"price":{"applicablePriceDiscounts":[],"value":"176","currency":"RUR"},"hid":"15756887","name":"Амлодипин Алкалоид таб., 10 мг, 30 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  • Рейтинг товара: 4.8 из 5
    на основе 5 оценок
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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
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  • Рейтинг товара: 4.8 из 5
    на основе 25 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 63 оценки
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-yya5oruueja/addToCartButton":{"offerId":"TlRhkwuJRWuGdfUHmBVXOQ","skuId":"453489075","pendingCartItem":{"productId":1401075757,"offerId":"TlRhkwuJRWuGdfUHmBVXOQ","showPlaceId":"OTNDnItfwRMjN9MRHuEMMhi59sH_lB2Zrl258kGsRB_nNJfhoUslxpxrUdNSw2fSVg27yHWRXZtoTYAYVvl6mNEWoMi-NvGa90R2f3lM6eHbfQw2LQnuUIYvsH2ws8w1FDRyLt9Ov5mlakyq-y3k9iPju-aZjURdWNmyZG9YvxUv2DuriqrSvS6qQ2Z5ymVxacown0Ta-KMg1NPnyOMH2g,,","feeShow":"OTNDnItfwRMjN9MRHuEMMhi59sH_lB2Zrl258kGsRB_nNJfhoUslxpxrUdNSw2fSVg27yHWRXZtoTYAYVvl6mNEWoMi-NvGa90R2f3lM6eHbfQw2LQnuUIYvsH2ws8w1FDRyLt9Ov5mlakyq-y3k9iPju-aZjURdWNmyZG9YvxUv2DuriqrSvS6qQ2Z5ymVxacown0Ta-KMg1NPnyOMH2g,,","skuId":"453489075","shopId":77075781,"price":{"applicablePriceDiscounts":[],"value":"338","currency":"RUR"},"hid":"15756887","name":"Лозартан таб. п/о плен., 50 мг, 90 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  • Рейтинг товара: 5 из 5
    на основе 2 оценки
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Инструкция

Показания к применению

Артериальная гипертензия (монотерапия или в комбинации с другими антигипертензивными средствами).
Стабильная стенокардия напряжения и вазоспастическая стенокардия (стенокардия Принцметала) (монотерапия или в комбинации с другими антиангинальными средствами).

Противопоказания

Повышенная чувствительность к амлодипину, производным дигидропиридина и другим компонентам препарата;
выраженная артериальная гипотензия (систолическое АД менее 90 мм рт.ст.);
коллапс, кардиогенный шок;
нестабильная стенокардия (за исключением стенокардии Принцметала);
клинически значимый стеноз аорты;
беременность и период лактации;
возраст до 18 лет (эффективность и безопасность не изучены);
непереносимость лактозы, дефицит лактазы или глюкозо-галактозная мальабсорбция.
С осторожностью:
Нарушениях функции печени, синдроме слабости синусового узла (выраженная брадикардия, тахикардия), хронической сердечной недостаточности неишемической этиологии III-1V функционального класса по классификации NYHA, артериальной гипотензии, аортальном стенозе, митральном стенозе, гипертрофической обструктивной кардиомиопатии (ГОКМП), остром инфаркте миокарда (и в течение 1 месяца после инфаркта миокарда), в пожилом возрасте.

Способ применения и дозы

Внутрь, начальная доза для лечения артериальной гипертензии и стенокардии составляет 5 мг препарата 1 раз в сутки. Доза максимально может быть увеличена до 10 мг 1 раз в сутки. При артериальной гипертензии поддерживающая доза может быть 2,5 - 5 мг (1/2 таблетки по 5 мг - 1 таблетка по 5 мг) в сутки.
У пациентов пожилого возраста может увеличиваться Т1/2 амлодипина и снижаться клиренс креатинина (КК). Изменения доз не требуется, но необходимо более тщательное наблюдение за пациентами.
Не требуется изменения дозы при одновременном назначении с тиазидными диуретиками, бета-адреноблокаторам и ингибиторами ангиотензинпревращающего фермента (АГ1Ф).
Нe требуется изменения дозы у пациентов с почечной недостаточностью.
Полная инструкция
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Амлодипин-Прана таб.
Амлодипин-Прана таб., 10 мг, 90 шт.
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Инструкция

198 ₽

Скидка: 20%
–20 %
Вместо:248 ₽
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4.9
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У продавца:44 оценки·7 отзывов
У всех продавцов:110 оценок·25 отзывов
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user avatar
3 месяца назад • Светлана Д. • Куплен на Маркете
Достоинства: Стандартная упаковка, стандартный препарат. Удобно, что забирала вместе с другими товарами, в аптеку идти не пришлось.
user avatar
8 месяцев назад • Людмила Васильева • Куплен на Маркете
Достоинства: Мне помогает от давления. Применяю давно.
user avatar
7 месяцев назад • Дафна • Куплен на Маркете
Достоинства: только плюс! для меня лучший препарат
Недостатки: не обнаружила
Комментарий: гипертоник с большим стажем. помогает
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