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Описание

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Ксантинола никотинат р-р для в/в введ. введ. и в/м введ. амп, 150 мг/мл, 2 мл, 10 шт.

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до 1,0 мл"},{"name":"Действующее вещество","value":"Ксантинола никотинат","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28709579"]}}},{"name":"Способ применения и дозы","value":"Внутривенно (струйно или капельно), внутримышечно.\u003Cbr /\u003E\nСтепень тяжести заболевания, состояние пациента и пути введения препарата оцениваются врачом.\nПри внутримышечном введении - по 2-6 мл 15% раствора ежедневно в течение 2-3 недель.\u003Cbr /\u003E\nПрепарат вводят внутривенно струйно медленно по 300 мг (2 мл препарата) 1-2 раза в сутки (пациент при этом должен находиться в горизонтальном положении). Длительность лечения составляет 5-10 дней.\u003Cbr /\u003E\nПри острых нарушениях периферического и мозгового кровообращения препарат вводят внутривенно капельно со скоростью 40 - 50 капель в минуту. Для этого 1500 мг (10 мл) препарата разводят в 200 - 500 мл 5% раствора декстрозы или в 200 мл изотонического раствора натрия хлорида, полученную инфузионную смесь вводят капельно в течение 1,5-4 часов. Инфузию можно повторять до 4 раз в сутки; длительность лечения составляет 5 - 10 дней.\u003Cbr /\u003E\nПациентам с имплантированным водителем ритма препарат назначают в более низкой дозе."},{"name":"Побочные действия","value":"Со стороны сердечно-сосудистой системы: возможно снижение артериального давления, головокружение, ощущение жара, покраснение кожных покровов.\u003Cbr /\u003E\nСо стороны пищеварительной системы: тошнота, диарея, анорексия, гастралгия, боли в животе, боли в эпигастрии.\u003Cbr /\u003E\nСо стороны нервной системы: головная боль.\u003Cbr /\u003E\nАллергические реакции: кожный зуд, крапивница, ангионевротический отек, анафилактический шок.\u003Cbr /\u003E\nПрочие: слабость, озноб, покалывание кожного покрова, особенно в области головы и шеи.\u003Cbr /\u003E Эти симптомы обычно исчезают через 10-20 минут, не требуют специального лечения и отказа от применения данного препарата.\u003Cbr /\u003E\nПри применении препаратов никотиновой кислоты может отмечаться ложное повышение концентрации катехоламинов в плазме крови и моче, а также может отмечаться ложноположительный результат определения глюкозы в моче с использованием пробы Бенедикта.\u003Cbr /\u003E\nПри длительном назначении в высоких дозах препарат вызывает изменение толерантности к глюкозе, повышение активности \"печеночных\" трансаминаз (ACT, АЛТ) в сыворотке крови, повышение активности щелочной фосфатазы в сыворотке крови, повышение содержания мочевой кислоты в сыворотке крови.\u003Cbr /\u003E\nПри появлении нежелательных эффектов, не описанных в данной инструкции, и усилении вышеуказанных побочных эффектов при терапии данным препаратом следует немедленно сообщить об этом лечащему врачу.\u003Cbr /\u003E"},{"name":"Фармакологическое действие","value":"Ксантинола никотинат сочетает свойства лекарственных средств группы теофиллина и никотиновой кислоты: оказывает антиагрегантное действие, расширяет периферические сосуды, улучшает коллатеральное кровообращение. Блокируя аденозиновые рецепторы и фосфодиэстеразу, увеличивает содержание циклического аденозинмонофосфата в клетке, субстратно стимулирует синтез никотинамидадениндинуклеотида (НАД) и никотинамидадениндинуклеотидфосфата (НАДО). Улучшает микроциркуляцию, оксигенацию и питание тканей. При продолжительном применении оказывает антиатеросклеротическое действие, активирует процессы фибринолиза, снижает концентрацию холестерина и атерогенных липидов, усиливает активность липопротеинлипазы, уменьшает вязкость крови, снижает агрегацию тромбоцитов.\u003Cbr /\u003E\nУменьшая общее периферическое сосудистое сопротивление, способствует увеличение минутного объема крови и усилению мозгового кровообращения, уменьшает выраженность последствий церебральной гипоксии."},{"name":"Фармакологическая группа","value":"вазодилатирующее средство"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["35947170:36763748"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"Хранить в защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Препарат малотоксичен. Острая передозировка ксантинола никотината сопровождается артериальной гипотензией, общей слабостью, головокружением, тахикардией, болями в животе и рвотой.\u003Cbr /\u003E\nПри появлении симптомов передозировки назначается симптоматическая терапия."},{"name":"Применение при беременности и кормлении грудью","value":"Не применять в I триместр беременности. Во втором и третьем триместре беременности применение препарата допустимо только при наличии абсолютных показаний в случае, если предполагаемая польза для матери превышает потенциальный риск для плода. Применение препарата в этом случае должно проводиться под тщательным наблюдением врача.\u003Cbr /\u003E\nПри необходимости приема препарата в период лактации необходимо прервать грудное вскармливание, т.к. никотиновая кислота выделяется в грудное молоко."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Большие дозы препарата могут вызвать головокружение, слабость и артериальную гипотензию, в связи с этим следует воздержаться от управления транспортным средством, работы с механизмами и занятиями другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Во втором и третьем триместре беременности и в период лактации применение препарата допустимо только при наличии абсолютных показаний и тщательном наблюдении врача.\u003Cbr /\u003E\nКсантинола никотинат вызывает \"никотиноподобный\" синдром, сопровождающийся гиперестезией слизистой оболочки полости носа и рта (обостряет чувствительность обонятельных и вкусовых рецепторов). В связи с этим запах и вкус принимаемых во время терапии алкогольных напитков воспринимается более резким и извращенным.\u003Cbr /\u003E\nПри сахарном диабете необходимо тщательно контролировать гликемию.\u003Cbr /\u003E\nИзбегать попадания препарата в глаза или на слизистые оболочки."},{"name":"Взаимодействие","value":"Во избежание резкого понижения артериального давления препарат нельзя применять одновременно с гипотензивными средствами, в том числе (бета-адреноблокаторов, альфа-адреноблокаторов, ганглиоблокаторов).\u003Cbr /\u003E\nНе применять одновременно с ингибиторами моноаминоксидазы и строфантином.\u003Cbr /\u003E\nОдновременное применение препаратов никотиновой кислоты в сочетании с ингибиторами ГМГ-КоА редуктазы (статинами) может увеличивать риск развития миопатии и рабдомиолиза.\u003Cbr /\u003E\nОдновременное употребление алкоголя может усилить выраженность побочного действия ксантинола никотината (ощущение жара, покраснение кожных покровов)."},{"name":"Регистрационный номер","value":"ЛП-003449"},{"name":"Дата государственной регистрации","value":"05.02.2021"},{"name":"Владелец регистрационного удостоверения","value":"Эллара","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313","7893318:16002682"]}}},{"name":"Изготовитель","value":"Эллара"},{"name":"Фасовщик","value":"Эллара"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Ксантинола никотинат","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["17796364:18007810"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"11692892967405855613":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"головной мозг, кровеносная система, кровеносные сосуды"},{"name":"Назначение","value":"атеросклероз сосудов головного мозга, болезнь Рейно, гипертриглицеридемия, диабетическая ангиопатия, лечение и профилактика нарушений мозгового кровообращения, облитерирующий атеросклероз, облитерирующий эндартериит, первичная гиперхолестеринемия, тромбофлебит, трофические язвы, цереброваскулярная недостаточность"},{"name":"Показания к применению","value":"В составе комплексной терапии: облитерирующий атеросклероз сосудов конечностей, болезнь Рейно, облитерирующий эндартериит, диабетическая ангиопатия, острый тромбофлебит (поверхностных и глубоких вен), трофические язвы голеней, цереброваскулярная недостаточность, атеросклероз сосудов головного мозга, нарушение мозгового кровообращения, атеросклероз коронарных артерий, гиперхолестеринемия, гипертриглицеридемия."},{"name":"Противопоказания","value":"Повышенная чувствительность к ксантинола никотинату или любому другому компоненту препарата, острая сердечная недостаточность или декомпенсированная хроническая сердечная недостаточность, острое кровотечение, острый инфаркт миокарда, митральный стеноз, язвенная болезнь желудка и 12-перстной кишки в фазе обострения, артериальная гипотензия, беременность (особенно в I триместре), период лактации, острая почечная недостаточность, глаукома, нестабильная стенокардия.\nДетский возраст (опыт применения отсутствует)."},{"name":"Состав","value":"Действующее вещество: ксантинола никотинат — 150 мг \u003Cbr\u003EВспомогательные вещества: вода для инъекций - до 1,0 мл"},{"name":"Действующее вещество","value":"Ксантинола никотинат"},{"name":"Способ применения и дозы","value":"Внутривенно (струйно или капельно), внутримышечно.\u003Cbr /\u003E\nСтепень тяжести заболевания, состояние пациента и пути введения препарата оцениваются врачом.\nПри внутримышечном введении - по 2-6 мл 15% раствора ежедневно в течение 2-3 недель.\u003Cbr /\u003E\nПрепарат вводят внутривенно струйно медленно по 300 мг (2 мл препарата) 1-2 раза в сутки (пациент при этом должен находиться в горизонтальном положении). Длительность лечения составляет 5-10 дней.\u003Cbr /\u003E\nПри острых нарушениях периферического и мозгового кровообращения препарат вводят внутривенно капельно со скоростью 40 - 50 капель в минуту. Для этого 1500 мг (10 мл) препарата разводят в 200 - 500 мл 5% раствора декстрозы или в 200 мл изотонического раствора натрия хлорида, полученную инфузионную смесь вводят капельно в течение 1,5-4 часов. Инфузию можно повторять до 4 раз в сутки; длительность лечения составляет 5 - 10 дней.\u003Cbr /\u003E\nПациентам с имплантированным водителем ритма препарат назначают в более низкой дозе."},{"name":"Побочные действия","value":"Со стороны сердечно-сосудистой системы: возможно снижение артериального давления, головокружение, ощущение жара, покраснение кожных покровов.\u003Cbr /\u003E\nСо стороны пищеварительной системы: тошнота, диарея, анорексия, гастралгия, боли в животе, боли в эпигастрии.\u003Cbr /\u003E\nСо стороны нервной системы: головная боль.\u003Cbr /\u003E\nАллергические реакции: кожный зуд, крапивница, ангионевротический отек, анафилактический шок.\u003Cbr /\u003E\nПрочие: слабость, озноб, покалывание кожного покрова, особенно в области головы и шеи.\u003Cbr /\u003E Эти симптомы обычно исчезают через 10-20 минут, не требуют специального лечения и отказа от применения данного препарата.\u003Cbr /\u003E\nПри применении препаратов никотиновой кислоты может отмечаться ложное повышение концентрации катехоламинов в плазме крови и моче, а также может отмечаться ложноположительный результат определения глюкозы в моче с использованием пробы Бенедикта.\u003Cbr /\u003E\nПри длительном назначении в высоких дозах препарат вызывает изменение толерантности к глюкозе, повышение активности \"печеночных\" трансаминаз (ACT, АЛТ) в сыворотке крови, повышение активности щелочной фосфатазы в сыворотке крови, повышение содержания мочевой кислоты в сыворотке крови.\u003Cbr /\u003E\nПри появлении нежелательных эффектов, не описанных в данной инструкции, и усилении вышеуказанных побочных эффектов при терапии данным препаратом следует немедленно сообщить об этом лечащему врачу.\u003Cbr /\u003E"},{"name":"Фармакологическое действие","value":"Ксантинола никотинат сочетает свойства лекарственных средств группы теофиллина и никотиновой кислоты: оказывает антиагрегантное действие, расширяет периферические сосуды, улучшает коллатеральное кровообращение. Блокируя аденозиновые рецепторы и фосфодиэстеразу, увеличивает содержание циклического аденозинмонофосфата в клетке, субстратно стимулирует синтез никотинамидадениндинуклеотида (НАД) и никотинамидадениндинуклеотидфосфата (НАДО). Улучшает микроциркуляцию, оксигенацию и питание тканей. При продолжительном применении оказывает антиатеросклеротическое действие, активирует процессы фибринолиза, снижает концентрацию холестерина и атерогенных липидов, усиливает активность липопротеинлипазы, уменьшает вязкость крови, снижает агрегацию тромбоцитов.\u003Cbr /\u003E\nУменьшая общее периферическое сосудистое сопротивление, способствует увеличение минутного объема крови и усилению мозгового кровообращения, уменьшает выраженность последствий церебральной гипоксии."},{"name":"Фармакологическая группа","value":"вазодилатирующее средство"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"Хранить в защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Препарат малотоксичен. Острая передозировка ксантинола никотината сопровождается артериальной гипотензией, общей слабостью, головокружением, тахикардией, болями в животе и рвотой.\u003Cbr /\u003E\nПри появлении симптомов передозировки назначается симптоматическая терапия."},{"name":"Применение при беременности и кормлении грудью","value":"Не применять в I триместр беременности. Во втором и третьем триместре беременности применение препарата допустимо только при наличии абсолютных показаний в случае, если предполагаемая польза для матери превышает потенциальный риск для плода. Применение препарата в этом случае должно проводиться под тщательным наблюдением врача.\u003Cbr /\u003E\nПри необходимости приема препарата в период лактации необходимо прервать грудное вскармливание, т.к. никотиновая кислота выделяется в грудное молоко."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Большие дозы препарата могут вызвать головокружение, слабость и артериальную гипотензию, в связи с этим следует воздержаться от управления транспортным средством, работы с механизмами и занятиями другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Во втором и третьем триместре беременности и в период лактации применение препарата допустимо только при наличии абсолютных показаний и тщательном наблюдении врача.\u003Cbr /\u003E\nКсантинола никотинат вызывает \"никотиноподобный\" синдром, сопровождающийся гиперестезией слизистой оболочки полости носа и рта (обостряет чувствительность обонятельных и вкусовых рецепторов). В связи с этим запах и вкус принимаемых во время терапии алкогольных напитков воспринимается более резким и извращенным.\u003Cbr /\u003E\nПри сахарном диабете необходимо тщательно контролировать гликемию.\u003Cbr /\u003E\nИзбегать попадания препарата в глаза или на слизистые оболочки."},{"name":"Взаимодействие","value":"Во избежание резкого понижения артериального давления препарат нельзя применять одновременно с гипотензивными средствами, в том числе (бета-адреноблокаторов, альфа-адреноблокаторов, ганглиоблокаторов).\u003Cbr /\u003E\nНе применять одновременно с ингибиторами моноаминоксидазы и строфантином.\u003Cbr /\u003E\nОдновременное применение препаратов никотиновой кислоты в сочетании с ингибиторами ГМГ-КоА редуктазы (статинами) может увеличивать риск развития миопатии и рабдомиолиза.\u003Cbr /\u003E\nОдновременное употребление алкоголя может усилить выраженность побочного действия ксантинола никотината (ощущение жара, покраснение кожных покровов)."},{"name":"Регистрационный номер","value":"ЛП-003449"},{"name":"Дата государственной регистрации","value":"05.02.2021"},{"name":"Владелец регистрационного удостоверения","value":"Эллара"},{"name":"Изготовитель","value":"Эллара"},{"name":"Фасовщик","value":"Эллара"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Ксантинола никотинат"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_2654644599340140420"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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  • Рейтинг товара: 5 из 5
    на основе 2 оценки
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  • {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-641x05qwpnf/addToCartButton":{"offerId":"0M_fdkiOCZK_6fSZGed1yQ","skuId":"227814104","pendingCartItem":{"productId":1778173808,"offerId":"0M_fdkiOCZK_6fSZGed1yQ","showPlaceId":"OTNDnItfwRMjN9MRHuEMMinnPuqzMCXcXePfMNiqgUsWg2BZONrlbq7TMoA5mlj5Yh9OoVuFBiD764nMFB-4NAqHZh0RbGNE9h_G836ZjmerTPlrWROyt5zfRm6GojJBa71GX3nPe4hXV5nRhtn0Q_wsW25HXlmhSEwZ0YIZW5YzCx0dgE5hjVUG7rXmCkkBa2u_rwLqj79QI3TWho1k4g,,","feeShow":"OTNDnItfwRMjN9MRHuEMMinnPuqzMCXcXePfMNiqgUsWg2BZONrlbq7TMoA5mlj5Yh9OoVuFBiD764nMFB-4NAqHZh0RbGNE9h_G836ZjmerTPlrWROyt5zfRm6GojJBa71GX3nPe4hXV5nRhtn0Q_wsW25HXlmhSEwZ0YIZW5YzCx0dgE5hjVUG7rXmCkkBa2u_rwLqj79QI3TWho1k4g,,","skuId":"227814104","shopId":55106433,"price":{"applicablePriceDiscounts":[],"value":"7482","currency":"RUR"},"hid":"15756887","name":"Вазостенон конц. д/приг. р-ра д/инф. / амп, 20 мкг/мл, 1 мл, 10 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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
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  • Рейтинг товара: 5 из 5
    на основе 2 оценки
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  • Рейтинг товара: 5 из 5
    на основе 3 оценки
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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
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Инструкция

Показания к применению

В составе комплексной терапии: облитерирующий атеросклероз сосудов конечностей, болезнь Рейно, облитерирующий эндартериит, диабетическая ангиопатия, острый тромбофлебит (поверхностных и глубоких вен), трофические язвы голеней, цереброваскулярная недостаточность, атеросклероз сосудов головного мозга, нарушение мозгового кровообращения, атеросклероз коронарных артерий, гиперхолестеринемия, гипертриглицеридемия.

Противопоказания

Повышенная чувствительность к ксантинола никотинату или любому другому компоненту препарата, острая сердечная недостаточность или декомпенсированная хроническая сердечная недостаточность, острое кровотечение, острый инфаркт миокарда, митральный стеноз, язвенная болезнь желудка и 12-перстной кишки в фазе обострения, артериальная гипотензия, беременность (особенно в I триместре), период лактации, острая почечная недостаточность, глаукома, нестабильная стенокардия. Детский возраст (опыт применения отсутствует).

Способ применения и дозы

Внутривенно (струйно или капельно), внутримышечно.
Степень тяжести заболевания, состояние пациента и пути введения препарата оцениваются врачом. При внутримышечном введении - по 2-6 мл 15% раствора ежедневно в течение 2-3 недель.
Препарат вводят внутривенно струйно медленно по 300 мг (2 мл препарата) 1-2 раза в сутки (пациент при этом должен находиться в горизонтальном положении). Длительность лечения составляет 5-10 дней.
При острых нарушениях периферического и мозгового кровообращения препарат вводят внутривенно капельно со скоростью 40 - 50 капель в минуту. Для этого 1500 мг (10 мл) препарата разводят в 200 - 500 мл 5% раствора декстрозы или в 200 мл изотонического раствора натрия хлорида, полученную инфузионную смесь вводят капельно в течение 1,5-4 часов. Инфузию можно повторять до 4 раз в сутки; длительность лечения составляет 5 - 10 дней.
Пациентам с имплантированным водителем ритма препарат назначают в более низкой дозе.
Полная инструкция
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Ксантинола никотинат р-р для в/в введ. введ. и в/м введ. амп
Ксантинола никотинат р-р для в/в введ. введ. и в/м введ. амп, 150 мг/мл, 2 мл, 10 шт.
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Инструкция

292 ₽

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3.7
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У продавца:3 оценки·0 отзывов
У всех продавцов:8 оценок·1 отзыв
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Заказывайте в новом приложении
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