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Описание

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Фталазол таб., 500 мг, 10 шт.

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Коротко о товаре

Артикул Маркета
4453166287
Действующее вещество
Форма выпуска
таблетки
Инструкция
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Средняя курсовая доза - 25-30 г. Через 5-6 дней проводят второй курс лечения: 1-2 день - по 1 г 5 раз в сутки (днем - через каждые 4 ч, ночью - через 8 ч), 3-4 день - по 1 г 4 раза в день (ночью не дают), 5 день - по 1 г 3 раза в день. Общая доза во втором цикле -21 г, при легком течении - 18 г. Высшие дозы для взрослых: разовая -2 г, суточная -7 г.\u003Cbr\u003EДетям старше 3 лет - по 0,25-0,5 г 4 раза в сутки.\u003Cbr\u003EПри других инфекциях взрослым в первые 2-3 дня назначают по 1-2 г каждые 4-6 ч, в следующие 2-3 дня - половинные дозы; детям - 0,1 г/кг/сут равными дозами через 4 ч с ночным перерывом, в следующие дни - по 0,2-0,5 г каждые 6-8 ч.\u003Cbr\u003EПри профилактике гнойных осложнений при оперативных вмешательствах на кишечнике взрослым в первые 2-3 дня назначают по 1 г 4 раза в сутки; в следующие 2-3 дня - половинные дозы по 0,5 г 4 раза в сутки. Лечение сочетают с назначением антибиотиков."},{"name":"Побочные действия","value":"Нарушения со стороны крови и лимфатической системы: в редких случаях - лейкопения, тромбоцитопения, агранулоцитоз, гемолиз эритроцитов. При длительном применении может возникнуть анемия вследствие дефицита пантотеновой и птероилглютаровой кислот, продуцируемых микробными клетками.\u003Cbr\u003EНарушения со стороны иммунной системы: лекарственная аллергия, в т.ч., кожные проявления лекарственной аллергии в виде разнообразных сыпей, вплоть до узловатой и многоформной экссудативной эритемы, в отдельных случаях - эпидермальный некролиз (синдром Лайела). В отдельных случаях возникает аллергический отек губ и лица, узелковый периартериит.\u003Cbr\u003EНарушения со стороны нервной системы: головная боль, головокружение, подавленное настроение.\u003Cbr\u003EНарушения со стороны сердца: миокардит, цианоз.\u003Cbr\u003EНарушения со стороны дыхательной системы, органов грудной клетки и средостения: эозинофильная пневмония.\u003Cbr\u003EНарушения со стороны желудочно-кишечного тракта: тошнота, рвота, понос, поражения полости рта (стоматит, гингивит, глоссит и другие), гастрит, недостаточность витаминов группы В (вследствие угнетения микрофлоры кишечника).\u003Cbr\u003EНарушения со стороны печени и желчевыводящих путей: холангит, гепатит.\u003Cbr\u003EНарушения со стороны почек и мочевыводящих путей: мочекаменная болезнь."},{"name":"Фармакологическое действие","value":"Фталазол, как и другие сульфаниламидные препараты, сходные по структуре с ПАБК (парааминобензойной кислотой), по принципу конкурентных взаимоотношений препятствует включению ее в синтез фолиевой кислоты микробной клетки. Это приводит к нарушению образования фолиевой кислоты, участвующей в синтезе пуриновых и пиримидиновых оснований, от которых зависит рост и развитие микроорганизмов.\u003Cbr\u003EНаиболее выраженное бактериостатическое действие фталазол оказывает на вегетативные формы микробов. Этот эффект развивается постепенно, так как в микробной клетке имеются некоторые запасы ПАБК. Кроме того, степень сродства фталазола с синтетазой дигидрофолиевой кислотой - ферментом, лимитирующим образование фолиевой кислоты, по сравнению с ПАБК значительно слабее. Поэтому фталазол нужно вводить в достаточно высоких дозах, препятствующих использованию микроорганизмами ПАБК, содержащейся в тканях. В противном случае могут образовываться устойчивые штаммы возбудителей, не поддающиеся в дальнейшем воздействию сульфаниламидных препаратов.\u003Cbr\u003EКроме антибактериального, фталазол, как и другие сульфаниламидные препараты, оказывает противовоспалительное действие, которое связывают с его способностью ограничивать миграцию лейкоцитов, уменьшать общее количество мигрирующих клеточных элементов и частично стимулировать выработку глюкокортикостероидов.\u003Cbr\u003EСпектр антимикробного действия фталазола, как и других сульфаниламидов, уже, чем антибиотиков. Сульфаниламиды оказывают бактериостатическое действие на Streptococcus spp., Neisseria meningitidis, Neisseria gonorrhoeae, Escherichia coli, Pseudomonas aeruginosa, Shigella dysenteriae, Proteus vulgaris."},{"name":"Фармакологическая группа","value":"противомикробное средство - сульфаниламид"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"antibiotiki-protivomikrobnye-i-protivoparazitarnye-sredstva","categoryId":"15756919","navnodeId":"72512","glfilters":["35947170:36763744"]}}},{"name":"Условия хранения","value":"В сухом, защищенном от света месте, при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Случаи передозировки препарата маловероятны, однако не рекомендуется принимать таблетки более 10 дней в больших дозах.\u003Cbr\u003EЛечение: отмена препарата, промывание желудка 2% раствором гидрокарбоната натрия и взвесью активированного угля; обильное питье 2% раствора натрия гидрокарбоната, форсированный диурез, гемодиализ."},{"name":"Применение при беременности и кормлении грудью","value":"Препарат легко проникает через плаценту, в грудное молоко. При беременности и в период грудного вскармливания применение препарата возможно только в том случае, если предполагаемая польза для матери превышает потенциальный риск для плода."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Во время лечения следует соблюдать осторожность при управлении транспортными средствами, а также занятие видами деятельности, требующими быстроты психомоторных реакций и точных движений."},{"name":"Особые указания","value":"При необходимости можно применять одновременно с сульфаниламидами или антибиотиками бактериостатического действия."},{"name":"Взаимодействие","value":"При применении фталазола совместно с другими лекарственными препаратами могут наблюдаться следующие взаимодействия:\u003Cbr\u003E- ПАСК (парааминосалициловая кислота) и барбитураты - усиливается активность сульфаниламидов;\u003Cbr\u003E- салицилаты - усиливается активность и токсичность;\u003Cbr\u003E- метотрексат и дифенин - усиливается токсичность;\u003Cbr\u003E- тиоацетазон, левомицетин - повышается возможность развития агранулоцитоза;\u003Cbr\u003E- нитрофураны - увеличивается риск возникновения анемии и метгемоглобинемии;\u003Cbr\u003E- антикоагулянты непрямого действия - усиливается антикоагулянтное действие;\u003Cbr\u003E- оксациллин - снижается активность антибиотика.\u003Cbr\u003EМиелотоксичные лекарственные средства усиливают проявления гематотоксичности препарата.\u003Cbr\u003EСовместное применение фталазола с кислотами и кислотореагирующими препаратами, гексаметилентетрамином, раствором эпинефрина нецелесообразно, так как они химически несовместимы.\u003Cbr\u003EПри применении фталазола с препаратами, содержащими эфиры парааминобензойной кислоты (новокаин, анестезин, дикаин), инактивируется антибактериальная активность сульфаниламида по конкурентному механизму.\u003Cbr\u003EЭффект усиливают антибиотики и хорошо всасывающиеся сульфаниламиды."},{"name":"Регистрационный номер","value":"P N003869/01"},{"name":"Дата государственной регистрации","value":"09.08.2021"},{"name":"Владелец регистрационного удостоверения","value":"Дальхимфарм","transition":{"type":"catalog","params":{"categorySlug":"antibiotiki-protivomikrobnye-i-protivoparazitarnye-sredstva","categoryId":"15756919","navnodeId":"72512","glfilters":["34324371:35649313","7893318:13877405"]}}},{"name":"Изготовитель","value":"Дальхимфарм"},{"name":"Фасовщик","value":"Дальхимфарм"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Фталазол","transition":{"type":"catalog","params":{"categorySlug":"antibiotiki-protivomikrobnye-i-protivoparazitarnye-sredstva","categoryId":"15756919","navnodeId":"72512","glfilters":["17796364:18025023"]}}},{"name":"Срок годности","value":"48 мес."}]}},"fullSpecsGrouped":{"7970165815866673758":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Назначение","value":"гастроэнтерит, дизентерия, колит, операции на кишечнике"},{"name":"Органы и системы","value":"кишечник"},{"name":"Показания к применению","value":"- Дизентерия (острая и хроническая формы в стадии обострения);\u003Cbr\u003E- колиты;\u003Cbr\u003E- гастроэнтериты;\u003Cbr\u003E- профилактика гнойных осложнений при оперативных вмешательствах на кишечнике."},{"name":"Противопоказания","value":"- Повышенная индивидуальная чувствительность к препаратам сульфаниламидного ряда;\u003Cbr\u003E- болезни системы крови;\u003Cbr\u003E- гипертиреоз;\u003Cbr\u003E- хроническая почечная недостаточность;\u003Cbr\u003E- гломерулонефрит;\u003Cbr\u003E- острый гепатит;\u003Cbr\u003E- кишечная непроходимость;\u003Cbr\u003E- детский возраст до 3 лет (для данной лекарственной формы)."},{"name":"Состав","value":"На одну таблетку:\u003Cbr\u003EДействующее вещество: фталилсульфатиазол - 500 мг\u003Cbr\u003EВспомогательные вещества: крахмал картофельный - 79 мг, тальк - 6 мг, кальция стеарат - 15 мг."},{"name":"Действующее вещество","value":"Фталилсульфатиазол"},{"name":"Способ применения и дозы","value":"Внутрь, при острой дизентерии взрослым в 1-2 день - по 1 г 6 раз в сутки, в 3-4 день - по 1 г 4 раза в сутки, в 5-6 день - по 1 г 3 раза в сутки. Средняя курсовая доза - 25-30 г. Через 5-6 дней проводят второй курс лечения: 1-2 день - по 1 г 5 раз в сутки (днем - через каждые 4 ч, ночью - через 8 ч), 3-4 день - по 1 г 4 раза в день (ночью не дают), 5 день - по 1 г 3 раза в день. Общая доза во втором цикле -21 г, при легком течении - 18 г. Высшие дозы для взрослых: разовая -2 г, суточная -7 г.\u003Cbr\u003EДетям старше 3 лет - по 0,25-0,5 г 4 раза в сутки.\u003Cbr\u003EПри других инфекциях взрослым в первые 2-3 дня назначают по 1-2 г каждые 4-6 ч, в следующие 2-3 дня - половинные дозы; детям - 0,1 г/кг/сут равными дозами через 4 ч с ночным перерывом, в следующие дни - по 0,2-0,5 г каждые 6-8 ч.\u003Cbr\u003EПри профилактике гнойных осложнений при оперативных вмешательствах на кишечнике взрослым в первые 2-3 дня назначают по 1 г 4 раза в сутки; в следующие 2-3 дня - половинные дозы по 0,5 г 4 раза в сутки. Лечение сочетают с назначением антибиотиков."},{"name":"Побочные действия","value":"Нарушения со стороны крови и лимфатической системы: в редких случаях - лейкопения, тромбоцитопения, агранулоцитоз, гемолиз эритроцитов. При длительном применении может возникнуть анемия вследствие дефицита пантотеновой и птероилглютаровой кислот, продуцируемых микробными клетками.\u003Cbr\u003EНарушения со стороны иммунной системы: лекарственная аллергия, в т.ч., кожные проявления лекарственной аллергии в виде разнообразных сыпей, вплоть до узловатой и многоформной экссудативной эритемы, в отдельных случаях - эпидермальный некролиз (синдром Лайела). В отдельных случаях возникает аллергический отек губ и лица, узелковый периартериит.\u003Cbr\u003EНарушения со стороны нервной системы: головная боль, головокружение, подавленное настроение.\u003Cbr\u003EНарушения со стороны сердца: миокардит, цианоз.\u003Cbr\u003EНарушения со стороны дыхательной системы, органов грудной клетки и средостения: эозинофильная пневмония.\u003Cbr\u003EНарушения со стороны желудочно-кишечного тракта: тошнота, рвота, понос, поражения полости рта (стоматит, гингивит, глоссит и другие), гастрит, недостаточность витаминов группы В (вследствие угнетения микрофлоры кишечника).\u003Cbr\u003EНарушения со стороны печени и желчевыводящих путей: холангит, гепатит.\u003Cbr\u003EНарушения со стороны почек и мочевыводящих путей: мочекаменная болезнь."},{"name":"Фармакологическое действие","value":"Фталазол, как и другие сульфаниламидные препараты, сходные по структуре с ПАБК (парааминобензойной кислотой), по принципу конкурентных взаимоотношений препятствует включению ее в синтез фолиевой кислоты микробной клетки. Это приводит к нарушению образования фолиевой кислоты, участвующей в синтезе пуриновых и пиримидиновых оснований, от которых зависит рост и развитие микроорганизмов.\u003Cbr\u003EНаиболее выраженное бактериостатическое действие фталазол оказывает на вегетативные формы микробов. Этот эффект развивается постепенно, так как в микробной клетке имеются некоторые запасы ПАБК. Кроме того, степень сродства фталазола с синтетазой дигидрофолиевой кислотой - ферментом, лимитирующим образование фолиевой кислоты, по сравнению с ПАБК значительно слабее. Поэтому фталазол нужно вводить в достаточно высоких дозах, препятствующих использованию микроорганизмами ПАБК, содержащейся в тканях. В противном случае могут образовываться устойчивые штаммы возбудителей, не поддающиеся в дальнейшем воздействию сульфаниламидных препаратов.\u003Cbr\u003EКроме антибактериального, фталазол, как и другие сульфаниламидные препараты, оказывает противовоспалительное действие, которое связывают с его способностью ограничивать миграцию лейкоцитов, уменьшать общее количество мигрирующих клеточных элементов и частично стимулировать выработку глюкокортикостероидов.\u003Cbr\u003EСпектр антимикробного действия фталазола, как и других сульфаниламидов, уже, чем антибиотиков. Сульфаниламиды оказывают бактериостатическое действие на Streptococcus spp., Neisseria meningitidis, Neisseria gonorrhoeae, Escherichia coli, Pseudomonas aeruginosa, Shigella dysenteriae, Proteus vulgaris."},{"name":"Фармакологическая группа","value":"противомикробное средство - сульфаниламид"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В сухом, защищенном от света месте, при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Случаи передозировки препарата маловероятны, однако не рекомендуется принимать таблетки более 10 дней в больших дозах.\u003Cbr\u003EЛечение: отмена препарата, промывание желудка 2% раствором гидрокарбоната натрия и взвесью активированного угля; обильное питье 2% раствора натрия гидрокарбоната, форсированный диурез, гемодиализ."},{"name":"Применение при беременности и кормлении грудью","value":"Препарат легко проникает через плаценту, в грудное молоко. При беременности и в период грудного вскармливания применение препарата возможно только в том случае, если предполагаемая польза для матери превышает потенциальный риск для плода."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Во время лечения следует соблюдать осторожность при управлении транспортными средствами, а также занятие видами деятельности, требующими быстроты психомоторных реакций и точных движений."},{"name":"Особые указания","value":"При необходимости можно применять одновременно с сульфаниламидами или антибиотиками бактериостатического действия."},{"name":"Взаимодействие","value":"При применении фталазола совместно с другими лекарственными препаратами могут наблюдаться следующие взаимодействия:\u003Cbr\u003E- ПАСК (парааминосалициловая кислота) и барбитураты - усиливается активность сульфаниламидов;\u003Cbr\u003E- салицилаты - усиливается активность и токсичность;\u003Cbr\u003E- метотрексат и дифенин - усиливается токсичность;\u003Cbr\u003E- тиоацетазон, левомицетин - повышается возможность развития агранулоцитоза;\u003Cbr\u003E- нитрофураны - увеличивается риск возникновения анемии и метгемоглобинемии;\u003Cbr\u003E- антикоагулянты непрямого действия - усиливается антикоагулянтное действие;\u003Cbr\u003E- оксациллин - снижается активность антибиотика.\u003Cbr\u003EМиелотоксичные лекарственные средства усиливают проявления гематотоксичности препарата.\u003Cbr\u003EСовместное применение фталазола с кислотами и кислотореагирующими препаратами, гексаметилентетрамином, раствором эпинефрина нецелесообразно, так как они химически несовместимы.\u003Cbr\u003EПри применении фталазола с препаратами, содержащими эфиры парааминобензойной кислоты (новокаин, анестезин, дикаин), инактивируется антибактериальная активность сульфаниламида по конкурентному механизму.\u003Cbr\u003EЭффект усиливают антибиотики и хорошо всасывающиеся сульфаниламиды."},{"name":"Регистрационный номер","value":"P N003869/01"},{"name":"Дата государственной регистрации","value":"09.08.2021"},{"name":"Владелец регистрационного удостоверения","value":"Дальхимфарм"},{"name":"Изготовитель","value":"Дальхимфарм"},{"name":"Фасовщик","value":"Дальхимфарм"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Фталазол"},{"name":"Срок годности","value":"48 мес."}]}],"transitionId":"tr_15026582304842097016"}}}}
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Инструкция

Показания к применению

- Дизентерия (острая и хроническая формы в стадии обострения);
- колиты;
- гастроэнтериты;
- профилактика гнойных осложнений при оперативных вмешательствах на кишечнике.

Противопоказания

- Повышенная индивидуальная чувствительность к препаратам сульфаниламидного ряда;
- болезни системы крови;
- гипертиреоз;
- хроническая почечная недостаточность;
- гломерулонефрит;
- острый гепатит;
- кишечная непроходимость;
- детский возраст до 3 лет (для данной лекарственной формы).

Способ применения и дозы

Внутрь, при острой дизентерии взрослым в 1-2 день - по 1 г 6 раз в сутки, в 3-4 день - по 1 г 4 раза в сутки, в 5-6 день - по 1 г 3 раза в сутки. Средняя курсовая доза - 25-30 г. Через 5-6 дней проводят второй курс лечения: 1-2 день - по 1 г 5 раз в сутки (днем - через каждые 4 ч, ночью - через 8 ч), 3-4 день - по 1 г 4 раза в день (ночью не дают), 5 день - по 1 г 3 раза в день. Общая доза во втором цикле -21 г, при легком течении - 18 г. Высшие дозы для взрослых: разовая -2 г, суточная -7 г.
Детям старше 3 лет - по 0,25-0,5 г 4 раза в сутки.
При других инфекциях взрослым в первые 2-3 дня назначают по 1-2 г каждые 4-6 ч, в следующие 2-3 дня - половинные дозы; детям - 0,1 г/кг/сут равными дозами через 4 ч с ночным перерывом, в следующие дни - по 0,2-0,5 г каждые 6-8 ч.
При профилактике гнойных осложнений при оперативных вмешательствах на кишечнике взрослым в первые 2-3 дня назначают по 1 г 4 раза в сутки; в следующие 2-3 дня - половинные дозы по 0,5 г 4 раза в сутки. Лечение сочетают с назначением антибиотиков.
Полная инструкция
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Фталазол таб.
Фталазол таб., 500 мг, 10 шт.
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Инструкция

180 ₽

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5.0
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У продавца:4 оценки·0 отзывов
У всех продавцов:43 оценки·12 отзывов
Написать отзыв
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