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Бетагистин Канон таб., 24 мг, 30 шт.

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Дозировка: 24 мг

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Количество штук в упаковке, шт.: 30

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Коротко о товаре

Артикул Маркета
3338088971
Действующее вещество
Возраст
от 18 лет
Инструкция
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Лечение длительное.\u003Cbr\u003EНе требуется коррекции дозы у пациентов пожилого возраста, а также у пациентов с печеночной и/или почечной недостаточностью.\u003Cbr\u003EУлучшение иногда наблюдается через несколько недель лечения; наилучшие результаты иногда достигаются после нескольких месяцев лечения."},{"name":"Побочные действия","value":"Классификация частоты развития побочных эффектов согласно рекомендациям Всемирной Организации Здравоохранения: очень часто (≥1/10), часто (от ≥1/100 до \u003C1/10), нечасто (от ≥1/1000 до \u003C1/100), редко (от ≥1/10000 до \u003C1/1000), очень редко (\u003C1/10000), включая отдельные сообщения; частота неизвестна - по имеющимся данным установить частоту возникновения не представляется возможным.\u003Cbr\u003EСо стороны пищеварительной системы:\u003Cbr\u003Eчасто - тошнота, диспепсия;\u003Cbr\u003Eчастота неизвестна - рвота, ощущение тяжести в эпигастрии, абдоминальная боль, вздутие живота.\u003Cbr\u003EСо стороны кожных покровов:\u003Cbr\u003Eчастота неизвестна - кожный зуд, сыпь, крапивница, отек Квинке.\u003Cbr\u003EАллергические реакции:\u003Cbr\u003Eчастота неизвестна - реакции повышенной чувствительности, в т.ч. анафилактические реакции.\u003Cbr\u003EСо стороны центральной нервной системы:\u003Cbr\u003Eчасто - головная боль."},{"name":"Фармакологическое действие","value":"Механизм действия бетагистина известен только частично. Существует несколько возможных гипотез, подтвержденных доклиническими и клиническими данными:\u003Cbr\u003EВлияние на гистаминергическую систему. Частичный агонист Н1-гистаминовых и антагонист Н3-гистаминовых рецепторов вестибулярных ядер центральной нервной системы, обладает незначительной активностью в отношении Н2-гистаминовых рецепторов. Бетагистин увеличивает обмен гистамина и его высвобождение путем блокирования пресинаптических Н3-гистаминовых рецепторов и снижения количества Н3-гистаминовых рецепторов.\u003Cbr\u003EУсиление кровотока кохлеарной области, а также всего головного мозга. Согласно доклиническим исследованиям, бетагистин улучшает кровообращение в сосудистой полоске внутреннего уха за счет расслабления прекапиллярных сфинктеров сосудов внутреннего уха. Также показано, что бетагистин усиливает мозговой кровоток у человека.\u003Cbr\u003EОблегчение процесса центральной вестибулярной компенсации. Бетагистин ускоряет восстановление вестибулярной функции у животных после односторонней вестибулярной нейрэктомии, ускоряя и облегчая нейтральную вестибулярную компенсацию за счет антагонизма с Н3-гистаминовыми рецепторами. Время восстановления после вестибулярной нейрэктомии у человека при лечении бетагистином также уменьшается.\u003Cbr\u003EВозбуждение нейронов в вестибулярных ядрах. Дозозависимо снижает генерацию потенциалов действия в нейронах латеральных и медиальных вестибулярных ядер. Фармакологические свойства, выявленные на животных, обеспечивают положительный терапевтический эффект бетагистина в вестибулярной системе. Эффективность бетагистина была продемонстрирована у пациентов с вестибулярным головокружением и синдромом Меньера, что проявлялось уменьшением выраженности и частоты головокружений."},{"name":"Фармакологическая группа","value":"гистамина препарат"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-nervnoi-sistemy","categoryId":"15756525","navnodeId":"72478","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"В сухом, защищенном от света месте при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: тошнота, абдоминальная боль, сонливость (при приеме в дозе до 640 мг), судороги, сердечно-легочные осложнения (при приеме в дозе более 640 мг или в сочетании с другими лекарственными препаратами).\u003Cbr\u003EЛечение: промывание желудка, прием активированного угля, симптоматическая терапия."},{"name":"Применение при беременности и кормлении грудью","value":"Прием бетагистина при беременности и в период грудного вскармливания противопоказан из-за отсутствия достаточного количества данных о его безопасности во время беременности и в период грудного вскармливания. Неизвестно, выделяется ли бетагистин с грудным молоком; если прием препарата необходим в период грудного вскармливания, кормление грудью необходимо прекратить."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Бетагистин показан для лечения синдрома Меньера, который характеризуется триадой основных симптомов: головокружением, снижением слуха, шумом в ушах, а также для симптоматического лечения вестибулярного головокружения. Оба состояния могут негативно влиять на способность управлять автомобилем и работать с механизмами. По результатам клинических исследований доказано, что влияние бетагистина на способность управлять транспортными средствами и работать с механизмами отсутствует или незначительно."},{"name":"Особые указания","value":"Терапевтический эффект в ряде случаев нарастает в течение нескольких месяцев от начала лечения.\u003Cbr\u003EУлучшение иногда наблюдается через несколько недель лечения; наилучшие результаты иногда достигаются после нескольких месяцев лечения.\u003Cbr\u003EУ пациентов с язвенной болезнью желудка или 12-перстной кишки (в анамнезе), бронхиальной астмой, артериальной гипотензией препарат следует применять с осторожностью и под контролем лечащего врача.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EЯзвенная болезнь желудка или 12-перстной кишки (в анамнезе), бронхиальная астма, пациенты с артериальной гипотензией."},{"name":"Взаимодействие","value":"Исследования in vivo, направленные на изучение взаимодействия с другими лекарственными препаратами, не проводились. Основываясь на данных in vitro, можно предположить отсутствие ингибирования активности изоферментов цитохрома Р450 in vivo.\u003Cbr\u003EДанные in vitro показали ингибирование метаболизма бетагистина под действием препаратов, которые ингибируют моноаминоксидазу (МАО), включая МАО подтипа В (например, селегинин). Следует соблюдать осторожность при одновременном назначении бетагистина и ингибиторов МАО (включая МАО-В).\u003Cbr\u003EБетагистин является аналогом гистамина, взаимодействие бетагистина с блокаторами H1-гистаминовых рецепторов теоретически может влиять на эффективность одного из этих лекарственных средств."},{"name":"Регистрационный номер","value":"ЛС-002330"},{"name":"Дата государственной регистрации","value":"09.08.2021"},{"name":"Владелец регистрационного удостоверения","value":"Канонфарма продакшн","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-nervnoi-sistemy","categoryId":"15756525","navnodeId":"72478","glfilters":["34324371:35649313","7893318:16146766"]}}},{"name":"Изготовитель","value":"Канонфарма продакшн"},{"name":"Фасовщик","value":"Канонфарма продакшн"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Бетагистин Канон","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-nervnoi-sistemy","categoryId":"15756525","navnodeId":"72478","glfilters":["17796364:18028717"]}}},{"name":"Срок годности","value":"24 мес."}]}},"fullSpecsGrouped":{"1484973585404755883":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"нервная система"},{"name":"Назначение","value":"болезнь и синдром Меньера, вертиго, головокружение, шум в ушах"},{"name":"Показания к применению","value":"лечение синдрома Меньера, характеризующегося головокружением (сопровождающимся тошнотой и рвотой), снижением слуха и шумом в ушах.\u003Cbr\u003Eсимптоматическое лечение вестибулярного головокружения (вертиго)."},{"name":"Противопоказания","value":"- повышенная чувствительность к бетагистина или к любому из компонентов препарата;\u003Cbr\u003E- дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция;\u003Cbr\u003E- феохромоцитома;\u003Cbr\u003E- беременность;\u003Cbr\u003E- период грудного вскармливания;\u003Cbr\u003E- возраст до 18 лет (эффективность и безопасность не установлены)."},{"name":"Состав","value":"1 таблетка содержит:\u003Cbr\u003Eактивное вещество: бетагистина дигидрохлорид 8 мг, 16 мг и 24 мг;\u003Cbr\u003Eвспомогательные вещества: коповидон 5,2 мг, 10,4 мг, 15,6 мг; лактозы моногидрат 41,6 мг, 83,2 мг, 124,8 мг; магния стеарат 1 мг, 2 мг, 3 мг; целлюлоза микрокристаллическая 64,2 мг, 128,4 мг, 192,6 мг."},{"name":"Действующее вещество","value":"Бетагистин"},{"name":"Способ применения и дозы","value":"Внутрь, во время еды.\u003Cbr\u003EТаблетки 8 мг: 1-2 таблетки 3 раза в день.\u003Cbr\u003EТаблетки 16 мг: ½ -1 таблетка 3 раза в день.\u003Cbr\u003EТаблетка 24 мг: по 1 таблетке 2 раза в день.\u003Cbr\u003EКурс лечения определяется индивидуально. Лечение длительное.\u003Cbr\u003EНе требуется коррекции дозы у пациентов пожилого возраста, а также у пациентов с печеночной и/или почечной недостаточностью.\u003Cbr\u003EУлучшение иногда наблюдается через несколько недель лечения; наилучшие результаты иногда достигаются после нескольких месяцев лечения."},{"name":"Побочные действия","value":"Классификация частоты развития побочных эффектов согласно рекомендациям Всемирной Организации Здравоохранения: очень часто (≥1/10), часто (от ≥1/100 до \u003C1/10), нечасто (от ≥1/1000 до \u003C1/100), редко (от ≥1/10000 до \u003C1/1000), очень редко (\u003C1/10000), включая отдельные сообщения; частота неизвестна - по имеющимся данным установить частоту возникновения не представляется возможным.\u003Cbr\u003EСо стороны пищеварительной системы:\u003Cbr\u003Eчасто - тошнота, диспепсия;\u003Cbr\u003Eчастота неизвестна - рвота, ощущение тяжести в эпигастрии, абдоминальная боль, вздутие живота.\u003Cbr\u003EСо стороны кожных покровов:\u003Cbr\u003Eчастота неизвестна - кожный зуд, сыпь, крапивница, отек Квинке.\u003Cbr\u003EАллергические реакции:\u003Cbr\u003Eчастота неизвестна - реакции повышенной чувствительности, в т.ч. анафилактические реакции.\u003Cbr\u003EСо стороны центральной нервной системы:\u003Cbr\u003Eчасто - головная боль."},{"name":"Фармакологическое действие","value":"Механизм действия бетагистина известен только частично. Существует несколько возможных гипотез, подтвержденных доклиническими и клиническими данными:\u003Cbr\u003EВлияние на гистаминергическую систему. Частичный агонист Н1-гистаминовых и антагонист Н3-гистаминовых рецепторов вестибулярных ядер центральной нервной системы, обладает незначительной активностью в отношении Н2-гистаминовых рецепторов. Бетагистин увеличивает обмен гистамина и его высвобождение путем блокирования пресинаптических Н3-гистаминовых рецепторов и снижения количества Н3-гистаминовых рецепторов.\u003Cbr\u003EУсиление кровотока кохлеарной области, а также всего головного мозга. Согласно доклиническим исследованиям, бетагистин улучшает кровообращение в сосудистой полоске внутреннего уха за счет расслабления прекапиллярных сфинктеров сосудов внутреннего уха. Также показано, что бетагистин усиливает мозговой кровоток у человека.\u003Cbr\u003EОблегчение процесса центральной вестибулярной компенсации. Бетагистин ускоряет восстановление вестибулярной функции у животных после односторонней вестибулярной нейрэктомии, ускоряя и облегчая нейтральную вестибулярную компенсацию за счет антагонизма с Н3-гистаминовыми рецепторами. Время восстановления после вестибулярной нейрэктомии у человека при лечении бетагистином также уменьшается.\u003Cbr\u003EВозбуждение нейронов в вестибулярных ядрах. Дозозависимо снижает генерацию потенциалов действия в нейронах латеральных и медиальных вестибулярных ядер. Фармакологические свойства, выявленные на животных, обеспечивают положительный терапевтический эффект бетагистина в вестибулярной системе. Эффективность бетагистина была продемонстрирована у пациентов с вестибулярным головокружением и синдромом Меньера, что проявлялось уменьшением выраженности и частоты головокружений."},{"name":"Фармакологическая группа","value":"гистамина препарат"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В сухом, защищенном от света месте при температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: тошнота, абдоминальная боль, сонливость (при приеме в дозе до 640 мг), судороги, сердечно-легочные осложнения (при приеме в дозе более 640 мг или в сочетании с другими лекарственными препаратами).\u003Cbr\u003EЛечение: промывание желудка, прием активированного угля, симптоматическая терапия."},{"name":"Применение при беременности и кормлении грудью","value":"Прием бетагистина при беременности и в период грудного вскармливания противопоказан из-за отсутствия достаточного количества данных о его безопасности во время беременности и в период грудного вскармливания. Неизвестно, выделяется ли бетагистин с грудным молоком; если прием препарата необходим в период грудного вскармливания, кормление грудью необходимо прекратить."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Бетагистин показан для лечения синдрома Меньера, который характеризуется триадой основных симптомов: головокружением, снижением слуха, шумом в ушах, а также для симптоматического лечения вестибулярного головокружения. Оба состояния могут негативно влиять на способность управлять автомобилем и работать с механизмами. По результатам клинических исследований доказано, что влияние бетагистина на способность управлять транспортными средствами и работать с механизмами отсутствует или незначительно."},{"name":"Особые указания","value":"Терапевтический эффект в ряде случаев нарастает в течение нескольких месяцев от начала лечения.\u003Cbr\u003EУлучшение иногда наблюдается через несколько недель лечения; наилучшие результаты иногда достигаются после нескольких месяцев лечения.\u003Cbr\u003EУ пациентов с язвенной болезнью желудка или 12-перстной кишки (в анамнезе), бронхиальной астмой, артериальной гипотензией препарат следует применять с осторожностью и под контролем лечащего врача.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EЯзвенная болезнь желудка или 12-перстной кишки (в анамнезе), бронхиальная астма, пациенты с артериальной гипотензией."},{"name":"Взаимодействие","value":"Исследования in vivo, направленные на изучение взаимодействия с другими лекарственными препаратами, не проводились. Основываясь на данных in vitro, можно предположить отсутствие ингибирования активности изоферментов цитохрома Р450 in vivo.\u003Cbr\u003EДанные in vitro показали ингибирование метаболизма бетагистина под действием препаратов, которые ингибируют моноаминоксидазу (МАО), включая МАО подтипа В (например, селегинин). Следует соблюдать осторожность при одновременном назначении бетагистина и ингибиторов МАО (включая МАО-В).\u003Cbr\u003EБетагистин является аналогом гистамина, взаимодействие бетагистина с блокаторами H1-гистаминовых рецепторов теоретически может влиять на эффективность одного из этих лекарственных средств."},{"name":"Регистрационный номер","value":"ЛС-002330"},{"name":"Дата государственной регистрации","value":"09.08.2021"},{"name":"Владелец регистрационного удостоверения","value":"Канонфарма продакшн"},{"name":"Изготовитель","value":"Канонфарма продакшн"},{"name":"Фасовщик","value":"Канонфарма продакшн"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Бетагистин Канон"},{"name":"Срок годности","value":"24 мес."}]}],"transitionId":"tr_5749771818020095465"}}}}
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Ещё может подойти

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Инструкция

Показания к применению

лечение синдрома Меньера, характеризующегося головокружением (сопровождающимся тошнотой и рвотой), снижением слуха и шумом в ушах.
симптоматическое лечение вестибулярного головокружения (вертиго).

Противопоказания

- повышенная чувствительность к бетагистина или к любому из компонентов препарата;
- дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция;
- феохромоцитома;
- беременность;
- период грудного вскармливания;
- возраст до 18 лет (эффективность и безопасность не установлены).

Способ применения и дозы

Внутрь, во время еды.
Таблетки 8 мг: 1-2 таблетки 3 раза в день.
Таблетки 16 мг: ½ -1 таблетка 3 раза в день.
Таблетка 24 мг: по 1 таблетке 2 раза в день.
Курс лечения определяется индивидуально. Лечение длительное.
Не требуется коррекции дозы у пациентов пожилого возраста, а также у пациентов с печеночной и/или почечной недостаточностью.
Улучшение иногда наблюдается через несколько недель лечения; наилучшие результаты иногда достигаются после нескольких месяцев лечения.
Полная инструкция
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Бетагистин Канон таб.
Бетагистин Канон таб., 24 мг, 30 шт.
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Инструкция

136 ₽

Скидка: 27%
–27 %
Вместо:186 ₽
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4.9
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У продавца:14 оценок·5 отзывов
У всех продавцов:51 оценка·13 отзывов
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user avatar
Месяц назад • наталия с. • Куплен на Маркете
Достоинства: постоянно его принимаю,помогает держать ровновесие
user avatar
3 месяца назад • Алексей Ногин • Куплен на Маркете
Достоинства: Удобная упаковка цена
user avatar
6 месяцев назад • Имя скрыто • Куплен на Маркете
Достоинства: реально помогают
Недостатки: нет
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