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Альфакальцидол Канон капс.
Альфакальцидол Канон капс., 30 шт.
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Инструкция

Цена с картой Яндекс Пэй:262₽/уп

Скидка: 17%
–17 %
Вместо: 265₽/уп315₽/уп
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Альфакальцидол Канон капс., 30 шт.
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Повышает абсорбцию кальция и фосфора в кишечнике, увеличивает их реабсорбцию в почках, восстанавливает положительный кальциевый баланс при лечении синдрома кальциевой мальабсорбции и снижает концентрацию в крови паратиреоидного гормона.\u003Cbr\u003EВоздействуя на обе части процесса костного ремоделирования—(резорбцию и синтез), альфакальцидол не только увеличивает минерализацию костной ткани, но и повышает ее упругость за счет стимулирования синтеза белков матрикса кости, костных морфогенетических белков, факторов роста кости, что способствует уменьшению частоты развития переломов.\u003Cbr\u003EУ пациентов пожилого возраста на фоне эндокринно-иммунной дисфункции, в том числе дефицита продукции D-гормона (кальцитриола), происходит снижение общей мышечной массы (саркопения) и появление синдрома мышечной слабости (вследствие нарушения нормального функционирования нервно-мышечного аппарата), что сопровождается повышением риска падений и обусловленных этим травм и переломов. В ряде исследований было показано значительное снижение частоты падений пожилых пациентов при применении альфакальцидола. Альфакальцидол стимулирует регенерацию мышечных волокон, что восстанавливает утраченный мышечный тонус."},{"description":"","filters":[{"id":50921473,"name":"Состав"}],"isMainProperty":false,"name":"Состав","value":"1 капсула 0,25 мкг содержит:\u003Cbr\u003Eдействующее вещество: альфакальцидол 0,25 мкг;\u003Cbr\u003Eвспомогательные вещества: арахиса масло 98,79975 мг, лимонная кислота (безводная) 0,01500 мг, пропилгаллат 0,02000 мг, альфа-токоферол 0,02000 мг, этиловый спирт (этанол) 1,14500 мг;\u003Cbr\u003Eкапсула мягкая желатиновая: сорбитол частично дегидратированный 12,45 мг, глицерол 18,38 мг, желатин 78,32 мг, краситель железа оксид красный 0,85 мг.\u003Cbr\u003E1 капсула 1 мкг содержит:\u003Cbr\u003Eдействующее вещество: альфакальцидол 1,00 мкг;\u003Cbr\u003Eвспомогательные вещества: арахиса масло 98,8000 мг, лимонная кислота (безводная) 0,01500 мг, пропилгаллат 0,02000 мг, альфа-токоферол 0,02000 мг, этиловый спирт (этанол) 1,14400 мг;\u003Cbr\u003Eкапсула мягкая желатиновая: сорбитол частично дегидратированный 12,39 мг, глицерол 18,67 мг, желатин 77,80 мг, краситель железа оксид желтый 0,08 мг, титана диоксид 1,06 мг."},{"description":"","filters":[{"id":50921347,"name":"Взаимодействие"}],"isMainProperty":false,"name":"Взаимодействие","value":"Индукторы микросомальных ферментов печени (в том числе фенитоин и фенобарбитал) снижают, а ингибиторы - повышают концентрацию альфакальцидола в плазме (возможно изменение его эффективности).\u003Cbr\u003EПри одновременном применении альфакальцидола с препаратами наперстянки повышается риск развития аритмии.\u003Cbr\u003EВсасывание альфакальцидола уменьшается при его совместном применении с колестирамином, колестиполом, минеральным маслом, сукральфатом, антацидами. Для снижения вероятности взаимодействия альфакальцидол следует применять за 1 час до или через 4-6 часов после приема вышеуказанных препаратов.\u003Cbr\u003EКальцитонин, производные этидроновой и памидроновой кислот, пликамицин, галлия нитрат и глюкокортикостероиды снижают эффект альфакальцидола.\u003Cbr\u003EАльфакальцидол увеличивает абсорбцию фосфорсодержащих препаратов и риск возникновения гиперфосфатемии.\u003Cbr\u003EОдновременное применение альфакальцидола с препаратами кальция, тиазидными диуретиками может вызвать гиперкальциемию за счет повышения абсорбции кальция в кишечнике, увеличения его реабсорбции в почках.\u003Cbr\u003EСочетанная терапия магнийсодержащими антацидами и витамином D может вызвать повышение содержания магния в крови, а алюминийсодержащими антацидами - алюминия в крови, особенно при ХПН.\u003Cbr\u003EОдновременное применение различных аналогов витамина D сопровождается аддитивным действием с развитием гиперкальциемии. Альфакальцидол не следует назначать одновременно с другими препаратами витамина D и его производными."},{"description":"","filters":[{"id":50921465,"name":"Показания к применению"}],"isMainProperty":false,"name":"Показания к применению","value":"Заболевания, вызванные нарушением обмена кальция и фосфора вследствие недостаточного эндогенного синтеза 1,25-дигидроксивитамина D3:\u003Cbr\u003E- остеопороз (в т.ч. постменопаузальный, сенильный, стероидный и др.);\u003Cbr\u003E- остеодистрофия при хронической почечной недостаточности (ХПН);\u003Cbr\u003E- гипопаратиреоз и псевдогипопаратиреоз;\u003Cbr\u003E- витамин D-резистентный рахит и остеомаляция."},{"description":"","filters":[{"id":50925451,"name":"Противопоказания"}],"isMainProperty":false,"name":"Противопоказания","value":"Гиперчувствительность к компонентам препарата, в том числе к арахису;\u003Cbr\u003E- гиперкальциемия;\u003Cbr\u003E- гиперфосфатемия;\u003Cbr\u003E- гипермагниемия;\u003Cbr\u003E- гипервитаминоз D;\u003Cbr\u003E- период беременности и грудного вскармливания;\u003Cbr\u003E- детский возраст до 12 лет;\u003Cbr\u003E- длительная иммобилизация;\u003Cbr\u003E- туберкулез легких (активная форма)."},{"description":"","filters":[{"id":50921469,"name":"Способ применения и дозы"}],"isMainProperty":false,"name":"Способ применения и дозы","value":"Препарат Альфакальцидол Канон принимают внутрь независимо от приема пищи, не разжевывая, запивая достаточным количеством жидкости, однократно в сутки. Длительность курса лечения определяется врачом индивидуально в каждом конкретном случае и зависит от характера заболевания и эффективности терапии.\u003Cbr\u003EВзрослые и дети с 12 лет\u003Cbr\u003EНачальная доза - 1 мкг в сутки.\u003Cbr\u003EПоддерживающая доза - 0,25-2 мкг в сутки.\u003Cbr\u003EПри рахите и остеомаляции: от 1 до 3 мкг в сутки; при гипопаратиреозе: 1-4 мкг в сутки; при остеодистрофии при ХПН: 0,5-2 мкг в сутки; при остеопорозе (в том числе постменопаузальном, сенильном, стероидном и др.): 0,5-1 мкг в сутки.\u003Cbr\u003EНачинать лечение рекомендуется с минимальных доз, контролируя 1 раз в неделю концентрацию кальция и фосфора в плазме крови. Дозу препарата можно повышать на 0,25 или 0,5 мкг/сут до стабилизации биохимических показателей. При достижении минимальной эффективной дозы рекомендуется контролировать концентрацию кальция в плазме крови каждые 3-5 недель."},{"description":"","filters":[{"id":50921474,"name":"Применение при беременности"}],"isMainProperty":false,"name":"Применение при беременности","value":"Гиперкальциемия у матери в период беременности, связанная с длительной передозировкой витамина D, может вызвать у плода повышение чувствительности к витамину D, подавление функции паращитовидной железы, синдром специфической эльфоподобной внешности, задержку умственного развития, аортальный стеноз.\u003Cbr\u003EПрепарат противопоказан к применению при беременности и в период грудного вскармливания."},{"description":"","filters":[{"id":50921464,"name":"Побочные действия"}],"isMainProperty":false,"name":"Побочные действия","value":"Наиболее распространенными нежелательными эффектами альфакальцидола являются: гиперкальциемия, гиперкальциурия и витамин D-зависимая токсичность.\u003Cbr\u003EНиже приводятся данные о неблагоприятных побочных реакциях, в зависимости от частоты их возникновения. Неблагоприятные побочные реакции, отличные от признаков гиперкальциемии, полученные как отдельные сообщения, также включены.\u003Cbr\u003EЧастота определяется как: очень часто - ≥1/10; часто - ≥1/100 и \u003C1/10; нечасто - ≥1/1000 и \u003C1/100; редко -≥1/10000 и \u003C1/1000; очень редко - \u003C1/10000 (включая отдельные сообщения); частота неизвестна (невозможно оценить на основании имеющихся данных).\u003Cbr\u003EСо стороны обмена веществ\u003Cbr\u003Eочень часто: гиперкальциемия;\u003Cbr\u003Eнечасто: метастатические кальцификации, гиперфосфатемия, высокое содержание кальциево-фосфатных соединений, анорексия;\u003Cbr\u003Eчастота неизвестна: гипермагниемия, сниженный аппетит, снижение массы тела, дегидратация, прекращение роста, альбуминурия, гиперхолестеринемия, повышение уровня ACT и АЛТ в сыворотке крови.\u003Cbr\u003EАллергические реакции\u003Cbr\u003Eчастота неизвестна: реакции гиперчувствительности с такими симптомами, как: лихорадка, озноб, крапивница и отек языка.\u003Cbr\u003EСо стороны нервной системы\u003Cbr\u003Eнечасто: головная боль, дизестезия, дисгевзия;\u003Cbr\u003Eочень редко: нарушения психики, галлюцинации, кома, апатия;\u003Cbr\u003Eчастота неизвестна: гипертермия.\u003Cbr\u003EСо стороны сердечно-сосудистой системы\u003Cbr\u003Eредко: тахикардия, повышение артериального давления.\u003Cbr\u003EСо стороны пищеварительной системы\u003Cbr\u003Eнечасто: тошнота, рвота, боль в животе, запор, диарея, диспепсия;\u003Cbr\u003Eочень редко: острый панкреатит;\u003Cbr\u003Eчастота неизвестна: изъязвление языка, изъязвление десен, полидипсия.\u003Cbr\u003EСо стороны кожных покровов\u003Cbr\u003Eчасто: кожный зуд;\u003Cbr\u003Eочень редко: мультиформная эритема, псориаз;\u003Cbr\u003Eчастота неизвестна: сыпь (эритематозная, макулопапулезная, пустулезная), эксфолиативный дерматит.\u003Cbr\u003EСо стороны органов чувств\u003Cbr\u003Eочень редко: кальциноз конъюнктивы и склеры.\u003Cbr\u003EСо стороны дыхательной системы\u003Cbr\u003Eчастота неизвестна: ринит.\u003Cbr\u003EСо стороны мочевыделителъной системы\u003Cbr\u003Eчасто: гиперкальциурия, повышение уровня креатинина и мочевины в сыворотке_крови: частота неизвестна: почечная недостаточность, нефрокальциноз, инфекции мочевыводящих путей.\u003Cbr\u003EСо стороны репродуктивной системы\u003Cbr\u003Eчастота неизвестна: снижение либидо.\u003Cbr\u003EПрочие\u003Cbr\u003Eредко: кальциноз, астения и повышенная утомляемость."},{"description":"","filters":[{"id":50921468,"name":"Передозировка"}],"isMainProperty":false,"name":"Передозировка","value":"Ранние симптомы гипервитаминоза витамина D (обусловленные гиперкальциемией): запор или диарея, сухость слизистой оболочки полости рта, головная боль, жажда, поллакиурия, никтурия, полиурия, анорексия, металлический привкус во рту, тошнота, рвота, общая слабость, гиперкальциурия.\u003Cbr\u003EПоздние симптомы гипервитаминоза витамина D: боль в костях, помутнение мочи (появление в моче гиалиновых цилиндров), повышение артериального давления, кожный зуд, светобоязнь, гиперемия конъюнктивы, аритмия, сонливость, миалгия, тошнота, рвота, снижение массы тела, редко - изменения психики и настроения, спутанность сознания.\u003Cbr\u003EСимптомы хронической интоксикации витамина D: кальциноз мягких тканей, кровеносных сосудов и внутренних органов (почек, легких), почечная и сердечно-сосудистая недостаточность, нарушение роста у детей.\u003Cbr\u003EУровень кальция в сыворотке крови нормализуется через 2-7 дней после прекращения приема препарата.\u003Cbr\u003EЛечение\u003Cbr\u003EГиперкальциемия лечится временным прекращением приема альфакальцидола, введением диеты с низким содержанием кальция и прекращением приема добавок кальция.\u003Cbr\u003EВ тяжелых случаях острой случайной передозировки и устойчивой гиперкальциемии следует предпринять общие поддерживающие мероприятия.\u003Cbr\u003EВ случае передозировки следует отменить препарат. В ранние сроки острой передозировки показано промывание желудка и/или прием внутрь минерального масла (вазелинового), способствующего уменьшению всасывания и увеличению выведения препарата через кишечник. В тяжелых случаях (уровень кальция в сыворотке крови \u003E3 ммоль/л) может потребоваться проведение поддерживающих лечебных мероприятий - гидратации с введением инфузионных солевых растворов (с целью форсированного диуреза), в некоторых случаях - назначение глюкокортикостероидных препаратов, петлевых диуретиков, бисфосфонатов, кальцитонина, перитонеального диализа или гемодиализа с применением диализата, не содержащего кальций. Обязателен контроле содержания электролитов в сыворотке крови (особенно кальция), функции почек и состояния сердца (по данным электрокардиограммы), особенно у пациентов, принимающих дигоксин или другие препараты наперстянки)."},{"description":"","filters":[{"id":50921467,"name":"Условия хранения"}],"isMainProperty":false,"name":"Условия хранения","value":"Хранить при температуре не выше 25 °C во вторичной упаковке (пачке картонной).\u003Cbr\u003EХранить в недоступном для детей месте."},{"description":"","filters":[{"id":50921466,"name":"Особые указания"}],"isMainProperty":false,"name":"Особые указания","value":"С осторожностью:\u003Cbr\u003EПри нефроуролитиазе, атеросклерозе, хронической сердечной недостаточности, хронической почечной недостаточности, туберкулезе, саркоидозе или других гранулематозах, органических поражениях сердца, у пациентов с печеночной недостаточностью, у пациентов, получающих тиазидные диуретики или сердечные гликозиды, у пациентов с повышенным риском развития гиперкальциемии; особенно, при наличии почечнокаменной болезни, заболеваниях желудочно-кишечного тракта (в том числе, язвенная болезнь желудка и 12-перстной кишки), гипотериозе, у детей старше 12 лет.\u003Cbr\u003EСледует обратить внимание на пациентов, принимающих сердечные гликозиды, так как гиперкальциемия может привести к развитию аритмии у таких пациентов.\u003Cbr\u003EСледует обратить внимание на пациентов, принимающих тиазидные диуретики, так как у таких пациентов может увеличиваться риск развития гиперкальциемии.\u003Cbr\u003EЭффективность альфакальцидола в целом сохраняется у пациентов со сниженной функцией печени. При тяжелой печеночной недостаточности концентрация активного метаболита 1,25-дигидроксивитамина D может уменьшаться за счет ослабления процесса гидроксилирования или ввиду снижения энтерогепатической циркуляции. В этом случае может потребоваться назначение препарата в более высоких дозах.\u003Cbr\u003EПри применении препарата у пожилых людей корректировки дозы не требуется.\u003Cbr\u003EПрепарат может способствовать развитию гиперкальциемии, поэтому пациентов следует информировать о клинических симптомах этого состояния (см. раздел «Передозировка»). Во время применения альфакальцидола необходимо регулярно контролировать концентрацию кальция, фосфатов, кальциево-фосфатных соединений, щелочной фосфатазы и уровень паратиреоидного гормона в сыворотке крови.\u003Cbr\u003EКонцентрацию кальция следует определять один раз в неделю или в месяц в зависимости от клинической ситуации. Более частое измерение содержания кальция требуется в начале лечения, особенно при состояниях без значительного поражения костей, например, гипопаратиреозе, и, если содержание кальция в плазме уже повышено, а также на более поздних этапах лечения при наличии признаков восстановления структуры костной ткани. Риск развития гиперкальциемии определяется такими факторами, как: степень деминерализации кости, функциональная способность почек и доза альфакальцидола. Появление гиперкальциемии может быть обусловлено тем, что доза препарата не снижается своевременно и адекватно при наличии биохимических признаков восстановления структуры костной ткани (нормализация щелочной фосфатазы в крови). Следует предотвращать развитие длительной гиперкальциемии, особенно при ХПН, ориентируясь на такие показатели, как концентрация в сыворотке крови кальция, щелочной фосфатазы, паратиреоидного гормона, количество кальция, выделяющегося с мочой, рентгенологические и биохимические данные.\u003Cbr\u003EПри развитии гиперкальциемии или стойком повышении уровня кальциево-фосфатных соединений, выходящего за пределы клинической нормы, препарат нужно немедленно отменить, по меньшей мере, до тех пор, пока данные показатели не нормализуются (обычно в течение одной недели), затем прием препарата можно возобновить в дозе, составляющей половину от предыдущей.\u003Cbr\u003EПациенты с выраженным поражением костей (в отличие от пациентов с почечной недостаточностью) могут переносить более высокие дозы препарата без признаков гиперкальциемии. Отсутствие быстрого повышения содержания кальция в сыворотке крови у пациентов с остеомаляцией не обязательно означает, что должна быть повышена доза препарата, так как кальций может проникать в деминерализованную кость за счет его возросшей абсорбции в кишечнике.\u003Cbr\u003EНеобходимо избегать чрезмерного подавления паратиреоидною гормона. Для пациентов, находящихся на диализе, уровень паратиреоидного гормона в сыворотке крови должен соответствовать действующим руководствам по лечению.\u003Cbr\u003EДля предотвращения развития гиперфосфатемии у пациентов с поражением костей почечного генеза, альфакацидол можно применять вместе с фосфатсвязывающими средствами.\u003Cbr\u003EПри остеопорозе применение альфакальцидола можно сочетать с эстрогенами и антирезорбтивными препаратами.\u003Cbr\u003EВ состав вспомогательных веществ препарата входит масло арахиса. 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Альфакальцидол стимулирует регенерацию мышечных волокон, что восстанавливает утраченный мышечный тонус."},{"description":"","filters":[{"id":50921473,"name":"Состав"}],"isMainProperty":false,"name":"Состав","value":"1 капсула 0,25 мкг содержит:\u003Cbr\u003Eдействующее вещество: альфакальцидол 0,25 мкг;\u003Cbr\u003Eвспомогательные вещества: арахиса масло 98,79975 мг, лимонная кислота (безводная) 0,01500 мг, пропилгаллат 0,02000 мг, альфа-токоферол 0,02000 мг, этиловый спирт (этанол) 1,14500 мг;\u003Cbr\u003Eкапсула мягкая желатиновая: сорбитол частично дегидратированный 12,45 мг, глицерол 18,38 мг, желатин 78,32 мг, краситель железа оксид красный 0,85 мг.\u003Cbr\u003E1 капсула 1 мкг содержит:\u003Cbr\u003Eдействующее вещество: альфакальцидол 1,00 мкг;\u003Cbr\u003Eвспомогательные вещества: арахиса масло 98,8000 мг, лимонная кислота (безводная) 0,01500 мг, пропилгаллат 0,02000 мг, альфа-токоферол 0,02000 мг, этиловый спирт (этанол) 1,14400 мг;\u003Cbr\u003Eкапсула мягкая желатиновая: сорбитол частично дегидратированный 12,39 мг, глицерол 18,67 мг, желатин 77,80 мг, краситель железа оксид желтый 0,08 мг, титана диоксид 1,06 мг."},{"description":"","filters":[{"id":50921347,"name":"Взаимодействие"}],"isMainProperty":false,"name":"Взаимодействие","value":"Индукторы микросомальных ферментов печени (в том числе фенитоин и фенобарбитал) снижают, а ингибиторы - повышают концентрацию альфакальцидола в плазме (возможно изменение его эффективности).\u003Cbr\u003EПри одновременном применении альфакальцидола с препаратами наперстянки повышается риск развития аритмии.\u003Cbr\u003EВсасывание альфакальцидола уменьшается при его совместном применении с колестирамином, колестиполом, минеральным маслом, сукральфатом, антацидами. Для снижения вероятности взаимодействия альфакальцидол следует применять за 1 час до или через 4-6 часов после приема вышеуказанных препаратов.\u003Cbr\u003EКальцитонин, производные этидроновой и памидроновой кислот, пликамицин, галлия нитрат и глюкокортикостероиды снижают эффект альфакальцидола.\u003Cbr\u003EАльфакальцидол увеличивает абсорбцию фосфорсодержащих препаратов и риск возникновения гиперфосфатемии.\u003Cbr\u003EОдновременное применение альфакальцидола с препаратами кальция, тиазидными диуретиками может вызвать гиперкальциемию за счет повышения абсорбции кальция в кишечнике, увеличения его реабсорбции в почках.\u003Cbr\u003EСочетанная терапия магнийсодержащими антацидами и витамином D может вызвать повышение содержания магния в крови, а алюминийсодержащими антацидами - алюминия в крови, особенно при ХПН.\u003Cbr\u003EОдновременное применение различных аналогов витамина D сопровождается аддитивным действием с развитием гиперкальциемии. Альфакальцидол не следует назначать одновременно с другими препаратами витамина D и его производными."},{"description":"","filters":[{"id":50921465,"name":"Показания к применению"}],"isMainProperty":false,"name":"Показания к применению","value":"Заболевания, вызванные нарушением обмена кальция и фосфора вследствие недостаточного эндогенного синтеза 1,25-дигидроксивитамина D3:\u003Cbr\u003E- остеопороз (в т.ч. постменопаузальный, сенильный, стероидный и др.);\u003Cbr\u003E- остеодистрофия при хронической почечной недостаточности (ХПН);\u003Cbr\u003E- гипопаратиреоз и псевдогипопаратиреоз;\u003Cbr\u003E- витамин D-резистентный рахит и остеомаляция."},{"description":"","filters":[{"id":50925451,"name":"Противопоказания"}],"isMainProperty":false,"name":"Противопоказания","value":"Гиперчувствительность к компонентам препарата, в том числе к арахису;\u003Cbr\u003E- гиперкальциемия;\u003Cbr\u003E- гиперфосфатемия;\u003Cbr\u003E- гипермагниемия;\u003Cbr\u003E- гипервитаминоз D;\u003Cbr\u003E- период беременности и грудного вскармливания;\u003Cbr\u003E- детский возраст до 12 лет;\u003Cbr\u003E- длительная иммобилизация;\u003Cbr\u003E- туберкулез легких (активная форма)."},{"description":"","filters":[{"id":50921469,"name":"Способ применения и дозы"}],"isMainProperty":false,"name":"Способ применения и дозы","value":"Препарат Альфакальцидол Канон принимают внутрь независимо от приема пищи, не разжевывая, запивая достаточным количеством жидкости, однократно в сутки. Длительность курса лечения определяется врачом индивидуально в каждом конкретном случае и зависит от характера заболевания и эффективности терапии.\u003Cbr\u003EВзрослые и дети с 12 лет\u003Cbr\u003EНачальная доза - 1 мкг в сутки.\u003Cbr\u003EПоддерживающая доза - 0,25-2 мкг в сутки.\u003Cbr\u003EПри рахите и остеомаляции: от 1 до 3 мкг в сутки; при гипопаратиреозе: 1-4 мкг в сутки; при остеодистрофии при ХПН: 0,5-2 мкг в сутки; при остеопорозе (в том числе постменопаузальном, сенильном, стероидном и др.): 0,5-1 мкг в сутки.\u003Cbr\u003EНачинать лечение рекомендуется с минимальных доз, контролируя 1 раз в неделю концентрацию кальция и фосфора в плазме крови. Дозу препарата можно повышать на 0,25 или 0,5 мкг/сут до стабилизации биохимических показателей. При достижении минимальной эффективной дозы рекомендуется контролировать концентрацию кальция в плазме крови каждые 3-5 недель."},{"description":"","filters":[{"id":50921474,"name":"Применение при беременности"}],"isMainProperty":false,"name":"Применение при беременности","value":"Гиперкальциемия у матери в период беременности, связанная с длительной передозировкой витамина D, может вызвать у плода повышение чувствительности к витамину D, подавление функции паращитовидной железы, синдром специфической эльфоподобной внешности, задержку умственного развития, аортальный стеноз.\u003Cbr\u003EПрепарат противопоказан к применению при беременности и в период грудного вскармливания."},{"description":"","filters":[{"id":50921464,"name":"Побочные действия"}],"isMainProperty":false,"name":"Побочные действия","value":"Наиболее распространенными нежелательными эффектами альфакальцидола являются: гиперкальциемия, гиперкальциурия и витамин D-зависимая токсичность.\u003Cbr\u003EНиже приводятся данные о неблагоприятных побочных реакциях, в зависимости от частоты их возникновения. Неблагоприятные побочные реакции, отличные от признаков гиперкальциемии, полученные как отдельные сообщения, также включены.\u003Cbr\u003EЧастота определяется как: очень часто - ≥1/10; часто - ≥1/100 и \u003C1/10; нечасто - ≥1/1000 и \u003C1/100; редко -≥1/10000 и \u003C1/1000; очень редко - \u003C1/10000 (включая отдельные сообщения); частота неизвестна (невозможно оценить на основании имеющихся данных).\u003Cbr\u003EСо стороны обмена веществ\u003Cbr\u003Eочень часто: гиперкальциемия;\u003Cbr\u003Eнечасто: метастатические кальцификации, гиперфосфатемия, высокое содержание кальциево-фосфатных соединений, анорексия;\u003Cbr\u003Eчастота неизвестна: гипермагниемия, сниженный аппетит, снижение массы тела, дегидратация, прекращение роста, альбуминурия, гиперхолестеринемия, повышение уровня ACT и АЛТ в сыворотке крови.\u003Cbr\u003EАллергические реакции\u003Cbr\u003Eчастота неизвестна: реакции гиперчувствительности с такими симптомами, как: лихорадка, озноб, крапивница и отек языка.\u003Cbr\u003EСо стороны нервной системы\u003Cbr\u003Eнечасто: головная боль, дизестезия, дисгевзия;\u003Cbr\u003Eочень редко: нарушения психики, галлюцинации, кома, апатия;\u003Cbr\u003Eчастота неизвестна: гипертермия.\u003Cbr\u003EСо стороны сердечно-сосудистой системы\u003Cbr\u003Eредко: тахикардия, повышение артериального давления.\u003Cbr\u003EСо стороны пищеварительной системы\u003Cbr\u003Eнечасто: тошнота, рвота, боль в животе, запор, диарея, диспепсия;\u003Cbr\u003Eочень редко: острый панкреатит;\u003Cbr\u003Eчастота неизвестна: изъязвление языка, изъязвление десен, полидипсия.\u003Cbr\u003EСо стороны кожных покровов\u003Cbr\u003Eчасто: кожный зуд;\u003Cbr\u003Eочень редко: мультиформная эритема, псориаз;\u003Cbr\u003Eчастота неизвестна: сыпь (эритематозная, макулопапулезная, пустулезная), эксфолиативный дерматит.\u003Cbr\u003EСо стороны органов чувств\u003Cbr\u003Eочень редко: кальциноз конъюнктивы и склеры.\u003Cbr\u003EСо стороны дыхательной системы\u003Cbr\u003Eчастота неизвестна: ринит.\u003Cbr\u003EСо стороны мочевыделителъной системы\u003Cbr\u003Eчасто: гиперкальциурия, повышение уровня креатинина и мочевины в сыворотке_крови: частота неизвестна: почечная недостаточность, нефрокальциноз, инфекции мочевыводящих путей.\u003Cbr\u003EСо стороны репродуктивной системы\u003Cbr\u003Eчастота неизвестна: снижение либидо.\u003Cbr\u003EПрочие\u003Cbr\u003Eредко: кальциноз, астения и повышенная утомляемость."},{"description":"","filters":[{"id":50921468,"name":"Передозировка"}],"isMainProperty":false,"name":"Передозировка","value":"Ранние симптомы гипервитаминоза витамина D (обусловленные гиперкальциемией): запор или диарея, сухость слизистой оболочки полости рта, головная боль, жажда, поллакиурия, никтурия, полиурия, анорексия, металлический привкус во рту, тошнота, рвота, общая слабость, гиперкальциурия.\u003Cbr\u003EПоздние симптомы гипервитаминоза витамина D: боль в костях, помутнение мочи (появление в моче гиалиновых цилиндров), повышение артериального давления, кожный зуд, светобоязнь, гиперемия конъюнктивы, аритмия, сонливость, миалгия, тошнота, рвота, снижение массы тела, редко - изменения психики и настроения, спутанность сознания.\u003Cbr\u003EСимптомы хронической интоксикации витамина D: кальциноз мягких тканей, кровеносных сосудов и внутренних органов (почек, легких), почечная и сердечно-сосудистая недостаточность, нарушение роста у детей.\u003Cbr\u003EУровень кальция в сыворотке крови нормализуется через 2-7 дней после прекращения приема препарата.\u003Cbr\u003EЛечение\u003Cbr\u003EГиперкальциемия лечится временным прекращением приема альфакальцидола, введением диеты с низким содержанием кальция и прекращением приема добавок кальция.\u003Cbr\u003EВ тяжелых случаях острой случайной передозировки и устойчивой гиперкальциемии следует предпринять общие поддерживающие мероприятия.\u003Cbr\u003EВ случае передозировки следует отменить препарат. В ранние сроки острой передозировки показано промывание желудка и/или прием внутрь минерального масла (вазелинового), способствующего уменьшению всасывания и увеличению выведения препарата через кишечник. В тяжелых случаях (уровень кальция в сыворотке крови \u003E3 ммоль/л) может потребоваться проведение поддерживающих лечебных мероприятий - гидратации с введением инфузионных солевых растворов (с целью форсированного диуреза), в некоторых случаях - назначение глюкокортикостероидных препаратов, петлевых диуретиков, бисфосфонатов, кальцитонина, перитонеального диализа или гемодиализа с применением диализата, не содержащего кальций. Обязателен контроле содержания электролитов в сыворотке крови (особенно кальция), функции почек и состояния сердца (по данным электрокардиограммы), особенно у пациентов, принимающих дигоксин или другие препараты наперстянки)."},{"description":"","filters":[{"id":50921467,"name":"Условия хранения"}],"isMainProperty":false,"name":"Условия хранения","value":"Хранить при температуре не выше 25 °C во вторичной упаковке (пачке картонной).\u003Cbr\u003EХранить в недоступном для детей месте."},{"description":"","filters":[{"id":50921466,"name":"Особые указания"}],"isMainProperty":false,"name":"Особые указания","value":"С осторожностью:\u003Cbr\u003EПри нефроуролитиазе, атеросклерозе, хронической сердечной недостаточности, хронической почечной недостаточности, туберкулезе, саркоидозе или других гранулематозах, органических поражениях сердца, у пациентов с печеночной недостаточностью, у пациентов, получающих тиазидные диуретики или сердечные гликозиды, у пациентов с повышенным риском развития гиперкальциемии; особенно, при наличии почечнокаменной болезни, заболеваниях желудочно-кишечного тракта (в том числе, язвенная болезнь желудка и 12-перстной кишки), гипотериозе, у детей старше 12 лет.\u003Cbr\u003EСледует обратить внимание на пациентов, принимающих сердечные гликозиды, так как гиперкальциемия может привести к развитию аритмии у таких пациентов.\u003Cbr\u003EСледует обратить внимание на пациентов, принимающих тиазидные диуретики, так как у таких пациентов может увеличиваться риск развития гиперкальциемии.\u003Cbr\u003EЭффективность альфакальцидола в целом сохраняется у пациентов со сниженной функцией печени. При тяжелой печеночной недостаточности концентрация активного метаболита 1,25-дигидроксивитамина D может уменьшаться за счет ослабления процесса гидроксилирования или ввиду снижения энтерогепатической циркуляции. В этом случае может потребоваться назначение препарата в более высоких дозах.\u003Cbr\u003EПри применении препарата у пожилых людей корректировки дозы не требуется.\u003Cbr\u003EПрепарат может способствовать развитию гиперкальциемии, поэтому пациентов следует информировать о клинических симптомах этого состояния (см. раздел «Передозировка»). Во время применения альфакальцидола необходимо регулярно контролировать концентрацию кальция, фосфатов, кальциево-фосфатных соединений, щелочной фосфатазы и уровень паратиреоидного гормона в сыворотке крови.\u003Cbr\u003EКонцентрацию кальция следует определять один раз в неделю или в месяц в зависимости от клинической ситуации. Более частое измерение содержания кальция требуется в начале лечения, особенно при состояниях без значительного поражения костей, например, гипопаратиреозе, и, если содержание кальция в плазме уже повышено, а также на более поздних этапах лечения при наличии признаков восстановления структуры костной ткани. Риск развития гиперкальциемии определяется такими факторами, как: степень деминерализации кости, функциональная способность почек и доза альфакальцидола. Появление гиперкальциемии может быть обусловлено тем, что доза препарата не снижается своевременно и адекватно при наличии биохимических признаков восстановления структуры костной ткани (нормализация щелочной фосфатазы в крови). Следует предотвращать развитие длительной гиперкальциемии, особенно при ХПН, ориентируясь на такие показатели, как концентрация в сыворотке крови кальция, щелочной фосфатазы, паратиреоидного гормона, количество кальция, выделяющегося с мочой, рентгенологические и биохимические данные.\u003Cbr\u003EПри развитии гиперкальциемии или стойком повышении уровня кальциево-фосфатных соединений, выходящего за пределы клинической нормы, препарат нужно немедленно отменить, по меньшей мере, до тех пор, пока данные показатели не нормализуются (обычно в течение одной недели), затем прием препарата можно возобновить в дозе, составляющей половину от предыдущей.\u003Cbr\u003EПациенты с выраженным поражением костей (в отличие от пациентов с почечной недостаточностью) могут переносить более высокие дозы препарата без признаков гиперкальциемии. Отсутствие быстрого повышения содержания кальция в сыворотке крови у пациентов с остеомаляцией не обязательно означает, что должна быть повышена доза препарата, так как кальций может проникать в деминерализованную кость за счет его возросшей абсорбции в кишечнике.\u003Cbr\u003EНеобходимо избегать чрезмерного подавления паратиреоидною гормона. Для пациентов, находящихся на диализе, уровень паратиреоидного гормона в сыворотке крови должен соответствовать действующим руководствам по лечению.\u003Cbr\u003EДля предотвращения развития гиперфосфатемии у пациентов с поражением костей почечного генеза, альфакацидол можно применять вместе с фосфатсвязывающими средствами.\u003Cbr\u003EПри остеопорозе применение альфакальцидола можно сочетать с эстрогенами и антирезорбтивными препаратами.\u003Cbr\u003EВ состав вспомогательных веществ препарата входит масло арахиса. 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