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Участвует в реакциях переноса ацильных групп, взаимодействует и восстанавливает эндогенный глутатион. АЛК способна захватывать свободные радикалы, регулировать связывание тяжёлых металлов. Основная функция α- липоевой кислоты - прямое участие в углеводном обмене, а именно, в аэробном метаболизме продукта гликолиза - пирувата. Таким образом, АЛК способствует ликвидации метаболического ацидоза. Играет важную роль в липидном обмене. Обладает положительным липотропным действием, облегчая перенос ацетата и жирных кислот из цитозоля в матрикс митохондрий для последующего окисления за счёт повышения выработки ко-энзима А. Снижает содержание холестерина и насыщенных жирных кислот в крови, предотвращая развитие атеросклероза и жировой дистрофии печени. Благодаря свойствам а-липоевой кислоты восстанавливать запасы глутатиона, предотвращать повреждение митохондрий, высвобождение цитохрома и гибель клеток, обусловленную воздействием фактора некроза опухоли (TNF-а), α-липоевая кислота применяется при лечении токсических заболеваний печени, в том числе эффективна на всех стадиях алкогольной болезни печени. Механизм защитного действия связан со снижением концентрации токсических продуктов метаболизма этанола, увеличением соотношения надн/над, снижением пероксидации липидов, повышением синтеза глутатиона, приводящим к преобладанию активности антиоксидантных систем над процессами свободнорадикального окисления (гепатопротекторное и дезинтоксикационное действие). Результаты рандомизированных контролируемых исследований показывают, что препараты альфа-липоевой кислоты улучшают гликемический профиль у лиц с метаболическими нарушениями, за счет увеличения утилизации глюкозы инсулинзависимыми и инсулиннезависимыми тканями, а также снижают уровень гликозилирования белков.
Рекомендации по применению:
Взрослым по 1 капсуле 2 раза в день перед едой. Продолжительность приема - 1 месяц. При необходимости курс приема можно повторить.
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