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Бикалутамид Канон таб. п/о плен., 150 мг, 30 шт.

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Дозировка: 150 мг

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Коротко о товаре

Артикул Маркета
4453168649
Действующее вещество
Возраст
от 18 лет
Инструкция
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железы","transition":{"type":"catalog","params":{"categorySlug":"protivoopukholevye-preparaty-i-immunomoduliatory","categoryId":"15756914","navnodeId":"72508","glfilters":["34045610:34516009"]}}},{"name":"Назначение","value":"противоопухолевая терапия, рак предстательной железы","transition":{"type":"catalog","params":{"categorySlug":"protivoopukholevye-preparaty-i-immunomoduliatory","categoryId":"15756914","navnodeId":"72508","glfilters":["36476390:36618162,36617629"]}}},{"name":"Показания к применению","value":"- Монотерапия или адъювантная терапия, в комбинации с аналогом гонадотропин- рилизинг-гормона (ГнРГ) или хирургической кастрацией, распространенного рака предстательной железы;\u003Cbr\u003E\n- лечение местнораспространенного рака предстательной железы (Т3-Т4, любая N, М0, Т1-Т2, N+, М0) в качестве монотерапии или адъювантной терапии в сочетании с радикальной простатэктомией или радиотерапией;\u003Cbr\u003E\n- лечение местнораспространенного неметастатического рака предстательной железы в случаях, когда хирургическая кастрация или другие препараты не эффективны или неприемлемы."},{"name":"Противопоказания","value":"- Повышенная чувствительность к бикалутамиду или другим компонентам препарата;\u003Cbr\u003E\n- дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция;\u003Cbr\u003E\n- женщины;\u003Cbr\u003E\n- детский возраст;\u003Cbr\u003E\n- одновременный прием с терфенадином, астемизолом и цизапридом."},{"name":"Состав","value":"1 таблетка, покрытая пленочной оболочкой, содержит:\u003Cbr /\u003EДозировка 50 мг\u003Cbr /\u003Eактивное вещество: бикалутамид 50 мг;\u003Cbr /\u003Eвспомогательные вещества: крахмал кукурузный 35 мг, кроскармеллоза натрия (примеллоза) 6,5 мг, лактозы моногидрат (сахар молочный) 44,3 мг, повидон 3,2 мг, натрия стеарилфумарат 1 мг;\u003Cbr /\u003Eсостав пленочной оболочки: Опадрай II белый 4 мг, в том числе: поливиниловый спирт 1,6 мг, макрогол (полиэтиленгликоль) 0,808 мг, тальк 0,592 мг, титана диоксид 1 мг.\u003Cbr /\u003EДозировка 150 мг\u003Cbr /\u003Eактивное вещество: бикалутамид 150 мг;\u003Cbr /\u003Eвспомогательные вещества: крахмал кукурузный 107 мг, кроскармеллоза натрия (примеллоза) 19,5 мг, лактозы моногидрат (сахар молочный) 132,9 мг, повидон 7,6 мг, натрия стеарилфумарат 3 мг;\u003Cbr /\u003Eсостав пленочной оболочки: Опадрай II белый 12 мг, в том числе: поливиниловый спирт 4,8 мг, макрогол (полиэтиленгликоль) 2,424 мг, тальк 1,776 мг, титана диоксид 3 мг.\u003Cbr /\u003E"},{"name":"Действующее вещество","value":"Бикалутамид","transition":{"type":"catalog","params":{"categorySlug":"protivoopukholevye-preparaty-i-immunomoduliatory","categoryId":"15756914","navnodeId":"72508","glfilters":["27144131:28709949"]}}},{"name":"Способ применения и дозы","value":"Взрослые мужчины, в том числе пожилые:\u003Cbr\u003E\nПри распространённом раке предстательной железы в комбинации с аналогом ГнРГ или хирургической кастрацией: внутрь по 50 мг один раз в сутки.\u003Cbr\u003E\nПри местнораспространенном раке предстательной железы: внутрь по 150 мг один раз в сутки.\u003Cbr\u003E\nБикалутамид следует принимать продолжительно, как минимум в течение 2 лет.\u003Cbr\u003E\nПри появлении признаков прогрессирования заболевания прием препарата следует прекратить."},{"name":"Побочные действия","value":"Нарушения со стороны иммунной системы: редко - реакции повышенной чувствительности, включая ангионевротический отек, крапивницу, кожная сыпь.\u003Cbr\u003E\nНарушения со стороны эндокринной системы: очень часто - гинекомастия (может сохраняться даже после прекращения терапии, особенно в случае приема препарата в течение длительного времени), болезненность грудных желез; часто - снижение полового влечения, эректильная дисфункция, снижение или повышение массы тела, гипергликемия, сахарный диабет.\u003Cbr\u003E\nНарушения со стороны нервной системы: часто - астенический синдром, головокружение, бессонница или сонливость, тревожность, снижение аппетита; редко - депрессия, \"приливы\" крови к лицу.\u003Cbr\u003E\nНарушения со стороны сердца: часто - стенокардия, развитие или усугубление сердечной недостаточности, повышение артериального давления.\u003Cbr\u003E\nНарушения со стороны дыхательной системы, органов грудной клетки и средостения: редко - боль в груди, кашель, фарингит, бронхит, пневмония, интерстициальные легочные заболевания (в том числе с фатальным исходом), ринит.\u003Cbr\u003E\nНарушения со стороны желудочно-кишечного тракта: часто - тошнота; редко - боль в животе, диспепсия, запор, диарея, рвота, метеоризм, желудочное кровотечение, сухость слизистой оболочки полости рта.\u003Cbr\u003E\nНарушения со стороны печени и желчевыводящих путей: редко - транзиторное повышение активности \"печеночных\" трансаминаз, холестаз, желтуха; очень редко - печеночная недостаточность (в том числе с фатальным исходом).\u003Cbr\u003E\nНарушения со стороны кожи и подкожных тканей: часто - алопеция, гирсутизм или восстановление роста волос, сухость кожи.\u003Cbr\u003E\nНарушения со стороны скелетно-мышечной и соединительной ткани: часто - миастения, миалгия, судороги, артрит, контрактуры суставов.\u003Cbr\u003E\nНарушения со стороны почек и мочевыводящих путей: нечасто - дизурия, полиурия, задержка мочи, периферические отеки; редко - гематурия.\u003Cbr\u003E\nОбщие расстройства и нарушение в месте введения: часто - лихорадка, гриппоподобный синдром, озноб, повышенное потоотделение, боль в тазовой области.\u003Cbr\u003E\nЛабораторные и инструментальные данные: часто: анемия.\u003Cbr\u003E\nНарушения со стороны иммунной системы: редко - реакции повышенной чувствительности, включая ангионевротический отек, крапивницу, кожная сыпь.\u003Cbr\u003E\nНарушения со стороны эндокринной системы: очень часто - гинекомастия (может сохраняться даже после прекращения терапии, особенно в случае приема препарата в течение длительного времени), болезненность грудных желез; часто - снижение полового влечения, эректильная дисфункция, снижение или повышение массы тела, гипергликемия, сахарный диабет.\u003Cbr\u003E\nНарушения со стороны нервной системы: часто - астенический синдром, головокружение, бессонница или сонливость, тревожность, снижение аппетита; редко - депрессия, \"приливы\" крови к лицу.\u003Cbr\u003E\nНарушения со стороны сердца: часто - стенокардия, развитие или усугубление сердечной недостаточности, повышение артериального давления.\u003Cbr\u003E\nНарушения со стороны дыхательной системы, органов грудной клетки и средостения: редко - боль в груди, кашель, фарингит, бронхит, пневмония, интерстициальные легочные заболевания (в том числе с фатальным исходом), ринит.\u003Cbr\u003E\nНарушения со стороны желудочно-кишечного тракта: часто - тошнота; редко - боль в животе, диспепсия, запор, диарея, рвота, метеоризм, желудочное кровотечение, сухость слизистой оболочки полости рта.\u003Cbr\u003E\nНарушения со стороны печени и желчевыводящих путей: редко - транзиторное повышение активности \"печеночных\" трансаминаз, холестаз, желтуха; очень редко - печеночная недостаточность (в том числе с фатальным исходом).\u003Cbr\u003E\nНарушения со стороны кожи и подкожных тканей: часто - алопеция, гирсутизм или восстановление роста волос, сухость кожи.\u003Cbr\u003E\nНарушения со стороны скелетно-мышечной и соединительной ткани: часто - миастения, миалгия, судороги, артрит, контрактуры суставов.\u003Cbr\u003E\nНарушения со стороны почек и мочевыводящих путей: нечасто - дизурия, полиурия, задержка мочи, периферические отеки; редко - гематурия.\u003Cbr\u003E\nОбщие расстройства и нарушение в месте введения: часто - лихорадка, гриппоподобный синдром, озноб, повышенное потоотделение, боль в тазовой области.\u003Cbr\u003E\nЛабораторные и инструментальные данные: часто: анемия."},{"name":"Фармакологическое действие","value":"Противоопухолевое средство, нестероидный антиандрогенный препарат - конкурентный антагонист эндогенных андрогенов. Связываясь с рецепторами на поверхности клеток органов-мишеней, делает их недоступными для андрогенов, повышая при этом концентрацию гормонов в плазме. Результатом этого является регрессия новообразований предстательной железы."},{"name":"Фармакологическая группа","value":"противоопухолевые средства","transition":{"type":"catalog","params":{"categorySlug":"protivoopukholevye-preparaty-i-immunomoduliatory","categoryId":"15756914","navnodeId":"72508","glfilters":["34045110:34518988"]}}},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"protivoopukholevye-preparaty-i-immunomoduliatory","categoryId":"15756914","navnodeId":"72508","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"В сухом, защищенном от света месте при температуре не выше 25 °С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Случаи передозировки у человека не описаны. Специфического антидота нет.\u003Cbr\u003E\nЛечение передозировки: симптоматическое, необходим мониторинг жизненно важных функций организма. Гемодиализ неэффективен, так как бикалутамид прочно связывается с белками плазмы и не выводится с мочой в неизмененном виде."},{"name":"Применение при беременности и кормлении грудью","value":"Бикалутамид Канон противопоказан женщинам и не должен назначаться беременным или в период лактации."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"При применении бикалутамида может наблюдаться сонливость и головокружение, в связи с чем следует соблюдать осторожность при управлении автотранспортом или иными движущимися механизмами."},{"name":"Особые указания","value":"Бикалутамид интенсивно метаболизируется в печени. Учитывая возможность замедления выведения бикалутамида и кумуляции бикалутамида у больных с выраженным нарушением функции печени, целесообразно периодически оценивать функцию печени. Большинство изменений функции печени встречаются в течение первых шести месяцев лечения препаратом.\u003Cbr\u003E\nБикалутамид следует применять с осторожностью у больных со средним и тяжелым нарушением функции печени.\u003Cbr\u003E\nТяжелые нарушения печени при использовании препарата возникают редко, сообщалось о случаях с фатальным исходом. В случае развития выраженных изменений функции печени и/или повышении функциональных проб более чем в 2 раза прием препарата необходимо прекратить.\u003Cbr\u003E\nПри совместном приеме с циклоспорином, после начала использования или отмены бикалутамида рекомендуется проводить тщательный контроль концентрации циклоспорина в плазме и состояния пациента.\u003Cbr\u003E\nУ пациентов с прогрессированием заболевания на фоне повышения концентрации простатспецифического антигена (АСА) необходимо рассмотреть вопрос о прекращении лечения бикалутамидом.\u003Cbr\u003E\nУчитывая возможность ингибирования препаратом активности цитохрома Р450 (изофермента CYP 3А4), следует проявлять осторожность при одновременном применении бикалутамида с препаратами, преимущественно метаболизирующимися с участием изофермента CYP 3А4. Рекомендуется регулярно контролировать протромбиновое время при назначении бикалутамида пациентам, получающим непрямые антикоагулянты кумаринового ряда.\u003Cbr\u003E\nУ пациентов, принимающих агонисты ГнРГ, наблюдалось снижение переносимости глюкозы. Этот эффект может приводить к развитию сахарного диабета или снижению толерантности к глюкозе у пациентов с сахарным диабетом. В связи с чем у пациентов, принимающих бикалутамид в комбинации с агонистами ГнРГ, необходимо контролировать концентрацию глюкозы в крови."},{"name":"Взаимодействие","value":"При применении бикалутамида в течение 28 дней на фоне приема мидазолама, АUC мидазолама увеличивалась на 80%.\u003Cbr\u003EПри одновременном применении бикалутамида с циклоспорином или блокаторами кальциевых каналов возможно потенцирование или развитие нежелательных реакций.\u003Cbr\u003EТеоретически возможно повышение концентрации бикалутамида в плазме крови при его одновременном применении с ингибиторами микросомальных ферментов печени, что может сопровождаться увеличением частоты возникновения нежелательных реакций.\u003Cbr\u003EИсследования in vitro показали, что бикалутамид может вытеснять антикоагулянт кумаринового ряда варфарин из участков связывания с белками плазмы."},{"name":"Регистрационный номер","value":"ЛП-001745"},{"name":"Дата государственной регистрации","value":"14.09.2021"},{"name":"Владелец регистрационного удостоверения","value":"Канонфарма продакшн","transition":{"type":"catalog","params":{"categorySlug":"protivoopukholevye-preparaty-i-immunomoduliatory","categoryId":"15756914","navnodeId":"72508","glfilters":["34324371:35649313","7893318:16146766"]}}},{"name":"Изготовитель","value":"Канонфарма продакшн"},{"name":"Фасовщик","value":"Канонфарма продакшн"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Бикалутамид Канон","transition":{"type":"catalog","params":{"categorySlug":"protivoopukholevye-preparaty-i-immunomoduliatory","categoryId":"15756914","navnodeId":"72508","glfilters":["17796364:18050513"]}}},{"name":"Срок годности","value":"37 мес."}]}},"fullSpecsGrouped":{"10079485356458830176":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"половые железы"},{"name":"Назначение","value":"противоопухолевая терапия, рак предстательной железы"},{"name":"Показания к применению","value":"- Монотерапия или адъювантная терапия, в комбинации с аналогом гонадотропин- рилизинг-гормона (ГнРГ) или хирургической кастрацией, распространенного рака предстательной железы;\u003Cbr\u003E\n- лечение местнораспространенного рака предстательной железы (Т3-Т4, любая N, М0, Т1-Т2, N+, М0) в качестве монотерапии или адъювантной терапии в сочетании с радикальной простатэктомией или радиотерапией;\u003Cbr\u003E\n- лечение местнораспространенного неметастатического рака предстательной железы в случаях, когда хирургическая кастрация или другие препараты не эффективны или неприемлемы."},{"name":"Противопоказания","value":"- Повышенная чувствительность к бикалутамиду или другим компонентам препарата;\u003Cbr\u003E\n- дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция;\u003Cbr\u003E\n- женщины;\u003Cbr\u003E\n- детский возраст;\u003Cbr\u003E\n- одновременный прием с терфенадином, астемизолом и цизапридом."},{"name":"Состав","value":"1 таблетка, покрытая пленочной оболочкой, содержит:\u003Cbr /\u003EДозировка 50 мг\u003Cbr /\u003Eактивное вещество: бикалутамид 50 мг;\u003Cbr /\u003Eвспомогательные вещества: крахмал кукурузный 35 мг, кроскармеллоза натрия (примеллоза) 6,5 мг, лактозы моногидрат (сахар молочный) 44,3 мг, повидон 3,2 мг, натрия стеарилфумарат 1 мг;\u003Cbr /\u003Eсостав пленочной оболочки: Опадрай II белый 4 мг, в том числе: поливиниловый спирт 1,6 мг, макрогол (полиэтиленгликоль) 0,808 мг, тальк 0,592 мг, титана диоксид 1 мг.\u003Cbr /\u003EДозировка 150 мг\u003Cbr /\u003Eактивное вещество: бикалутамид 150 мг;\u003Cbr /\u003Eвспомогательные вещества: крахмал кукурузный 107 мг, кроскармеллоза натрия (примеллоза) 19,5 мг, лактозы моногидрат (сахар молочный) 132,9 мг, повидон 7,6 мг, натрия стеарилфумарат 3 мг;\u003Cbr /\u003Eсостав пленочной оболочки: Опадрай II белый 12 мг, в том числе: поливиниловый спирт 4,8 мг, макрогол (полиэтиленгликоль) 2,424 мг, тальк 1,776 мг, титана диоксид 3 мг.\u003Cbr /\u003E"},{"name":"Действующее вещество","value":"Бикалутамид"},{"name":"Способ применения и дозы","value":"Взрослые мужчины, в том числе пожилые:\u003Cbr\u003E\nПри распространённом раке предстательной железы в комбинации с аналогом ГнРГ или хирургической кастрацией: внутрь по 50 мг один раз в сутки.\u003Cbr\u003E\nПри местнораспространенном раке предстательной железы: внутрь по 150 мг один раз в сутки.\u003Cbr\u003E\nБикалутамид следует принимать продолжительно, как минимум в течение 2 лет.\u003Cbr\u003E\nПри появлении признаков прогрессирования заболевания прием препарата следует прекратить."},{"name":"Побочные действия","value":"Нарушения со стороны иммунной системы: редко - реакции повышенной чувствительности, включая ангионевротический отек, крапивницу, кожная сыпь.\u003Cbr\u003E\nНарушения со стороны эндокринной системы: очень часто - гинекомастия (может сохраняться даже после прекращения терапии, особенно в случае приема препарата в течение длительного времени), болезненность грудных желез; часто - снижение полового влечения, эректильная дисфункция, снижение или повышение массы тела, гипергликемия, сахарный диабет.\u003Cbr\u003E\nНарушения со стороны нервной системы: часто - астенический синдром, головокружение, бессонница или сонливость, тревожность, снижение аппетита; редко - депрессия, \"приливы\" крови к лицу.\u003Cbr\u003E\nНарушения со стороны сердца: часто - стенокардия, развитие или усугубление сердечной недостаточности, повышение артериального давления.\u003Cbr\u003E\nНарушения со стороны дыхательной системы, органов грудной клетки и средостения: редко - боль в груди, кашель, фарингит, бронхит, пневмония, интерстициальные легочные заболевания (в том числе с фатальным исходом), ринит.\u003Cbr\u003E\nНарушения со стороны желудочно-кишечного тракта: часто - тошнота; редко - боль в животе, диспепсия, запор, диарея, рвота, метеоризм, желудочное кровотечение, сухость слизистой оболочки полости рта.\u003Cbr\u003E\nНарушения со стороны печени и желчевыводящих путей: редко - транзиторное повышение активности \"печеночных\" трансаминаз, холестаз, желтуха; очень редко - печеночная недостаточность (в том числе с фатальным исходом).\u003Cbr\u003E\nНарушения со стороны кожи и подкожных тканей: часто - алопеция, гирсутизм или восстановление роста волос, сухость кожи.\u003Cbr\u003E\nНарушения со стороны скелетно-мышечной и соединительной ткани: часто - миастения, миалгия, судороги, артрит, контрактуры суставов.\u003Cbr\u003E\nНарушения со стороны почек и мочевыводящих путей: нечасто - дизурия, полиурия, задержка мочи, периферические отеки; редко - гематурия.\u003Cbr\u003E\nОбщие расстройства и нарушение в месте введения: часто - лихорадка, гриппоподобный синдром, озноб, повышенное потоотделение, боль в тазовой области.\u003Cbr\u003E\nЛабораторные и инструментальные данные: часто: анемия.\u003Cbr\u003E\nНарушения со стороны иммунной системы: редко - реакции повышенной чувствительности, включая ангионевротический отек, крапивницу, кожная сыпь.\u003Cbr\u003E\nНарушения со стороны эндокринной системы: очень часто - гинекомастия (может сохраняться даже после прекращения терапии, особенно в случае приема препарата в течение длительного времени), болезненность грудных желез; часто - снижение полового влечения, эректильная дисфункция, снижение или повышение массы тела, гипергликемия, сахарный диабет.\u003Cbr\u003E\nНарушения со стороны нервной системы: часто - астенический синдром, головокружение, бессонница или сонливость, тревожность, снижение аппетита; редко - депрессия, \"приливы\" крови к лицу.\u003Cbr\u003E\nНарушения со стороны сердца: часто - стенокардия, развитие или усугубление сердечной недостаточности, повышение артериального давления.\u003Cbr\u003E\nНарушения со стороны дыхательной системы, органов грудной клетки и средостения: редко - боль в груди, кашель, фарингит, бронхит, пневмония, интерстициальные легочные заболевания (в том числе с фатальным исходом), ринит.\u003Cbr\u003E\nНарушения со стороны желудочно-кишечного тракта: часто - тошнота; редко - боль в животе, диспепсия, запор, диарея, рвота, метеоризм, желудочное кровотечение, сухость слизистой оболочки полости рта.\u003Cbr\u003E\nНарушения со стороны печени и желчевыводящих путей: редко - транзиторное повышение активности \"печеночных\" трансаминаз, холестаз, желтуха; очень редко - печеночная недостаточность (в том числе с фатальным исходом).\u003Cbr\u003E\nНарушения со стороны кожи и подкожных тканей: часто - алопеция, гирсутизм или восстановление роста волос, сухость кожи.\u003Cbr\u003E\nНарушения со стороны скелетно-мышечной и соединительной ткани: часто - миастения, миалгия, судороги, артрит, контрактуры суставов.\u003Cbr\u003E\nНарушения со стороны почек и мочевыводящих путей: нечасто - дизурия, полиурия, задержка мочи, периферические отеки; редко - гематурия.\u003Cbr\u003E\nОбщие расстройства и нарушение в месте введения: часто - лихорадка, гриппоподобный синдром, озноб, повышенное потоотделение, боль в тазовой области.\u003Cbr\u003E\nЛабораторные и инструментальные данные: часто: анемия."},{"name":"Фармакологическое действие","value":"Противоопухолевое средство, нестероидный антиандрогенный препарат - конкурентный антагонист эндогенных андрогенов. Связываясь с рецепторами на поверхности клеток органов-мишеней, делает их недоступными для андрогенов, повышая при этом концентрацию гормонов в плазме. Результатом этого является регрессия новообразований предстательной железы."},{"name":"Фармакологическая группа","value":"противоопухолевые средства"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В сухом, защищенном от света месте при температуре не выше 25 °С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Случаи передозировки у человека не описаны. Специфического антидота нет.\u003Cbr\u003E\nЛечение передозировки: симптоматическое, необходим мониторинг жизненно важных функций организма. Гемодиализ неэффективен, так как бикалутамид прочно связывается с белками плазмы и не выводится с мочой в неизмененном виде."},{"name":"Применение при беременности и кормлении грудью","value":"Бикалутамид Канон противопоказан женщинам и не должен назначаться беременным или в период лактации."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"При применении бикалутамида может наблюдаться сонливость и головокружение, в связи с чем следует соблюдать осторожность при управлении автотранспортом или иными движущимися механизмами."},{"name":"Особые указания","value":"Бикалутамид интенсивно метаболизируется в печени. Учитывая возможность замедления выведения бикалутамида и кумуляции бикалутамида у больных с выраженным нарушением функции печени, целесообразно периодически оценивать функцию печени. Большинство изменений функции печени встречаются в течение первых шести месяцев лечения препаратом.\u003Cbr\u003E\nБикалутамид следует применять с осторожностью у больных со средним и тяжелым нарушением функции печени.\u003Cbr\u003E\nТяжелые нарушения печени при использовании препарата возникают редко, сообщалось о случаях с фатальным исходом. В случае развития выраженных изменений функции печени и/или повышении функциональных проб более чем в 2 раза прием препарата необходимо прекратить.\u003Cbr\u003E\nПри совместном приеме с циклоспорином, после начала использования или отмены бикалутамида рекомендуется проводить тщательный контроль концентрации циклоспорина в плазме и состояния пациента.\u003Cbr\u003E\nУ пациентов с прогрессированием заболевания на фоне повышения концентрации простатспецифического антигена (АСА) необходимо рассмотреть вопрос о прекращении лечения бикалутамидом.\u003Cbr\u003E\nУчитывая возможность ингибирования препаратом активности цитохрома Р450 (изофермента CYP 3А4), следует проявлять осторожность при одновременном применении бикалутамида с препаратами, преимущественно метаболизирующимися с участием изофермента CYP 3А4. Рекомендуется регулярно контролировать протромбиновое время при назначении бикалутамида пациентам, получающим непрямые антикоагулянты кумаринового ряда.\u003Cbr\u003E\nУ пациентов, принимающих агонисты ГнРГ, наблюдалось снижение переносимости глюкозы. Этот эффект может приводить к развитию сахарного диабета или снижению толерантности к глюкозе у пациентов с сахарным диабетом. В связи с чем у пациентов, принимающих бикалутамид в комбинации с агонистами ГнРГ, необходимо контролировать концентрацию глюкозы в крови."},{"name":"Взаимодействие","value":"При применении бикалутамида в течение 28 дней на фоне приема мидазолама, АUC мидазолама увеличивалась на 80%.\u003Cbr\u003EПри одновременном применении бикалутамида с циклоспорином или блокаторами кальциевых каналов возможно потенцирование или развитие нежелательных реакций.\u003Cbr\u003EТеоретически возможно повышение концентрации бикалутамида в плазме крови при его одновременном применении с ингибиторами микросомальных ферментов печени, что может сопровождаться увеличением частоты возникновения нежелательных реакций.\u003Cbr\u003EИсследования in vitro показали, что бикалутамид может вытеснять антикоагулянт кумаринового ряда варфарин из участков связывания с белками плазмы."},{"name":"Регистрационный номер","value":"ЛП-001745"},{"name":"Дата государственной регистрации","value":"14.09.2021"},{"name":"Владелец регистрационного удостоверения","value":"Канонфарма продакшн"},{"name":"Изготовитель","value":"Канонфарма продакшн"},{"name":"Фасовщик","value":"Канонфарма продакшн"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Бикалутамид Канон"},{"name":"Срок годности","value":"37 мес."}]}],"transitionId":"tr_16160773360870634339"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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    на основе 24 оценки
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  • Рейтинг товара: 5 из 5
    на основе 2 оценки
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  • {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-j1kjlpshv0l/addToCartButton":{"offerId":"X2vBO80FeArtyNM2YBEqTw","skuId":"101333037763","pendingCartItem":{"productId":186939279,"offerId":"X2vBO80FeArtyNM2YBEqTw","showPlaceId":"OTNDnItfwRMjN9MRHuEMMsL7W7eICv7ZxrtvmnVpgs9FN2bRwbsEyLXDM4RtW_X2VaGSTTop0Nd2rPV0AbwEUjrHpOGdZb5aGunw7i7PBuIC4CY7qVfvDq318t3EGDdcUb0NwTQmb8ORp6FkypU3yfuF9hDTX_NHDg5um0sUqcoZiMxVPX3WrDzLZ2MGorQxZ5rgHeObcc3KzbMtI0osIA,,","feeShow":"OTNDnItfwRMjN9MRHuEMMsL7W7eICv7ZxrtvmnVpgs9FN2bRwbsEyLXDM4RtW_X2VaGSTTop0Nd2rPV0AbwEUjrHpOGdZb5aGunw7i7PBuIC4CY7qVfvDq318t3EGDdcUb0NwTQmb8ORp6FkypU3yfuF9hDTX_NHDg5um0sUqcoZiMxVPX3WrDzLZ2MGorQxZ5rgHeObcc3KzbMtI0osIA,,","skuId":"101333037763","shopId":77075781,"price":{"applicablePriceDiscounts":[],"value":"4105","currency":"RUR"},"hid":"15756914","name":"Золадекс капс. для п/к введ. пролонг. действ. шприц-аппликатор, 3.6 мг, 1 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  • Рейтинг товара: 4.8 из 5
    на основе 12 оценок
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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
    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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
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  • Рейтинг товара: 4.8 из 5
    на основе 9 оценок
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Инструкция

Показания к применению

- Монотерапия или адъювантная терапия, в комбинации с аналогом гонадотропин- рилизинг-гормона (ГнРГ) или хирургической кастрацией, распространенного рака предстательной железы;
- лечение местнораспространенного рака предстательной железы (Т3-Т4, любая N, М0, Т1-Т2, N+, М0) в качестве монотерапии или адъювантной терапии в сочетании с радикальной простатэктомией или радиотерапией;
- лечение местнораспространенного неметастатического рака предстательной железы в случаях, когда хирургическая кастрация или другие препараты не эффективны или неприемлемы.

Противопоказания

- Повышенная чувствительность к бикалутамиду или другим компонентам препарата;
- дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция;
- женщины;
- детский возраст;
- одновременный прием с терфенадином, астемизолом и цизапридом.

Способ применения и дозы

Взрослые мужчины, в том числе пожилые:
При распространённом раке предстательной железы в комбинации с аналогом ГнРГ или хирургической кастрацией: внутрь по 50 мг один раз в сутки.
При местнораспространенном раке предстательной железы: внутрь по 150 мг один раз в сутки.
Бикалутамид следует принимать продолжительно, как минимум в течение 2 лет.
При появлении признаков прогрессирования заболевания прием препарата следует прекратить.
Полная инструкция
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Бикалутамид Канон таб. п/о плен.
Бикалутамид Канон таб. п/о плен., 150 мг, 30 шт.
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Инструкция

1 828 ₽

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5.0
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У продавца:2 оценки·2 отзыва
У всех продавцов:19 оценок·4 отзыва
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user avatar
3 месяца назад • Александр Николаев • Куплен на Маркете
Достоинства: То, что нужно для лечения. Без рецепта!!!
Недостатки: нет
user avatar
4 месяца назад • Сергей М. • Куплен на Маркете
Достоинства: нормальный товар, недорого.
Недостатки: не выявлено
Посмотреть все отзывы на Маркете
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  • Бикалутамид таб. п/о плен., 50 мг, 30 шт.
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  • Таблетница органайзер на неделю, контейнер для таблеток, бокс, на 7 дней, 4 приема, 28 ячеек
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  • Таблетница из 14 секций на семь дней Утро-вечер
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  • Бикалутамид-тева таб. п/о плен., 50 мг, 28 шт.
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  • Лефлуномид Канон таб. п/о плен., 10 мг, 30 шт.
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  • Таблетница на 7 дней 3 приема черная
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    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:78049719_6/content/content/toggleWishlist":{"skuId":"102841232117","productId":78049719,"offerId":"KeGl1bzVQDEMw7c2ZkEbJg","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQkP3TjdDcqZUFEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIVCLfjmyUQ9dXCjv8CGJL29wcgzc49","sign":"ZD2h1PQX42pcASWT1tNWCGpHSTirFlrCDggKTTMO3gE="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:78049719_6/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Золадекс капс. для п/к введ. пролонг. действ. шприц-аппликатор, 3.6 мг, 1 шт.
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  • Реклама
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  • Таблетница органайзер на неделю утро / день / вечер; Органайзер для таблеток на 7 дней; Карманная аптечка
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  • Меркаптопурин таб., 50 мг, 25 шт.
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  • Аромазин таб. п/о, 25 мг, 30 шт.
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  • Таблетница компактная /органайзер аптечка/ контейнер для таблеток БАД Panda_Home (синего цвета)
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  • Лестродекс таб. п/о плен., 2.5 мг, 30 шт.
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  • Диферелин лиоф. д/приг. сусп. для в/м введ. пролонг. действ. фл., 11.25 мг, 1 шт.
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:186487587_14/content/content/gallery":{"title":"Диферелин лиоф. д/приг. сусп. для в/м введ. пролонг. действ. фл., 11.25 мг, 1 шт.","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/1478677/img_id489634863997861206.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/1478677/img_id489634863997861206.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/1478677/img_id489634863997861206.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/1478677/img_id489634863997861206.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/1478677/img_id489634863997861206.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/1478677/img_id489634863997861206.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"},{"src":"https://avatars.mds.yandex.net/get-mpic/5350118/img_id3598348887976603607.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/5350118/img_id3598348887976603607.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/5350118/img_id3598348887976603607.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/5350118/img_id3598348887976603607.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/5350118/img_id3598348887976603607.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/5350118/img_id3598348887976603607.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"}],"firstImageLazyLoading":false,"baobabClientData":{"realTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQkP3TjdDcqZUFEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIWCKOm9lgQkcTXwPkCGPvd0Acg8tzBBw==","sign":"uXgPYDJy8lwVf1JbSfK+tju2lF8oYYt/EFTeBbNy2cM="},"target":"model_card"},"isNoPicturePadding":true}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:186487587_14/content/content/gallery":{"name":"@marketfront/SnippetConstructor/Gallery"}}}
    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:186487587_14/content/content/toggleWishlist":{"skuId":"101335818769","productId":186487587,"offerId":"zaUIbzR_GiAgfL8RXwx2uQ","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQkP3TjdDcqZUFEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIWCKOm9lgQkcTXwPkCGPvd0Acg8tzBBw==","sign":"uXgPYDJy8lwVf1JbSfK+tju2lF8oYYt/EFTeBbNy2cM="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:186487587_14/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Таблетница - брелок на день, 1 раздел, контейнер для таблеток металлический маленький (черный матовый)
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1880169529_15/content/content/gallery":{"title":"Таблетница - брелок на день, 1 раздел, контейнер для таблеток металлический маленький (черный матовый)","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/4732637/img_id4653985497778709236.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/4732637/img_id4653985497778709236.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/4732637/img_id4653985497778709236.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/4732637/img_id4653985497778709236.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/4732637/img_id4653985497778709236.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/4732637/img_id4653985497778709236.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 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  • Курадерм крем, 10 мл
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  • Бикана таб. п/о плен., 50 мг, 28 шт.
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  • Лефлуномид таб. п/о плен., 20 мг, 30 шт.
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  • Таблетница на 7 дней Органайзер для лекарств
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  • Таблетница на 7 дней Органайзер для лекарств
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  • Реклама
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  • Таблетница на 7 дней / органайзер / бокс / контейнер на неделю для хранения таблеток и лекарств 4 приема Clear Daswerk
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  • Таблетница, контейнер для лекарств, органайзер для таблеток, маленькая
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