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Описание

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Эритромицин таб. п/о кш/раств., 250 мг, 10 шт.

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конъюнктивит новорожденных, пневмония у детей, мочеполовые инфекции у беременных, вызванные Chlamydia trachomatis;\u003Cbr /\u003E- Первичный сифилис (у пациентов с аллергией к пенициллинам), неосложненный хламидиоз у взрослых (с локализацией в нижних отделах мочеполовых путей и прямой кишки) при непереносимости или неэффективности тетрациклинов и др;\u003Cbr /\u003E- Инфекции ЛОР-органов (тонзиллит, отит, синусит);\u003Cbr /\u003E- Инфекции желчевыводящих путей (холецистит);\u003Cbr /\u003E- Инфекции верхних и нижних дыхательных путей (трахеит, бронхит, пневмония);\u003Cbr /\u003E- Инфекции кожи и мягких тканей (гнойничковые заболевания кожи, в т.ч. юношеские угри, инфицированные раны, пролежни, ожоги II-III ст, трофические язвы);\u003Cbr /\u003E- Инфекции слизистой оболочки глаз;\u003Cbr /\u003E- Профилактика обострений стрептококковой инфекции (тонзиллит, фарингит) у больных ревматизмом;\u003Cbr /\u003E- Профилактика инфекционных осложнений при лечебных и диагностических процедурах (в т.ч. предоперационная подготовка кишечника, стоматологические вмешательства, эндоскопия, у больных с пороками сердца)."},{"name":"Противопоказания","value":"- повышенная чувствительность к эритромицину, другим компонентам препарата;\u003Cbr /\u003E- потеря слуха;\u003Cbr /\u003E- одновременный прием терфенадина, эрготамина, дигидроэрготамина, астемизола, цизапридина, пимозида;\u003Cbr /\u003E- детский возраст до 3-х лет;\u003Cbr /\u003E- период грудного вскармливания;\u003Cbr /\u003E- непереносимость лактозы, дефицит лактазы, глюкогалактозная мальабсорбция."},{"name":"Состав","value":"На одну таблетку.\u003Cbr /\u003EДействующее вещество:\u003Cbr /\u003EЭритромицин в пересчете на 100% вещество\t- 100 мг\t- 250 мг\u003Cbr /\u003EВспомогательные вещества ядра:\u003Cbr /\u003Eжелатин\t- 3,1 мг - 7,0 мг\u003Cbr /\u003Eкальция стеарат - 1,95 мг - 4,4 мг\u003Cbr /\u003Eполисорбат 80 (твин 80) - 0,4 мг - 1,05 мг\u003Cbr /\u003Eлактозы моногидрат (сахар молочный)\t- 20,28 мг\t- 45,76 мг\u003Cbr /\u003Eкарбоксиметилкрахмал натрия (примогель), тип А\t- 7,8 мг\t- 17,6 мг\u003Cbr /\u003Eкрахмал картофельный\t- до 195 мг\t- до 440 мг\u003Cbr /\u003EВспомогательные вещества оболочки:\u003Cbr /\u003Eметакриловой кислоты и этилакрилата сополимер (1:1) (колликут МАЕ 100Р) - 8,5 мг - 18,41 мг\u003Cbr /\u003Eтальк - 2,7 мг\t- 5,84 мг\u003Cbr /\u003Eповидон К-30\t- 1,62 мг\t- 3,52 мг\u003Cbr /\u003Eтитана диоксид\t- 0,48 мг\t- 1,05 мг\u003Cbr /\u003Eполисорбат 80 (твин 80)\t- 1,7 мг\t- 3,68 мг"},{"name":"Действующее вещество","value":"Эритромицин","transition":{"type":"catalog","params":{"categorySlug":"antibiotiki-protivomikrobnye-i-protivoparazitarnye-sredstva","categoryId":"15756919","navnodeId":"72512","glfilters":["27144131:28710518"]}}},{"name":"Способ применения и дозы","value":"Внутрь.\u003Cbr /\u003EРазовая доза для взрослых и подростков старше 14 лет составляет 0,25-0,5 г, суточная - 1-2 г. Интервал между назначением - 6 ч. При тяжелых инфекциях суточная доза может быть увеличена до 4 г.\u003Cbr /\u003EДетям от 3-х до 14 лет, в зависимости от возраста, массы тела и тяжести инфекции - по 30-50 мг/кг/сут в 2-4 приема. В случае тяжелых инфекций, доза может быть удвоена.\u003Cbr /\u003EДля лечения дифтерийного носительства - по 0,25 г 2 раза в сутки. Курсовая доза для лечения первичного сифилиса - 30-40 г, продолжительность лечения - 10-15 дней.\u003Cbr /\u003EПри амебной дизентерии взрослым - по 0,25 г 4 раза в сутки, детям - по 30-50 мг/кг/сут; продолжительность курса - 10-14 дней.\u003Cbr /\u003EПри легионеллезе - по 0,5-1 г 4 раза в сутки в течение 14 дней.\u003Cbr /\u003EПри гонорее - по 0,5 г каждые 6 ч в течение 3 дней, далее по 0,25 г каждые 6 ч в течение 7 дней.\u003Cbr /\u003EДля предоперационной подготовки кишечника с целью профилактики инфекционных осложнений - внутрь, по 1 г за 19 ч, 18 ч и 9 ч до начала операции (всего 3 г).\u003Cbr /\u003EДля профилактики стрептококковой инфекции (при тонзиллите, фарингите) взрослым - 20-50 мг/кг/сут, детям - 20-30 мг/кг/сут, продолжительность курса - не менее 10 дней.\u003Cbr /\u003EДля профилактики септического эндокардита у больных с пороками сердца - по 1 г для взрослых и по 20 мг/кг - для детей, за 1 ч до лечебной или диагностической процедуры, далее по 0,5 г - для взрослых и 10 мг/кг для детей, повторно через 6 ч.\u003Cbr /\u003EПри коклюше - 40-50 мг/кг/сут в течение 5-14 дней.\u003Cbr /\u003EПри пневмонии у детей - 50 мг/кг/сут в 4 приема, в течение не менее 3 нед.\u003Cbr /\u003EПри мочеполовых инфекциях во время беременности - 0,5 г 4 раза в день в течение не менее 7 дней или (при плохой переносимости такой дозы) - по 0,25 г 4 раза в сутки в течение не менее 14 дней.\u003Cbr /\u003EУ взрослых, при неосложненном хламидиозе и непереносимости тетрациклинов - по 0,5 г 4 раза в сутки в течение не менее 7 дней."},{"name":"Побочные действия","value":"Реакции гиперчувствительности: кожные аллергические реакции (крапивница, др. формы сыпи), эозинофилия, редко - анафилактический шок.\u003Cbr /\u003EТошнота, рвота, гастралгия, тенезмы, абдоминальные боли, диарея, дисбактериоз, редко - кандидоз полости рта, псевдомембранозный энтероколит (как во время лечения, так и после него), нарушение функции печени, холестатическая желтуха, повышение активности \"печеночных\" трансаминаз, панкреатит, снижение слуха и/или шум в ушах (при применении высоких доз - более 4 г/сут, снижение слуха после отмены препарата обычно обратимо).\u003Cbr /\u003EРедко - тахикардия, удлинение интервала QT на ЭКГ, желудочковые аритмии, включая желудочковую тахикардию (типа \"пируэт\"), у больных с удлиненным интервалом QT."},{"name":"Фармакологическое действие","value":"Бактериостатический антибиотик из группы макролидов, обратимо связывается с 50S субъединицей рибосом в ее донорской части, что нарушает образование пептидных связей между молекулами аминокислот и блокирует синтез белков микроорганизмов (не влияет на синтез нуклеиновых кислот). При применении в высоких дозах может проявлять бактерицидное действие.\u003Cbr /\u003EСпектр действия включает грамположительные (Staphylococcus spp., продуцирующие и не продуцирующие пенициллиназу, в т.ч. Staphylococcus aureus; Streptococcus spp. (в т.ч. Streptococcus pneumoniae, Streptococcus pyogenes), альфа-гемолитический стрептококк (группы Viridans), Bacillus anthracis, Corynebacterium diphtheriae, Corynebacterium minutissimum) и грамотрицательные микроорганизмы (Neisseria gonorrhoeae, Haemophilus influenzae, Bordetella pertussis, Brucella spp., Legionella spp., в т.ч. Legionella pneumophila) и другие микроорганизмы: Mycoplasma spp. (в т.ч. Mycoplasma pneumoniae), Chlamydia spp. (в т.ч. Chlamydia trachomatis), Treponema spp., Rickettsia spp., Entamoeba histolytica, Listeria monocytogenes.\u003Cbr /\u003EУстойчивы грамотрицательные палочки: Escherichia coli, Pseudomonas aeruginosa, а также Shigella spp., Salmonella spp. и др.\u003Cbr /\u003EК группе чувствительных относятся микроорганизмы, рост которых задерживается при концентрации антибиотика менее 0,5 мг/л, среднечувствительных - 1-6 мг/л, умеренно устойчивых и устойчивых - 6-8 мг/л."},{"name":"Фармакологическая группа","value":"антибиотик-макролид"},{"name":"Форма выпуска","value":"таблетки, покрытые кишечнорастворимой оболочкой"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"antibiotiki-protivomikrobnye-i-protivoparazitarnye-sredstva","categoryId":"15756919","navnodeId":"72512","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 3 лет"},{"name":"Условия хранения","value":"При температуре не выше 25 °С.\u003Cbr /\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: нарушение функции печени, вплоть до острой печеночной недостаточности, потеря слуха.\u003Cbr /\u003EЛечение: активированный уголь, тщательный контроль за состоянием дыхательной системы. Промывание желудка эффективно при приеме дозы, пятикратно превышающей среднюю терапевтическую. Гемодиализ, перитонеальный диализ, форсированный диурез неэффективны."},{"name":"Применение при беременности и кормлении грудью","value":"Применение препарата при беременности возможно только в том случае, когда ожидаемая польза для матери превышает потенциальный риск для плода.\u003Cbr /\u003EНа период лечения эритромицином грудное вскармливание необходимо приостановить."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо соблюдать осторожность при управлении автотранспортом и занятии потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"С осторожностью:\u003Cbr /\u003EПрием эритромицина может вызывать удлинение интервала Q-T, аритмия (в том\u003Cbr /\u003Eчисле в анамнезе), желтуха (в том числе в анамнезе), печеночная и/или почечная недостаточность, одновременный прием гепатотоксичных препаратов, миастения-gravis.\u003Cbr /\u003EСледует соблюдать осторожность “при совместном \"назначении эритромицина и колхицина.\u003Cbr\u003EПри длительной терапии необходимо осуществлять контроль лабораторных показателей функции печени.\u003Cbr /\u003EСимптомы холестатической желтухи могут развиться через несколько дней после начала терапии, однако риск развития повышается после 7-14 дней непрерывной терапии. Вероятность развития ототоксического эффекта выше у больных с почечной и печеночной недостаточностью, а также у пожилых пациентов.\u003Cbr /\u003EМожет помешать определению катехоламинов в моче и активности \"печеночных\" трансаминаз в крови (колориметрическое определение с помощью дефинилгидразина). При одновременном приёме колхицина и эритромицина необходима коррекция Дозы колхицина и тщательный контроль состояния пациента с целью выявления признаков токсичности.\u003Cbr /\u003EПри совместном применении со статинами, возможно развитие рабдомиолиза и псевдомембранозного колита.\u003Cbr /\u003EИмеются сведения о развитии интерстициального нефрита на фоне лечения эритромицином.\u003Cbr /\u003EПри проявлении симптоматики данного заболевания, необходимо принять соответствующие меры."},{"name":"Взаимодействие","value":"Препараты, блокирующие канальцевую секрецию, удлиняет период полувыведения эритромицина.\u003Cbr /\u003EСнижает бактерицидное действие (антагонизм) беталактамных антибиотиков (пенициллины, цефалоспорины, карбопенемы), линкомицина, клиндамицина, хлорамфеникола, стрептомицина, тетрациклинов, колистина.\u003Cbr /\u003EПри одновременном приеме с препаратами, метаболизм которых осуществляется в печени (теофиллина, карбамазепина, вальпроевой кислоты, гексобарбитала, фенитоина, альфентанила, дизопирамида, ловастатина, бромокриптина), может повышаться концентрация этих препаратов в плазме (является ингибитором микросомальных ферментов печени).\u003Cbr /\u003EПри взаимодействии с теофиллином может потребоваться снижение дозы теофиллина, одновременно может снижаться концентрация эритромицина, что может привести к субтерапевтическим концентрациям эритромицина и уменьшению его эффекта. Усиливает нефротоксичность циклоспорина (особенно у больных с сопутствующей почечной недостаточностью).\u003Cbr /\u003EСнижает клиренс триазолама и мидазолама, в связи с чем может усиливать фармакологические эффекты бензодиазепинов.\u003Cbr /\u003EПри одновременном приеме с терфенадином или астемизолом - возможность развития аритмий, с дигидроэрготамином или негидрированнымй алкалоидами спорыньи - сужение сосудов до спазма, дизестезии.\u003Cbr /\u003EЗамедляет элиминацию (усиливает, эффект) метилпреднизолона, фелодипина и антикоагулянтов кумаринового ряда.\u003Cbr /\u003EПри совместном назначении с ловастатином и другими ингибиторами ГМГ-КоА-редуктазы повышается риск развития рабдомиолиза.\u003Cbr /\u003EПовышает биодоступность дигоксина. Снижает эффективность гормональной контрацепции.\u003Cbr /\u003EПри одновременном приеме с лекарственными препаратами, метаболизм которых осуществляется в печени (аценокумарол, астемизол, цилостазол, циклоспорин, дигидроэрготамин, эрготамин, омепразол, хинидин, рифабутин, такрослимус, терфенадин, винбластин и противогрибковые препараты такие как, флуконазол, кетоконазол и интраконазол) в плазме повышается концентрация этих лекарственных препаратов.\u003Cbr /\u003EОдновременное применение эритромицина с эрготамином ассоциировано с риском развития острой токсичности, проявляющейся спазмом сосудов, ишемией конечностей и других органов, включая центральную нервную систему. В связи с этим эритромицин противопоказан пациентам, принимающим эрготамин.\u003Cbr /\u003EПри одновременном приеме с эритромицином возможно повышение уровня цизаприда которое может привести к удлинению интервала QTc, возможно развитие аритмии (мерцание и трепетание желудочков), желудочковой тахикардии типа \"пируэт\".\u003Cbr /\u003EПри совместном приеме с верапамилом и другими блокаторами медленных кальциевых каналов наблюдается гипотония, брадиаритмия и лактоацидоз.\u003Cbr /\u003EЛекарственные препараты, являющиеся индуктарами изоферментов CYP3A4 (такие как, рифампицин, фенитоин, карбамазепин, фенобарбитал, зверобой продырявленный) могут индуцировать метаболизм эритромицина, что может привести к субтерапевтическим концентрациям эритромицина и уменьшению его эффекта. Взаимодействие сохраняется в течение 2 недель после прекращения лечения индуктарами CYP3A4.\u003Cbr /\u003EВзаимодействие эритромицина с колхицином может увеличивать токсичность и приводит к значительному повышению концентрации последнего в плазме крови ввиду способности эритромицина ингибировать CYP3A4.\u003Cbr /\u003EЭритромицин изменяет метаболизм мизоластина.\u003Cbr /\u003EПри совместном приеме с пимозидом возможно развитие аритмии (мерцание и трепетание желудочков), желудочковой тахикардии типа \"пируэт\", остановки сердца, вплоть до смертельного исхода.\u003Cbr /\u003EИнгибиторы протеазы: ингибируют метаболизм эритромицина, необходимо наблюдение за концентрацией эритромицина в плазме.\u003Cbr /\u003EЦиметидин ингибирует метаболизм эритромицина, что может привести к увеличенной плазменной концентрации эритромицина.\u003Cbr /\u003EЭритромицин снижает клиренс зопиклона и таким образом может увеличить фармакодинамические эффекты этого препарата."},{"name":"Регистрационный номер","value":"ЛСР-009305/08"},{"name":"Дата государственной регистрации","value":"19.11.2018"},{"name":"Владелец регистрационного удостоверения","value":"Биосинтез","transition":{"type":"catalog","params":{"categorySlug":"antibiotiki-protivomikrobnye-i-protivoparazitarnye-sredstva","categoryId":"15756919","navnodeId":"72512","glfilters":["34324371:35649313","7893318:16002664"]}}},{"name":"Изготовитель","value":"Биосинтез"},{"name":"Фасовщик","value":"Биосинтез"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Эритромицин","transition":{"type":"catalog","params":{"categorySlug":"antibiotiki-protivomikrobnye-i-protivoparazitarnye-sredstva","categoryId":"15756919","navnodeId":"72512","glfilters":["17796364:17880285"]}}},{"name":"Срок годности","value":"1 г."}]}},"fullSpecsGrouped":{"1424409196122535144":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Назначение","value":"бактериальные инфекции, бактериальные инфекции верхних отделов дыхательных путей и ЛОР-органов, бактериальные инфекции желчных путей, бактериальные инфекции кожи и мягких тканей, бактериальные инфекции нижних отделов дыхательных путей, бактериальные одонтогенные инфекции"},{"name":"Органы и системы","value":"выделительная система, дыхательная система, желчный пузырь и желчевыводящие пути, легкие, почки"},{"name":"Показания к применению","value":"- Бактериальные инфекции, вызванные чувствительной микрофлорой: дифтерия (в т.ч. бактерионосительство), коклюш (в т.ч. профилактика), трахома, бруцеллез, болезнь легионеров, эритразма, листериоз, скарлатина, амебная дизентерия, гонорея; конъюнктивит новорожденных, пневмония у детей, мочеполовые инфекции у беременных, вызванные Chlamydia trachomatis;\u003Cbr /\u003E- Первичный сифилис (у пациентов с аллергией к пенициллинам), неосложненный хламидиоз у взрослых (с локализацией в нижних отделах мочеполовых путей и прямой кишки) при непереносимости или неэффективности тетрациклинов и др;\u003Cbr /\u003E- Инфекции ЛОР-органов (тонзиллит, отит, синусит);\u003Cbr /\u003E- Инфекции желчевыводящих путей (холецистит);\u003Cbr /\u003E- Инфекции верхних и нижних дыхательных путей (трахеит, бронхит, пневмония);\u003Cbr /\u003E- Инфекции кожи и мягких тканей (гнойничковые заболевания кожи, в т.ч. юношеские угри, инфицированные раны, пролежни, ожоги II-III ст, трофические язвы);\u003Cbr /\u003E- Инфекции слизистой оболочки глаз;\u003Cbr /\u003E- Профилактика обострений стрептококковой инфекции (тонзиллит, фарингит) у больных ревматизмом;\u003Cbr /\u003E- Профилактика инфекционных осложнений при лечебных и диагностических процедурах (в т.ч. предоперационная подготовка кишечника, стоматологические вмешательства, эндоскопия, у больных с пороками сердца)."},{"name":"Противопоказания","value":"- повышенная чувствительность к эритромицину, другим компонентам препарата;\u003Cbr /\u003E- потеря слуха;\u003Cbr /\u003E- одновременный прием терфенадина, эрготамина, дигидроэрготамина, астемизола, цизапридина, пимозида;\u003Cbr /\u003E- детский возраст до 3-х лет;\u003Cbr /\u003E- период грудного вскармливания;\u003Cbr /\u003E- непереносимость лактозы, дефицит лактазы, глюкогалактозная мальабсорбция."},{"name":"Состав","value":"На одну таблетку.\u003Cbr /\u003EДействующее вещество:\u003Cbr /\u003EЭритромицин в пересчете на 100% вещество\t- 100 мг\t- 250 мг\u003Cbr /\u003EВспомогательные вещества ядра:\u003Cbr /\u003Eжелатин\t- 3,1 мг - 7,0 мг\u003Cbr /\u003Eкальция стеарат - 1,95 мг - 4,4 мг\u003Cbr /\u003Eполисорбат 80 (твин 80) - 0,4 мг - 1,05 мг\u003Cbr /\u003Eлактозы моногидрат (сахар молочный)\t- 20,28 мг\t- 45,76 мг\u003Cbr /\u003Eкарбоксиметилкрахмал натрия (примогель), тип А\t- 7,8 мг\t- 17,6 мг\u003Cbr /\u003Eкрахмал картофельный\t- до 195 мг\t- до 440 мг\u003Cbr /\u003EВспомогательные вещества оболочки:\u003Cbr /\u003Eметакриловой кислоты и этилакрилата сополимер (1:1) (колликут МАЕ 100Р) - 8,5 мг - 18,41 мг\u003Cbr /\u003Eтальк - 2,7 мг\t- 5,84 мг\u003Cbr /\u003Eповидон К-30\t- 1,62 мг\t- 3,52 мг\u003Cbr /\u003Eтитана диоксид\t- 0,48 мг\t- 1,05 мг\u003Cbr /\u003Eполисорбат 80 (твин 80)\t- 1,7 мг\t- 3,68 мг"},{"name":"Действующее вещество","value":"Эритромицин"},{"name":"Способ применения и дозы","value":"Внутрь.\u003Cbr /\u003EРазовая доза для взрослых и подростков старше 14 лет составляет 0,25-0,5 г, суточная - 1-2 г. Интервал между назначением - 6 ч. При тяжелых инфекциях суточная доза может быть увеличена до 4 г.\u003Cbr /\u003EДетям от 3-х до 14 лет, в зависимости от возраста, массы тела и тяжести инфекции - по 30-50 мг/кг/сут в 2-4 приема. В случае тяжелых инфекций, доза может быть удвоена.\u003Cbr /\u003EДля лечения дифтерийного носительства - по 0,25 г 2 раза в сутки. Курсовая доза для лечения первичного сифилиса - 30-40 г, продолжительность лечения - 10-15 дней.\u003Cbr /\u003EПри амебной дизентерии взрослым - по 0,25 г 4 раза в сутки, детям - по 30-50 мг/кг/сут; продолжительность курса - 10-14 дней.\u003Cbr /\u003EПри легионеллезе - по 0,5-1 г 4 раза в сутки в течение 14 дней.\u003Cbr /\u003EПри гонорее - по 0,5 г каждые 6 ч в течение 3 дней, далее по 0,25 г каждые 6 ч в течение 7 дней.\u003Cbr /\u003EДля предоперационной подготовки кишечника с целью профилактики инфекционных осложнений - внутрь, по 1 г за 19 ч, 18 ч и 9 ч до начала операции (всего 3 г).\u003Cbr /\u003EДля профилактики стрептококковой инфекции (при тонзиллите, фарингите) взрослым - 20-50 мг/кг/сут, детям - 20-30 мг/кг/сут, продолжительность курса - не менее 10 дней.\u003Cbr /\u003EДля профилактики септического эндокардита у больных с пороками сердца - по 1 г для взрослых и по 20 мг/кг - для детей, за 1 ч до лечебной или диагностической процедуры, далее по 0,5 г - для взрослых и 10 мг/кг для детей, повторно через 6 ч.\u003Cbr /\u003EПри коклюше - 40-50 мг/кг/сут в течение 5-14 дней.\u003Cbr /\u003EПри пневмонии у детей - 50 мг/кг/сут в 4 приема, в течение не менее 3 нед.\u003Cbr /\u003EПри мочеполовых инфекциях во время беременности - 0,5 г 4 раза в день в течение не менее 7 дней или (при плохой переносимости такой дозы) - по 0,25 г 4 раза в сутки в течение не менее 14 дней.\u003Cbr /\u003EУ взрослых, при неосложненном хламидиозе и непереносимости тетрациклинов - по 0,5 г 4 раза в сутки в течение не менее 7 дней."},{"name":"Побочные действия","value":"Реакции гиперчувствительности: кожные аллергические реакции (крапивница, др. формы сыпи), эозинофилия, редко - анафилактический шок.\u003Cbr /\u003EТошнота, рвота, гастралгия, тенезмы, абдоминальные боли, диарея, дисбактериоз, редко - кандидоз полости рта, псевдомембранозный энтероколит (как во время лечения, так и после него), нарушение функции печени, холестатическая желтуха, повышение активности \"печеночных\" трансаминаз, панкреатит, снижение слуха и/или шум в ушах (при применении высоких доз - более 4 г/сут, снижение слуха после отмены препарата обычно обратимо).\u003Cbr /\u003EРедко - тахикардия, удлинение интервала QT на ЭКГ, желудочковые аритмии, включая желудочковую тахикардию (типа \"пируэт\"), у больных с удлиненным интервалом QT."},{"name":"Фармакологическое действие","value":"Бактериостатический антибиотик из группы макролидов, обратимо связывается с 50S субъединицей рибосом в ее донорской части, что нарушает образование пептидных связей между молекулами аминокислот и блокирует синтез белков микроорганизмов (не влияет на синтез нуклеиновых кислот). При применении в высоких дозах может проявлять бактерицидное действие.\u003Cbr /\u003EСпектр действия включает грамположительные (Staphylococcus spp., продуцирующие и не продуцирующие пенициллиназу, в т.ч. Staphylococcus aureus; Streptococcus spp. (в т.ч. Streptococcus pneumoniae, Streptococcus pyogenes), альфа-гемолитический стрептококк (группы Viridans), Bacillus anthracis, Corynebacterium diphtheriae, Corynebacterium minutissimum) и грамотрицательные микроорганизмы (Neisseria gonorrhoeae, Haemophilus influenzae, Bordetella pertussis, Brucella spp., Legionella spp., в т.ч. Legionella pneumophila) и другие микроорганизмы: Mycoplasma spp. (в т.ч. Mycoplasma pneumoniae), Chlamydia spp. (в т.ч. Chlamydia trachomatis), Treponema spp., Rickettsia spp., Entamoeba histolytica, Listeria monocytogenes.\u003Cbr /\u003EУстойчивы грамотрицательные палочки: Escherichia coli, Pseudomonas aeruginosa, а также Shigella spp., Salmonella spp. и др.\u003Cbr /\u003EК группе чувствительных относятся микроорганизмы, рост которых задерживается при концентрации антибиотика менее 0,5 мг/л, среднечувствительных - 1-6 мг/л, умеренно устойчивых и устойчивых - 6-8 мг/л."},{"name":"Фармакологическая группа","value":"антибиотик-макролид"},{"name":"Форма выпуска","value":"таблетки, покрытые кишечнорастворимой оболочкой"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 3 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"При температуре не выше 25 °С.\u003Cbr /\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: нарушение функции печени, вплоть до острой печеночной недостаточности, потеря слуха.\u003Cbr /\u003EЛечение: активированный уголь, тщательный контроль за состоянием дыхательной системы. Промывание желудка эффективно при приеме дозы, пятикратно превышающей среднюю терапевтическую. Гемодиализ, перитонеальный диализ, форсированный диурез неэффективны."},{"name":"Применение при беременности и кормлении грудью","value":"Применение препарата при беременности возможно только в том случае, когда ожидаемая польза для матери превышает потенциальный риск для плода.\u003Cbr /\u003EНа период лечения эритромицином грудное вскармливание необходимо приостановить."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо соблюдать осторожность при управлении автотранспортом и занятии потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"С осторожностью:\u003Cbr /\u003EПрием эритромицина может вызывать удлинение интервала Q-T, аритмия (в том\u003Cbr /\u003Eчисле в анамнезе), желтуха (в том числе в анамнезе), печеночная и/или почечная недостаточность, одновременный прием гепатотоксичных препаратов, миастения-gravis.\u003Cbr /\u003EСледует соблюдать осторожность “при совместном \"назначении эритромицина и колхицина.\u003Cbr\u003EПри длительной терапии необходимо осуществлять контроль лабораторных показателей функции печени.\u003Cbr /\u003EСимптомы холестатической желтухи могут развиться через несколько дней после начала терапии, однако риск развития повышается после 7-14 дней непрерывной терапии. Вероятность развития ототоксического эффекта выше у больных с почечной и печеночной недостаточностью, а также у пожилых пациентов.\u003Cbr /\u003EМожет помешать определению катехоламинов в моче и активности \"печеночных\" трансаминаз в крови (колориметрическое определение с помощью дефинилгидразина). При одновременном приёме колхицина и эритромицина необходима коррекция Дозы колхицина и тщательный контроль состояния пациента с целью выявления признаков токсичности.\u003Cbr /\u003EПри совместном применении со статинами, возможно развитие рабдомиолиза и псевдомембранозного колита.\u003Cbr /\u003EИмеются сведения о развитии интерстициального нефрита на фоне лечения эритромицином.\u003Cbr /\u003EПри проявлении симптоматики данного заболевания, необходимо принять соответствующие меры."},{"name":"Взаимодействие","value":"Препараты, блокирующие канальцевую секрецию, удлиняет период полувыведения эритромицина.\u003Cbr /\u003EСнижает бактерицидное действие (антагонизм) беталактамных антибиотиков (пенициллины, цефалоспорины, карбопенемы), линкомицина, клиндамицина, хлорамфеникола, стрептомицина, тетрациклинов, колистина.\u003Cbr /\u003EПри одновременном приеме с препаратами, метаболизм которых осуществляется в печени (теофиллина, карбамазепина, вальпроевой кислоты, гексобарбитала, фенитоина, альфентанила, дизопирамида, ловастатина, бромокриптина), может повышаться концентрация этих препаратов в плазме (является ингибитором микросомальных ферментов печени).\u003Cbr /\u003EПри взаимодействии с теофиллином может потребоваться снижение дозы теофиллина, одновременно может снижаться концентрация эритромицина, что может привести к субтерапевтическим концентрациям эритромицина и уменьшению его эффекта. Усиливает нефротоксичность циклоспорина (особенно у больных с сопутствующей почечной недостаточностью).\u003Cbr /\u003EСнижает клиренс триазолама и мидазолама, в связи с чем может усиливать фармакологические эффекты бензодиазепинов.\u003Cbr /\u003EПри одновременном приеме с терфенадином или астемизолом - возможность развития аритмий, с дигидроэрготамином или негидрированнымй алкалоидами спорыньи - сужение сосудов до спазма, дизестезии.\u003Cbr /\u003EЗамедляет элиминацию (усиливает, эффект) метилпреднизолона, фелодипина и антикоагулянтов кумаринового ряда.\u003Cbr /\u003EПри совместном назначении с ловастатином и другими ингибиторами ГМГ-КоА-редуктазы повышается риск развития рабдомиолиза.\u003Cbr /\u003EПовышает биодоступность дигоксина. Снижает эффективность гормональной контрацепции.\u003Cbr /\u003EПри одновременном приеме с лекарственными препаратами, метаболизм которых осуществляется в печени (аценокумарол, астемизол, цилостазол, циклоспорин, дигидроэрготамин, эрготамин, омепразол, хинидин, рифабутин, такрослимус, терфенадин, винбластин и противогрибковые препараты такие как, флуконазол, кетоконазол и интраконазол) в плазме повышается концентрация этих лекарственных препаратов.\u003Cbr /\u003EОдновременное применение эритромицина с эрготамином ассоциировано с риском развития острой токсичности, проявляющейся спазмом сосудов, ишемией конечностей и других органов, включая центральную нервную систему. В связи с этим эритромицин противопоказан пациентам, принимающим эрготамин.\u003Cbr /\u003EПри одновременном приеме с эритромицином возможно повышение уровня цизаприда которое может привести к удлинению интервала QTc, возможно развитие аритмии (мерцание и трепетание желудочков), желудочковой тахикардии типа \"пируэт\".\u003Cbr /\u003EПри совместном приеме с верапамилом и другими блокаторами медленных кальциевых каналов наблюдается гипотония, брадиаритмия и лактоацидоз.\u003Cbr /\u003EЛекарственные препараты, являющиеся индуктарами изоферментов CYP3A4 (такие как, рифампицин, фенитоин, карбамазепин, фенобарбитал, зверобой продырявленный) могут индуцировать метаболизм эритромицина, что может привести к субтерапевтическим концентрациям эритромицина и уменьшению его эффекта. Взаимодействие сохраняется в течение 2 недель после прекращения лечения индуктарами CYP3A4.\u003Cbr /\u003EВзаимодействие эритромицина с колхицином может увеличивать токсичность и приводит к значительному повышению концентрации последнего в плазме крови ввиду способности эритромицина ингибировать CYP3A4.\u003Cbr /\u003EЭритромицин изменяет метаболизм мизоластина.\u003Cbr /\u003EПри совместном приеме с пимозидом возможно развитие аритмии (мерцание и трепетание желудочков), желудочковой тахикардии типа \"пируэт\", остановки сердца, вплоть до смертельного исхода.\u003Cbr /\u003EИнгибиторы протеазы: ингибируют метаболизм эритромицина, необходимо наблюдение за концентрацией эритромицина в плазме.\u003Cbr /\u003EЦиметидин ингибирует метаболизм эритромицина, что может привести к увеличенной плазменной концентрации эритромицина.\u003Cbr /\u003EЭритромицин снижает клиренс зопиклона и таким образом может увеличить фармакодинамические эффекты этого препарата."},{"name":"Регистрационный номер","value":"ЛСР-009305/08"},{"name":"Дата государственной регистрации","value":"19.11.2018"},{"name":"Владелец регистрационного удостоверения","value":"Биосинтез"},{"name":"Изготовитель","value":"Биосинтез"},{"name":"Фасовщик","value":"Биосинтез"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Эритромицин"},{"name":"Срок годности","value":"1 г."}]}],"transitionId":"tr_3427282536900830127"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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Инструкция

Показания к применению

- Бактериальные инфекции, вызванные чувствительной микрофлорой: дифтерия (в т.ч. бактерионосительство), коклюш (в т.ч. профилактика), трахома, бруцеллез, болезнь легионеров, эритразма, листериоз, скарлатина, амебная дизентерия, гонорея; конъюнктивит новорожденных, пневмония у детей, мочеполовые инфекции у беременных, вызванные Chlamydia trachomatis;
- Первичный сифилис (у пациентов с аллергией к пенициллинам), неосложненный хламидиоз у взрослых (с локализацией в нижних отделах мочеполовых путей и прямой кишки) при непереносимости или неэффективности тетрациклинов и др;
- Инфекции ЛОР-органов (тонзиллит, отит, синусит);
- Инфекции желчевыводящих путей (холецистит);
- Инфекции верхних и нижних дыхательных путей (трахеит, бронхит, пневмония);
- Инфекции кожи и мягких тканей (гнойничковые заболевания кожи, в т.ч. юношеские угри, инфицированные раны, пролежни, ожоги II-III ст, трофические язвы);
- Инфекции слизистой оболочки глаз;
- Профилактика обострений стрептококковой инфекции (тонзиллит, фарингит) у больных ревматизмом;
- Профилактика инфекционных осложнений при лечебных и диагностических процедурах (в т.ч. предоперационная подготовка кишечника, стоматологические вмешательства, эндоскопия, у больных с пороками сердца).

Противопоказания

- повышенная чувствительность к эритромицину, другим компонентам препарата;
- потеря слуха;
- одновременный прием терфенадина, эрготамина, дигидроэрготамина, астемизола, цизапридина, пимозида;
- детский возраст до 3-х лет;
- период грудного вскармливания;
- непереносимость лактозы, дефицит лактазы, глюкогалактозная мальабсорбция.

Способ применения и дозы

Внутрь.
Разовая доза для взрослых и подростков старше 14 лет составляет 0,25-0,5 г, суточная - 1-2 г. Интервал между назначением - 6 ч. При тяжелых инфекциях суточная доза может быть увеличена до 4 г.
Детям от 3-х до 14 лет, в зависимости от возраста, массы тела и тяжести инфекции - по 30-50 мг/кг/сут в 2-4 приема. В случае тяжелых инфекций, доза может быть удвоена.
Для лечения дифтерийного носительства - по 0,25 г 2 раза в сутки. Курсовая доза для лечения первичного сифилиса - 30-40 г, продолжительность лечения - 10-15 дней.
При амебной дизентерии взрослым - по 0,25 г 4 раза в сутки, детям - по 30-50 мг/кг/сут; продолжительность курса - 10-14 дней.
При легионеллезе - по 0,5-1 г 4 раза в сутки в течение 14 дней.
При гонорее - по 0,5 г каждые 6 ч в течение 3 дней, далее по 0,25 г каждые 6 ч в течение 7 дней.
Для предоперационной подготовки кишечника с целью профилактики инфекционных осложнений - внутрь, по 1 г за 19 ч, 18 ч и 9 ч до начала операции (всего 3 г).
Для профилактики стрептококковой инфекции (при тонзиллите, фарингите) взрослым - 20-50 мг/кг/сут, детям - 20-30 мг/кг/сут, продолжительность курса - не менее 10 дней.
Для профилактики септического эндокардита у больных с пороками сердца - по 1 г для взрослых и по 20 мг/кг - для детей, за 1 ч до лечебной или диагностической процедуры, далее по 0,5 г - для взрослых и 10 мг/кг для детей, повторно через 6 ч.
При коклюше - 40-50 мг/кг/сут в течение 5-14 дней.
При пневмонии у детей - 50 мг/кг/сут в 4 приема, в течение не менее 3 нед.
При мочеполовых инфекциях во время беременности - 0,5 г 4 раза в день в течение не менее 7 дней или (при плохой переносимости такой дозы) - по 0,25 г 4 раза в сутки в течение не менее 14 дней.
У взрослых, при неосложненном хламидиозе и непереносимости тетрациклинов - по 0,5 г 4 раза в сутки в течение не менее 7 дней.
Полная инструкция
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Эритромицин таб. п/о кш/раств.
Эритромицин таб. п/о кш/раств., 250 мг, 10 шт.
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Инструкция

154 ₽

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5.0
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  • Тройчатка Эвалар капс., 40 шт.
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  • Black Walnut Hulls капс., 100 г, 100 шт.
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  • Таблетница - брелок на день, 1 раздел, контейнер для таблеток металлический маленький (черный матовый)
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  • Таблетница органайзер на неделю утро / день / вечер; Органайзер для таблеток на 7 дней; Карманная аптечка
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  • Контейнер для хранения/таблетница/кейс для таблеток
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  • Таблетница компактная /органайзер аптечка/ контейнер для таблеток БАД Panda_Home (синего цвета)
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    Реклама
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  • Таблетница на 7 дней / органайзер / бокс / контейнер на неделю для хранения таблеток и лекарств 4 приема Clear Daswerk
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  • Таблетница с делителем (резаком) и размельчителем таблеток. Органайзер - таблеторезка с фиксатором, 3 в 1. 12x6,5x2 см, серый.
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  • Таблетница Органайзер на 7 дней с делениями x1
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  • {"widgets":{"@yandex-market/LazyLoader-market":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator":{"widgetName":"@marketfront/RecomLayout","widgetId":"ServerListRendererForSerp_RecommendationRoll","options":{"resolverParams":{"resources":{"garsons":[{"count":24,"limit":24,"params":{"cartProductIds":[],"snippetTypes":["product","product-block","category-block","advertisement","media-incut","promo-trigger","media-adv-banner-single","media-adv-banner-double","media-adv-carousel"],"program":"remix_desktop_model_card","hyperid":1434054579},"id":"RemixData"}],"shuffle":{"mode":"exclusive"}},"limit":24},"id":"RecommendationRoll","slotOptions":{"dynamic":true},"className":"","needToProvideData":true,"wrapperProps":{},"widgetOptions":{"config":{"pictureBlock":{"maxGalleryImagesCount":5},"descriptionBlock":{"order":1,"titleRowCount":"2"},"offerBlock":{"withGreenPrice":true,"order":2,"price":{"wrap":true,"overflow":"hidden"}}},"galleryImageSize":250},"layoutOptions":{"needFallbackOnError":true,"needFallbackOnEmpty":false,"countInRows":6},"isChefRemixExp":false},"slotOptions":{"dynamic":true},"placeholder":"Invisible","infinite":true,"cspNonce":"lm+5YUckEloUsizGsNrd6Q==","renderStrategy":"append","renderedOnce":true}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator":{"name":"@yandex-market/LazyLoader-market"}}}
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