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Эзлор таб. п/о плен.
Эзлор таб. п/о плен., 5мг, 10 шт.
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Инструкция

Цена с картой Яндекс Пэй:288

Скидка: 1%
–1 %
Вместо: 291
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Описание

лекарственный препарат, назначение: аллергический ринит, крапивница

Инструкция

Общие характеристики

Тип препарата
Органы и системы
Назначение
Показания к применению
Аллергический ринит (устранение или облегчение чиханья, заложенности носа, выделения слизи из носа, зуда в носу, зуда неба, зуда и покраснения глаз, слезотечения); крапивница (уменьшение или устранение кожного зуда, сыпи).
Противопоказания
Повышенная чувствительность к какому-либо из компонентов, входящих в состав препарата; беременность и лактация; возраст до 12 лет; непереносимость лактозы, недостаточность лактазы или синдром глюкозо-галактозной мальабсорбции.
Состав
Одна таблетка содержит:
активное вещество: дезлоратадин 5,0 мг;
вспомогательные вещества (ядро): лактозы моногидрат (сахар молочный) 70,0 мг; целлюлоза микрокристаллическая 12,1 мг; повидон (поливинилпирролидон) 3,0 мг; магния стеарат 0,9 мг; кроскармеллоза натрия 4,0 мг;
вспомогательные вещества (оболочка): опадрай II 85F48105 Белый 3,0 мг, в т.ч. (поливиниловый спирт 1,407 мг; макрогол 3350 0,708 мг; тальк 0,522 мг; титана диоксид 0,363 мг).
Действующее вещество
Способ применения и дозы
Таблетку следует проглатывать целиком, не разжевывая, запивая небольшим количеством воды. Препарат принимать желательно в одно и то же время суток, независимо от времени приема пищи.
Взрослым и подросткам в возрасте от 12 лет - по 1 таблетке (5 мг) 1 раз в сутки.
Побочные действия
Частота развития побочных эффектов классифицирована согласно рекомендациям Всемирной организации здравоохранения: очень часто - не менее 10%; часто - не менее - 1%, но менее 10%; нечасто - не менее 0,1%, но менее 1%; редко - не менее 0,01%, но менее 0,1%; очень редко - менее 0,01%.
Со стороны иммунной системы: очень редко - сыпь, в том числе крапивница, ангионевротический отек, крапивница, диспноэ, анафилактический шок.
Со стороны центральной нервной системы: нечасто - головная боль; очень редко - головокружение, сонливость, бессонница, психомоторная гиперактивность, судороги, галлюцинации.
Со стороны сердечно-сосудистой системы: очень редко -тахикардия, ощущение сердцебиения.
Со стороны желудочно-кишечного тракта: нечасто - сухость во рту; очень редко - тошнота, рвота, диспепсия, диарея, боль в животе, повышение активности "печеночных" ферментов, повышение концентрации билирубина, гепатит.
Со стороны костно-мышечной системы и соединительной ткани: очень редко - миалгия.
Прочие: часто - повышенная утомляемость.
Фармакологическое действие
Блокатор H1-гистаминовых рецепторов (длительного действия). Является первичным активным метаболитом лоратадина. Ингибирует каскад реакций аллергического воспаления, в том числе высвобождение противовоспалительных цитокинов, включая интерлейкины ИЛ-4, ИЛ-6, ИЛ-8, ИЛ-13, высвобождение провоспалительных хемокинов (RANTES), продукцию супероксидных анионов активированными полиморфноядерными нейтрофилами, адгезию и хемотаксис эозинофилов, выделение молекул адгезии, таких как Р-селектин, IgE-опосредованное высвобождение гистамина, простагландина D2 и лейкотриена С4. Таким образом, предупреждает развитие и облегчает течение аллергических реакций, обладает противозудным и противоэкссудативным действием, уменьшает проницаемость капилляров, предупреждает развитие отека тканей, спазма гладкой мускулатуры.
Препарат не оказывает воздействия на центральную нервную систему, практически не обладает седативным эффектом (не вызывает сонливости) и не влияет на скорость психомоторных реакций. Не вызывает удлинения интервала QT на ЭКГ.
Действие лекарственного препарата начинается в течение 30 минут после приема внутрь и продолжается в течение 24 часов.
Фармакологическая группа
H1-антигистаминные средства
Форма выпуска
таблетки
Способ применения/введения
Минимальный возраст применения
от 12 лет
Продолжительность действия
24 часа

Дополнительно

Условия хранения
В защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте.
Передозировка
Симптомы: прием дозы, превышающей рекомендованную в 5 раз, не приводил к появлению каких-либо симптомов. В ходе клинических исследований ежедневное применение у взрослых и подростков дезлоратадина в дозе до 20 мг в течение 14 дней не сопровождалось статистически или клинически значимыми изменениями со стороны сердечно-сосудистой системы. В клинико-фармакологическом исследовании применения дезлоратадина в дозе 45 мг в сутки (в 9 раз выше рекомендованной) в течение 10 дней не вызывало удлинение интервала QT и не сопровождалось появлениями серьезных побочных эффектов.
Лечение: при случайном приеме внутрь большого количества препарата - промывание желудка, прием активированного угля; при необходимости - симптоматическая терапия. Дезлоратадин не выводится при гемодиализе, эффективность перитонеального диализа не установлена.
Применение при беременности и кормлении грудью
Применение препарата при беременности противопоказано в связи с отсутствием клинических данных о безопасности его применения во время беременности.
Влияние на способность управлять транспортом и механизмами
В рекомендованной дозе препарат не влияет на способность к вождению транспортных средств или управлению механизмами.
Особые указания
Влияние на способность управлять трансп. ср. и мех.:
В рекомендованной дозе препарат не влияет на способность к вождению транспортных средств или управлению механизмами.
Взаимодействие
Взаимодействия с другими лекарственными средствами не выявлено.
Прием пищи не оказывает влияния на эффективность препарата.
Дезлоратадин не усиливает действие алкоголя на центральную нервную систему.
Источник
Регистрационный номер
ЛП-002161
Дата государственной регистрации
27.07.2018
Владелец регистрационного удостоверения
Изготовитель
ОЗОН
Фасовщик
ОЗОН
Страна бренда
Россия
Страна-производитель
Россия
Название препарата
Срок годности
35 мес.
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