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Описание

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Галидор р-р для в/в и в/м введ. амп., 25 мг/мл, 2 мл, 10 шт.

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У продавца: 
нет • На Маркете: 4.1
(9)
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Тяжелая дыхательная, почечная или печеночная недостаточность.\u003Cbr\u003EДекомпенсированная сердечная недостаточность, острый инфаркт миокарда, атриовентрикулярная блокада.\u003Cbr\u003EЭпилепсия и другие формы спазмофилии.\u003Cbr\u003EНедавно перенесенный геморрагический инсульт.\u003Cbr\u003EЧерепно-мозговая травма (в течении последних 12 месяцев).\u003Cbr\u003EБеременность и кормление грудью."},{"name":"Состав","value":"Каждая ампула объемом 2 мл содержит 50 мг активного вещества бенциклана фумарата, а также вспомогательные вещества: натрия хлорид для парентеральных лекарственных форм 8 мг и воду для инъекций до 2 мл."},{"name":"Действующее вещество","value":"Бенциклан","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28709508"]}}},{"name":"Способ применения и дозы","value":"Раствор для в/в инъекций (после разведения) или инфузии.\u003Cbr\u003EСосудистые заболевания\u003Cbr\u003EИнфузия: При сосудистых заболеваниях препарат может применяться в суточной дозе 200 мг, разделенной на 2 инфузии. 100 мг (4 мл) препарата разводят в 100 - 200 мл изотонического раствора NaCl. Препарат вводится внутривенно-капельно в течение 1 часа 2 раза в сутки.\u003Cbr\u003EУстранения спазма внутренних органов\u003Cbr\u003EИнъекции: В острых случаях вводят в вену медленно 2-4 ампулы (4-8 мл) препарата, разведенного солевым раствором до 10 - 20 мл или глубоко внутримышечно 2 мл.\u003Cbr\u003EКурс лечения 2-3 недели, при необходимости, с последующим переводом пациента на прием препарата Галидор таблетки."},{"name":"Побочные действия","value":"Желудочно-кишечные: сухость во рту, боль в животе, чувство сытости, тошнота, рвота.\u003Cbr\u003EЦентральная нервная система: беспокойство, головная боль, головокружение, нарушение походки, тремор, бессонница, расстройства памяти, редко - преходящее спутанное состояние сознания, галлюцинации, очень редко - симптомы очагового поражения ЦНС.\u003Cbr\u003EСердечно-сосудистые: иногда может возникать предсердная или желудочковая тахиаритмия (особенно при совместном введении с другими проаритмогенными препаратами).\u003Cbr\u003EЛабораторные показатели: преходящее повышение активности аспарат-аминотрансферазы и аламин-аминотрансферазы, уменьшение количества белых кровяных клеток.\u003Cbr\u003EДругие: общее недомогание, увеличение веса тела, аллергические реакции, редко - тромбофлебит при внутривенном введении."},{"name":"Фармакологическое действие","value":"Бенциклан - миотропный спазмолитик с выраженным вазодилатирующим действием. Сосудорасширяющее действие бенциклана в основном связано с его способностью блокировать кальциевые каналы, антисеротониновым действием, и в меньшей степени - с блокадой симпатических ганглиев. Кроме того, бенциклан обладает спазмолитическим действием на висцеральную мускулатуру (желудочно-кишечного тракта, мочеполовых органов, органов дыхания). Препарат вызывает некоторое повышение частоты сердечных сокращений. Известно также его слабое транквилизирующее действие.\u003Cbr\u003EМеханизм действия\u003Cbr\u003EБенциклан может вызывать дозозависимое подавление Na/K -зависимой АТФазы и агрегации тромбоцитов и эритроцитов, а также повышение эластичности эритроцитов. Эти эффекты наблюдаются в основном в периферических сосудах, коронарных артериях и мозговых сосудах."},{"name":"Фармакологическая группа","value":"спазмолитическое средство"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["35947170:36763748"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"Хранить при температуре 15-25° С в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: учащение сердечных сокращений, снижение артериального давления, предрасположенность к коллапсу, недержание мочи, сонливость, беспокойство, а в тяжелых случаях - эпилептиформные судорожные припадки. Значительная передозировка может вызвать тонические и клонические судороги.\u003Cbr\u003EЛечение: Специфический антидот не известен. При передозировке следует применять симптоматическое лечение. Для лечения судорожных припадков рекомендуется применять бензодиазепины. Данных о возможном выведении бенциклана посредством диализа нет."},{"name":"Применение при беременности и кормлении грудью","value":"Данные доклинических исследований не выявили никаких эмбриотоксических или тератогенных эффектов. Однако, достаточных достоверных исследований о применении препарата во время беременности и кормления грудью у человека проведено не было. Поэтому введение препарата пациенткам в первом триместре беременности не рекомендуется. В период лактации следует воздержаться от назначения препарата, либо решить вопрос о прекращении грудного вскармливания во время лечения."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В начале курса лечения вождение транспортных средств и выполнение работ с повышенным риском несчастных случаев требует особой осторожности."},{"name":"Особые указания","value":"Места инъекций следует периодически менять, т.к. препарат может вызвать повреждение эндотелия сосудов и тромбофлебит.\u003Cbr\u003EСледует воздерживаться от парентерального введения препарата больным с тяжелой сердечнососудистой или дыхательной недостаточностью, предрасположенным к коллапсу, а также с гипертрофией предстательной железы и задержкой мочи (степень задержки повышается при расслаблении мышц мочевого пузыря).\u003Cbr\u003EПри длительной терапии бенцикланом рекомендуется регулярное проведение лабораторных исследований (не реже одного раза в 2 месяца)."},{"name":"Взаимодействие","value":"Следует соблюдать осторожность при комбинации со следующими средствами:\u003Cbr\u003E- анестетиками и седативными - их эффекты могут усиливаться;\u003Cbr\u003E- симпатомиметиками - из-за риска предсердных и желудочковых тахиаритмий;\u003Cbr\u003E- средствами, снижающими уровень калия крови - из-за возможной суммации проаритмогенных эффектов;\u003Cbr\u003E- препаратами наперстянки - повышается риск аритмии при передозировке наперстянки;\u003Cbr\u003E- бета-блокаторами - из-за противоположности хронотропных эффектов (отрицательный у бета-блокаторов и положительный у бенциклана) может возникнуть необходимость подбора дозировки бета-блокатора;\u003Cbr\u003E- блокаторами кальциевых каналов и другими антигипертензивными препаратами - из-за возможности усиления их эффекта;\u003Cbr\u003E- лекарственными средствами, вызывающих побочные эффекты в виде спазмофилии - из-за возможности суммации этих эффектов;\u003Cbr\u003E- аспирин - из-за усиления торможения агрегации тромбоцитов."},{"name":"Регистрационный номер","value":"П N012430/01"},{"name":"Дата государственной регистрации","value":"14.12.2017"},{"name":"Владелец регистрационного удостоверения","value":"Egis Pharmaceuticals","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313","7893318:16002706"]}}},{"name":"Изготовитель","value":"Фармацевтический завод ЭГИС"},{"name":"Фасовщик","value":"Фармацевтический завод ЭГИС"},{"name":"Страна бренда","value":"Венгрия"},{"name":"Страна-производитель","value":"Венгрия"},{"name":"Название препарата","value":"Галидор","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["17796364:18042661"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"17262310207481774287":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"выделительная система, кровеносные сосуды, пищеварительная система"},{"name":"Назначение","value":"болезнь Рейно, гастроэнтерит, желудочно-кишечные спазмы, желчекаменная болезнь, ишемический инсульт, мочекаменная болезнь, острые нарушения мозгового кровообращения, спазмы гладкой мускулатуры внутренних органов, хронические облитерирующие заболевания артерий, язва желудка, язвенная болезнь желудка и двенадцатиперстной кишки"},{"name":"Показания к применению","value":"Сосудистые заболевания\u003Cbr\u003EЗаболевания периферических сосудов: болезнь Рейно, другие заболевания с акроцианозом и спазмом сосудов, а также хронические облитерирующие заболевания артерий.\u003Cbr\u003EЗаболевания мозговых сосудов: в комплексной терапии острой и хронической церебральной ишемии.\u003Cbr\u003EУстранения спазма внутренних органов\u003Cbr\u003EЖелудочно-кишечные заболевания: гастроэнтериты различной этиологии (особенно инфекционные), инфекционные и воспалительные колиты, функциональные заболевания толстого кишечника, тенезмы, послеоперационный метеоризм, холецистит, желчнокаменная болезнь, состояние после холецистэктомии, нарушения моторики при дискинезии сфинктера Одди, язва желудка или двенадцатиперстной кишки - в сочетании с другими лекарственными препаратами.\u003Cbr\u003EУрологические синдромы: спазмы и тенезмы мочевого пузыря, сопутствующая терапия мочекаменной болезни (в сочетании с аналгетиками при почечной колике), подготовка к инструментальным методам исследования."},{"name":"Противопоказания","value":"Повышенная чувствительность к активному или любому другому компоненту препарата. Тяжелая дыхательная, почечная или печеночная недостаточность.\u003Cbr\u003EДекомпенсированная сердечная недостаточность, острый инфаркт миокарда, атриовентрикулярная блокада.\u003Cbr\u003EЭпилепсия и другие формы спазмофилии.\u003Cbr\u003EНедавно перенесенный геморрагический инсульт.\u003Cbr\u003EЧерепно-мозговая травма (в течении последних 12 месяцев).\u003Cbr\u003EБеременность и кормление грудью."},{"name":"Состав","value":"Каждая ампула объемом 2 мл содержит 50 мг активного вещества бенциклана фумарата, а также вспомогательные вещества: натрия хлорид для парентеральных лекарственных форм 8 мг и воду для инъекций до 2 мл."},{"name":"Действующее вещество","value":"Бенциклан"},{"name":"Способ применения и дозы","value":"Раствор для в/в инъекций (после разведения) или инфузии.\u003Cbr\u003EСосудистые заболевания\u003Cbr\u003EИнфузия: При сосудистых заболеваниях препарат может применяться в суточной дозе 200 мг, разделенной на 2 инфузии. 100 мг (4 мл) препарата разводят в 100 - 200 мл изотонического раствора NaCl. Препарат вводится внутривенно-капельно в течение 1 часа 2 раза в сутки.\u003Cbr\u003EУстранения спазма внутренних органов\u003Cbr\u003EИнъекции: В острых случаях вводят в вену медленно 2-4 ампулы (4-8 мл) препарата, разведенного солевым раствором до 10 - 20 мл или глубоко внутримышечно 2 мл.\u003Cbr\u003EКурс лечения 2-3 недели, при необходимости, с последующим переводом пациента на прием препарата Галидор таблетки."},{"name":"Побочные действия","value":"Желудочно-кишечные: сухость во рту, боль в животе, чувство сытости, тошнота, рвота.\u003Cbr\u003EЦентральная нервная система: беспокойство, головная боль, головокружение, нарушение походки, тремор, бессонница, расстройства памяти, редко - преходящее спутанное состояние сознания, галлюцинации, очень редко - симптомы очагового поражения ЦНС.\u003Cbr\u003EСердечно-сосудистые: иногда может возникать предсердная или желудочковая тахиаритмия (особенно при совместном введении с другими проаритмогенными препаратами).\u003Cbr\u003EЛабораторные показатели: преходящее повышение активности аспарат-аминотрансферазы и аламин-аминотрансферазы, уменьшение количества белых кровяных клеток.\u003Cbr\u003EДругие: общее недомогание, увеличение веса тела, аллергические реакции, редко - тромбофлебит при внутривенном введении."},{"name":"Фармакологическое действие","value":"Бенциклан - миотропный спазмолитик с выраженным вазодилатирующим действием. Сосудорасширяющее действие бенциклана в основном связано с его способностью блокировать кальциевые каналы, антисеротониновым действием, и в меньшей степени - с блокадой симпатических ганглиев. Кроме того, бенциклан обладает спазмолитическим действием на висцеральную мускулатуру (желудочно-кишечного тракта, мочеполовых органов, органов дыхания). Препарат вызывает некоторое повышение частоты сердечных сокращений. Известно также его слабое транквилизирующее действие.\u003Cbr\u003EМеханизм действия\u003Cbr\u003EБенциклан может вызывать дозозависимое подавление Na/K -зависимой АТФазы и агрегации тромбоцитов и эритроцитов, а также повышение эластичности эритроцитов. Эти эффекты наблюдаются в основном в периферических сосудах, коронарных артериях и мозговых сосудах."},{"name":"Фармакологическая группа","value":"спазмолитическое средство"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"Хранить при температуре 15-25° С в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: учащение сердечных сокращений, снижение артериального давления, предрасположенность к коллапсу, недержание мочи, сонливость, беспокойство, а в тяжелых случаях - эпилептиформные судорожные припадки. Значительная передозировка может вызвать тонические и клонические судороги.\u003Cbr\u003EЛечение: Специфический антидот не известен. При передозировке следует применять симптоматическое лечение. Для лечения судорожных припадков рекомендуется применять бензодиазепины. Данных о возможном выведении бенциклана посредством диализа нет."},{"name":"Применение при беременности и кормлении грудью","value":"Данные доклинических исследований не выявили никаких эмбриотоксических или тератогенных эффектов. Однако, достаточных достоверных исследований о применении препарата во время беременности и кормления грудью у человека проведено не было. Поэтому введение препарата пациенткам в первом триместре беременности не рекомендуется. В период лактации следует воздержаться от назначения препарата, либо решить вопрос о прекращении грудного вскармливания во время лечения."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В начале курса лечения вождение транспортных средств и выполнение работ с повышенным риском несчастных случаев требует особой осторожности."},{"name":"Особые указания","value":"Места инъекций следует периодически менять, т.к. препарат может вызвать повреждение эндотелия сосудов и тромбофлебит.\u003Cbr\u003EСледует воздерживаться от парентерального введения препарата больным с тяжелой сердечнососудистой или дыхательной недостаточностью, предрасположенным к коллапсу, а также с гипертрофией предстательной железы и задержкой мочи (степень задержки повышается при расслаблении мышц мочевого пузыря).\u003Cbr\u003EПри длительной терапии бенцикланом рекомендуется регулярное проведение лабораторных исследований (не реже одного раза в 2 месяца)."},{"name":"Взаимодействие","value":"Следует соблюдать осторожность при комбинации со следующими средствами:\u003Cbr\u003E- анестетиками и седативными - их эффекты могут усиливаться;\u003Cbr\u003E- симпатомиметиками - из-за риска предсердных и желудочковых тахиаритмий;\u003Cbr\u003E- средствами, снижающими уровень калия крови - из-за возможной суммации проаритмогенных эффектов;\u003Cbr\u003E- препаратами наперстянки - повышается риск аритмии при передозировке наперстянки;\u003Cbr\u003E- бета-блокаторами - из-за противоположности хронотропных эффектов (отрицательный у бета-блокаторов и положительный у бенциклана) может возникнуть необходимость подбора дозировки бета-блокатора;\u003Cbr\u003E- блокаторами кальциевых каналов и другими антигипертензивными препаратами - из-за возможности усиления их эффекта;\u003Cbr\u003E- лекарственными средствами, вызывающих побочные эффекты в виде спазмофилии - из-за возможности суммации этих эффектов;\u003Cbr\u003E- аспирин - из-за усиления торможения агрегации тромбоцитов."},{"name":"Регистрационный номер","value":"П N012430/01"},{"name":"Дата государственной регистрации","value":"14.12.2017"},{"name":"Владелец регистрационного удостоверения","value":"Egis Pharmaceuticals"},{"name":"Изготовитель","value":"Фармацевтический завод ЭГИС"},{"name":"Фасовщик","value":"Фармацевтический завод ЭГИС"},{"name":"Страна бренда","value":"Венгрия"},{"name":"Страна-производитель","value":"Венгрия"},{"name":"Название препарата","value":"Галидор"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_610802420701947141"}}}}
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Инструкция

Показания к применению

Сосудистые заболевания
Заболевания периферических сосудов: болезнь Рейно, другие заболевания с акроцианозом и спазмом сосудов, а также хронические облитерирующие заболевания артерий.
Заболевания мозговых сосудов: в комплексной терапии острой и хронической церебральной ишемии.
Устранения спазма внутренних органов
Желудочно-кишечные заболевания: гастроэнтериты различной этиологии (особенно инфекционные), инфекционные и воспалительные колиты, функциональные заболевания толстого кишечника, тенезмы, послеоперационный метеоризм, холецистит, желчнокаменная болезнь, состояние после холецистэктомии, нарушения моторики при дискинезии сфинктера Одди, язва желудка или двенадцатиперстной кишки - в сочетании с другими лекарственными препаратами.
Урологические синдромы: спазмы и тенезмы мочевого пузыря, сопутствующая терапия мочекаменной болезни (в сочетании с аналгетиками при почечной колике), подготовка к инструментальным методам исследования.

Противопоказания

Повышенная чувствительность к активному или любому другому компоненту препарата. Тяжелая дыхательная, почечная или печеночная недостаточность.
Декомпенсированная сердечная недостаточность, острый инфаркт миокарда, атриовентрикулярная блокада.
Эпилепсия и другие формы спазмофилии.
Недавно перенесенный геморрагический инсульт.
Черепно-мозговая травма (в течении последних 12 месяцев).
Беременность и кормление грудью.

Способ применения и дозы

Раствор для в/в инъекций (после разведения) или инфузии.
Сосудистые заболевания
Инфузия: При сосудистых заболеваниях препарат может применяться в суточной дозе 200 мг, разделенной на 2 инфузии. 100 мг (4 мл) препарата разводят в 100 - 200 мл изотонического раствора NaCl. Препарат вводится внутривенно-капельно в течение 1 часа 2 раза в сутки.
Устранения спазма внутренних органов
Инъекции: В острых случаях вводят в вену медленно 2-4 ампулы (4-8 мл) препарата, разведенного солевым раствором до 10 - 20 мл или глубоко внутримышечно 2 мл.
Курс лечения 2-3 недели, при необходимости, с последующим переводом пациента на прием препарата Галидор таблетки.
Полная инструкция
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Галидор р-р для в/в и в/м введ. амп.
Галидор р-р для в/в и в/м введ. амп., 25 мг/мл, 2 мл, 10 шт.
У продавца: 
нет • На Маркете: 4.1
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Инструкция

767 ₽

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