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Кеторол Экспресс таб. дисперг., 10 мг, 20 шт.

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полное или неполное сочетание бронхиальной астмы, рецидивирующего полипоза носа и околоносовых пазух и непереносимости ацетилсалициловой кислоты или других НПВП (в том числе в анамнезе); эрозивно-язвенные поражения ЖКТ, активное желудочно-кишечное кровотечение; воспалительные заболевания кишечника (в том числе язвенный колит, болезнь Крона); заболевания костного мозга и крови (лейкопения, в том числе в анамнезе; тромбоцитопения; гипокоагуляция, в том числе гемофилия), миелосупрессия, кровотечения или высокий риск их развития; тяжелая почечная недостаточность (клиренс креатинина (КК) менее 30 мл/мин), подтвержденная гиперкалиемия; тяжелая печеночная недостаточность или активное заболевание печени; состояние после проведения аортокоронарного шунтирования; профилактическое обезболивание перед и во время обширных оперативных вмешательств из-за высокого риска кровотечения; активные цереброваскулярные заболевания (в том числе внутричерепное кровоизлияние или подозрение на него); беременность; период родов; период грудного вскармливания; детский возраст до 16 лет (безопасность и эффективность применения не установлены); одновременное применение с пробенецидом; одновременное применение с пентоксифиллином; одновременное применение с ацетилсалициловой кислотой и другими НПВП (включая селективные ингибиторы ЦОГ-2); одновременное применение с солями лития, одновременное применение с антикоагулянтами (включая варфарин и гепарин)."},{"name":"Состав","value":"Каждая таблетка, диспергируемая в полости рта, содержит:\u003Cbr\u003EДействующее вещество: кеторолака трометамин (кеторолака трометамол) 10,000 мг;\u003Cbr\u003EВспомогательные вещества: целлюлоза микрокристаллическая (Avicel PH101), кремния диоксид, бутилгидроксианизол, маннитол, кросповидон (тип А), сукралоза, ароматизатор мятный, краситель хинолиновый желтый (Е104), магния стеарат."},{"name":"Действующее вещество","value":"Кеторолак","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-travm-boli-v-myshtsakh-i-sustavakh","categoryId":"15756903","navnodeId":"25542230","glfilters":["27144131:28709744"]}}},{"name":"Способ применения и дозы","value":"Положить таблетку на язык, где она сразу же начнет растворяться. Держать во рту в течение нескольких секунд до полного растворения, при желании можно запить жидкостью.\u003Cbr\u003EПрием таблеток, диспергируемых в полости рта, не требует обязательного запивания водой, не влияет на увеличение продукции слюны, позволяет принимать препарат пациентам с отклонениями в акте глотания при поведенческих и неврологических нарушениях.\u003Cbr\u003EКеторол Экспресс применяют внутрь однократно или повторно в зависимости от тяжести болевого синдрома.\u003Cbr\u003EОднократная доза - 10 мг. при повторном приеме рекомендуется принимать по 10 мг до 4-х раз в сутки, в зависимости от выраженности боли; максимальная суточная доза не должна превышать 40 мг.\u003Cbr\u003EПри приеме внутрь продолжительность курса не должна превышать 5 дней.\u003Cbr\u003EДля снижения риска развития нежелательных явлений следует применять минимальную эффективную дозу кеторолака минимально возможным коротким курсом.\u003Cbr\u003EПри переходе с парентерального введения препарата на его прием внутрь суммарная суточная доза обеих лекарственных форм в день перевода не должна превышать 90 мг для пациентов с 16 до 65 лет и 60 мг - для пациентов старше 65 лет или с нарушенной функцией почек. При этом доза препарата в таблетках в день перехода не должна превышать 30 мг."},{"name":"Побочные действия","value":"Частота побочных эффектов классифицируется в зависимости от частоты встречаемости случая; часто (1-10%), нечасто (0,1-1%), редко (0,01-0,1%). очень редко (менее 0,01%) и частота неизвестна, включая отдельные сообщения.\u003Cbr\u003EСо стороны пищеварительной системы\u003Cbr\u003EЧасто (особенно у пожилых пациентов старше 65 лет. имеющих в анамнезе эрозивноязвенные поражения ЖКТ) - гастралгия, диарея; нечасто - стоматит, метеоризм, запор, рвота, ощущение переполнения желудка; редко - тошнота, эрозивно-язвенные поражения ЖКТ (в том числе с перфорацией и/или кровотечением - абдоминальная боль, спазм или жжение в эпигастральной области, мелена, рвота по типу \"кофейной гущи\", тошнота, изжога), холестатическая желтуха, гепатит, гепатомегалия, острый панкреатит.\u003Cbr\u003EСо стороны мочевыделительной системы\u003Cbr\u003EРедко - острая почечная недостаточность, боль в пояснице, гематурия, азотемия, гемолитико-уремический синдром (гемолитическая анемия, почечная недостаточность, тромбоцитопения, пурпура), частое мочеиспускание, олигурия, полиурия, интерстициальный нефрит, отеки почечного генеза; частота неизвестна - задержка мочеиспускания.\u003Cbr\u003EСо стороны органов чувств\u003Cbr\u003EРедко - снижение слуха, звон в ушах, нарушение зрения (в том числе нечеткость зрительного восприятия); частота неизвестна - нарушение вкуса.\u003Cbr\u003EСо стороны дыхательной системы\u003Cbr\u003EРедко - бронхоспазм или диспноэ, ринит, отек гортани (одышка, затруднение дыхания).\u003Cbr\u003EСо стороны центральной нервной системы\u003Cbr\u003EЧасто - головная боль, головокружение, сонливость; редко - асептический менингит (лихорадка, сильная головная боль, судороги, ригидность мышц шеи и/или спины), гиперактивность (изменение настроения, беспокойство), галлюцинации, депрессия, психоз.\u003Cbr\u003EСо стороны сердечно-сосудистой системы\u003Cbr\u003EНечасто - повышение артериального давления; редко - отек легких, обморочные состояния.\u003Cbr\u003EСо стороны органов кроветворения\u003Cbr\u003EРедко - анемия, эозинофилия, лейкопения.\u003Cbr\u003EСо стороны системы гемостаза\u003Cbr\u003EРедко - кровотечение из послеоперационной раны, носовое кровотечение, ректальное кровотечение.\u003Cbr\u003EСо стороны кожных покровов\u003Cbr\u003EНечасто - кожная сыпь (включая макулопапулезную сыпь), пурпура; редко - эксфолиативный дерматит (лихорадка с ознобом или без, покраснение, уплотнение или шелушение кожи, опухание и/или болезненность небных миндалин), крапивница, синдром Стивенса-Джонсона, синдром Лайелла.\u003Cbr\u003EАллергические реакции\u003Cbr\u003EРедко - анафилаксия или анафилактоидные реакции (изменение цвета кожи лица, кожная сыпь, крапивница, кожный зуд, тахипноэ или диспноэ, отеки век, отек языка, периорбитальный отек, одышка, затрудненное дыхание, тяжесть в грудной клетке, свистящее дыхание).\u003Cbr\u003EПрочие\u003Cbr\u003EЧасто - отеки (лица, голеней, лодыжек, пальцев, ступней, повышение массы тела); нечасто - повышенная потливость; редко - лихорадка; частота неизвестна - гиперкалиемия, гипонатриемия."},{"name":"Фармакологическое действие","value":"Нестероидный противовоспалительный препарат (НПВП), оказывает выраженное анальгезирующее действие, обладает противовоспалительным и умеренным жаропонижающим действием. Механизм действия связан с неселективным угнетением активности циклооксигеназы (ЦОГ) - ЦОГ-1 и ЦОГ-2, катализирующей образование простагландинов из арахидоновой кислоты, играющих важную роль в патогенезе воспаления, боли и лихорадки.\u003Cbr\u003EКеторолак представляет собой рацемическую смесь [-]S и [+]R энантиомеров, при этом обезболивающее действие обусловлено [-]S формой.\u003Cbr\u003EПо силе анальгезирующего эффекта кеторолак сопоставим с морфином, значительно превосходя другие НПВП. Препарат не влияет на опиоидные рецепторы, не угнетает дыхания, не вызывает лекарственной зависимости, не обладает седативным и анксиолитическим действием.\u003Cbr\u003EПосле приема внутрь начало обезболивающего действия отмечается через 1 ч, максимальный эффект достигается через 1-2 ч."},{"name":"Фармакологическая группа","value":"нестероидный противовоспалительный препарат (НПВП)"},{"name":"Форма выпуска","value":"таблетки диспергируемые"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-travm-boli-v-myshtsakh-i-sustavakh","categoryId":"15756903","navnodeId":"25542230","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 16 лет"},{"name":"Условия хранения","value":"При температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: боль в животе, тошнота, рвота, эрозивно-язвенное поражение ЖКТ, нарушение функции почек, метаболический ацидоз.\u003Cbr\u003EЛечение: промывание желудка, введение адсорбентов (активированный уголь) и проведение симптоматической терапии (поддержание жизненно важных функций организма). Гемодиализ малоэффективен."},{"name":"Применение при беременности и кормлении грудью","value":"Беременность\u003Cbr\u003EПротивопоказано применение препарата в период беременности (неблагоприятное влияние на сердечно-сосудистую систему плода - преждевременное закрытие аортального протока), во время родов и в раннем послеродовом периоде (ингибируя синтез простагландинов, кеторолак может отрицательно повлиять на кровообращение плода и ослабить сократительную деятельность матки, что повышает риск маточных кровотечений).\u003Cbr\u003EПериод грудного вскармливания\u003Cbr\u003EПрименение кеторолака в период грудного вскармливания противопоказано. Кеторолак приникает в материнское молоко."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо соблюдать осторожность при вождении автотранспорта и занятии другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Выбор лекарственной формы препарата зависит от степени выраженности болевого синдрома и состояния пациента. Препарат Кеторол выпускается в следующих лекарственных формах: гель для наружного применения: таблетки, покрытые пленочной оболочкой; таблетки, диспергируемые в полости рта; раствор для внутривенного и внутримышечного введения.\u003Cbr\u003EПеред применением препарата необходимо выяснить вопрос о предшествующей аллергии на препарат или другие НПВП. Из-за риска развития аллергических реакций прием первой дозы проводят под тщательным наблюдением врача.\u003Cbr\u003EКеторолак подавляет агрегацию тромбоцитов и увеличивает время свертывания крови. Влияние на агрегацию тромбоцитов прекращается через 24-48 ч после приема препарата. Пациентам с нарушением свертывания крови назначают препарат только при постоянном контроле числа тромбоцитов, что особенно важно в послеоперационном периоде, когда требуется тщательный контроль гемостаза.\u003Cbr\u003EГиповолемия повышает риск развития нефротоксических побочных реакций.\u003Cbr\u003EПри необходимости можно применять в комбинации с наркотическими анальгетиками. Не применять с парацетамолом более 2 дней.\u003Cbr\u003EРиск развития нежелательных реакций возрастает при удлинении курса лечения и повышении пероральной дозы кеторолака более 40 мг/сут.\u003Cbr\u003EОдновременный прием кеторолака с пробенецидом, пентоксифиллином, ацетилсалициловой кислотой и другими НПВП (включая ингибиторы ЦОГ-2), солями лития, антикоагулянтами (включая варфарин и гепарин) противопоказан.\u003Cbr\u003EПротивопоказано применение кеторолака для профилактического обезболивания перед и во время обширных оперативных вмешательств из-за высокого риска кровотечения.\u003Cbr\u003EКеторолак не рекомендуется применять в качестве средства для премедикации и поддерживающей анестезии.\u003Cbr\u003EПри применении кеторолака сообщалось о случаях задержки жидкости, повышении артериального давления и отеках.\u003Cbr\u003EНеобходимо соблюдать осторожность при назначении пациентам с сердечной недостаточностью, артериальной гипертензией.\u003Cbr\u003EОдновременное применение кеторолака с другими НПВП может приводить к таким нарушениям, как декомпенсация сердечной недостаточности и повышение артериального давления.\u003Cbr\u003EПо данным клинических исследований, использование некоторых НПВП в высоких дозах может привести к увеличению риска артериальных тромботических осложнений (например, инфаркт миокарда, инсульт). Несмотря на то, что о подобных осложнениях при применении кеторолака не сообщалось, существующих данных недостаточно для исключения риска таких осложнений.\u003Cbr\u003EДля снижения риска развития НПВП-индуцированной гастропатии рекомендовано применение антацидных лекарственных средств, мизопростола, а также препаратов, снижающих желудочную секрецию (блокаторов Н-рецепторов гистамина, ингибиторов протоновой помпы). Для снижения риска развития нежелательных явлений следует применять минимальную эффективную дозу кеторолака минимально возможным коротким курсом.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EБронхиальная астма; наличие факторов, повышающих токсичность в отношении ЖКТ: алкоголизм, табакокурение и холецистит; послеоперационный период; хроническая сердечная недостаточность; отечный синдром; артериальная гипертензия; почечная недостаточность средней степени тяжести (клиренс креатинина 30-60 мл/мин); холестаз; активный гепатит; сепсис; системная красная волчанка; ишемическая болезнь сердца; цереброваскулярные заболевания; дислипидемия/гиперлипидемия; сахарный диабет; заболевания периферических артерии; язвенные поражения ЖКТ в анамнезе; наличие инфекции Helicobacter pylori; длительное применение НПВП; тяжелые соматические заболевания: заболевания щитовидной железы; туберкулез; одновременный прием пероральных глюкокортикостероидов (в том числе преднизолона), антиагрегантов (в том числе клопидогрела), селективных ингибиторов обратного захвата серотонина (в том числе циталопрама, флуоксетина, пароксетина, сергралина); пожилой возраст (старше 65 лет)."},{"name":"Взаимодействие","value":"Одновременное применение кеторолака с ацетилсалициловой кислотой или другими НПВП, препаратами кальция, глюкокортикостероидами, этанолом, кортикотропином может привести к существенному увеличению риска побочных реакций, в том числе образованию язв ЖКТ и развитию желудочно-кишечных кровотечений.\u003Cbr\u003EПри одновременном применении кеторолака с другими НПВП (включая ингибиторы ЦОГ-2) может наблюдаться задержка жидкости, декомпенсация сердечной деятельности, повышение артериального давления.\u003Cbr\u003EОдновременное применение кеторолака с непрямыми антикоагулянтами, тромболитиками, антиагрегантами, цефоперазоном, цефотетаном и пентоксифиллином повышает риск кровотечения.\u003Cbr\u003EПробенецид уменьшает плазменный клиренс и объем распределения кеторолака, повышает его концентрацию в плазме крови и увеличивает его T1/2.\u003Cbr\u003EСовместное применение кеторолака с вальпроатом вызывает нарушение агрегации тромбоцитов.\u003Cbr\u003EПри применении кеторолака с другими нефротоксичными лекарственными средствами (в том числе с препаратами золота) повышается риск развития нефротоксичности. Совместное применение с парацетамолом повышает нефротоксичность кеторолака.\u003Cbr\u003EЛекарственные средства, блокирующие канальцевую секрецию, снижают клиренс кеторолака и повышают его концентрацию в плазме крови.\u003Cbr\u003EСовместное применение кеторолака с метотрексатом повышает гепато- и нефротоксичность метотрексата. Совместное применение кеторолака и метотрексата возможно только при применении низких доз последнего. Возможно уменьшение клиренса метотрексата (необходимо контролировать концентрацию метотрексата в плазме крови).\u003Cbr\u003EНа фоне применения кеторолака возможно уменьшение клиренса лития, увеличение его концентрации в плазме крови и усиление токсического действия лития. Одновременное применение с солями лития противопоказано.\u003Cbr\u003EКеторолак снижает эффект гипотензивных и диуретических препаратов (снижается синтез простагландинов в почках).\u003Cbr\u003EКеторолак усиливает эффект наркотических анальгетиков. При комбинировании с опиоидными анальгетиками дозы последних могут быть существенно снижены. Кеторолак усиливает гипогликемическое действие инсулина и пероральных гипогликемических препаратов, в связи с чем необходим перерасчет дозы указанных препаратов.\u003Cbr\u003EКеторолак повышает концентрацию в плазме крови верапамила и нифедипина. Одновременное применение НПВП и мифепристона может снижать эффективность мифепристона. НПВП не рекомендуется применять в течение 8-12 дней после применения мифепристона.\u003Cbr\u003EОдновременное применение НПВП и циклоспорина увеличивает риск развития нефротоксичности.\u003Cbr\u003EОдновременное применение НПВП и антибиотиков хинолонового ряда увеличивает риск развития судорог.\u003Cbr\u003EОдновременное применение НПВП и такролимуса увеличивает риск развития нефротоксичности.\u003Cbr\u003EОдновременное применение НПВП и зидовудина увеличивает риск развития гематологической токсичности.\u003Cbr\u003EПри одновременном применении с дигоксином кеторолак не нарушает связывание дигоксина с белками плазмы крови. Терапевтические концентрации дигоксина не влияют на связывание кеторолака с белками плазмы крови.\u003Cbr\u003EАнтацидные средства не влияют на всасывание кеторолака.\u003Cbr\u003EМиелотоксичные лекарственные средства усиливают проявления гематотоксичности кеторолака."},{"name":"Регистрационный номер","value":"ЛП-004929"},{"name":"Дата государственной регистрации","value":"01.11.2019"},{"name":"Владелец регистрационного удостоверения","value":"Dr. Reddy's Laboratories","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-travm-boli-v-myshtsakh-i-sustavakh","categoryId":"15756903","navnodeId":"25542230","glfilters":["34324371:35649313","7893318:16077120"]}}},{"name":"Изготовитель","value":"Dr. Reddy's"},{"name":"Фасовщик","value":"Dr. Reddy's"},{"name":"Страна бренда","value":"Индия"},{"name":"Страна-производитель","value":"Индия"},{"name":"Название препарата","value":"Кеторол","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-travm-boli-v-myshtsakh-i-sustavakh","categoryId":"15756903","navnodeId":"25542230","glfilters":["17796364:18042643"]}}},{"name":"Срок годности","value":"23 мес."}]}},"fullSpecsGrouped":{"16515396006892066594":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"опорно-двигательная система"},{"name":"Назначение","value":"артралгия, болевой синдром средней и высокой интенсивности различной этиологии, боль в мышцах, боль в суставах, интенсивный хронический болевой синдром, миалгия, невралгия, посттравматический болевой синдром, радикулит, растяжения, ревматоидный артрит, сопровождающая терапия онкологических заболеваний"},{"name":"Показания к применению","value":"Болевой синдром сильной и умеренной выраженности: травмы, зубная боль, боли в послеоперационном периоде, онкологические заболевания, миалгия, артралгия. невралгия, радикулит, вывихи, растяжения, ревматические заболевания.\u003Cbr\u003EПредназначен для симптоматической терапии, уменьшения интенсивности боли и воспаления на момент использования, не влияет на прогрессирование заболевания."},{"name":"Противопоказания","value":"Гиперчувствительность (в том числе к другим ННВП); полное или неполное сочетание бронхиальной астмы, рецидивирующего полипоза носа и околоносовых пазух и непереносимости ацетилсалициловой кислоты или других НПВП (в том числе в анамнезе); эрозивно-язвенные поражения ЖКТ, активное желудочно-кишечное кровотечение; воспалительные заболевания кишечника (в том числе язвенный колит, болезнь Крона); заболевания костного мозга и крови (лейкопения, в том числе в анамнезе; тромбоцитопения; гипокоагуляция, в том числе гемофилия), миелосупрессия, кровотечения или высокий риск их развития; тяжелая почечная недостаточность (клиренс креатинина (КК) менее 30 мл/мин), подтвержденная гиперкалиемия; тяжелая печеночная недостаточность или активное заболевание печени; состояние после проведения аортокоронарного шунтирования; профилактическое обезболивание перед и во время обширных оперативных вмешательств из-за высокого риска кровотечения; активные цереброваскулярные заболевания (в том числе внутричерепное кровоизлияние или подозрение на него); беременность; период родов; период грудного вскармливания; детский возраст до 16 лет (безопасность и эффективность применения не установлены); одновременное применение с пробенецидом; одновременное применение с пентоксифиллином; одновременное применение с ацетилсалициловой кислотой и другими НПВП (включая селективные ингибиторы ЦОГ-2); одновременное применение с солями лития, одновременное применение с антикоагулянтами (включая варфарин и гепарин)."},{"name":"Состав","value":"Каждая таблетка, диспергируемая в полости рта, содержит:\u003Cbr\u003EДействующее вещество: кеторолака трометамин (кеторолака трометамол) 10,000 мг;\u003Cbr\u003EВспомогательные вещества: целлюлоза микрокристаллическая (Avicel PH101), кремния диоксид, бутилгидроксианизол, маннитол, кросповидон (тип А), сукралоза, ароматизатор мятный, краситель хинолиновый желтый (Е104), магния стеарат."},{"name":"Действующее вещество","value":"Кеторолак"},{"name":"Способ применения и дозы","value":"Положить таблетку на язык, где она сразу же начнет растворяться. Держать во рту в течение нескольких секунд до полного растворения, при желании можно запить жидкостью.\u003Cbr\u003EПрием таблеток, диспергируемых в полости рта, не требует обязательного запивания водой, не влияет на увеличение продукции слюны, позволяет принимать препарат пациентам с отклонениями в акте глотания при поведенческих и неврологических нарушениях.\u003Cbr\u003EКеторол Экспресс применяют внутрь однократно или повторно в зависимости от тяжести болевого синдрома.\u003Cbr\u003EОднократная доза - 10 мг. при повторном приеме рекомендуется принимать по 10 мг до 4-х раз в сутки, в зависимости от выраженности боли; максимальная суточная доза не должна превышать 40 мг.\u003Cbr\u003EПри приеме внутрь продолжительность курса не должна превышать 5 дней.\u003Cbr\u003EДля снижения риска развития нежелательных явлений следует применять минимальную эффективную дозу кеторолака минимально возможным коротким курсом.\u003Cbr\u003EПри переходе с парентерального введения препарата на его прием внутрь суммарная суточная доза обеих лекарственных форм в день перевода не должна превышать 90 мг для пациентов с 16 до 65 лет и 60 мг - для пациентов старше 65 лет или с нарушенной функцией почек. При этом доза препарата в таблетках в день перехода не должна превышать 30 мг."},{"name":"Побочные действия","value":"Частота побочных эффектов классифицируется в зависимости от частоты встречаемости случая; часто (1-10%), нечасто (0,1-1%), редко (0,01-0,1%). очень редко (менее 0,01%) и частота неизвестна, включая отдельные сообщения.\u003Cbr\u003EСо стороны пищеварительной системы\u003Cbr\u003EЧасто (особенно у пожилых пациентов старше 65 лет. имеющих в анамнезе эрозивноязвенные поражения ЖКТ) - гастралгия, диарея; нечасто - стоматит, метеоризм, запор, рвота, ощущение переполнения желудка; редко - тошнота, эрозивно-язвенные поражения ЖКТ (в том числе с перфорацией и/или кровотечением - абдоминальная боль, спазм или жжение в эпигастральной области, мелена, рвота по типу \"кофейной гущи\", тошнота, изжога), холестатическая желтуха, гепатит, гепатомегалия, острый панкреатит.\u003Cbr\u003EСо стороны мочевыделительной системы\u003Cbr\u003EРедко - острая почечная недостаточность, боль в пояснице, гематурия, азотемия, гемолитико-уремический синдром (гемолитическая анемия, почечная недостаточность, тромбоцитопения, пурпура), частое мочеиспускание, олигурия, полиурия, интерстициальный нефрит, отеки почечного генеза; частота неизвестна - задержка мочеиспускания.\u003Cbr\u003EСо стороны органов чувств\u003Cbr\u003EРедко - снижение слуха, звон в ушах, нарушение зрения (в том числе нечеткость зрительного восприятия); частота неизвестна - нарушение вкуса.\u003Cbr\u003EСо стороны дыхательной системы\u003Cbr\u003EРедко - бронхоспазм или диспноэ, ринит, отек гортани (одышка, затруднение дыхания).\u003Cbr\u003EСо стороны центральной нервной системы\u003Cbr\u003EЧасто - головная боль, головокружение, сонливость; редко - асептический менингит (лихорадка, сильная головная боль, судороги, ригидность мышц шеи и/или спины), гиперактивность (изменение настроения, беспокойство), галлюцинации, депрессия, психоз.\u003Cbr\u003EСо стороны сердечно-сосудистой системы\u003Cbr\u003EНечасто - повышение артериального давления; редко - отек легких, обморочные состояния.\u003Cbr\u003EСо стороны органов кроветворения\u003Cbr\u003EРедко - анемия, эозинофилия, лейкопения.\u003Cbr\u003EСо стороны системы гемостаза\u003Cbr\u003EРедко - кровотечение из послеоперационной раны, носовое кровотечение, ректальное кровотечение.\u003Cbr\u003EСо стороны кожных покровов\u003Cbr\u003EНечасто - кожная сыпь (включая макулопапулезную сыпь), пурпура; редко - эксфолиативный дерматит (лихорадка с ознобом или без, покраснение, уплотнение или шелушение кожи, опухание и/или болезненность небных миндалин), крапивница, синдром Стивенса-Джонсона, синдром Лайелла.\u003Cbr\u003EАллергические реакции\u003Cbr\u003EРедко - анафилаксия или анафилактоидные реакции (изменение цвета кожи лица, кожная сыпь, крапивница, кожный зуд, тахипноэ или диспноэ, отеки век, отек языка, периорбитальный отек, одышка, затрудненное дыхание, тяжесть в грудной клетке, свистящее дыхание).\u003Cbr\u003EПрочие\u003Cbr\u003EЧасто - отеки (лица, голеней, лодыжек, пальцев, ступней, повышение массы тела); нечасто - повышенная потливость; редко - лихорадка; частота неизвестна - гиперкалиемия, гипонатриемия."},{"name":"Фармакологическое действие","value":"Нестероидный противовоспалительный препарат (НПВП), оказывает выраженное анальгезирующее действие, обладает противовоспалительным и умеренным жаропонижающим действием. Механизм действия связан с неселективным угнетением активности циклооксигеназы (ЦОГ) - ЦОГ-1 и ЦОГ-2, катализирующей образование простагландинов из арахидоновой кислоты, играющих важную роль в патогенезе воспаления, боли и лихорадки.\u003Cbr\u003EКеторолак представляет собой рацемическую смесь [-]S и [+]R энантиомеров, при этом обезболивающее действие обусловлено [-]S формой.\u003Cbr\u003EПо силе анальгезирующего эффекта кеторолак сопоставим с морфином, значительно превосходя другие НПВП. Препарат не влияет на опиоидные рецепторы, не угнетает дыхания, не вызывает лекарственной зависимости, не обладает седативным и анксиолитическим действием.\u003Cbr\u003EПосле приема внутрь начало обезболивающего действия отмечается через 1 ч, максимальный эффект достигается через 1-2 ч."},{"name":"Фармакологическая группа","value":"нестероидный противовоспалительный препарат (НПВП)"},{"name":"Форма выпуска","value":"таблетки диспергируемые"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 16 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"При температуре не выше 25 °С.\u003Cbr\u003EХранить в недоступном для детей месте."},{"name":"Передозировка","value":"Симптомы: боль в животе, тошнота, рвота, эрозивно-язвенное поражение ЖКТ, нарушение функции почек, метаболический ацидоз.\u003Cbr\u003EЛечение: промывание желудка, введение адсорбентов (активированный уголь) и проведение симптоматической терапии (поддержание жизненно важных функций организма). Гемодиализ малоэффективен."},{"name":"Применение при беременности и кормлении грудью","value":"Беременность\u003Cbr\u003EПротивопоказано применение препарата в период беременности (неблагоприятное влияние на сердечно-сосудистую систему плода - преждевременное закрытие аортального протока), во время родов и в раннем послеродовом периоде (ингибируя синтез простагландинов, кеторолак может отрицательно повлиять на кровообращение плода и ослабить сократительную деятельность матки, что повышает риск маточных кровотечений).\u003Cbr\u003EПериод грудного вскармливания\u003Cbr\u003EПрименение кеторолака в период грудного вскармливания противопоказано. Кеторолак приникает в материнское молоко."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо соблюдать осторожность при вождении автотранспорта и занятии другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Выбор лекарственной формы препарата зависит от степени выраженности болевого синдрома и состояния пациента. Препарат Кеторол выпускается в следующих лекарственных формах: гель для наружного применения: таблетки, покрытые пленочной оболочкой; таблетки, диспергируемые в полости рта; раствор для внутривенного и внутримышечного введения.\u003Cbr\u003EПеред применением препарата необходимо выяснить вопрос о предшествующей аллергии на препарат или другие НПВП. Из-за риска развития аллергических реакций прием первой дозы проводят под тщательным наблюдением врача.\u003Cbr\u003EКеторолак подавляет агрегацию тромбоцитов и увеличивает время свертывания крови. Влияние на агрегацию тромбоцитов прекращается через 24-48 ч после приема препарата. Пациентам с нарушением свертывания крови назначают препарат только при постоянном контроле числа тромбоцитов, что особенно важно в послеоперационном периоде, когда требуется тщательный контроль гемостаза.\u003Cbr\u003EГиповолемия повышает риск развития нефротоксических побочных реакций.\u003Cbr\u003EПри необходимости можно применять в комбинации с наркотическими анальгетиками. Не применять с парацетамолом более 2 дней.\u003Cbr\u003EРиск развития нежелательных реакций возрастает при удлинении курса лечения и повышении пероральной дозы кеторолака более 40 мг/сут.\u003Cbr\u003EОдновременный прием кеторолака с пробенецидом, пентоксифиллином, ацетилсалициловой кислотой и другими НПВП (включая ингибиторы ЦОГ-2), солями лития, антикоагулянтами (включая варфарин и гепарин) противопоказан.\u003Cbr\u003EПротивопоказано применение кеторолака для профилактического обезболивания перед и во время обширных оперативных вмешательств из-за высокого риска кровотечения.\u003Cbr\u003EКеторолак не рекомендуется применять в качестве средства для премедикации и поддерживающей анестезии.\u003Cbr\u003EПри применении кеторолака сообщалось о случаях задержки жидкости, повышении артериального давления и отеках.\u003Cbr\u003EНеобходимо соблюдать осторожность при назначении пациентам с сердечной недостаточностью, артериальной гипертензией.\u003Cbr\u003EОдновременное применение кеторолака с другими НПВП может приводить к таким нарушениям, как декомпенсация сердечной недостаточности и повышение артериального давления.\u003Cbr\u003EПо данным клинических исследований, использование некоторых НПВП в высоких дозах может привести к увеличению риска артериальных тромботических осложнений (например, инфаркт миокарда, инсульт). Несмотря на то, что о подобных осложнениях при применении кеторолака не сообщалось, существующих данных недостаточно для исключения риска таких осложнений.\u003Cbr\u003EДля снижения риска развития НПВП-индуцированной гастропатии рекомендовано применение антацидных лекарственных средств, мизопростола, а также препаратов, снижающих желудочную секрецию (блокаторов Н-рецепторов гистамина, ингибиторов протоновой помпы). Для снижения риска развития нежелательных явлений следует применять минимальную эффективную дозу кеторолака минимально возможным коротким курсом.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EБронхиальная астма; наличие факторов, повышающих токсичность в отношении ЖКТ: алкоголизм, табакокурение и холецистит; послеоперационный период; хроническая сердечная недостаточность; отечный синдром; артериальная гипертензия; почечная недостаточность средней степени тяжести (клиренс креатинина 30-60 мл/мин); холестаз; активный гепатит; сепсис; системная красная волчанка; ишемическая болезнь сердца; цереброваскулярные заболевания; дислипидемия/гиперлипидемия; сахарный диабет; заболевания периферических артерии; язвенные поражения ЖКТ в анамнезе; наличие инфекции Helicobacter pylori; длительное применение НПВП; тяжелые соматические заболевания: заболевания щитовидной железы; туберкулез; одновременный прием пероральных глюкокортикостероидов (в том числе преднизолона), антиагрегантов (в том числе клопидогрела), селективных ингибиторов обратного захвата серотонина (в том числе циталопрама, флуоксетина, пароксетина, сергралина); пожилой возраст (старше 65 лет)."},{"name":"Взаимодействие","value":"Одновременное применение кеторолака с ацетилсалициловой кислотой или другими НПВП, препаратами кальция, глюкокортикостероидами, этанолом, кортикотропином может привести к существенному увеличению риска побочных реакций, в том числе образованию язв ЖКТ и развитию желудочно-кишечных кровотечений.\u003Cbr\u003EПри одновременном применении кеторолака с другими НПВП (включая ингибиторы ЦОГ-2) может наблюдаться задержка жидкости, декомпенсация сердечной деятельности, повышение артериального давления.\u003Cbr\u003EОдновременное применение кеторолака с непрямыми антикоагулянтами, тромболитиками, антиагрегантами, цефоперазоном, цефотетаном и пентоксифиллином повышает риск кровотечения.\u003Cbr\u003EПробенецид уменьшает плазменный клиренс и объем распределения кеторолака, повышает его концентрацию в плазме крови и увеличивает его T1/2.\u003Cbr\u003EСовместное применение кеторолака с вальпроатом вызывает нарушение агрегации тромбоцитов.\u003Cbr\u003EПри применении кеторолака с другими нефротоксичными лекарственными средствами (в том числе с препаратами золота) повышается риск развития нефротоксичности. Совместное применение с парацетамолом повышает нефротоксичность кеторолака.\u003Cbr\u003EЛекарственные средства, блокирующие канальцевую секрецию, снижают клиренс кеторолака и повышают его концентрацию в плазме крови.\u003Cbr\u003EСовместное применение кеторолака с метотрексатом повышает гепато- и нефротоксичность метотрексата. Совместное применение кеторолака и метотрексата возможно только при применении низких доз последнего. Возможно уменьшение клиренса метотрексата (необходимо контролировать концентрацию метотрексата в плазме крови).\u003Cbr\u003EНа фоне применения кеторолака возможно уменьшение клиренса лития, увеличение его концентрации в плазме крови и усиление токсического действия лития. Одновременное применение с солями лития противопоказано.\u003Cbr\u003EКеторолак снижает эффект гипотензивных и диуретических препаратов (снижается синтез простагландинов в почках).\u003Cbr\u003EКеторолак усиливает эффект наркотических анальгетиков. При комбинировании с опиоидными анальгетиками дозы последних могут быть существенно снижены. Кеторолак усиливает гипогликемическое действие инсулина и пероральных гипогликемических препаратов, в связи с чем необходим перерасчет дозы указанных препаратов.\u003Cbr\u003EКеторолак повышает концентрацию в плазме крови верапамила и нифедипина. Одновременное применение НПВП и мифепристона может снижать эффективность мифепристона. НПВП не рекомендуется применять в течение 8-12 дней после применения мифепристона.\u003Cbr\u003EОдновременное применение НПВП и циклоспорина увеличивает риск развития нефротоксичности.\u003Cbr\u003EОдновременное применение НПВП и антибиотиков хинолонового ряда увеличивает риск развития судорог.\u003Cbr\u003EОдновременное применение НПВП и такролимуса увеличивает риск развития нефротоксичности.\u003Cbr\u003EОдновременное применение НПВП и зидовудина увеличивает риск развития гематологической токсичности.\u003Cbr\u003EПри одновременном применении с дигоксином кеторолак не нарушает связывание дигоксина с белками плазмы крови. Терапевтические концентрации дигоксина не влияют на связывание кеторолака с белками плазмы крови.\u003Cbr\u003EАнтацидные средства не влияют на всасывание кеторолака.\u003Cbr\u003EМиелотоксичные лекарственные средства усиливают проявления гематотоксичности кеторолака."},{"name":"Регистрационный номер","value":"ЛП-004929"},{"name":"Дата государственной регистрации","value":"01.11.2019"},{"name":"Владелец регистрационного удостоверения","value":"Dr. Reddy's Laboratories"},{"name":"Изготовитель","value":"Dr. Reddy's"},{"name":"Фасовщик","value":"Dr. Reddy's"},{"name":"Страна бренда","value":"Индия"},{"name":"Страна-производитель","value":"Индия"},{"name":"Название препарата","value":"Кеторол"},{"name":"Срок годности","value":"23 мес."}]}],"transitionId":"tr_5063965807702418361"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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Цена с картой Яндекс Пэй:83₽/шт

Скидка: 38%
–38 %
Вместо: 84₽/шт134₽/шт
  • 26-28 июня, самовывоз  0 ₽
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Инструкция

Показания к применению

Болевой синдром сильной и умеренной выраженности: травмы, зубная боль, боли в послеоперационном периоде, онкологические заболевания, миалгия, артралгия. невралгия, радикулит, вывихи, растяжения, ревматические заболевания.
Предназначен для симптоматической терапии, уменьшения интенсивности боли и воспаления на момент использования, не влияет на прогрессирование заболевания.

Противопоказания

Гиперчувствительность (в том числе к другим ННВП); полное или неполное сочетание бронхиальной астмы, рецидивирующего полипоза носа и околоносовых пазух и непереносимости ацетилсалициловой кислоты или других НПВП (в том числе в анамнезе); эрозивно-язвенные поражения ЖКТ, активное желудочно-кишечное кровотечение; воспалительные заболевания кишечника (в том числе язвенный колит, болезнь Крона); заболевания костного мозга и крови (лейкопения, в том числе в анамнезе; тромбоцитопения; гипокоагуляция, в том числе гемофилия), миелосупрессия, кровотечения или высокий риск их развития; тяжелая почечная недостаточность (клиренс креатинина (КК) менее 30 мл/мин), подтвержденная гиперкалиемия; тяжелая печеночная недостаточность или активное заболевание печени; состояние после проведения аортокоронарного шунтирования; профилактическое обезболивание перед и во время обширных оперативных вмешательств из-за высокого риска кровотечения; активные цереброваскулярные заболевания (в том числе внутричерепное кровоизлияние или подозрение на него); беременность; период родов; период грудного вскармливания; детский возраст до 16 лет (безопасность и эффективность применения не установлены); одновременное применение с пробенецидом; одновременное применение с пентоксифиллином; одновременное применение с ацетилсалициловой кислотой и другими НПВП (включая селективные ингибиторы ЦОГ-2); одновременное применение с солями лития, одновременное применение с антикоагулянтами (включая варфарин и гепарин).

Способ применения и дозы

Положить таблетку на язык, где она сразу же начнет растворяться. Держать во рту в течение нескольких секунд до полного растворения, при желании можно запить жидкостью.
Прием таблеток, диспергируемых в полости рта, не требует обязательного запивания водой, не влияет на увеличение продукции слюны, позволяет принимать препарат пациентам с отклонениями в акте глотания при поведенческих и неврологических нарушениях.
Кеторол Экспресс применяют внутрь однократно или повторно в зависимости от тяжести болевого синдрома.
Однократная доза - 10 мг. при повторном приеме рекомендуется принимать по 10 мг до 4-х раз в сутки, в зависимости от выраженности боли; максимальная суточная доза не должна превышать 40 мг.
При приеме внутрь продолжительность курса не должна превышать 5 дней.
Для снижения риска развития нежелательных явлений следует применять минимальную эффективную дозу кеторолака минимально возможным коротким курсом.
При переходе с парентерального введения препарата на его прием внутрь суммарная суточная доза обеих лекарственных форм в день перевода не должна превышать 90 мг для пациентов с 16 до 65 лет и 60 мг - для пациентов старше 65 лет или с нарушенной функцией почек. При этом доза препарата в таблетках в день перехода не должна превышать 30 мг.
Полная инструкция
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Кеторол Экспресс таб. дисперг.
Кеторол Экспресс таб. дисперг., 10 мг, 20 шт.
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Инструкция

Цена с картой Яндекс Пэй:83₽/шт

Скидка: 38%
–38 %
Вместо: 84₽/шт134₽/шт
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4.9
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У продавца:33 оценки·3 отзыва
У всех продавцов:292 оценки·117 отзывов
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user avatar
2 недели назад • Вера Николаевна • Куплен на Маркете
Достоинства: не надо запивать, быстро рассацивается на языке. при спазме помогает.
Недостатки: ? у каждого свои нюансы.
Комментарий: принимать без фанатизма.
user avatar
Неделю назад • Valentina Tarasova • Куплен на Маркете
Достоинства: боль снимает быстро
user avatar
Год назад • Имя скрыто • Куплен на Маркете
Достоинства: Единственный препарат, который помогает при болях
Недостатки: Выпускается по рецепту
Посмотреть все отзывы на Маркете
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  • Vitamin D3, 2000 ME, 30 мл, 30 г, 30 шт.
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  • Omega-3 капс., 1000 мг, 100 мл, 30 шт.
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  • Gummies B Complex со вкусом клубники, 220 г, 45 шт., клубника
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  • Таблетница Пилюля Трансформер
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  • Эвалар Чай Эвалар БИО при повышенном содержании мочевой кислоты, 20 фильтр-пакетов
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  • Бинт эластичный самофиксирующийся / бандажная лента для животных, для перевязок, для тату, 5 см х 4,5 м, черный, 1 шт
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  • Эвалар чай Турбослим Очищение ф/п, 2 г, 20 шт.
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  • MAXLER USA Glucosamine-Chondroitin-MSM (90 таблеток)
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  • Препарат для укрепления связок и суставов Universal Nutrition Animal Flex, 44 шт.
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:873692947_12/content/content/gallery":{"title":"Препарат для укрепления связок и суставов Universal Nutrition Animal Flex, 44 шт.","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/12505310/img_id7218260310259548828.png/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/12505310/img_id7218260310259548828.png/120x160 120w, https://avatars.mds.yandex.net/get-mpic/12505310/img_id7218260310259548828.png/180x240 180w, https://avatars.mds.yandex.net/get-mpic/12505310/img_id7218260310259548828.png/240x320 240w, https://avatars.mds.yandex.net/get-mpic/12505310/img_id7218260310259548828.png/300x400 300w, https://avatars.mds.yandex.net/get-mpic/12505310/img_id7218260310259548828.png/600x800 600w","sizes":"(max-width: 1456px) 15vw, 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  • Магне-В6 р-р д/вн. приема амп., 10 шт.
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  • Бинт когезивный (самофиксирующийся) "Вариант", 4м х 6см , белый, 2 шт. в наборе
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  • Марлевый Бинт медицинский стерильный Вариант 5 м х 10 см ГОСТ, 5 шт. в наборе
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  • Таблетница из 14 секций на семь дней Утро-вечер
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  • Марля медицинская повышенной плотности, отрез 3 метра
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