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Описание

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Мезатон р-р д/ин. . амп., 10 мг/мл, 1 мл, 10 шт.

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У продавца: 
нет • На Маркете: 4.8
(12)
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Коротко о товаре

Инструкция
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При необходимости введение повторяют.\u003Cbr\u003EВнутривенно капельно - 1 мл 1% раствора в 250-500 мл 5% раствора декстрозы.\u003Cbr\u003EПодкожно или внутримышечно, взрослым - 0,3-1 мл 1% раствора 2-3 раза в день; детям старше 15 лет при артериальной гипотензии во время спинномозговой анестезии - 0,5-1 мг/кг.\u003Cbr\u003EДля сужения сосудов слизистых оболочек и уменьшения воспалительных явлений смазывают или закапывают(концентрации раствора - 0,125%, 0,25%, 0,5%, 1%).\u003Cbr\u003EПри местной анестезии добавляют по 0,3-0,5 мл 1% раствора на 10 мл раствора анестетика.\u003Cbr\u003EВысшие дозы для взрослых: подкожно и внутримышечно: разовая - 10 мг, суточная - 50 мг; внутривенно: разовая - 5 мг, суточная - 25 мг."},{"name":"Побочные действия","value":"Со стороны сердечно-сосудистой системы: повышение артериального давления, сердцебиение, фибрилляция желудочков сердца, аритмия, брадикардия, кардиалгия.\u003Cbr\u003EСо стороны ЦНС: головокружение, чувство страха, бессонница, беспокойство, слабость, головная боль, тремор, парестезии, судороги, кровоизлияние в мозг.\u003Cbr\u003EПрочие: бледность кожи лица, ишемия кожи в месте инъекции, в единичных случаях возможны некроз и образование струпа при попадании в ткани или при подкожных инъекциях, аллергические реакции."},{"name":"Фармакологическое действие","value":"Альфа1-адреностимулятор, мало влияющий на бета-адренорецепторы сердца; не является катехоламином (содержит лишь одну гидроксильную гpyппy в ароматическом ядре). Вызывает сужение артериол и повышение артериального давления (с возможной рефлекторной брадикардией). По сравнению с норэпинефрином и эпинефрином менее резко повышает артериальное давление, но действует более длительно (слабее подвержен действию катехол-О-метилтрансферазы); не вызывает увеличения минутного объема крови.\u003Cbr\u003EДействие начинается сразу после введения и продолжается в течение 5-20 мин (после внутривенного введения), 50 мин (при подкожном введении), 1-2 ч (после внутримышечного введения)."},{"name":"Фармакологическая группа","value":"альфа-адреномиметики"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["35947170:36763748"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"Хранить в сухом, защищенном от света и недоступном для детей месте при температуре не выше 25 °С."},{"name":"Передозировка","value":"Симптомы: желудочковая экстрасистолия, короткие пароксизмы желудочковой тахикардии, ощущение тяжести в голове и конечностях, значительное повышение АД.\u003Cbr\u003EЛечение: внутривенное введение альфа-адреноблокаторов (фентоламин) и бета-адреноблокаторов (при нарушениях сердечного ритма)."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо воздержаться от управления транспортными средствами и занятий потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"В период лечения следует контролировать показатели ЭКГ, АД, минутного объема крови, кровообращение в конечностях и в месте инъекции.\u003Cbr\u003EУ больных с артериальной гипертензией в случае медикаментозного коллапса достаточно поддерживать систолическое артериальное давление на уровне, ниже привычного на 30-40 мм рт.ст.\u003Cbr\u003EПеред началом или во время терапии шоковых состояний обязательна коррекция гиповолемии, гипоксии, ацидоза и гиперкапнии.\u003Cbr\u003EРезкое повышение артериального давления, выраженная брадикардия или тахикардия, стойкие нарушения ритма сердца требуют прекращения лечения.\u003Cbr\u003EДля предотвращения повторного снижения АД после отмены препарата дозу следует уменьшать постепенно, особенно после длительной инфузии.\u003Cbr\u003EИнфузию возобновляют, если систолическое артериальное давление снижается до 70-80 мм рт.ст.\u003Cbr\u003EСледует иметь в виду, что использование вазоконстрикторов во время родов для коррекции артериальной гипотензии или в качестве добавок к местным анестетикам па фоне средств, стимулирующих родовую деятельность (вазопрессина, эрготамина, эргометрина, метилэргометрина), может повлечь стойкое повышение артериального давления в послеродовом периоде.\u003Cbr\u003EС возрастом снижается количество адренорецепторов, чувствительных к фенилэфрину. Ингибиторы моноаминоксидазы, повышая прессорный эффект симпатомиметиков, могут обусловливать возникновение головных болей, аритмии, рвоты, гипертонического криза, поэтому при приеме пациентами ингибиторов моноаминоксидазы в предшествующие 2-3 недели дозы симпатомиметиков должны быть снижены."},{"name":"Взаимодействие","value":"Мезатон снижает антигипертензивный эффект диуретиков и антигипертензивных лекарственных средств (метилдопы, мекамиламина, гуанадрела, гуанетидина).\u003Cbr\u003EФенотиазины, альфа-адреноблокаторы (фентоламин), фуросемид и прочие диуретики снижают гинертензивный эффект.\u003Cbr\u003EИнгибиторы моноаминоксидазы (фуразолидон, прокарбазин, селегилин), окситоцин, алкалоиды спорыньи, трициклические антидепрессанты, метилфенидат, адреностимуляторы усиливают прессорный эффект и аритмогенность фенилэфрина.\u003Cbr\u003EБета-адреноблокаторы уменьшают кардиостимулирующую активность, на фоне резерпина - возможна артериальная гипертензия (в результате истощения запасов катехоламинов в адренергических окончаниях повышается чувствительность к адреномиметикам). Ингаляционные анестетики (хлороформ, энфлуран, галотан, изофлуран, метоксифлуран) увеличивают риск появления тяжелой предсердной и желудочковой аритмии, поскольку резко повышают чувствительность миокарда к симпатомиметикам.\u003Cbr\u003EЭргометрин, эрготамин, метилэргометрин, окситоцин, доксапрам увеличивают выраженность вазоконстрикторного эффекта.\u003Cbr\u003EСнижает антиангинальный эффект нитратов, которые, в свою очередь, могут снизить прессорный эффект симпатомиметиков и риск возникновения артериальной гипотензии (одновременное применение возможно в зависимости от достижения необходимого терапевтического эффекта).\u003Cbr\u003EТиреоидные гормоны увеличивают (взаимно) эффект и связанный с ним риск возникновения коронарной недостаточности (особенно при коронарном атеросклерозе)."},{"name":"Регистрационный номер","value":"ЛП-004206"},{"name":"Дата государственной регистрации","value":"21.03.2017"},{"name":"Владелец регистрационного удостоверения","value":"Дальхимфарм","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313","7893318:13877405"]}}},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Мезатон","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["17796364:18017750"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"2295457930010299002":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"кровеносные сосуды, сердце"},{"name":"Назначение","value":"артериальная гипотония, острая сердечно-сосудистая недостаточность, шок различного генеза"},{"name":"Показания к применению","value":"Парентерально:\u003Cbr\u003E— артериальная гипотензия;\u003Cbr\u003E— шоковые состояния (в т.ч. травматический, токсический);\u003Cbr\u003E— сосудистая недостаточность (в т.ч. на фоне передозировки вазодилататоров);\u003Cbr\u003E— в качестве вазоконстриктора при проведении местной анестезии.\u003Cbr\u003EИнтраназально:\u003Cbr\u003E— вазомоторный и аллергический ринит."},{"name":"Противопоказания","value":"— повышенная чувствительность к препарату;\u003Cbr\u003E— гипертрофическая обструктнвная кардиомиопатия;\u003Cbr\u003E— феохромоцитома;\u003Cbr\u003E— фибрилляция желудочков.\u003Cbr\u003EС осторожностью:\u003Cbr\u003EМетаболический ацидоз, гиперкапния, гипоксия, фибрилляция предсердий, закрытоугольная глаукома, артериальная гипертензия, гипертензия в малом круге кровообращения, гиповолемия, тяжелый стеноз устья аорты, острый инфаркт миокарда, тахиаритмия, желудочковая аритмия, окклюзионные заболевания сосудов (в т.ч. в анамнезе) - артериальная тромбоэмболия, атеросклероз, облитерирующий тромбангиит (болезнь Бюргера), болезнь Рейно, склонность сосудов к спазмам (в т.ч. при отморожении), диабетический эндартериит, тиреотоксикоз, сахарный диабет, порфирия, дефицит глюкозо-6-фосфатдегидрогеназы, совместное применение ингибиторов моноаминоксидазы, при общем наркозе (фторотановый), нарушениях функции почек, пожилой возраст, возраст до 18 лет (эффективность и безопасность не установлены)."},{"name":"Состав","value":"Действующее вещество: фенилэфрина гидрохлорид 10 мг."},{"name":"Действующее вещество","value":"Фенилэфрин"},{"name":"Способ применения и дозы","value":"Внутривенно медленно, при коллапсе - 0,1-0,3-0,5 мл 1% раствора, разведя в 20 мл 5% раствора декстрозы или 0,9% раствора натрия хлорида. При необходимости введение повторяют.\u003Cbr\u003EВнутривенно капельно - 1 мл 1% раствора в 250-500 мл 5% раствора декстрозы.\u003Cbr\u003EПодкожно или внутримышечно, взрослым - 0,3-1 мл 1% раствора 2-3 раза в день; детям старше 15 лет при артериальной гипотензии во время спинномозговой анестезии - 0,5-1 мг/кг.\u003Cbr\u003EДля сужения сосудов слизистых оболочек и уменьшения воспалительных явлений смазывают или закапывают(концентрации раствора - 0,125%, 0,25%, 0,5%, 1%).\u003Cbr\u003EПри местной анестезии добавляют по 0,3-0,5 мл 1% раствора на 10 мл раствора анестетика.\u003Cbr\u003EВысшие дозы для взрослых: подкожно и внутримышечно: разовая - 10 мг, суточная - 50 мг; внутривенно: разовая - 5 мг, суточная - 25 мг."},{"name":"Побочные действия","value":"Со стороны сердечно-сосудистой системы: повышение артериального давления, сердцебиение, фибрилляция желудочков сердца, аритмия, брадикардия, кардиалгия.\u003Cbr\u003EСо стороны ЦНС: головокружение, чувство страха, бессонница, беспокойство, слабость, головная боль, тремор, парестезии, судороги, кровоизлияние в мозг.\u003Cbr\u003EПрочие: бледность кожи лица, ишемия кожи в месте инъекции, в единичных случаях возможны некроз и образование струпа при попадании в ткани или при подкожных инъекциях, аллергические реакции."},{"name":"Фармакологическое действие","value":"Альфа1-адреностимулятор, мало влияющий на бета-адренорецепторы сердца; не является катехоламином (содержит лишь одну гидроксильную гpyппy в ароматическом ядре). Вызывает сужение артериол и повышение артериального давления (с возможной рефлекторной брадикардией). По сравнению с норэпинефрином и эпинефрином менее резко повышает артериальное давление, но действует более длительно (слабее подвержен действию катехол-О-метилтрансферазы); не вызывает увеличения минутного объема крови.\u003Cbr\u003EДействие начинается сразу после введения и продолжается в течение 5-20 мин (после внутривенного введения), 50 мин (при подкожном введении), 1-2 ч (после внутримышечного введения)."},{"name":"Фармакологическая группа","value":"альфа-адреномиметики"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"Хранить в сухом, защищенном от света и недоступном для детей месте при температуре не выше 25 °С."},{"name":"Передозировка","value":"Симптомы: желудочковая экстрасистолия, короткие пароксизмы желудочковой тахикардии, ощущение тяжести в голове и конечностях, значительное повышение АД.\u003Cbr\u003EЛечение: внутривенное введение альфа-адреноблокаторов (фентоламин) и бета-адреноблокаторов (при нарушениях сердечного ритма)."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения необходимо воздержаться от управления транспортными средствами и занятий потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"В период лечения следует контролировать показатели ЭКГ, АД, минутного объема крови, кровообращение в конечностях и в месте инъекции.\u003Cbr\u003EУ больных с артериальной гипертензией в случае медикаментозного коллапса достаточно поддерживать систолическое артериальное давление на уровне, ниже привычного на 30-40 мм рт.ст.\u003Cbr\u003EПеред началом или во время терапии шоковых состояний обязательна коррекция гиповолемии, гипоксии, ацидоза и гиперкапнии.\u003Cbr\u003EРезкое повышение артериального давления, выраженная брадикардия или тахикардия, стойкие нарушения ритма сердца требуют прекращения лечения.\u003Cbr\u003EДля предотвращения повторного снижения АД после отмены препарата дозу следует уменьшать постепенно, особенно после длительной инфузии.\u003Cbr\u003EИнфузию возобновляют, если систолическое артериальное давление снижается до 70-80 мм рт.ст.\u003Cbr\u003EСледует иметь в виду, что использование вазоконстрикторов во время родов для коррекции артериальной гипотензии или в качестве добавок к местным анестетикам па фоне средств, стимулирующих родовую деятельность (вазопрессина, эрготамина, эргометрина, метилэргометрина), может повлечь стойкое повышение артериального давления в послеродовом периоде.\u003Cbr\u003EС возрастом снижается количество адренорецепторов, чувствительных к фенилэфрину. Ингибиторы моноаминоксидазы, повышая прессорный эффект симпатомиметиков, могут обусловливать возникновение головных болей, аритмии, рвоты, гипертонического криза, поэтому при приеме пациентами ингибиторов моноаминоксидазы в предшествующие 2-3 недели дозы симпатомиметиков должны быть снижены."},{"name":"Взаимодействие","value":"Мезатон снижает антигипертензивный эффект диуретиков и антигипертензивных лекарственных средств (метилдопы, мекамиламина, гуанадрела, гуанетидина).\u003Cbr\u003EФенотиазины, альфа-адреноблокаторы (фентоламин), фуросемид и прочие диуретики снижают гинертензивный эффект.\u003Cbr\u003EИнгибиторы моноаминоксидазы (фуразолидон, прокарбазин, селегилин), окситоцин, алкалоиды спорыньи, трициклические антидепрессанты, метилфенидат, адреностимуляторы усиливают прессорный эффект и аритмогенность фенилэфрина.\u003Cbr\u003EБета-адреноблокаторы уменьшают кардиостимулирующую активность, на фоне резерпина - возможна артериальная гипертензия (в результате истощения запасов катехоламинов в адренергических окончаниях повышается чувствительность к адреномиметикам). Ингаляционные анестетики (хлороформ, энфлуран, галотан, изофлуран, метоксифлуран) увеличивают риск появления тяжелой предсердной и желудочковой аритмии, поскольку резко повышают чувствительность миокарда к симпатомиметикам.\u003Cbr\u003EЭргометрин, эрготамин, метилэргометрин, окситоцин, доксапрам увеличивают выраженность вазоконстрикторного эффекта.\u003Cbr\u003EСнижает антиангинальный эффект нитратов, которые, в свою очередь, могут снизить прессорный эффект симпатомиметиков и риск возникновения артериальной гипотензии (одновременное применение возможно в зависимости от достижения необходимого терапевтического эффекта).\u003Cbr\u003EТиреоидные гормоны увеличивают (взаимно) эффект и связанный с ним риск возникновения коронарной недостаточности (особенно при коронарном атеросклерозе)."},{"name":"Регистрационный номер","value":"ЛП-004206"},{"name":"Дата государственной регистрации","value":"21.03.2017"},{"name":"Владелец регистрационного удостоверения","value":"Дальхимфарм"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Мезатон"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_5"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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Еще может подойти

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Инструкция

Показания к применению

Парентерально:
— артериальная гипотензия;
— шоковые состояния (в т.ч. травматический, токсический);
— сосудистая недостаточность (в т.ч. на фоне передозировки вазодилататоров);
— в качестве вазоконстриктора при проведении местной анестезии.
Интраназально:
— вазомоторный и аллергический ринит.

Противопоказания

— повышенная чувствительность к препарату;
— гипертрофическая обструктнвная кардиомиопатия;
— феохромоцитома;
— фибрилляция желудочков.
С осторожностью:
Метаболический ацидоз, гиперкапния, гипоксия, фибрилляция предсердий, закрытоугольная глаукома, артериальная гипертензия, гипертензия в малом круге кровообращения, гиповолемия, тяжелый стеноз устья аорты, острый инфаркт миокарда, тахиаритмия, желудочковая аритмия, окклюзионные заболевания сосудов (в т.ч. в анамнезе) - артериальная тромбоэмболия, атеросклероз, облитерирующий тромбангиит (болезнь Бюргера), болезнь Рейно, склонность сосудов к спазмам (в т.ч. при отморожении), диабетический эндартериит, тиреотоксикоз, сахарный диабет, порфирия, дефицит глюкозо-6-фосфатдегидрогеназы, совместное применение ингибиторов моноаминоксидазы, при общем наркозе (фторотановый), нарушениях функции почек, пожилой возраст, возраст до 18 лет (эффективность и безопасность не установлены).

Способ применения и дозы

Внутривенно медленно, при коллапсе - 0,1-0,3-0,5 мл 1% раствора, разведя в 20 мл 5% раствора декстрозы или 0,9% раствора натрия хлорида. При необходимости введение повторяют.
Внутривенно капельно - 1 мл 1% раствора в 250-500 мл 5% раствора декстрозы.
Подкожно или внутримышечно, взрослым - 0,3-1 мл 1% раствора 2-3 раза в день; детям старше 15 лет при артериальной гипотензии во время спинномозговой анестезии - 0,5-1 мг/кг.
Для сужения сосудов слизистых оболочек и уменьшения воспалительных явлений смазывают или закапывают(концентрации раствора - 0,125%, 0,25%, 0,5%, 1%).
При местной анестезии добавляют по 0,3-0,5 мл 1% раствора на 10 мл раствора анестетика.
Высшие дозы для взрослых: подкожно и внутримышечно: разовая - 10 мг, суточная - 50 мг; внутривенно: разовая - 5 мг, суточная - 25 мг.
Полная инструкция
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Мезатон р-р д/ин. . амп.
Мезатон р-р д/ин. . амп., 10 мг/мл, 1 мл, 10 шт.
У продавца: 
нет • На Маркете: 4.8
(12)
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Инструкция

113 ₽

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  • Фуросемид р-р для в/в введ. и в/м введ. амп., 10 мг/мл, 2 мл, 10 шт.
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  • Викасол р-р для в/м введ. введ., 10 мг/мл, 1 мл, 10 шт.
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  • Пентоксифиллин р-р д/ин. амп., 20 мг/мл, 5 мл, 10 шт.
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  • Кальция хлорид р-р для в/в введ. введ., 100 мг/мл, 10 мл, 10 шт.
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  • Стелфрин р-р д/ин. амп., 10 мг/мл, 1 мл, 10 шт.
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  • {"widgets":{"@yandex-market/LazyLoader-market":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator":{"widgetName":"@marketfront/RecomLayout","widgetId":"ServerListRendererForSerp_RecommendationRoll","options":{"resolverParams":{"resources":{"garsons":[{"count":24,"limit":24,"params":{"cartProductIds":[],"snippetTypes":["product","product-block","category-block","advertisement","media-incut","promo-trigger","media-adv-banner-single","media-adv-banner-double","media-adv-carousel"],"program":"remix_desktop_model_card","hyperid":"1778174037"},"id":"RemixData"}],"shuffle":{"mode":"exclusive"}},"limit":24},"id":"RecommendationRoll","slotOptions":{"dynamic":true},"className":"","needToProvideData":true,"wrapperProps":{},"widgetOptions":{"config":{"pictureBlock":{"maxGalleryImagesCount":5},"descriptionBlock":{"order":1,"titleRowCount":"2"},"offerBlock":{"withGreenPrice":true,"order":2,"price":{"wrap":true,"overflow":"hidden"}}},"galleryImageSize":250},"layoutOptions":{"needFallbackOnError":true,"needFallbackOnEmpty":false,"countInRows":6},"isChefRemixExp":false},"slotOptions":{"dynamic":true},"placeholder":"Invisible","infinite":true,"cspNonce":"yYGQp2RgLj9ToTcUF94Fyw==","renderStrategy":"append","renderedOnce":true}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator":{"name":"@yandex-market/LazyLoader-market"}}}
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