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Описание

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Моксонидин-СЗ таб. п/о плен., 0.3 мг, 28 шт.

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Дозировка: 0.3 мг

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Количество штук в упаковке, шт.: 28

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Коротко о товаре

Инструкция
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;\u003Cbr\u003E- выраженная брадикардия (частота сердечных сокращений покоя менее 50 уд/мин); ;\u003Cbr\u003E- атриовентрикулярная блокада II и III степени; ;\u003Cbr\u003E- выраженные нарушения ритма сердца; ;\u003Cbr\u003E- острая и хроническая сердечная недостаточность (III-IV функциональный класс по классификации NYHA); ;\u003Cbr\u003E- одновременное применение с трициклическими антидепрессантами (см. раздел \"Взаимодействие с другими лекарственными препаратами\");;\u003Cbr\u003E- тяжелая почечная недостаточность (КК менее 30 мл/мин); ;\u003Cbr\u003E- гемодиализ; ;\u003Cbr\u003E- период лактации; ;\u003Cbr\u003E- наследственная непереносимость лактозы, дефицит лактазы или мальабсорбция глюкозы-галактозы; ;\u003Cbr\u003E- возраст старше 75 лет; ;\u003Cbr\u003E- возраст до 18 лет (в связи с отсутствием данных по безопасности и эффективности)."},{"name":"Состав","value":"1 таблетка, покрытая пленочной оболочкой, содержит:\u003Cbr\u003Eдозировка 0,2 мг:\u003Cbr\u003Eдействующее вещество: моксонидин - 0,2 мг\u003Cbr\u003Eвспомогательные вещества (ядро): кроскармеллоза натрия (примеллоза) -19,5 мг; лактозы моногидрат (лактопресс)(сахар молочный) - 47,7 мг; целлюлоза микрокристаллическая 102-25,0 мг; повидон К30 (поливинилпирролидон среднемолекулярный) - 6,2 мг; кремния диоксид коллоидный (аэросил) - 0,4 мг; натрия стеарилфумарат - 1,0 мг;\u003Cbr\u003Eвспомогательные вещества (оболочка): гипромеллоза - 1,60 мг; полисорбат-80 (твин-80) - 0,46 мг; тальк - 0,45 мг; титана диоксид Е171 - 0,488 мг; алюминиевый лак на основе красителя кармуазин - 0,002 мг.\u003Cbr\u003Eдозировка 0,3 мг:\u003Cbr\u003Eдействующее вещество: моксонидин - 0,3 мг\u003Cbr\u003Eвспомогательные вещества (ядро): кроскармеллоза натрия (примеллоза) - 19,5 мг; лактозы моногидрат (лактопресс) (сахар молочный) - 47,6 мг; целлюлоза микрокристаллическая 102 - 25,0 мг; повидон К30 (поливинилпирролидон среднемолекулярный) - 6,2 мг; кремния диоксид коллоидный (аэросил) - 0,4 мг; натрия стеарилфумарат - 1,0 мг;\u003Cbr\u003Eвспомогательные вещества (оболочка): гипромеллоза - 1,60 мг; полисорбат-80 (твин-80) - 0,64 мг; тальк - 0,45 мг; титана диоксид Е171 - 0,30 мг; алюминиевый лак на основе красителя кармуазин - 0,01 мг.\u003Cbr\u003Eдозировка 0,4 мг:\u003Cbr\u003Eдействующее вещество: моксонидин - 0,4 мг\u003Cbr\u003Eвспомогательные вещества (ядро): кроскармеллоза натрия (примеллоза) - 19,5 мг; лактозы моногидрат (лактопресс) (сахар молочный) - 47,5 мг; целлюлоза микрокристаллическая 102 - 25,0 мг; повидон К30 (поливинилпирролидон среднемолекулярный) - 6,2 мг; кремния диоксид коллоидный (аэросил) - 0,4 мг; натрия стеарилфумарат - 1,0 мг;\u003Cbr\u003Eвспомогательные вещества (оболочка): гипромеллоза - 1,60 мг; полисорбат-80 (твин-80) - 0,64 мг; тальк - 0,45 мг; титана диоксид Е171 - 0,29 мг; алюминиевый лак на основе красителя кармуазин - 0,02 мг."},{"name":"Действующее вещество","value":"Моксонидин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28709517"]}}},{"name":"Способ применения и дозы","value":"Внутрь, независимо от приема пищи.\u003Cbr\u003EВ большинстве случаев начальная доза препарата Моксонидин-СЗ составляет 0,2 мг в сутки. Максимальная разовая доза составляет 0,4 мг. Максимальная суточная доза, которую следует разделить на 2 приема, составляет 0,6 мг. Необходима индивидуальная коррекция суточной дозы в зависимости от переносимости пациентом проводимой терапии.\u003Cbr\u003EКоррекция дозы для пациентов с печеночной недостаточностью не требуется. Начальная доза для пациентов с умеренной или тяжелой почечной недостаточностью составляет 0,2 мг/сутки.\u003Cbr\u003EВ случае необходимости и при хорошей переносимости суточная доза может быть увеличена до максимальной 0,4 мг.\u003Cbr\u003EПациентам с почечной недостаточностью рекомендуется осторожный подбор дозы, особенно в начале лечения. Начальная доза должна составлять 0,2 мг в сутки. В случае необходимости и при хорошей переносимости суточная доза препарата может быть увеличена максимум до 0,4 мг для пациентов с умеренной почечной недостаточностью (КК более 30 мл/мин, но менее 60 мл/мин) и 0,3 мг для пациентов с тяжелой почечной недостаточностью (КК менее 30 мл/мин)."},{"name":"Побочные действия","value":"Наиболее частые побочные эффекты у пациентов, принимающих моксонидин: сухость во рту, головокружение, астения и сонливость. Эти симптомы часто уменьшаются по прошествии первых недель терапии.\u003Cbr\u003EУ пациентов, принимавших участие в плацебо-контролируемых клинических исследованиях моксонидина, отмечены следующие побочные эффекты.\u003Cbr\u003EЧастота побочных эффектов, приведенных ниже, определялась соответственно следующему: очень часто (\u003E1/10); часто (\u003E1/100, \u003C1/10); нечасто (\u003E1/1000, \u003C1/100); включая отдельные сообщения. \u003Cbr\u003EСо стороны центральной нервной системы:\u003Cbr\u003EЧасто: головная боль*, головокружение (вертиго), сонливость. \u003Cbr\u003EНечасто: обморок*.\u003Cbr\u003EСо стороны сердечно-сосудистой системы: \u003Cbr\u003EНечасто: выраженное снижение АД, ортостатическая гипотензия*, брадикардия. \u003Cbr\u003EСо стороны желудочно-кишечного тракта: \u003Cbr\u003EОчень часто: сухость слизистой оболочки полости рта. \u003Cbr\u003EЧасто: диарея, тошнота, рвота, диспепсия. \u003Cbr\u003EСо стороны кожи и подкожных тканей: \u003Cbr\u003EЧасто: кожная сыпь, зуд. \u003Cbr\u003EНечасто: ангионевротический отек. \u003Cbr\u003EНарушения психики: \u003Cbr\u003EЧасто: бессонница. \u003Cbr\u003EНечасто: нервозность. \u003Cbr\u003EСо стороны органа слуха и лабиринтные нарушения: \u003Cbr\u003EНечасто: звон в ушах. \u003Cbr\u003EСо стороны скелетно-мышечной и соединительной ткани: \u003Cbr\u003EЧасто: боль в спине. \u003Cbr\u003EНечасто: боль в области шеи. \u003Cbr\u003EОбщие расстройства и нарушения в месте введения: \u003Cbr\u003EЧасто: астения. \u003Cbr\u003EНечасто: периферические отеки. \u003Cbr\u003E(* - частота сопоставима с плацебо)."},{"name":"Фармакологическое действие","value":"Моксонидин является гипотензивным средством с центральным механизмом действия. В стволовых структурах мозга (ростральный слой боковых желудочков) моксонидин селективно стимулирует имидазолин-чувствительные рецепторы, принимающие участие в тонической и рефлекторной регуляции симпатической нервной системы. Стимуляция имидазолиновых рецепторов снижает периферическую симпатическую активность и артериальное давление (АД).\u003Cbr\u003EМоксонидин отличается от других симпатолитических гипотензивных средств более низким сродством к α2-адренорецепторам, что объясняет меньшую вероятность развития седативного эффекта и сухости во рту.\u003Cbr\u003EПрием моксонидина приводит к снижению системного сосудистого сопротивления и АД.\u003Cbr\u003EМоксонидин улучшает на 21% индекс чувствительности к инсулину (в сравнении с плацебо) у пациентов с ожирением, инсулинрезистентностью и умеренной степенью артериальной гипертензии."},{"name":"Фармакологическая группа","value":"гипотензивное средство центрального действия"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"В защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Имеются сообщения о нескольких случаях передозировки без летального исхода, когда одномоментно применялись дозы до 19,6 мг. \u003Cbr\u003EСимптомы: головная боль, седативный эффект, выраженное снижение АД, головокружение, астения, брадикардия, сухость слизистой оболочки полости рта, рвота, повышенная утомляемость, боль в эпигастральной области, угнетение дыхания и нарушение сознания. Кроме того, возможны также кратковременное повышение АД, тахикардия и гипергликемия, как было показано в нескольких исследованиях по изучению высоких доз на животных. \u003Cbr\u003EЛечение\u003Cbr\u003EСпецифического антидота не существует. В случае выраженного снижения АД может потребоваться восстановление объема циркулирующей крови за счет введения жидкости и допамина (инъекционно). \u003Cbr\u003EБрадикардия может быть купирована атропином (инъекционное введение). \u003Cbr\u003EВ тяжелых случаях передозировки рекомендуется тщательно контролировать нарушения сознания и не допускать угнетения дыхания. \u003Cbr\u003EАнтагонисты альфа-адренорецепторов могут уменьшать или устранять парадоксальные гипертензивные эффекты при передозировке моксонидином. \u003Cbr\u003E"},{"name":"Применение при беременности и кормлении грудью","value":"Клинические данные о применении Моксонидина-СЗ у беременных отсутствуют. В ходе исследований на животных было установлено эмбриотоксическое действие препарата.\u003Cbr\u003EМоксонидин-СЗ следует назначать беременным, только после тщательной оценки соотношения риска и пользы, когда польза для матери превышает потенциальный риск для плода.\u003Cbr\u003EПериод лактации\u003Cbr\u003EМоксонидин-СЗ проникает в грудное молоко и поэтому не должен назначаться во время кормления грудью. \u003Cbr\u003EМоксонидин-СПри необходимости применения Моксонидина-СЗ в период лактации, грудное вскармливание необходимо прекратить."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Исследования влияния препарата на способность управлять автомобилем и другими механизмами не проводились. Имеются сообщения о сонливости и головокружении в период лечения моксонидином. Это следует учитывать при выполнении вышеуказанных действий."},{"name":"Особые указания","value":"Во время лечения необходим регулярный контроль АД.\u003Cbr\u003E\n\u003Cbr\u003E\nВ постмаркетинговом наблюдении зафиксированы случаи атриовентрикулярной блокады различной степени тяжести у пациентов, принимающих моксонидин. Связь между приемом препарата Моксонидин-СЗ и замедлением атриовентрикулярной проводимости не может быть полностью исключена. Таким образом, при лечении пациентов с вероятной предрасположенностью к развитию атриовентрикулярной блокады рекомендуется соблюдать осторожность.\u003Cbr\u003E\n\u003Cbr\u003E\nПри необходимости отмены одновременного принимаемых бета-адреноблокаторов и препарата Моксонидин-СЗ сначала отменяют бета-адреноблокаторы и лишь через несколько дней Моксонидин-СЗ.\u003Cbr\u003E\n\u003Cbr\u003E\nВ настоящее время нет подтверждений того, что прекращение приема препарата Моксонидин-СЗ приводит к повышению АД.\u003Cbr\u003E\n\u003Cbr\u003E\nОднако не рекомендуется прекращать прием препарата Моксонидин-СЗ резко, вместо этого следует постепенно уменьшать дозу препарата в течении двух недель.\u003Cbr\u003E\n\u003Cbr\u003E\nУ пациентов пожилого возраста может быть повышен риск развития сердечно-сосудистых осложнений вследствие применения гипотензивных препаратов, поэтому терапию препаратом Моксонидин-СЗ следует начинать с минимальной дозы."},{"name":"Взаимодействие","value":"Совместное применение моксонидина с другими гипотензивными средствами приводит к аддитивному эффекту.\u003Cbr\u003EТрициклические антидепрессанты могут снижать эффективность гипотензивных средств центрального действия, в связи с чем не рекомендуется их прием совместно с моксонидином.\u003Cbr\u003EМоксонидин может усиливать действие трициклических антидепрессантов, транквилизаторов, этанола, седативных и снотворных средств. .\u003Cbr\u003EМоксонидин способен умеренно улучшать ослабленные когнитивные функции у пациентов, получающих лоразепам.\u003Cbr\u003EМоксонидин может усиливать седативный эффект производных бензодиазепина при их одновременном назначении.\u003Cbr\u003EМоксонидин выделяется путем канальцевой секреции. Поэтому не исключено его взаимодействие с другими препаратами, выделяющимися путем канальцевой секреции."},{"name":"Регистрационный номер","value":"ЛП-002321"},{"name":"Дата государственной регистрации","value":"11.01.2023"},{"name":"Владелец регистрационного удостоверения","value":"Северная Звезда","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313","7893318:16002862"]}}},{"name":"Изготовитель","value":"Северная Звезда"},{"name":"Фасовщик","value":"Северная Звезда"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Моксонидин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["17796364:17893175"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"11834337183523510350":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"кровеносная система, кровеносные сосуды, сердце"},{"name":"Назначение","value":"артериальная гипертензия, гипертония, нормализация артериального давления, эссенциальная гипертензия"},{"name":"Показания к применению","value":"Артериальная гипертензия."},{"name":"Противопоказания","value":"- Повышенная чувствительность к активному веществу и другим компонентам препарата;\u003Cbr\u003E- синдром слабости синусового узла; ;\u003Cbr\u003E- выраженная брадикардия (частота сердечных сокращений покоя менее 50 уд/мин); ;\u003Cbr\u003E- атриовентрикулярная блокада II и III степени; ;\u003Cbr\u003E- выраженные нарушения ритма сердца; ;\u003Cbr\u003E- острая и хроническая сердечная недостаточность (III-IV функциональный класс по классификации NYHA); ;\u003Cbr\u003E- одновременное применение с трициклическими антидепрессантами (см. раздел \"Взаимодействие с другими лекарственными препаратами\");;\u003Cbr\u003E- тяжелая почечная недостаточность (КК менее 30 мл/мин); ;\u003Cbr\u003E- гемодиализ; ;\u003Cbr\u003E- период лактации; ;\u003Cbr\u003E- наследственная непереносимость лактозы, дефицит лактазы или мальабсорбция глюкозы-галактозы; ;\u003Cbr\u003E- возраст старше 75 лет; ;\u003Cbr\u003E- возраст до 18 лет (в связи с отсутствием данных по безопасности и эффективности)."},{"name":"Состав","value":"1 таблетка, покрытая пленочной оболочкой, содержит:\u003Cbr\u003Eдозировка 0,2 мг:\u003Cbr\u003Eдействующее вещество: моксонидин - 0,2 мг\u003Cbr\u003Eвспомогательные вещества (ядро): кроскармеллоза натрия (примеллоза) -19,5 мг; лактозы моногидрат (лактопресс)(сахар молочный) - 47,7 мг; целлюлоза микрокристаллическая 102-25,0 мг; повидон К30 (поливинилпирролидон среднемолекулярный) - 6,2 мг; кремния диоксид коллоидный (аэросил) - 0,4 мг; натрия стеарилфумарат - 1,0 мг;\u003Cbr\u003Eвспомогательные вещества (оболочка): гипромеллоза - 1,60 мг; полисорбат-80 (твин-80) - 0,46 мг; тальк - 0,45 мг; титана диоксид Е171 - 0,488 мг; алюминиевый лак на основе красителя кармуазин - 0,002 мг.\u003Cbr\u003Eдозировка 0,3 мг:\u003Cbr\u003Eдействующее вещество: моксонидин - 0,3 мг\u003Cbr\u003Eвспомогательные вещества (ядро): кроскармеллоза натрия (примеллоза) - 19,5 мг; лактозы моногидрат (лактопресс) (сахар молочный) - 47,6 мг; целлюлоза микрокристаллическая 102 - 25,0 мг; повидон К30 (поливинилпирролидон среднемолекулярный) - 6,2 мг; кремния диоксид коллоидный (аэросил) - 0,4 мг; натрия стеарилфумарат - 1,0 мг;\u003Cbr\u003Eвспомогательные вещества (оболочка): гипромеллоза - 1,60 мг; полисорбат-80 (твин-80) - 0,64 мг; тальк - 0,45 мг; титана диоксид Е171 - 0,30 мг; алюминиевый лак на основе красителя кармуазин - 0,01 мг.\u003Cbr\u003Eдозировка 0,4 мг:\u003Cbr\u003Eдействующее вещество: моксонидин - 0,4 мг\u003Cbr\u003Eвспомогательные вещества (ядро): кроскармеллоза натрия (примеллоза) - 19,5 мг; лактозы моногидрат (лактопресс) (сахар молочный) - 47,5 мг; целлюлоза микрокристаллическая 102 - 25,0 мг; повидон К30 (поливинилпирролидон среднемолекулярный) - 6,2 мг; кремния диоксид коллоидный (аэросил) - 0,4 мг; натрия стеарилфумарат - 1,0 мг;\u003Cbr\u003Eвспомогательные вещества (оболочка): гипромеллоза - 1,60 мг; полисорбат-80 (твин-80) - 0,64 мг; тальк - 0,45 мг; титана диоксид Е171 - 0,29 мг; алюминиевый лак на основе красителя кармуазин - 0,02 мг."},{"name":"Действующее вещество","value":"Моксонидин"},{"name":"Способ применения и дозы","value":"Внутрь, независимо от приема пищи.\u003Cbr\u003EВ большинстве случаев начальная доза препарата Моксонидин-СЗ составляет 0,2 мг в сутки. Максимальная разовая доза составляет 0,4 мг. Максимальная суточная доза, которую следует разделить на 2 приема, составляет 0,6 мг. Необходима индивидуальная коррекция суточной дозы в зависимости от переносимости пациентом проводимой терапии.\u003Cbr\u003EКоррекция дозы для пациентов с печеночной недостаточностью не требуется. Начальная доза для пациентов с умеренной или тяжелой почечной недостаточностью составляет 0,2 мг/сутки.\u003Cbr\u003EВ случае необходимости и при хорошей переносимости суточная доза может быть увеличена до максимальной 0,4 мг.\u003Cbr\u003EПациентам с почечной недостаточностью рекомендуется осторожный подбор дозы, особенно в начале лечения. Начальная доза должна составлять 0,2 мг в сутки. В случае необходимости и при хорошей переносимости суточная доза препарата может быть увеличена максимум до 0,4 мг для пациентов с умеренной почечной недостаточностью (КК более 30 мл/мин, но менее 60 мл/мин) и 0,3 мг для пациентов с тяжелой почечной недостаточностью (КК менее 30 мл/мин)."},{"name":"Побочные действия","value":"Наиболее частые побочные эффекты у пациентов, принимающих моксонидин: сухость во рту, головокружение, астения и сонливость. Эти симптомы часто уменьшаются по прошествии первых недель терапии.\u003Cbr\u003EУ пациентов, принимавших участие в плацебо-контролируемых клинических исследованиях моксонидина, отмечены следующие побочные эффекты.\u003Cbr\u003EЧастота побочных эффектов, приведенных ниже, определялась соответственно следующему: очень часто (\u003E1/10); часто (\u003E1/100, \u003C1/10); нечасто (\u003E1/1000, \u003C1/100); включая отдельные сообщения. \u003Cbr\u003EСо стороны центральной нервной системы:\u003Cbr\u003EЧасто: головная боль*, головокружение (вертиго), сонливость. \u003Cbr\u003EНечасто: обморок*.\u003Cbr\u003EСо стороны сердечно-сосудистой системы: \u003Cbr\u003EНечасто: выраженное снижение АД, ортостатическая гипотензия*, брадикардия. \u003Cbr\u003EСо стороны желудочно-кишечного тракта: \u003Cbr\u003EОчень часто: сухость слизистой оболочки полости рта. \u003Cbr\u003EЧасто: диарея, тошнота, рвота, диспепсия. \u003Cbr\u003EСо стороны кожи и подкожных тканей: \u003Cbr\u003EЧасто: кожная сыпь, зуд. \u003Cbr\u003EНечасто: ангионевротический отек. \u003Cbr\u003EНарушения психики: \u003Cbr\u003EЧасто: бессонница. \u003Cbr\u003EНечасто: нервозность. \u003Cbr\u003EСо стороны органа слуха и лабиринтные нарушения: \u003Cbr\u003EНечасто: звон в ушах. \u003Cbr\u003EСо стороны скелетно-мышечной и соединительной ткани: \u003Cbr\u003EЧасто: боль в спине. \u003Cbr\u003EНечасто: боль в области шеи. \u003Cbr\u003EОбщие расстройства и нарушения в месте введения: \u003Cbr\u003EЧасто: астения. \u003Cbr\u003EНечасто: периферические отеки. \u003Cbr\u003E(* - частота сопоставима с плацебо)."},{"name":"Фармакологическое действие","value":"Моксонидин является гипотензивным средством с центральным механизмом действия. В стволовых структурах мозга (ростральный слой боковых желудочков) моксонидин селективно стимулирует имидазолин-чувствительные рецепторы, принимающие участие в тонической и рефлекторной регуляции симпатической нервной системы. Стимуляция имидазолиновых рецепторов снижает периферическую симпатическую активность и артериальное давление (АД).\u003Cbr\u003EМоксонидин отличается от других симпатолитических гипотензивных средств более низким сродством к α2-адренорецепторам, что объясняет меньшую вероятность развития седативного эффекта и сухости во рту.\u003Cbr\u003EПрием моксонидина приводит к снижению системного сосудистого сопротивления и АД.\u003Cbr\u003EМоксонидин улучшает на 21% индекс чувствительности к инсулину (в сравнении с плацебо) у пациентов с ожирением, инсулинрезистентностью и умеренной степенью артериальной гипертензии."},{"name":"Фармакологическая группа","value":"гипотензивное средство центрального действия"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"Имеются сообщения о нескольких случаях передозировки без летального исхода, когда одномоментно применялись дозы до 19,6 мг. \u003Cbr\u003EСимптомы: головная боль, седативный эффект, выраженное снижение АД, головокружение, астения, брадикардия, сухость слизистой оболочки полости рта, рвота, повышенная утомляемость, боль в эпигастральной области, угнетение дыхания и нарушение сознания. Кроме того, возможны также кратковременное повышение АД, тахикардия и гипергликемия, как было показано в нескольких исследованиях по изучению высоких доз на животных. \u003Cbr\u003EЛечение\u003Cbr\u003EСпецифического антидота не существует. В случае выраженного снижения АД может потребоваться восстановление объема циркулирующей крови за счет введения жидкости и допамина (инъекционно). \u003Cbr\u003EБрадикардия может быть купирована атропином (инъекционное введение). \u003Cbr\u003EВ тяжелых случаях передозировки рекомендуется тщательно контролировать нарушения сознания и не допускать угнетения дыхания. \u003Cbr\u003EАнтагонисты альфа-адренорецепторов могут уменьшать или устранять парадоксальные гипертензивные эффекты при передозировке моксонидином. \u003Cbr\u003E"},{"name":"Применение при беременности и кормлении грудью","value":"Клинические данные о применении Моксонидина-СЗ у беременных отсутствуют. В ходе исследований на животных было установлено эмбриотоксическое действие препарата.\u003Cbr\u003EМоксонидин-СЗ следует назначать беременным, только после тщательной оценки соотношения риска и пользы, когда польза для матери превышает потенциальный риск для плода.\u003Cbr\u003EПериод лактации\u003Cbr\u003EМоксонидин-СЗ проникает в грудное молоко и поэтому не должен назначаться во время кормления грудью. \u003Cbr\u003EМоксонидин-СПри необходимости применения Моксонидина-СЗ в период лактации, грудное вскармливание необходимо прекратить."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Исследования влияния препарата на способность управлять автомобилем и другими механизмами не проводились. Имеются сообщения о сонливости и головокружении в период лечения моксонидином. Это следует учитывать при выполнении вышеуказанных действий."},{"name":"Особые указания","value":"Во время лечения необходим регулярный контроль АД.\u003Cbr\u003E\n\u003Cbr\u003E\nВ постмаркетинговом наблюдении зафиксированы случаи атриовентрикулярной блокады различной степени тяжести у пациентов, принимающих моксонидин. Связь между приемом препарата Моксонидин-СЗ и замедлением атриовентрикулярной проводимости не может быть полностью исключена. Таким образом, при лечении пациентов с вероятной предрасположенностью к развитию атриовентрикулярной блокады рекомендуется соблюдать осторожность.\u003Cbr\u003E\n\u003Cbr\u003E\nПри необходимости отмены одновременного принимаемых бета-адреноблокаторов и препарата Моксонидин-СЗ сначала отменяют бета-адреноблокаторы и лишь через несколько дней Моксонидин-СЗ.\u003Cbr\u003E\n\u003Cbr\u003E\nВ настоящее время нет подтверждений того, что прекращение приема препарата Моксонидин-СЗ приводит к повышению АД.\u003Cbr\u003E\n\u003Cbr\u003E\nОднако не рекомендуется прекращать прием препарата Моксонидин-СЗ резко, вместо этого следует постепенно уменьшать дозу препарата в течении двух недель.\u003Cbr\u003E\n\u003Cbr\u003E\nУ пациентов пожилого возраста может быть повышен риск развития сердечно-сосудистых осложнений вследствие применения гипотензивных препаратов, поэтому терапию препаратом Моксонидин-СЗ следует начинать с минимальной дозы."},{"name":"Взаимодействие","value":"Совместное применение моксонидина с другими гипотензивными средствами приводит к аддитивному эффекту.\u003Cbr\u003EТрициклические антидепрессанты могут снижать эффективность гипотензивных средств центрального действия, в связи с чем не рекомендуется их прием совместно с моксонидином.\u003Cbr\u003EМоксонидин может усиливать действие трициклических антидепрессантов, транквилизаторов, этанола, седативных и снотворных средств. .\u003Cbr\u003EМоксонидин способен умеренно улучшать ослабленные когнитивные функции у пациентов, получающих лоразепам.\u003Cbr\u003EМоксонидин может усиливать седативный эффект производных бензодиазепина при их одновременном назначении.\u003Cbr\u003EМоксонидин выделяется путем канальцевой секреции. Поэтому не исключено его взаимодействие с другими препаратами, выделяющимися путем канальцевой секреции."},{"name":"Регистрационный номер","value":"ЛП-002321"},{"name":"Дата государственной регистрации","value":"11.01.2023"},{"name":"Владелец регистрационного удостоверения","value":"Северная Звезда"},{"name":"Изготовитель","value":"Северная Звезда"},{"name":"Фасовщик","value":"Северная Звезда"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Моксонидин"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_198702039780574641"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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Инструкция

Показания к применению

Артериальная гипертензия.

Противопоказания

- Повышенная чувствительность к активному веществу и другим компонентам препарата;
- синдром слабости синусового узла; ;
- выраженная брадикардия (частота сердечных сокращений покоя менее 50 уд/мин); ;
- атриовентрикулярная блокада II и III степени; ;
- выраженные нарушения ритма сердца; ;
- острая и хроническая сердечная недостаточность (III-IV функциональный класс по классификации NYHA); ;
- одновременное применение с трициклическими антидепрессантами (см. раздел "Взаимодействие с другими лекарственными препаратами");;
- тяжелая почечная недостаточность (КК менее 30 мл/мин); ;
- гемодиализ; ;
- период лактации; ;
- наследственная непереносимость лактозы, дефицит лактазы или мальабсорбция глюкозы-галактозы; ;
- возраст старше 75 лет; ;
- возраст до 18 лет (в связи с отсутствием данных по безопасности и эффективности).

Способ применения и дозы

Внутрь, независимо от приема пищи.
В большинстве случаев начальная доза препарата Моксонидин-СЗ составляет 0,2 мг в сутки. Максимальная разовая доза составляет 0,4 мг. Максимальная суточная доза, которую следует разделить на 2 приема, составляет 0,6 мг. Необходима индивидуальная коррекция суточной дозы в зависимости от переносимости пациентом проводимой терапии.
Коррекция дозы для пациентов с печеночной недостаточностью не требуется. Начальная доза для пациентов с умеренной или тяжелой почечной недостаточностью составляет 0,2 мг/сутки.
В случае необходимости и при хорошей переносимости суточная доза может быть увеличена до максимальной 0,4 мг.
Пациентам с почечной недостаточностью рекомендуется осторожный подбор дозы, особенно в начале лечения. Начальная доза должна составлять 0,2 мг в сутки. В случае необходимости и при хорошей переносимости суточная доза препарата может быть увеличена максимум до 0,4 мг для пациентов с умеренной почечной недостаточностью (КК более 30 мл/мин, но менее 60 мл/мин) и 0,3 мг для пациентов с тяжелой почечной недостаточностью (КК менее 30 мл/мин).
Полная инструкция
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Моксонидин-СЗ таб. п/о плен.
Моксонидин-СЗ таб. п/о плен., 0.3 мг, 28 шт.
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Инструкция

153 ₽

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4.7
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У продавца:18 оценок·5 отзывов
У всех продавцов:283 оценки·100 отзывов
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user avatar
3 месяца назад • Наталия Сорокина • Куплен на Маркете
Достоинства: это "Скорая помощь" при повышении давления.
Недостатки: резко снимать давление не рекомендуется
Комментарий: в зависимости от давления, беру дозу. В основном по половинке таблетки
user avatar
2 месяца назад • НИНА М. • Куплен на Маркете
Комментарий: цена, действие таблеток, все устраивает, покупала уже раньше. упаковка 60 таблеток тоже отлично.!
user avatar
4 месяца назад • Татьяна Иванова • Куплен на Маркете
Достоинства: Снижает давление
Недостатки: Не заметила
Комментарий: Лучше принимать ,по назначению врача !
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  • Милурит таб., 100 мг, 100 шт.
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  • Пенталгин таб. п/о плен., 24 шт.
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  • Глицин таб. подъязыч., 100 мг, 50 шт.
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  • Метформин таб., 1000 мг, 60 шт.
    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:998360039_4/content/content/toggleWishlist":{"skuId":"228004261","productId":998360039,"offerId":"FagKxhlRduDDZkmBz02OKA","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgsQt9WV7tmv2biIARIaChhyZW1peF9kZXNrdG9wX21vZGVsX2NhcmQyFQjnh4fcAxClo9xsGISpsggg3tnBBw==","sign":"S9lozuQXp/3FRIQLRgHk3HgBoDIo3qyEUbLMWiMLz2M="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:998360039_4/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Мексидол таб. п/о плен., 125 мг, 30 шт.
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    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1404748441_5/content/content/toggleWishlist":{"skuId":"227814286","productId":1404748441,"offerId":"iIgpwbogG37ZliD9Uhh9hA","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgsQt9WV7tmv2biIARIaChhyZW1peF9kZXNrdG9wX21vZGVsX2NhcmQyFQiZheudBRCO19BsGK3t/AUg7dnBBw==","sign":"z+WjM/x+WVJ3OsmJlZUWZ1NeBJHJsEhPJkvQ7aG9UnE="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1404748441_5/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Нольпаза таб. п/о плен. кш/раств., 40 мг, 14 шт.
    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1400799737_6/content/content/toggleWishlist":{"skuId":"661169004","productId":1400799737,"offerId":"fXv6gncbpCir9a5J0pFu4Q","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgsQt9WV7tmv2biIARIaChhyZW1peF9kZXNrdG9wX21vZGVsX2NhcmQyFgj5g/qbBRDsxqK7Ahi21YcEINrZwQc=","sign":"KfM2u6ZjJbmRPcZt/q3wVJnL/xSBXcnk+dEFPEWfC5w="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1400799737_6/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Парацетамол таб., 500 мг, 10 шт.
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  • {"widgets":{"@light/BannerCurtain":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_101_8/content/content/content/bannerCurtain":{"advertisementId":2110601,"impression":"/safeclick/data=SpQw45JhDGE6zDtOdUQO_D_IQ2AhH2r2VgiqFExVJ6IGvi1QmFllDe4jTHBtocvd1DIfzUb-25MlldusLA2_2EViREf3-jOk6HhGjofP_luMOXFJAvmXJZefHL0SqXgrMGw347y8-AkPly466_aiI8BkBU59o-Jvguol2-dGtBnGGtZJvRcP-rWcrSODIBfvZajyAnVbzfiQLzSwlrxTaUuWmub9hCyzIODTPoZDQy9jegIcnUvAsXlR8joulwpzbSOY4v0lbZXHbm1hgLLnrOM9zuKKEF-yucOBcvgFvtkJyN2MEZshP_Ac-cNM_v62RUwedPmGIUmib0R19CV0Orv3oEwSSVccapOCSM3vIL4aGex6rOzCqtw3BPuCnaWO20k7gP5jilWXktwvrFs_mxQwwauyvcMACOfaelnpYh3Yyf8l_8dxkqDn7NDlj4Uyi0QAUoO4Wx-zbVJrvINB8Gk-OoTm5e_3GN7q9xrDRfsz5uzuWtHKbjMqMLg_o_VExBLeZ5Q-Z9k7n-DRdrYmaZeITmEHk_jBZVodZgnyEjwDXp7clv5H7mjH3mbSJ4niuSOaCx6fL78jcU69LWB50jkCV4NJ5Q6MLJWLZz4vEm3zPJvL312fJTKMT7My2GWYutcDPo_fD_mGKwhpDg5ah7RDmWwIbKbWJqc9myRKDS3j1JFL9e_Pbw5x55oZYN0xnenxSYdgqedogFmoNL2W-VGIuYuCoNgobMJLQRzHhXDf07yv8zrTwCDzXOy7BJNTXlJ86GmmoEas0gnojpS19spxmGoy4jYCxtJC2a8D5nMRbvSOcyR79aBOJjuUSl4Lhzy0-TsZyEBWNEp4DEo4cYH_ZlL_0AErG4-WJGAMXsICXc0mt1WqfwvWWDO1mQ1wDA2HaLto1Jzqbe0J2_C0bmHyaISMZ_Excg-VhW4JMeok_6-oci8_DbHfCW6DvZC4j1_1H55DsLJqyGxFlxfREc0mHkcO2WVxhftkIDlVMyDFPNEt51j_0NG_2cFfxdeo6o5d4G5UK4k8m_MlXjiFBiRCdLTmNgyIdeBc5jq9okexF4jKWNzAUp3KTHUA_c21btVk3yQgYuz-N4TnnXfNlQ,,/b64e=1/sign=efc1833f5001c426fa522057d3c8c36f/keyno=MARKET_1/*"}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_101_8/content/content/content/bannerCurtain":{"name":"@light/BannerCurtain"}}}
    {"widgets":{"@monetize/Kebab":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_101_8/content/content/content/kebab":{"adLabel":{"adLabelText":"Реклама","advertizer":"Общество с ограниченной ответственностью Джонсон & Джонсон, ИНН 7725216105, ID #e-1g-100171-VND-ADV","adLabel":1},"advertisementId":2110601}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_101_8/content/content/content/kebab":{"name":"@monetize/Kebab"}}}
    Реклама
    {"widgets":{"@light/AdLabel":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_101_8/content/content/content/adLabel":{"adLabel":{"adLabelText":"Реклама","advertizer":"Общество с ограниченной ответственностью Джонсон & Джонсон, ИНН 7725216105, ID #e-1g-100171-VND-ADV","adLabel":1},"advertisementId":2110601,"allowDebug":false,"borderRadius":5,"indents":6}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_101_8/content/content/content/adLabel":{"name":"@light/AdLabel"}}}
    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  • Эвалар Чай Эвалар БИО при повышенном содержании мочевой кислоты, 20 фильтр-пакетов
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  • Панангин таб. п/о плен., 50 шт.
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    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1464857415_10/content/content/toggleWishlist":{"skuId":"101480589776","productId":1464857415,"offerId":"G0EhRoiY-IjqMviR_7IeOQ","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgsQt9WV7tmv2biIARIaChhyZW1peF9kZXNrdG9wX21vZGVsX2NhcmQyFwjH5r+6BRDQ09uF+gIYrav8BiCc/qMY","sign":"juS4FzQrwLyIK2KZ7pWR6yk1ymlkB3pWWM79Bk1104g="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1464857415_10/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Салфетка для стимуляции дыхания с нашатырем 3*6 см ( 20 штук)
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  • Фенибут таб., 250 мг, 20 шт.
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    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1404748601_12/content/content/toggleWishlist":{"skuId":"265134532","productId":1404748601,"offerId":"X-n7dCzvPCf7BgXye7boWA","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgsQt9WV7tmv2biIARIaChhyZW1peF9kZXNrdG9wX21vZGVsX2NhcmQyFQi5huudBRDEw7Z+GLPg0Acg7dnBBw==","sign":"Ddi4yCnKCeIQDgaIuXy1zL8KxaSXAeO4J78OzI4pX/0="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1404748601_12/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Риностоп капли наз., 0.05%, 10 мл
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  • БиоГая Пробиотик капли детск. фл., 5 мл, 1 уп.
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    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:997279548_14/content/content/toggleWishlist":{"skuId":"101370161396","productId":997279548,"offerId":"DNTgLfhb2SFZHNJpMz1ccg","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgsQt9WV7tmv2biIARIaChhyZW1peF9kZXNrdG9wX21vZGVsX2NhcmQyFwi8jsXbAxD00YfR+QIY9N/5ByDa2cEH","sign":"X1mzVbB0IZ2bgnLSwl3nSA/XbV6xGIJj7K9M3ArkMCc="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:997279548_14/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Ревмафлекс капс., 60 шт., нейтральный, 1 уп.
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  • Силденафил-СЗ таб. п/о плен., 100 мг, 10 шт.
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  • Vitamin D3, 5000 МЕ, 0.1 мл, 240 шт.
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