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Описание

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Онглиза таб. п/о плен., 5 мг, 30 шт.

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Коротко о товаре

Артикул Маркета
3123204729
Действующее вещество
Возраст
от 18 лет
Инструкция
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С осторожностью следует назначать препарат при почечной недостаточности умеренной и тяжелой степени, пожилым пациентам, а также совместно с производными сульфонилмочевины. Применение при беременности и кормлении грудью В связи с тем, что применение саксаглиптина при беременности не изучено, не следует назначать препарат в этот период. Неизвестно, проникает ли саксаглиптин в грудное молоко. В связи с тем, что не исключена возможность проникновения саксаглиптина в грудное молоко, следует прекратить грудное вскармливание на период лечения саксаглиптином или отменить терапию, учитывая соотношение риска для ребенка и пользы для матери. Применение при нарушениях функции печени При нарушении функции печени легкой, умеренной и тяжелой степени коррекции дозы не требуется. Применение при нарушениях функции почек Для пациентов с почечной недостаточностью легкой степени (КК \u003E50 мл/мин) коррекции дозы не требуется. Для пациентов с умеренной или тяжелой почечной недостаточностью (КК \u003C50 мл/мин), а также для пациентов на гемодиализе рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут. Препарат следует принимать по окончании сеанса гемодиализа. Применение саксаглиптина у пациентов на перитонеальном диализе не изучено. Перед началом терапии саксаглиптином и в процессе лечения рекомендуется проводить оценку функции почек."},{"name":"Состав","value":"Действующее вещество: саксаглиптин (в виде саксаглиптина гидрохлорида)\u003Cbr\u003EВспомогательные вещества: лактозы моногидрат — 99 мг*; МКЦ — 90 мг; кроскармеллоза натрия — 10 мг; магния стеарат — 1 мг**; 1М раствор хлористоводородной кислоты*** — q.s.; Opadry II белый — 26 мг (спирт поливиниловый — 40%, титана диоксид — 25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%); Opadry II желтый — 7 мг (спирт поливиниловый — 40%, титана диоксид — 24,25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%, краситель оксид железа желтый (E172) — 0,75%) (для дозировки 2,5 мг); Opadry II розовый — 7 мг (спирт поливиниловый — 40%, титана диоксид — 24,25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%, краситель оксид железа красный (E172) — 0,75%) (для дозировки 5 мг); чернила Opacode синий — q.s.\u003Cbr/\u003E"},{"name":"Действующее вещество","value":"Саксаглиптин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-sakharnogo-diabeta","categoryId":"15756510","navnodeId":"72472","glfilters":["27144131:28709725"]}}},{"name":"Способ применения и дозы","value":"Препарат назначают внутрь, независимо от приема пищи. При монотерапии рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут. При комбинированной терапии рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут в комбинации с метформином, тиазолидиндионами или производными сульфонилмочевины. При стартовой комбинированной терапии с метформином рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут, начальная доза метформина - 500 мг/сут. В случае неадекватного ответа доза метформина может быть увеличена. При пропуске приема препарата Онглиза пропущенную таблетку следует принять сразу, как только пациент об этом вспомнит, однако не следует принимать двойную дозу препарата в течение одних суток. Для пациентов с почечной недостаточностью легкой степени (КК \u003E50 мл/мин) коррекции дозы не требуется. Для пациентов с умеренной или тяжелой почечной недостаточностью (КК ≤50 мл/мин), а также для пациентов, находящихся на гемодиализе, рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут. Препарат следует принимать по окончании сеанса гемодиализа. Применение саксаглиптина у пациентов, находящихся на перитонеальном диализе, не изучено. Перед началом терапии саксаглиптином и в процессе лечения рекомендуется проводить оценку функции почек. При нарушении функции печени легкой, умеренной и тяжелой степени коррекции дозы не требуется. Коррекции дозы у пожилых пациентов не требуется. Однако при выборе дозы следует учитывать, что у этой категории пациентов более вероятно снижение функции почек. Безопасность и эффективность применения препарата у пациентов младше 18 лет не изучалась. При одновременном применении с мощными ингибиторами CYP 3A4/5, такими как кетоконазол, атазанавир, кларитромицин, индинавир, итраконазол, нефазодон, нелфинавир, ритонавир, саквинавир и телитромицин, рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут."},{"name":"Побочные действия","value":"Общая частота нежелательных явлений при приеме препарата Онглиза 5 мг в режиме монотерапии и в режиме добавления к терапии метформином, тиазолидиндионом или глибенкламидом была сопоставима с таковой в группе плацебо. Шкала частоты побочных реакций: очень часто (≥1/10); часто (≥1/100, \u003C1/10); нечасто (≥1/1000, \u003C1/100); редко (≥1/10 000, \u003C1/1000); очень редко (\u003C1/10 000). Частота реакций гиперчувствительности, отмеченных к 24 неделе терапии, составила 1.5% у пациентов, получавших препарат Онглиза 5 мг, и 0.4% у пациентов, получавших плацебо. Реакции гиперчувствительности, возникшие у пациентов, принимавших препарат Онглиза, не требовали госпитализации и были расценены лечащими врачами как не представлявшие угрозу жизни. Побочные эффекты препарата Онглиза при комбинированной терапии В исследовании по комбинированному применению саксаглиптина и глибенкламида частота подтвержденных эпизодов гипогликемии в группе саксаглиптина 5 мг (0.8%) и плацебо (0.7%) статистически не различалась. Частота подтвержденных эпизодов гипогликемии у пациентов, получавших препарат Онглиза 5 мг в ходе двух исследованиях саксаглиптина в режиме монотерапии, исследовании по комбинированной терапии саксаглиптином и метформином, а также в исследовании по комбинированному применению саксаглиптина и тиазолидиндионов, была сопоставима с таковой на фоне плацебо. В исследовании по применению саксаглиптина совместно с тиазолидиндионами частота периферических отеков была выше в группе саксаглиптина 5 мг по сравнению с группой плацебо (8.1% и 4.3% соответственно). Периферические отеки были слабо или умеренно выраженными и не приводили к прекращению лечения. Частота периферических отеков у пациентов, принимавших препарат Онглиза в дозе 5 мг в ходе клинических исследований монотерапии саксаглиптина и комбинированной терапии с метформином или глибенкламидом, была сопоставима с таковой на фоне плацебо (1.7% и 2.4% соответственно). При стартовой комбинированной терапии саксаглиптином в дозе 5 мг и метформином часто отмечались случаи назофарингита и головной боли. Частота назофарингита была выше на фоне комбинированной терапии (6.9%) по сравнению с монотерапией саксаглиптином 10 мг (4.2%) и метформином (4%). Головная боль была чаще в группе пациентов на комбинированной терапии метформином и саксаглиптином 5 мг (7.5%) по сравнению с группами монотерапии саксаглиптином 10 мг (6.3%) и метформином (5.2%). Лабораторные исследования: в клинических исследованиях частота изменений лабораторных показателей при приеме саксаглиптина в дозе 5 мг и плацебо была сопоставимой. Отмечалось небольшое снижение числа лимфоцитов, при этом среднее абсолютное число лимфоцитов оставалось стабильным и в пределах нормальных значений при ежедневном приеме саксаглиптина продолжительностью до 102 недель. Уменьшение количества лимфоцитов не сопровождалось клинически значимыми нежелательными реакциями. Клиническое значение уменьшения числа лимфоцитов на фоне терапии саксаглиптином не известно."},{"name":"Фармакологическое действие","value":"Саксаглиптин - мощный селективный обратимый конкурентный ингибитор дипептидилпептидазы-4 (ДПП-4). У пациентов с сахарным диабетом 2 типа прием саксаглиптина приводит к подавлению активности фермента ДПП-4 в течение 24 ч. После приема глюкозы внутрь ингибирование ДПП-4 приводит к 2-3 кратному увеличению концентрации глюкагоноподобного пептида-1 (ГПП-1) и глюкозозависимого инсулинотропного полипептида (ГИП), уменьшению концентрации глюкагона и усилению глюкозозависимой ответной реакции бета-клеток, что приводит к повышению концентрации инсулина и С-пептида. Высвобождение инсулина бета-клетками поджелудочной железы и снижение высвобождения глюкагона из панкреатических альфа-клеток приводит к снижению гликемии натощак и постпрандиальной гликемии. Эффективность и безопасность применения саксаглиптина при приеме в дозах 2.5 мг, 5 мг и 10 мг 1 раз/сут изучены в шести двойных слепых плацебо-контролируемых исследованиях с участием 4148 пациентов с сахарным диабетом 2 типа. Прием препарата сопровождался статистически значимым улучшением показателей гликозилированного гемоглобина (HbA1c), глюкозы плазмы крови натощак (ГПН) и постпрандиальной глюкозы (ППГ) плазмы крови по сравнению с контролем. Пациентам, у которых целевой уровень гликемии не удалось достигнуть при приеме саксаглиптина в виде монотерапии, дополнительно назначался метформин, глибенкламид или тиазолидиндионы. При приеме саксаглиптина в дозе 5 мг снижение HbA1c было отмечено через 4 недели и ГПН - через 2 недели. В группе пациентов, получавших саксаглиптин в комбинации с метформином, глибенкламидом или тиазолидиндионами, снижение HbA1c также отмечалось через 4 недели и ГПН - через 2 недели. Влияние саксаглиптина на липидный профиль сходно с таковым плацебо. На фоне терапии саксаглиптином не отмечено увеличения массы тела."},{"name":"Фармакологическая группа","value":"гипогликемическое средство - дипептидилпептидазы-4 ингибитор"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-sakharnogo-diabeta","categoryId":"15756510","navnodeId":"72472","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"Препарат следует хранить в недоступном для детей месте при температуре не выше 30°С. Срок годности - 3 года. Не применять по истечении срока годности, указанного на упаковке."},{"name":"Передозировка","value":"Симптомы интоксикации не описаны при длительном приеме препарата в дозах, до 80 раз превышающих рекомендованные. Лечение: в случае передозировки следует применять симптоматическую терапию. Саксаглиптин и его основной метаболит выводятся из организма при помощи гемодиализа (скорость выведения: 23% дозы за 4 ч)."},{"name":"Применение при беременности и кормлении грудью","value":"Противопоказан."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Исследований по изучению влияния саксаглиптина на способность к вождению автотранспорта и управлению механизмами не проводилось. Следует учитывать, что саксаглиптин может вызывать головокружение."},{"name":"Особые указания","value":"Применение препарата Онглиза в комбинации с инсулином, а так же в составе тройной терапии с метформином и тиазолидиндионами или метформином и производными сульфонилмочевины, не изучалось. Пациенты с нарушением функции почек Рекомендуется коррекция дозы для пациентов с умеренной и тяжелой степенью почечной недостаточностью, а также для пациентов, находящихся на гемодиализе. Перед началом терапии и периодически в процессе лечения препаратом рекомендуется проводить оценку функции почек. Применение в комбинации с препаратами, которые могут вызвать гипогликемию Производные сульфонилмочевины могут вызвать гипогликемию, поэтому для уменьшения риска гипогликемии при одновременном применении с препаратом Онглиза может потребоваться снижение дозы производных сульфонилмочевины. Реакции гиперчувствительности Препарат не следует назначать пациентам, у которых были отмечены серьезные реакции гиперчувствительности при применении других ингибиторов ДПП-4. Пациенты пожилого возраста По данным клинических исследований, показатели эффективности и безопасности у пациентов в возрасте 65 лет и старше не отличались от аналогичных показателей у пациентов более молодого возраста. Однако нельзя исключить повышенную индивидуальную чувствительность к саксаглиптину у некоторых пациентов пожилого возраста. Саксаглиптин и его основной метаболит частично выводятся почками, поэтому необходимо учитывать, что у пациентов пожилого возраста более вероятно снижение функции почек. Препарат Онглиза содержит лактозу. Пациенты с врожденной непереносимостью галактозы, лактазной недостаточностью и глюкозо-галактозной мальабсорбцией не должны принимать этот препарат."},{"name":"Взаимодействие","value":"Анализ данных клинических исследований позволяет предполагать, что риск клинически значимых взаимодействий саксаглиптина с другими лекарственными средствами при их совместном применении невелик. Метаболизм саксаглиптина преимущественно опосредован системой изоферментов цитохрома Р450 3А4/5 (CYP3A4/5). В исследованиях in vitro было показано, что саксаглиптин и его основной метаболит не ингибируют изоферменты CYP 1A2, 2А6, 2В6, 2С9, 2С19, 2D6, 2Е1 и 3А4 и не индуцируют изоферменты CYP 1A2, 2В6, 2С9, и ЗА4. В исследованиях с участием здоровых добровольцев фармакокинетические показатели саксаглиптина и его основного метаболита значимо не изменялись под влиянием метформина, глибенкламида, пиоглитазона, дигоксина, симвастатина, дилтиазема, кетоконазола, омепразола, комбинации алюминия гидроксида, магния гидроксида и симетикона, а также фамотидина. Саксаглиптин значимо не изменяет фармакокинетические показатели метформина, глибенкламида, пиоглитазона, дигоксина, симвастатина, дилтиазема или кетоконазола. Влияние индукторов изоферментов CYP 3A4/5 на фармакокинетику саксаглиптина не изучено. Однако совместное применение саксаглиптина и индукторов изоферментов CYP 3A4/5, таких как карбамазепин, дексаметазон, фенобарбитал, фенитоин и рифампицин, могут приводить к уменьшению концентрации саксаглиптина в плазме и увеличению концентрации его основного метаболита. Изучения влияния курения, диетического питания, приема растительных препаратов и употребления алкоголя на терапию саксаглиптином не проводилось."},{"name":"Регистрационный номер","value":"ЛCP-008697/10"},{"name":"Дата государственной регистрации","value":"28.08.2018"},{"name":"Владелец регистрационного удостоверения","value":"AstraZeneca","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-sakharnogo-diabeta","categoryId":"15756510","navnodeId":"72472","glfilters":["34324371:35649313","7893318:16002703"]}}},{"name":"Изготовитель","value":"АстраЗенека Фармасьютикалз"},{"name":"Фасовщик","value":"АстраЗенека ЮК Лимитед"},{"name":"Страна-производитель","value":"США"},{"name":"Название препарата","value":"Онглиза","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-sakharnogo-diabeta","categoryId":"15756510","navnodeId":"72472","glfilters":["17796364:18045539"]}}},{"name":"Срок годности","value":"35 мес."}]}},"fullSpecsGrouped":{"2836316094464485862":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"эндокринная система"},{"name":"Назначение","value":"сахарный диабет 2 типа"},{"name":"Показания к применению","value":"Сахарный диабет 2 типа в дополнение к диете и физическим упражнениям для улучшения гликемического контроля в качестве: — монотерапии; — стартовой комбинированной терапии с метформином; — добавления к монотерапии метформином, тиазолидиндионами, производными сульфониломочевины, при отсутствии адекватного гликемического контроля на данной терапии."},{"name":"Противопоказания","value":"— сахарный диабет 1 типа (применение не изучено); — применение совместно с инсулином (не изучено); — диабетический кетоацидоз; — врожденные непереносимость галактозы, лактазная недостаточность и глюкозо- галактозная мальабсорбция; — беременность; — лактация; — возраст до 18 лет (безопасность и эффективность не изучены); — повышенная индивидуальная чувствительность к любому компоненту препарата. С осторожностью следует назначать препарат при почечной недостаточности умеренной и тяжелой степени, пожилым пациентам, а также совместно с производными сульфонилмочевины. Применение при беременности и кормлении грудью В связи с тем, что применение саксаглиптина при беременности не изучено, не следует назначать препарат в этот период. Неизвестно, проникает ли саксаглиптин в грудное молоко. В связи с тем, что не исключена возможность проникновения саксаглиптина в грудное молоко, следует прекратить грудное вскармливание на период лечения саксаглиптином или отменить терапию, учитывая соотношение риска для ребенка и пользы для матери. Применение при нарушениях функции печени При нарушении функции печени легкой, умеренной и тяжелой степени коррекции дозы не требуется. Применение при нарушениях функции почек Для пациентов с почечной недостаточностью легкой степени (КК \u003E50 мл/мин) коррекции дозы не требуется. Для пациентов с умеренной или тяжелой почечной недостаточностью (КК \u003C50 мл/мин), а также для пациентов на гемодиализе рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут. Препарат следует принимать по окончании сеанса гемодиализа. Применение саксаглиптина у пациентов на перитонеальном диализе не изучено. Перед началом терапии саксаглиптином и в процессе лечения рекомендуется проводить оценку функции почек."},{"name":"Состав","value":"Действующее вещество: саксаглиптин (в виде саксаглиптина гидрохлорида)\u003Cbr\u003EВспомогательные вещества: лактозы моногидрат — 99 мг*; МКЦ — 90 мг; кроскармеллоза натрия — 10 мг; магния стеарат — 1 мг**; 1М раствор хлористоводородной кислоты*** — q.s.; Opadry II белый — 26 мг (спирт поливиниловый — 40%, титана диоксид — 25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%); Opadry II желтый — 7 мг (спирт поливиниловый — 40%, титана диоксид — 24,25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%, краситель оксид железа желтый (E172) — 0,75%) (для дозировки 2,5 мг); Opadry II розовый — 7 мг (спирт поливиниловый — 40%, титана диоксид — 24,25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%, краситель оксид железа красный (E172) — 0,75%) (для дозировки 5 мг); чернила Opacode синий — q.s.\u003Cbr/\u003E"},{"name":"Действующее вещество","value":"Саксаглиптин"},{"name":"Способ применения и дозы","value":"Препарат назначают внутрь, независимо от приема пищи. При монотерапии рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут. При комбинированной терапии рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут в комбинации с метформином, тиазолидиндионами или производными сульфонилмочевины. При стартовой комбинированной терапии с метформином рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут, начальная доза метформина - 500 мг/сут. В случае неадекватного ответа доза метформина может быть увеличена. При пропуске приема препарата Онглиза пропущенную таблетку следует принять сразу, как только пациент об этом вспомнит, однако не следует принимать двойную дозу препарата в течение одних суток. Для пациентов с почечной недостаточностью легкой степени (КК \u003E50 мл/мин) коррекции дозы не требуется. Для пациентов с умеренной или тяжелой почечной недостаточностью (КК ≤50 мл/мин), а также для пациентов, находящихся на гемодиализе, рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут. Препарат следует принимать по окончании сеанса гемодиализа. Применение саксаглиптина у пациентов, находящихся на перитонеальном диализе, не изучено. Перед началом терапии саксаглиптином и в процессе лечения рекомендуется проводить оценку функции почек. При нарушении функции печени легкой, умеренной и тяжелой степени коррекции дозы не требуется. Коррекции дозы у пожилых пациентов не требуется. Однако при выборе дозы следует учитывать, что у этой категории пациентов более вероятно снижение функции почек. Безопасность и эффективность применения препарата у пациентов младше 18 лет не изучалась. При одновременном применении с мощными ингибиторами CYP 3A4/5, такими как кетоконазол, атазанавир, кларитромицин, индинавир, итраконазол, нефазодон, нелфинавир, ритонавир, саквинавир и телитромицин, рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут."},{"name":"Побочные действия","value":"Общая частота нежелательных явлений при приеме препарата Онглиза 5 мг в режиме монотерапии и в режиме добавления к терапии метформином, тиазолидиндионом или глибенкламидом была сопоставима с таковой в группе плацебо. Шкала частоты побочных реакций: очень часто (≥1/10); часто (≥1/100, \u003C1/10); нечасто (≥1/1000, \u003C1/100); редко (≥1/10 000, \u003C1/1000); очень редко (\u003C1/10 000). Частота реакций гиперчувствительности, отмеченных к 24 неделе терапии, составила 1.5% у пациентов, получавших препарат Онглиза 5 мг, и 0.4% у пациентов, получавших плацебо. Реакции гиперчувствительности, возникшие у пациентов, принимавших препарат Онглиза, не требовали госпитализации и были расценены лечащими врачами как не представлявшие угрозу жизни. Побочные эффекты препарата Онглиза при комбинированной терапии В исследовании по комбинированному применению саксаглиптина и глибенкламида частота подтвержденных эпизодов гипогликемии в группе саксаглиптина 5 мг (0.8%) и плацебо (0.7%) статистически не различалась. Частота подтвержденных эпизодов гипогликемии у пациентов, получавших препарат Онглиза 5 мг в ходе двух исследованиях саксаглиптина в режиме монотерапии, исследовании по комбинированной терапии саксаглиптином и метформином, а также в исследовании по комбинированному применению саксаглиптина и тиазолидиндионов, была сопоставима с таковой на фоне плацебо. В исследовании по применению саксаглиптина совместно с тиазолидиндионами частота периферических отеков была выше в группе саксаглиптина 5 мг по сравнению с группой плацебо (8.1% и 4.3% соответственно). Периферические отеки были слабо или умеренно выраженными и не приводили к прекращению лечения. Частота периферических отеков у пациентов, принимавших препарат Онглиза в дозе 5 мг в ходе клинических исследований монотерапии саксаглиптина и комбинированной терапии с метформином или глибенкламидом, была сопоставима с таковой на фоне плацебо (1.7% и 2.4% соответственно). При стартовой комбинированной терапии саксаглиптином в дозе 5 мг и метформином часто отмечались случаи назофарингита и головной боли. Частота назофарингита была выше на фоне комбинированной терапии (6.9%) по сравнению с монотерапией саксаглиптином 10 мг (4.2%) и метформином (4%). Головная боль была чаще в группе пациентов на комбинированной терапии метформином и саксаглиптином 5 мг (7.5%) по сравнению с группами монотерапии саксаглиптином 10 мг (6.3%) и метформином (5.2%). Лабораторные исследования: в клинических исследованиях частота изменений лабораторных показателей при приеме саксаглиптина в дозе 5 мг и плацебо была сопоставимой. Отмечалось небольшое снижение числа лимфоцитов, при этом среднее абсолютное число лимфоцитов оставалось стабильным и в пределах нормальных значений при ежедневном приеме саксаглиптина продолжительностью до 102 недель. Уменьшение количества лимфоцитов не сопровождалось клинически значимыми нежелательными реакциями. Клиническое значение уменьшения числа лимфоцитов на фоне терапии саксаглиптином не известно."},{"name":"Фармакологическое действие","value":"Саксаглиптин - мощный селективный обратимый конкурентный ингибитор дипептидилпептидазы-4 (ДПП-4). У пациентов с сахарным диабетом 2 типа прием саксаглиптина приводит к подавлению активности фермента ДПП-4 в течение 24 ч. После приема глюкозы внутрь ингибирование ДПП-4 приводит к 2-3 кратному увеличению концентрации глюкагоноподобного пептида-1 (ГПП-1) и глюкозозависимого инсулинотропного полипептида (ГИП), уменьшению концентрации глюкагона и усилению глюкозозависимой ответной реакции бета-клеток, что приводит к повышению концентрации инсулина и С-пептида. Высвобождение инсулина бета-клетками поджелудочной железы и снижение высвобождения глюкагона из панкреатических альфа-клеток приводит к снижению гликемии натощак и постпрандиальной гликемии. Эффективность и безопасность применения саксаглиптина при приеме в дозах 2.5 мг, 5 мг и 10 мг 1 раз/сут изучены в шести двойных слепых плацебо-контролируемых исследованиях с участием 4148 пациентов с сахарным диабетом 2 типа. Прием препарата сопровождался статистически значимым улучшением показателей гликозилированного гемоглобина (HbA1c), глюкозы плазмы крови натощак (ГПН) и постпрандиальной глюкозы (ППГ) плазмы крови по сравнению с контролем. Пациентам, у которых целевой уровень гликемии не удалось достигнуть при приеме саксаглиптина в виде монотерапии, дополнительно назначался метформин, глибенкламид или тиазолидиндионы. При приеме саксаглиптина в дозе 5 мг снижение HbA1c было отмечено через 4 недели и ГПН - через 2 недели. В группе пациентов, получавших саксаглиптин в комбинации с метформином, глибенкламидом или тиазолидиндионами, снижение HbA1c также отмечалось через 4 недели и ГПН - через 2 недели. Влияние саксаглиптина на липидный профиль сходно с таковым плацебо. На фоне терапии саксаглиптином не отмечено увеличения массы тела."},{"name":"Фармакологическая группа","value":"гипогликемическое средство - дипептидилпептидазы-4 ингибитор"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"Препарат следует хранить в недоступном для детей месте при температуре не выше 30°С. Срок годности - 3 года. Не применять по истечении срока годности, указанного на упаковке."},{"name":"Передозировка","value":"Симптомы интоксикации не описаны при длительном приеме препарата в дозах, до 80 раз превышающих рекомендованные. Лечение: в случае передозировки следует применять симптоматическую терапию. Саксаглиптин и его основной метаболит выводятся из организма при помощи гемодиализа (скорость выведения: 23% дозы за 4 ч)."},{"name":"Применение при беременности и кормлении грудью","value":"Противопоказан."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Исследований по изучению влияния саксаглиптина на способность к вождению автотранспорта и управлению механизмами не проводилось. Следует учитывать, что саксаглиптин может вызывать головокружение."},{"name":"Особые указания","value":"Применение препарата Онглиза в комбинации с инсулином, а так же в составе тройной терапии с метформином и тиазолидиндионами или метформином и производными сульфонилмочевины, не изучалось. Пациенты с нарушением функции почек Рекомендуется коррекция дозы для пациентов с умеренной и тяжелой степенью почечной недостаточностью, а также для пациентов, находящихся на гемодиализе. Перед началом терапии и периодически в процессе лечения препаратом рекомендуется проводить оценку функции почек. Применение в комбинации с препаратами, которые могут вызвать гипогликемию Производные сульфонилмочевины могут вызвать гипогликемию, поэтому для уменьшения риска гипогликемии при одновременном применении с препаратом Онглиза может потребоваться снижение дозы производных сульфонилмочевины. Реакции гиперчувствительности Препарат не следует назначать пациентам, у которых были отмечены серьезные реакции гиперчувствительности при применении других ингибиторов ДПП-4. Пациенты пожилого возраста По данным клинических исследований, показатели эффективности и безопасности у пациентов в возрасте 65 лет и старше не отличались от аналогичных показателей у пациентов более молодого возраста. Однако нельзя исключить повышенную индивидуальную чувствительность к саксаглиптину у некоторых пациентов пожилого возраста. Саксаглиптин и его основной метаболит частично выводятся почками, поэтому необходимо учитывать, что у пациентов пожилого возраста более вероятно снижение функции почек. Препарат Онглиза содержит лактозу. Пациенты с врожденной непереносимостью галактозы, лактазной недостаточностью и глюкозо-галактозной мальабсорбцией не должны принимать этот препарат."},{"name":"Взаимодействие","value":"Анализ данных клинических исследований позволяет предполагать, что риск клинически значимых взаимодействий саксаглиптина с другими лекарственными средствами при их совместном применении невелик. Метаболизм саксаглиптина преимущественно опосредован системой изоферментов цитохрома Р450 3А4/5 (CYP3A4/5). В исследованиях in vitro было показано, что саксаглиптин и его основной метаболит не ингибируют изоферменты CYP 1A2, 2А6, 2В6, 2С9, 2С19, 2D6, 2Е1 и 3А4 и не индуцируют изоферменты CYP 1A2, 2В6, 2С9, и ЗА4. В исследованиях с участием здоровых добровольцев фармакокинетические показатели саксаглиптина и его основного метаболита значимо не изменялись под влиянием метформина, глибенкламида, пиоглитазона, дигоксина, симвастатина, дилтиазема, кетоконазола, омепразола, комбинации алюминия гидроксида, магния гидроксида и симетикона, а также фамотидина. Саксаглиптин значимо не изменяет фармакокинетические показатели метформина, глибенкламида, пиоглитазона, дигоксина, симвастатина, дилтиазема или кетоконазола. Влияние индукторов изоферментов CYP 3A4/5 на фармакокинетику саксаглиптина не изучено. Однако совместное применение саксаглиптина и индукторов изоферментов CYP 3A4/5, таких как карбамазепин, дексаметазон, фенобарбитал, фенитоин и рифампицин, могут приводить к уменьшению концентрации саксаглиптина в плазме и увеличению концентрации его основного метаболита. Изучения влияния курения, диетического питания, приема растительных препаратов и употребления алкоголя на терапию саксаглиптином не проводилось."},{"name":"Регистрационный номер","value":"ЛCP-008697/10"},{"name":"Дата государственной регистрации","value":"28.08.2018"},{"name":"Владелец регистрационного удостоверения","value":"AstraZeneca"},{"name":"Изготовитель","value":"АстраЗенека Фармасьютикалз"},{"name":"Фасовщик","value":"АстраЗенека ЮК Лимитед"},{"name":"Страна-производитель","value":"США"},{"name":"Название препарата","value":"Онглиза"},{"name":"Срок годности","value":"35 мес."}]}],"transitionId":"tr_6"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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Для пациентов с умеренной или тяжелой почечной недостаточностью (КК \u003C50 мл/мин), а также для пациентов на гемодиализе рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут. Препарат следует принимать по окончании сеанса гемодиализа. Применение саксаглиптина у пациентов на перитонеальном диализе не изучено. Перед началом терапии саксаглиптином и в процессе лечения рекомендуется проводить оценку функции почек."},{"description":"","filters":[{"id":15768292,"name":"Состав"}],"isMainProperty":false,"name":"Состав","value":"Действующее вещество: саксаглиптин (в виде саксаглиптина гидрохлорида)\u003Cbr\u003EВспомогательные вещества: лактозы моногидрат — 99 мг*; МКЦ — 90 мг; кроскармеллоза натрия — 10 мг; магния стеарат — 1 мг**; 1М раствор хлористоводородной кислоты*** — q.s.; Opadry II белый — 26 мг (спирт поливиниловый — 40%, титана диоксид — 25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%); Opadry II желтый — 7 мг (спирт поливиниловый — 40%, титана диоксид — 24,25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%, краситель оксид железа желтый (E172) — 0,75%) (для дозировки 2,5 мг); Opadry II розовый — 7 мг (спирт поливиниловый — 40%, титана диоксид — 24,25%, макрогол (ПЭГ 3350) — 20,2%, тальк — 14,8%, краситель оксид железа красный (E172) — 0,75%) (для дозировки 5 мг); чернила Opacode синий — q.s.\u003Cbr/\u003E"},{"description":"","filters":[{"id":27144131,"name":"Действующее вещество"}],"isMainProperty":false,"name":"Действующее вещество","value":"Саксаглиптин"},{"description":"","filters":[{"id":15768000,"name":"Способ применения и дозы"}],"isMainProperty":false,"name":"Способ применения и дозы","value":"Препарат назначают внутрь, независимо от приема пищи. При монотерапии рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут. При комбинированной терапии рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут в комбинации с метформином, тиазолидиндионами или производными сульфонилмочевины. При стартовой комбинированной терапии с метформином рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут, начальная доза метформина - 500 мг/сут. В случае неадекватного ответа доза метформина может быть увеличена. При пропуске приема препарата Онглиза пропущенную таблетку следует принять сразу, как только пациент об этом вспомнит, однако не следует принимать двойную дозу препарата в течение одних суток. Для пациентов с почечной недостаточностью легкой степени (КК \u003E50 мл/мин) коррекции дозы не требуется. Для пациентов с умеренной или тяжелой почечной недостаточностью (КК ≤50 мл/мин), а также для пациентов, находящихся на гемодиализе, рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут. Препарат следует принимать по окончании сеанса гемодиализа. Применение саксаглиптина у пациентов, находящихся на перитонеальном диализе, не изучено. Перед началом терапии саксаглиптином и в процессе лечения рекомендуется проводить оценку функции почек. При нарушении функции печени легкой, умеренной и тяжелой степени коррекции дозы не требуется. Коррекции дозы у пожилых пациентов не требуется. Однако при выборе дозы следует учитывать, что у этой категории пациентов более вероятно снижение функции почек. Безопасность и эффективность применения препарата у пациентов младше 18 лет не изучалась. При одновременном применении с мощными ингибиторами CYP 3A4/5, такими как кетоконазол, атазанавир, кларитромицин, индинавир, итраконазол, нефазодон, нелфинавир, ритонавир, саквинавир и телитромицин, рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут."},{"description":"","filters":[{"id":15767998,"name":"Побочные действия"}],"isMainProperty":false,"name":"Побочные действия","value":"Общая частота нежелательных явлений при приеме препарата Онглиза 5 мг в режиме монотерапии и в режиме добавления к терапии метформином, тиазолидиндионом или глибенкламидом была сопоставима с таковой в группе плацебо. Шкала частоты побочных реакций: очень часто (≥1/10); часто (≥1/100, \u003C1/10); нечасто (≥1/1000, \u003C1/100); редко (≥1/10 000, \u003C1/1000); очень редко (\u003C1/10 000). Частота реакций гиперчувствительности, отмеченных к 24 неделе терапии, составила 1.5% у пациентов, получавших препарат Онглиза 5 мг, и 0.4% у пациентов, получавших плацебо. Реакции гиперчувствительности, возникшие у пациентов, принимавших препарат Онглиза, не требовали госпитализации и были расценены лечащими врачами как не представлявшие угрозу жизни. Побочные эффекты препарата Онглиза при комбинированной терапии В исследовании по комбинированному применению саксаглиптина и глибенкламида частота подтвержденных эпизодов гипогликемии в группе саксаглиптина 5 мг (0.8%) и плацебо (0.7%) статистически не различалась. Частота подтвержденных эпизодов гипогликемии у пациентов, получавших препарат Онглиза 5 мг в ходе двух исследованиях саксаглиптина в режиме монотерапии, исследовании по комбинированной терапии саксаглиптином и метформином, а также в исследовании по комбинированному применению саксаглиптина и тиазолидиндионов, была сопоставима с таковой на фоне плацебо. В исследовании по применению саксаглиптина совместно с тиазолидиндионами частота периферических отеков была выше в группе саксаглиптина 5 мг по сравнению с группой плацебо (8.1% и 4.3% соответственно). Периферические отеки были слабо или умеренно выраженными и не приводили к прекращению лечения. Частота периферических отеков у пациентов, принимавших препарат Онглиза в дозе 5 мг в ходе клинических исследований монотерапии саксаглиптина и комбинированной терапии с метформином или глибенкламидом, была сопоставима с таковой на фоне плацебо (1.7% и 2.4% соответственно). При стартовой комбинированной терапии саксаглиптином в дозе 5 мг и метформином часто отмечались случаи назофарингита и головной боли. Частота назофарингита была выше на фоне комбинированной терапии (6.9%) по сравнению с монотерапией саксаглиптином 10 мг (4.2%) и метформином (4%). Головная боль была чаще в группе пациентов на комбинированной терапии метформином и саксаглиптином 5 мг (7.5%) по сравнению с группами монотерапии саксаглиптином 10 мг (6.3%) и метформином (5.2%). Лабораторные исследования: в клинических исследованиях частота изменений лабораторных показателей при приеме саксаглиптина в дозе 5 мг и плацебо была сопоставимой. Отмечалось небольшое снижение числа лимфоцитов, при этом среднее абсолютное число лимфоцитов оставалось стабильным и в пределах нормальных значений при ежедневном приеме саксаглиптина продолжительностью до 102 недель. Уменьшение количества лимфоцитов не сопровождалось клинически значимыми нежелательными реакциями. Клиническое значение уменьшения числа лимфоцитов на фоне терапии саксаглиптином не известно."},{"description":"","filters":[{"id":15768001,"name":"Фармакологическое действие"}],"isMainProperty":false,"name":"Фармакологическое действие","value":"Саксаглиптин - мощный селективный обратимый конкурентный ингибитор дипептидилпептидазы-4 (ДПП-4). У пациентов с сахарным диабетом 2 типа прием саксаглиптина приводит к подавлению активности фермента ДПП-4 в течение 24 ч. После приема глюкозы внутрь ингибирование ДПП-4 приводит к 2-3 кратному увеличению концентрации глюкагоноподобного пептида-1 (ГПП-1) и глюкозозависимого инсулинотропного полипептида (ГИП), уменьшению концентрации глюкагона и усилению глюкозозависимой ответной реакции бета-клеток, что приводит к повышению концентрации инсулина и С-пептида. Высвобождение инсулина бета-клетками поджелудочной железы и снижение высвобождения глюкагона из панкреатических альфа-клеток приводит к снижению гликемии натощак и постпрандиальной гликемии. Эффективность и безопасность применения саксаглиптина при приеме в дозах 2.5 мг, 5 мг и 10 мг 1 раз/сут изучены в шести двойных слепых плацебо-контролируемых исследованиях с участием 4148 пациентов с сахарным диабетом 2 типа. Прием препарата сопровождался статистически значимым улучшением показателей гликозилированного гемоглобина (HbA1c), глюкозы плазмы крови натощак (ГПН) и постпрандиальной глюкозы (ППГ) плазмы крови по сравнению с контролем. Пациентам, у которых целевой уровень гликемии не удалось достигнуть при приеме саксаглиптина в виде монотерапии, дополнительно назначался метформин, глибенкламид или тиазолидиндионы. При приеме саксаглиптина в дозе 5 мг снижение HbA1c было отмечено через 4 недели и ГПН - через 2 недели. В группе пациентов, получавших саксаглиптин в комбинации с метформином, глибенкламидом или тиазолидиндионами, снижение HbA1c также отмечалось через 4 недели и ГПН - через 2 недели. Влияние саксаглиптина на липидный профиль сходно с таковым плацебо. На фоне терапии саксаглиптином не отмечено увеличения массы тела."},{"description":"","filters":[{"id":34045110,"name":"Фармакологическая группа"}],"isMainProperty":false,"name":"Фармакологическая группа","value":"гипогликемическое средство - дипептидилпептидазы-4 ингибитор"},{"description":"","filters":[{"id":27141511,"name":"Форма выпуска для карточки"}],"isMainProperty":false,"name":"Форма выпуска","value":"таблетки"},{"description":"","filters":[{"id":35947170,"name":"Способ применения/введения"}],"isMainProperty":false,"name":"Способ применения/введения","value":"пероральный"},{"description":"","filters":[{"id":23679511,"name":"Минимальный возраст применения"},{"id":16082123,"name":"С рождения"}],"isMainProperty":false,"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","specs":[{"description":"","filters":[{"id":15767999,"name":"Условия хранения"}],"isMainProperty":false,"name":"Условия хранения","value":"Препарат следует хранить в недоступном для детей месте при температуре не выше 30°С. Срок годности - 3 года. Не применять по истечении срока годности, указанного на упаковке."},{"description":"","filters":[{"id":15768014,"name":"Передозировка"}],"isMainProperty":false,"name":"Передозировка","value":"Симптомы интоксикации не описаны при длительном приеме препарата в дозах, до 80 раз превышающих рекомендованные. Лечение: в случае передозировки следует применять симптоматическую терапию. Саксаглиптин и его основной метаболит выводятся из организма при помощи гемодиализа (скорость выведения: 23% дозы за 4 ч)."},{"description":"","filters":[{"id":15768015,"name":"Применение при беременности и кормлении грудью"}],"isMainProperty":false,"name":"Применение при беременности и кормлении грудью","value":"Противопоказан."},{"description":"","filters":[{"id":17360993,"name":"Влияние на способность управлять транспортом и механизмами"}],"isMainProperty":false,"name":"Влияние на способность управлять транспортом и механизмами","value":"Исследований по изучению влияния саксаглиптина на способность к вождению автотранспорта и управлению механизмами не проводилось. Следует учитывать, что саксаглиптин может вызывать головокружение."},{"description":"","filters":[{"id":15771167,"name":"Особые указания"}],"isMainProperty":false,"name":"Особые указания","value":"Применение препарата Онглиза в комбинации с инсулином, а так же в составе тройной терапии с метформином и тиазолидиндионами или метформином и производными сульфонилмочевины, не изучалось. Пациенты с нарушением функции почек Рекомендуется коррекция дозы для пациентов с умеренной и тяжелой степенью почечной недостаточностью, а также для пациентов, находящихся на гемодиализе. Перед началом терапии и периодически в процессе лечения препаратом рекомендуется проводить оценку функции почек. Применение в комбинации с препаратами, которые могут вызвать гипогликемию Производные сульфонилмочевины могут вызвать гипогликемию, поэтому для уменьшения риска гипогликемии при одновременном применении с препаратом Онглиза может потребоваться снижение дозы производных сульфонилмочевины. Реакции гиперчувствительности Препарат не следует назначать пациентам, у которых были отмечены серьезные реакции гиперчувствительности при применении других ингибиторов ДПП-4. Пациенты пожилого возраста По данным клинических исследований, показатели эффективности и безопасности у пациентов в возрасте 65 лет и старше не отличались от аналогичных показателей у пациентов более молодого возраста. Однако нельзя исключить повышенную индивидуальную чувствительность к саксаглиптину у некоторых пациентов пожилого возраста. Саксаглиптин и его основной метаболит частично выводятся почками, поэтому необходимо учитывать, что у пациентов пожилого возраста более вероятно снижение функции почек. Препарат Онглиза содержит лактозу. Пациенты с врожденной непереносимостью галактозы, лактазной недостаточностью и глюкозо-галактозной мальабсорбцией не должны принимать этот препарат."},{"description":"","filters":[{"id":15768012,"name":"Взаимодействие"}],"isMainProperty":false,"name":"Взаимодействие","value":"Анализ данных клинических исследований позволяет предполагать, что риск клинически значимых взаимодействий саксаглиптина с другими лекарственными средствами при их совместном применении невелик. Метаболизм саксаглиптина преимущественно опосредован системой изоферментов цитохрома Р450 3А4/5 (CYP3A4/5). В исследованиях in vitro было показано, что саксаглиптин и его основной метаболит не ингибируют изоферменты CYP 1A2, 2А6, 2В6, 2С9, 2С19, 2D6, 2Е1 и 3А4 и не индуцируют изоферменты CYP 1A2, 2В6, 2С9, и ЗА4. В исследованиях с участием здоровых добровольцев фармакокинетические показатели саксаглиптина и его основного метаболита значимо не изменялись под влиянием метформина, глибенкламида, пиоглитазона, дигоксина, симвастатина, дилтиазема, кетоконазола, омепразола, комбинации алюминия гидроксида, магния гидроксида и симетикона, а также фамотидина. Саксаглиптин значимо не изменяет фармакокинетические показатели метформина, глибенкламида, пиоглитазона, дигоксина, симвастатина, дилтиазема или кетоконазола. Влияние индукторов изоферментов CYP 3A4/5 на фармакокинетику саксаглиптина не изучено. Однако совместное применение саксаглиптина и индукторов изоферментов CYP 3A4/5, таких как карбамазепин, дексаметазон, фенобарбитал, фенитоин и рифампицин, могут приводить к уменьшению концентрации саксаглиптина в плазме и увеличению концентрации его основного метаболита. 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    на основе 7 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 42 оценки
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  • Рейтинг товара: 4.9 из 5
    на основе 51 оценка
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  • Рейтинг товара: 5 из 5
    на основе 9 оценок
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-rbxzt6q7ejr/addToCartButton":{"offerId":"UluZuqARy0U5ev0Jp2_3lQ","skuId":"101372359736","pendingCartItem":{"productId":452780010,"offerId":"UluZuqARy0U5ev0Jp2_3lQ","showPlaceId":"OTNDnItfwRMjN9MRHuEMMpWcb_h8lSoGzExwC2WjBqBHHEYeagY5P5pKFHVkIt6eMXdAi7-DoZE8isL1AEb9VbKSOTyZTMI5eHwenzGS3Not7vaOPzsQsOntu7eyQUAZWbjWFZEdGxM4csMY4kJbyaQ0OE-HcDk6Q7buGBY-9ZQpe_FOsFbJvyr9_EatmFJNWeOBrNNE4nbEiXmh8SH3UQ,,","feeShow":"OTNDnItfwRMjN9MRHuEMMpWcb_h8lSoGzExwC2WjBqBHHEYeagY5P5pKFHVkIt6eMXdAi7-DoZE8isL1AEb9VbKSOTyZTMI5eHwenzGS3Not7vaOPzsQsOntu7eyQUAZWbjWFZEdGxM4csMY4kJbyaQ0OE-HcDk6Q7buGBY-9ZQpe_FOsFbJvyr9_EatmFJNWeOBrNNE4nbEiXmh8SH3UQ,,","skuId":"101372359736","shopId":55106433,"price":{"applicablePriceDiscounts":[],"value":"1311","currency":"RUR"},"hid":"15756510","name":"Кселевия таб. п/о плен., 100 мг, 28 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  • Рейтинг товара: 5 из 5
    на основе 4 оценки
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  • Рейтинг товара: 5 из 5
    на основе 25 оценок
    {"widgets":{"@light/AddToCartButtonSnippet":{"/content/page/fancyPage/kkmCarousel/kkmCarousel/content/content/slot-lg69au89rpe/addToCartButton":{"offerId":"3D0HwagYW0A5aqWv3paKCg","skuId":"186960543","pendingCartItem":{"productId":998360018,"offerId":"3D0HwagYW0A5aqWv3paKCg","showPlaceId":"OTNDnItfwRMjN9MRHuEMMpWcb_h8lSoG9LvfLRm-wTrSFKb2PsIp8WAkPuT4vhsYiU6Zc2IEtZsElIYtUlyiEO1SNJsFwkv_dts5cCuKgjSG2Y20RSAc1BJJQ4o16mQMEOGmhVTjSyYZCmItaICA-7qmrdpYCfNEYkNSzH_41dbzHvBs-ofP2H9vLBwj2UsmzP8WtteZwMj9UE-ndrc24Q,,","feeShow":"OTNDnItfwRMjN9MRHuEMMpWcb_h8lSoG9LvfLRm-wTrSFKb2PsIp8WAkPuT4vhsYiU6Zc2IEtZsElIYtUlyiEO1SNJsFwkv_dts5cCuKgjSG2Y20RSAc1BJJQ4o16mQMEOGmhVTjSyYZCmItaICA-7qmrdpYCfNEYkNSzH_41dbzHvBs-ofP2H9vLBwj2UsmzP8WtteZwMj9UE-ndrc24Q,,","skuId":"186960543","shopId":55106433,"price":{"applicablePriceDiscounts":[],"value":"3001","currency":"RUR"},"hid":"15756510","name":"Джардинс таб. п/о плен., 10 мг, 30 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  • Рейтинг товара: 4.3 из 5
    на основе 6 оценок
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  • Рейтинг товара: 4.8 из 5
    на основе 37 оценок
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  • Рейтинг товара: 5 из 5
    на основе 1 оценка
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  • Рейтинг товара: 5 из 5
    на основе 10 оценок
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  • Рейтинг товара: 4.9 из 5
    на основе 17 оценок
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Инструкция

Показания к применению

Сахарный диабет 2 типа в дополнение к диете и физическим упражнениям для улучшения гликемического контроля в качестве: — монотерапии; — стартовой комбинированной терапии с метформином; — добавления к монотерапии метформином, тиазолидиндионами, производными сульфониломочевины, при отсутствии адекватного гликемического контроля на данной терапии.

Противопоказания

— сахарный диабет 1 типа (применение не изучено); — применение совместно с инсулином (не изучено); — диабетический кетоацидоз; — врожденные непереносимость галактозы, лактазная недостаточность и глюкозо- галактозная мальабсорбция; — беременность; — лактация; — возраст до 18 лет (безопасность и эффективность не изучены); — повышенная индивидуальная чувствительность к любому компоненту препарата. С осторожностью следует назначать препарат при почечной недостаточности умеренной и тяжелой степени, пожилым пациентам, а также совместно с производными сульфонилмочевины. Применение при беременности и кормлении грудью В связи с тем, что применение саксаглиптина при беременности не изучено, не следует назначать препарат в этот период. Неизвестно, проникает ли саксаглиптин в грудное молоко. В связи с тем, что не исключена возможность проникновения саксаглиптина в грудное молоко, следует прекратить грудное вскармливание на период лечения саксаглиптином или отменить терапию, учитывая соотношение риска для ребенка и пользы для матери. Применение при нарушениях функции печени При нарушении функции печени легкой, умеренной и тяжелой степени коррекции дозы не требуется. Применение при нарушениях функции почек Для пациентов с почечной недостаточностью легкой степени (КК >50 мл/мин) коррекции дозы не требуется. Для пациентов с умеренной или тяжелой почечной недостаточностью (КК <50 мл/мин), а также для пациентов на гемодиализе рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут. Препарат следует принимать по окончании сеанса гемодиализа. Применение саксаглиптина у пациентов на перитонеальном диализе не изучено. Перед началом терапии саксаглиптином и в процессе лечения рекомендуется проводить оценку функции почек.

Способ применения и дозы

Препарат назначают внутрь, независимо от приема пищи. При монотерапии рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут. При комбинированной терапии рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут в комбинации с метформином, тиазолидиндионами или производными сульфонилмочевины. При стартовой комбинированной терапии с метформином рекомендуемая доза саксаглиптина составляет 5 мг 1 раз/сут, начальная доза метформина - 500 мг/сут. В случае неадекватного ответа доза метформина может быть увеличена. При пропуске приема препарата Онглиза пропущенную таблетку следует принять сразу, как только пациент об этом вспомнит, однако не следует принимать двойную дозу препарата в течение одних суток. Для пациентов с почечной недостаточностью легкой степени (КК >50 мл/мин) коррекции дозы не требуется. Для пациентов с умеренной или тяжелой почечной недостаточностью (КК ≤50 мл/мин), а также для пациентов, находящихся на гемодиализе, рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут. Препарат следует принимать по окончании сеанса гемодиализа. Применение саксаглиптина у пациентов, находящихся на перитонеальном диализе, не изучено. Перед началом терапии саксаглиптином и в процессе лечения рекомендуется проводить оценку функции почек. При нарушении функции печени легкой, умеренной и тяжелой степени коррекции дозы не требуется. Коррекции дозы у пожилых пациентов не требуется. Однако при выборе дозы следует учитывать, что у этой категории пациентов более вероятно снижение функции почек. Безопасность и эффективность применения препарата у пациентов младше 18 лет не изучалась. При одновременном применении с мощными ингибиторами CYP 3A4/5, такими как кетоконазол, атазанавир, кларитромицин, индинавир, итраконазол, нефазодон, нелфинавир, ритонавир, саквинавир и телитромицин, рекомендуемая доза препарата Онглиза составляет 2.5 мг 1 раз/сут.
Полная инструкция
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Онглиза таб. п/о плен.
Онглиза таб. п/о плен., 5 мг, 30 шт.
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Инструкция

1 927 ₽

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Рекомендуем

  • Тражента таб. п/о плен., 5 мг, 30 шт.
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778172426_0/content/content/gallery":{"title":"Тражента таб. п/о плен., 5 мг, 30 шт.","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/4547325/img_id2037737004470465190.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/4547325/img_id2037737004470465190.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/4547325/img_id2037737004470465190.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/4547325/img_id2037737004470465190.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/4547325/img_id2037737004470465190.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/4547325/img_id2037737004470465190.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"},{"src":"https://avatars.mds.yandex.net/get-mpic/7980098/img_id524715313743819845.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/7980098/img_id524715313743819845.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/7980098/img_id524715313743819845.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/7980098/img_id524715313743819845.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/7980098/img_id524715313743819845.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/7980098/img_id524715313743819845.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"},{"src":"https://avatars.mds.yandex.net/get-mpic/5221145/img_id2546290492035387161.png/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/5221145/img_id2546290492035387161.png/120x160 120w, https://avatars.mds.yandex.net/get-mpic/5221145/img_id2546290492035387161.png/180x240 180w, https://avatars.mds.yandex.net/get-mpic/5221145/img_id2546290492035387161.png/240x320 240w, https://avatars.mds.yandex.net/get-mpic/5221145/img_id2546290492035387161.png/300x400 300w, https://avatars.mds.yandex.net/get-mpic/5221145/img_id2546290492035387161.png/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"}],"firstImageLazyLoading":false,"baobabClientData":{"realTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQoOaY89+QkoctEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIVCIqE888GEM/vjFkYxrTeByDe2cEH","sign":"QyEfJZ8iwurv57QpdkmxigRU9vKtZbOJ6bf6ueEnVPg="},"target":"model_card"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778172426_0/content/content/gallery":{"name":"@marketfront/SnippetConstructor/Gallery"}}}
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  • Галвус таб., 50 мг, 28 шт.
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778172503_1/content/content/gallery":{"title":"Галвус таб., 50 мг, 28 шт.","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/3721790/img_id4300994414509827340.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/3721790/img_id4300994414509827340.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/3721790/img_id4300994414509827340.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/3721790/img_id4300994414509827340.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/3721790/img_id4300994414509827340.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/3721790/img_id4300994414509827340.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"},{"src":"https://avatars.mds.yandex.net/get-mpic/6439030/img_id99763880341409280.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/6439030/img_id99763880341409280.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/6439030/img_id99763880341409280.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/6439030/img_id99763880341409280.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/6439030/img_id99763880341409280.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/6439030/img_id99763880341409280.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"},{"src":"https://avatars.mds.yandex.net/get-mpic/2008488/img_id1526409001436819087.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/2008488/img_id1526409001436819087.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/2008488/img_id1526409001436819087.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/2008488/img_id1526409001436819087.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/2008488/img_id1526409001436819087.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/2008488/img_id1526409001436819087.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"}],"firstImageLazyLoading":false,"baobabClientData":{"realTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQoOaY89+QkoctEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIXCNeE888GEL/oje37AhiQ1aEFIN7ZwQc=","sign":"4Dp7BFdjNkaCF20+B2UTNUnyQ7onaiItSipdmy0UMY8="},"target":"model_card"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778172503_1/content/content/gallery":{"name":"@marketfront/SnippetConstructor/Gallery"}}}
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  • Асиглия таб. п/о плен., 100 мг, 28 шт.
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  • Кселевия таб. п/о плен., 100 мг, 28 шт.
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:452780010_3/content/content/gallery":{"title":"Кселевия таб. п/о плен., 100 мг, 28 шт.","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/4291905/img_id5430983895986366822.png/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/4291905/img_id5430983895986366822.png/120x160 120w, https://avatars.mds.yandex.net/get-mpic/4291905/img_id5430983895986366822.png/180x240 180w, https://avatars.mds.yandex.net/get-mpic/4291905/img_id5430983895986366822.png/240x320 240w, https://avatars.mds.yandex.net/get-mpic/4291905/img_id5430983895986366822.png/300x400 300w, https://avatars.mds.yandex.net/get-mpic/4291905/img_id5430983895986366822.png/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"},{"src":"https://avatars.mds.yandex.net/get-mpic/5283489/img_id5737538834515318540.png/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/5283489/img_id5737538834515318540.png/120x160 120w, https://avatars.mds.yandex.net/get-mpic/5283489/img_id5737538834515318540.png/180x240 180w, https://avatars.mds.yandex.net/get-mpic/5283489/img_id5737538834515318540.png/240x320 240w, https://avatars.mds.yandex.net/get-mpic/5283489/img_id5737538834515318540.png/300x400 300w, https://avatars.mds.yandex.net/get-mpic/5283489/img_id5737538834515318540.png/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"}],"firstImageLazyLoading":false,"baobabClientData":{"realTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQoOaY89+QkoctEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIXCOq/89cBELjojdL5Ahin3dAHIN7ZwQc=","sign":"pdg2ke2P9W6Kl5fnXET/OJWTp+ySNVWcM1zTzginHm8="},"target":"model_card"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:452780010_3/content/content/gallery":{"name":"@marketfront/SnippetConstructor/Gallery"}}}
    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:452780010_3/content/content/toggleWishlist":{"skuId":"101372359736","productId":452780010,"offerId":"UluZuqARy0U5ev0Jp2_3lQ","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQoOaY89+QkoctEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIXCOq/89cBELjojdL5Ahin3dAHIN7ZwQc=","sign":"pdg2ke2P9W6Kl5fnXET/OJWTp+ySNVWcM1zTzginHm8="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:452780010_3/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Випидия таб. п/о плен., 25 мг, 28 шт.
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  • Джардинс таб. п/о плен., 10 мг, 30 шт.
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    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:998360018_5/content/content/toggleWishlist":{"skuId":"186960543","productId":998360018,"offerId":"3D0HwagYW0A5aqWv3paKCg","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQoOaY89+QkoctEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIVCNKHh9wDEJ+Vk1kYxrTeByDe2cEH","sign":"k+9s944Z4xhRGiX1/QEbPXk4a4CBS9k0htA9+Txbhg4="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:998360018_5/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Сигдуо Лонг таб. п/о плен. с модиф. высв., 10 мг+1000 мг, 30 шт.
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    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:998360070_6/content/content/toggleWishlist":{"skuId":"655917651","productId":998360070,"offerId":"-T_1T7RootNRGwkM29UdSw","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQoOaY89+QkoctEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIWCIaIh9wDENOE4rgCGI/d0Acg3tnBBw==","sign":"Si2TK0O6NQ3cQklLggexcPi2yyUyBxmxMKOnOZ/ORls="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:998360070_6/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Сиофор таб. п/о плен., 1000 мг, 60 шт.
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  • Таблетница пенал - органайзер ABORNS на неделю 7 ячеек 7 дней
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  • Таблетница из 14 секций на семь дней Утро-вечер
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1883422910_9/content/content/gallery":{"title":"Таблетница из 14 секций на семь дней Утро-вечер","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/2017291/img_id609256476390730612.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/2017291/img_id609256476390730612.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/2017291/img_id609256476390730612.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/2017291/img_id609256476390730612.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/2017291/img_id609256476390730612.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/2017291/img_id609256476390730612.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 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  • VETTA / Таблетница-органайзер для таблеток аптечка для лекарств карманная в дорогу с разделителем на 14 секций, на неделю 7 дней, утро вечер
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  • Таблетница на 7 дней Органайзер для лекарств
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  • Таблетница на 7 дней Органайзер для лекарств
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  • Таблетница на 7 дней/контейнер для таблеток и витаминов на 7 дней, Immunit
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  • Синджарди таб. п/о плен., 1000 мг+5 мг, 60 шт.
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  • Таблетница на 7 дней / органайзер / бокс / контейнер на неделю для хранения таблеток и лекарств 4 приема Clear Daswerk
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  • Таблетница пенал - органайзер ABORNS на неделю 7 ячеек 7 дней
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  • Таблетница на 7 дней / органайзер / бокс / контейнер на неделю для хранения таблеток и лекарств 1 прием Компактный, Daswerk
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  • Таблетница на день мини для капсул контейнер для таблеток белый
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  • Форсига таб. п/о плен., 10 мг, 90 шт.
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  • Таблетница органайзер на неделю утро / день / вечер; Органайзер для таблеток на 7 дней; Карманная аптечка
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  • Таблетница / органайзер для хранения лекарств на неделю 7 дней/ контейнер для бисера, 15*3*2 см, прозрачная
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