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Описание

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Протамина сульфат р-р для в/в введ. введ., 10 мг/мл, 5 мл, 5 шт.

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У продавца: 
нет • На Маркете: 5.0
(1)
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Коротко о товаре

Артикул Маркета
2228054976
Рецептурный препарат
Действующее вещество
Инструкция
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Скорость введения не должна превышать 5 мг в минуту (например, 50 мг препарата вводить в течение 10 минут), так как более быстрое введение может вызвать анафилактоидную реакцию. Доза препарата зависит от способа введения гепарина. Вычисленную дозу растворяют в 300-500 мл 0,9% раствора натрия хлорида. Не следует вводить более 150 мг протамина сульфата в течение часа. \u003Cbr\u003E\n При болюсных инъекциях гепарина доза протамина сульфата уменьшается в зависимости от времени, прошедшего от введения гепарина, так как последний непрерывно удаляется из организма. 2. Если гепарин вводился внутривенно капельно, необходимо прекратить его инфузию и ввести 25-30 мг протамина сульфата.\u003Cbr\u003E\n При подкожных инъекциях гепарина доза протамина сульфата составляет 1-1,5 мг на каждые 100 ME гепарина. Первые 25-50 мг протамина сульфата следует ввести внутривенно медленно, а оставшуюся дозу - внутривенно капельно в течение 8-16 часов. Возможно дробное введение протамина сульфата, что требует контроля активированного частичного тромбопластинового времени (АЧТВ). Например, если введено подкожно 20000 ME гепарина, через 2 часа происходит резорбция гепарина из комплексов с протамином по 3333 ME гепарина, в связи с этим следующая доза протамина сульфата составляет 33 мг.\u003Cbr\u003EВ случае использования экстракорпорального кровообращения при оперативном вмешательстве доза протамина сульфата составляет 1,5 мг на каждые 100 ME гепарина. При определении дозы протамина необходимо учитывать путь введения гепарина. Максимальная длительность лечения 3 дня."},{"name":"Побочные действия","value":"Со стороны сердечно-сосудистой системы: брадикардия, артериальная гипотензия.\u003Cbr\u003EСо стороны пищеварительной системы: тошнота, рвота.\u003Cbr\u003EАллергические реакции: кожная сыпь, зуд.\u003Cbr\u003EПрочие: ощущение жара, гиперемия кожи, чувство нехватки воздуха (при чрезмерно быстром введении)."},{"name":"Фармакологическое действие","value":"Протамина сульфат является специфическим антагонистом гепарина. 1 мг протамина сульфата нейтрализует 80-120 ЕД гепарина в крови. Комплексообразование обусловлено обилием катионных групп (за счет аргинина), которые связываются с анионными центрами гепарина. Действие препарата после внутривенного введения наступает мгновенно и продолжается в течение 2 часов. После внутривенного введения образуется комплекс протамин-гепарин, который может разрушаться с высвобождением гепарина. При передозировке может снижать свертываемость крови, т.к. сам протамина сульфат проявляет антикоагулянтную активность. Исследования фармакокинетики не проводились."},{"name":"Фармакологическая группа","value":"гемостатическое средство"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный","transition":{"type":"catalog","params":{"categorySlug":"vaktsiny-syvorotki-fagi-toksiny","categoryId":"15756921","navnodeId":"72514","glfilters":["35947170:36763748"]}}},{"name":"Комплектация","value":"в комплекте с ножом ампульным или скарификатором, если необходим для ампул данного типа"},{"name":"Условия хранения","value":"В защищенном от света месте, при температуре 4-25 град.(не замораживать)"},{"name":"Передозировка","value":"Может сопровождаться кровотечением, т.к. протамин обладает собственной антикоагулянтной активностью. Лечение - симптоматическое. Взаимодействие с другими лекарственными препаратами Несовместим с цефалоспоринами и пенициллинами. Является антагонистом низко молекулярных гепаринов. Может повышать интенсивность и длительность действия недеполяризующих миорелаксантов."},{"name":"Применение при беременности и кормлении грудью","value":"Возможно, если ожидаемый эффект терапии превышает потенциальный риск для плода."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Нет данных."},{"name":"Особые указания","value":"Введение проводят под контролем свертываемости крови. Перед введением следует убедиться в адекватности объема крови больного (гиповолемия увеличивает риск коллапса)."},{"name":"Взаимодействие","value":"Несовместим с цефалоспоринами и пенициллинами. Является антагонистом низкомолекулярных гепаринов. Может повышать интенсивность и длительность действия недеполяризующих миорелаксантов."},{"name":"Регистрационный номер","value":"ЛCP-004846/10"},{"name":"Дата государственной регистрации","value":"26.03.2021"},{"name":"Владелец регистрационного удостоверения","value":"Эллара","transition":{"type":"catalog","params":{"categorySlug":"vaktsiny-syvorotki-fagi-toksiny","categoryId":"15756921","navnodeId":"72514","glfilters":["34324371:35649313","7893318:16002682"]}}},{"name":"Изготовитель","value":"Эллара"},{"name":"Фасовщик","value":"Эллара"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Протамина сульфат","transition":{"type":"catalog","params":{"categorySlug":"vaktsiny-syvorotki-fagi-toksiny","categoryId":"15756921","navnodeId":"72514","glfilters":["17796364:18012112"]}}},{"name":"Срок годности","value":"1274 дн."}]}},"fullSpecsGrouped":{"5941191353791319720":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"кровеносная система, кровеносные сосуды"},{"name":"Назначение","value":"остановка кровотечения"},{"name":"Показания к применению","value":"Кровотечения вследствие передозировки гепарина;\u003Cbr\u003Eперед операцией у больных, которые принимают гепарин с лечебной целью;\u003Cbr\u003Eпосле операций на сердце и кровеносных сосудах с экстракорпоральным кровообращением;\u003Cbr\u003Eгипергепаринемия."},{"name":"Противопоказания","value":"- Повышенная чувствительность к компонентам препарата;\u003Cbr\u003E\n- идиопатическая или врожденная гипергепаринемия (в таких случаях препарат не эффективен и может усилить кровоточивость);\u003Cbr\u003E- выраженная артериальная гипотензия;\u003Cbr\u003E- тромбоцитопения;\u003Cbr\u003E- недостаточность коры надпочечников;\u003Cbr\u003E- прием больными инсулинов, содержащих протамина сульфат, а также других лекарственных средств, содержащих протамина сульфат;\u003Cbr\u003E- аллергические реакции на рыбу в анамнезе.\u003Cbr\u003EОпыт медицинского применения у детей ограничен."},{"name":"Состав","value":"1 мл препарата содержит: протамина сульфат - 10 мг; вода для инъекций до 1 мл."},{"name":"Действующее вещество","value":"Протамина сульфат"},{"name":"Способ применения и дозы","value":"Раствор протамина сульфата вводят медленно внутривенно струйно или капельно. Скорость введения не должна превышать 5 мг в минуту (например, 50 мг препарата вводить в течение 10 минут), так как более быстрое введение может вызвать анафилактоидную реакцию. Доза препарата зависит от способа введения гепарина. Вычисленную дозу растворяют в 300-500 мл 0,9% раствора натрия хлорида. Не следует вводить более 150 мг протамина сульфата в течение часа. \u003Cbr\u003E\n При болюсных инъекциях гепарина доза протамина сульфата уменьшается в зависимости от времени, прошедшего от введения гепарина, так как последний непрерывно удаляется из организма. 2. Если гепарин вводился внутривенно капельно, необходимо прекратить его инфузию и ввести 25-30 мг протамина сульфата.\u003Cbr\u003E\n При подкожных инъекциях гепарина доза протамина сульфата составляет 1-1,5 мг на каждые 100 ME гепарина. Первые 25-50 мг протамина сульфата следует ввести внутривенно медленно, а оставшуюся дозу - внутривенно капельно в течение 8-16 часов. Возможно дробное введение протамина сульфата, что требует контроля активированного частичного тромбопластинового времени (АЧТВ). Например, если введено подкожно 20000 ME гепарина, через 2 часа происходит резорбция гепарина из комплексов с протамином по 3333 ME гепарина, в связи с этим следующая доза протамина сульфата составляет 33 мг.\u003Cbr\u003EВ случае использования экстракорпорального кровообращения при оперативном вмешательстве доза протамина сульфата составляет 1,5 мг на каждые 100 ME гепарина. При определении дозы протамина необходимо учитывать путь введения гепарина. Максимальная длительность лечения 3 дня."},{"name":"Побочные действия","value":"Со стороны сердечно-сосудистой системы: брадикардия, артериальная гипотензия.\u003Cbr\u003EСо стороны пищеварительной системы: тошнота, рвота.\u003Cbr\u003EАллергические реакции: кожная сыпь, зуд.\u003Cbr\u003EПрочие: ощущение жара, гиперемия кожи, чувство нехватки воздуха (при чрезмерно быстром введении)."},{"name":"Фармакологическое действие","value":"Протамина сульфат является специфическим антагонистом гепарина. 1 мг протамина сульфата нейтрализует 80-120 ЕД гепарина в крови. Комплексообразование обусловлено обилием катионных групп (за счет аргинина), которые связываются с анионными центрами гепарина. Действие препарата после внутривенного введения наступает мгновенно и продолжается в течение 2 часов. После внутривенного введения образуется комплекс протамин-гепарин, который может разрушаться с высвобождением гепарина. При передозировке может снижать свертываемость крови, т.к. сам протамина сульфат проявляет антикоагулянтную активность. Исследования фармакокинетики не проводились."},{"name":"Фармакологическая группа","value":"гемостатическое средство"},{"name":"Форма выпуска","value":"раствор для инъекций"},{"name":"Способ применения/введения","value":"парентеральный"},{"name":"Комплектация","value":"в комплекте с ножом ампульным или скарификатором, если необходим для ампул данного типа"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В защищенном от света месте, при температуре 4-25 град.(не замораживать)"},{"name":"Передозировка","value":"Может сопровождаться кровотечением, т.к. протамин обладает собственной антикоагулянтной активностью. Лечение - симптоматическое. Взаимодействие с другими лекарственными препаратами Несовместим с цефалоспоринами и пенициллинами. Является антагонистом низко молекулярных гепаринов. Может повышать интенсивность и длительность действия недеполяризующих миорелаксантов."},{"name":"Применение при беременности и кормлении грудью","value":"Возможно, если ожидаемый эффект терапии превышает потенциальный риск для плода."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Нет данных."},{"name":"Особые указания","value":"Введение проводят под контролем свертываемости крови. Перед введением следует убедиться в адекватности объема крови больного (гиповолемия увеличивает риск коллапса)."},{"name":"Взаимодействие","value":"Несовместим с цефалоспоринами и пенициллинами. Является антагонистом низкомолекулярных гепаринов. Может повышать интенсивность и длительность действия недеполяризующих миорелаксантов."},{"name":"Регистрационный номер","value":"ЛCP-004846/10"},{"name":"Дата государственной регистрации","value":"26.03.2021"},{"name":"Владелец регистрационного удостоверения","value":"Эллара"},{"name":"Изготовитель","value":"Эллара"},{"name":"Фасовщик","value":"Эллара"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Протамина сульфат"},{"name":"Срок годности","value":"1274 дн."}]}],"transitionId":"tr_188735844395762847"}}}}
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

Где купить

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Ещё может подойти

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Инструкция

Показания к применению

Кровотечения вследствие передозировки гепарина;
перед операцией у больных, которые принимают гепарин с лечебной целью;
после операций на сердце и кровеносных сосудах с экстракорпоральным кровообращением;
гипергепаринемия.

Противопоказания

- Повышенная чувствительность к компонентам препарата;
- идиопатическая или врожденная гипергепаринемия (в таких случаях препарат не эффективен и может усилить кровоточивость);
- выраженная артериальная гипотензия;
- тромбоцитопения;
- недостаточность коры надпочечников;
- прием больными инсулинов, содержащих протамина сульфат, а также других лекарственных средств, содержащих протамина сульфат;
- аллергические реакции на рыбу в анамнезе.
Опыт медицинского применения у детей ограничен.

Способ применения и дозы

Раствор протамина сульфата вводят медленно внутривенно струйно или капельно. Скорость введения не должна превышать 5 мг в минуту (например, 50 мг препарата вводить в течение 10 минут), так как более быстрое введение может вызвать анафилактоидную реакцию. Доза препарата зависит от способа введения гепарина. Вычисленную дозу растворяют в 300-500 мл 0,9% раствора натрия хлорида. Не следует вводить более 150 мг протамина сульфата в течение часа.
При болюсных инъекциях гепарина доза протамина сульфата уменьшается в зависимости от времени, прошедшего от введения гепарина, так как последний непрерывно удаляется из организма. 2. Если гепарин вводился внутривенно капельно, необходимо прекратить его инфузию и ввести 25-30 мг протамина сульфата.
При подкожных инъекциях гепарина доза протамина сульфата составляет 1-1,5 мг на каждые 100 ME гепарина. Первые 25-50 мг протамина сульфата следует ввести внутривенно медленно, а оставшуюся дозу - внутривенно капельно в течение 8-16 часов. Возможно дробное введение протамина сульфата, что требует контроля активированного частичного тромбопластинового времени (АЧТВ). Например, если введено подкожно 20000 ME гепарина, через 2 часа происходит резорбция гепарина из комплексов с протамином по 3333 ME гепарина, в связи с этим следующая доза протамина сульфата составляет 33 мг.
В случае использования экстракорпорального кровообращения при оперативном вмешательстве доза протамина сульфата составляет 1,5 мг на каждые 100 ME гепарина. При определении дозы протамина необходимо учитывать путь введения гепарина. Максимальная длительность лечения 3 дня.
Полная инструкция
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Протамина сульфат р-р для в/в введ. введ.
Протамина сульфат р-р для в/в введ. введ., 10 мг/мл, 5 мл, 5 шт.
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  • Иммуновенин лиоф. д/приг. р-ра д/инф., 50 мг/мл, 25 мл
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778177310_2/content/content/gallery":{"title":"Иммуновенин лиоф. д/приг. р-ра д/инф., 50 мг/мл, 25 мл","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/1349652/img_id4008250513111243060.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/1349652/img_id4008250513111243060.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/1349652/img_id4008250513111243060.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/1349652/img_id4008250513111243060.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/1349652/img_id4008250513111243060.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/1349652/img_id4008250513111243060.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"},{"src":"https://avatars.mds.yandex.net/get-mpic/5256693/img_id5510280671472984466.jpeg/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/5256693/img_id5510280671472984466.jpeg/120x160 120w, https://avatars.mds.yandex.net/get-mpic/5256693/img_id5510280671472984466.jpeg/180x240 180w, https://avatars.mds.yandex.net/get-mpic/5256693/img_id5510280671472984466.jpeg/240x320 240w, https://avatars.mds.yandex.net/get-mpic/5256693/img_id5510280671472984466.jpeg/300x400 300w, https://avatars.mds.yandex.net/get-mpic/5256693/img_id5510280671472984466.jpeg/600x800 600w","sizes":"(max-width: 1456px) 15vw, 217px"}],"firstImageLazyLoading":false,"baobabClientData":{"realTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQ39yAoPCcp5oYEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIVCJ6q888GEIf23mwYjODQByD53MEH","sign":"2FCTc+N039zfUi2vlOQ3RV+CawZPyKhQzkx1az4CzWY="},"target":"model_card"},"isNoPicturePadding":true}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778177310_2/content/content/gallery":{"name":"@marketfront/SnippetConstructor/Gallery"}}}
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  • Унитиол р-р для в/м введ. введ. и п/к, 50 мг/мл, 5 мл, 10 шт.
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  • Регевак В сусп. для в/м введ., 20 мкг/мл, 0.5 мл, 10 шт.
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  • Налоксон р-р д/ин. амп., 0.4 мг/мл, 1 мл, 10 шт.
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  • Иммуноглобулин человека против клещевого энцефалита р-р для в/м введ. введ., 1 мл, 10 шт.
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  • Лейковорин-ЛЭНС р-р для в/в и в/м введ. фл, 5 мг/мл, 5 мл, 5 шт.
    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778176467_7/content/content/toggleWishlist":{"skuId":"835907068","productId":1778176467,"offerId":"r3Q-Raqhv1h8ZQHeXAgBdg","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQ39yAoPCcp5oYEhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIWCNOj888GEPzby44DGNrUoQUg+dzBBw==","sign":"FYDOcS3QcR/o9lk2QtDIixYCiOwtB69XzzS0GmVK1q0="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778176467_7/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Реклама
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  • Превенар 13 сусп. для в/м введ., 0.5 мл/доза, 0.5 мл, 1 шт.
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  • Джадену таб. п/о плен., 180 мг, 90 шт.
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  • Клебсифаг р-р д/вн. приема, мест. и нар.прим. фл., 20 мл, 4 шт.
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