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Описание

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Силденафил таб. п/о плен., 50 мг, 4 шт.

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Коротко о товаре

Артикул Маркета
2228004388
Действующее вещество
Возраст
от 18 лет
Инструкция
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Разовая доза составляет 50 мг. С учетом эффективности и переносимости доза может быть увеличена до 100 мг или снижена до 25 мг. Максимальная разовая доза составляет 100 мг. Максимальная частота применения - 1 раз/сут. Для пожилых пациентов в возрасте старше 65 лет и при сопутствующих нарушениях функции почек или печени доза составляет 25 мг.\u003Cbr\u003EЛегочная гипертензия: внутрь по 20 мг 3 раза/сут с интервалом около 6-8 ч независимо от приема пищи. Максимальная суточная доза составляет 60 мг. Пациентам с нарушением функции почек коррекция дозы не требуется, однако при плохой переносимости дозу снижают до 20 мг 2 раза/сут."},{"name":"Побочные действия","value":"Со стороны ЦНС: возможны головная боль, приливы, головокружение, бессонница.\u003Cbr\u003EСо стороны пищеварительной системы: возможны диспепсия, астения, диарея, боли в животе, тошнота.\u003Cbr\u003EСо стороны костно-мышечной системы: артралгии, миалгии, повышение мышечного тонуса.\u003Cbr\u003EСо стороны дыхательной системы: заложенность носа, фарингит, ринит, синусит, инфекции дыхательных путей, нарушение дыхания.\u003Cbr\u003EСо стороны органа зрения: изменение зрения (легкое и преходящее; главным образом изменение цвета объектов, а также усиленное восприятие света и нарушение четкости зрения), конъюнктивит.\u003Cbr\u003EПрочие: возможны гриппоподобный синдром, развитие инфекционных заболеваний, симптомы вазодилатации, боли в спине, сыпь, инфекции мочевыводящих путей, нарушения функции предстательной железы; в единичных случаях - приапизм."},{"name":"Фармакологическое действие","value":"Селективный ингибитор циклогуанозинмонофосфат (цГМФ)-специфической ФДЭ5. ФДЭ5, ответственная за распад цГМФ, содержится не только в кавернозном теле полового члена, но и в сосудах легких.\u003Cbr\u003EВосстанавливает нарушенную эректильную функцию и обеспечивает естественный ответ на сексуальное возбуждение. Силденафил не оказывает прямого расслабляющего влияния на кавернозное тело, но активно усиливает расслабляющий эффект окиси азота на эту ткань. При сексуальном возбуждении локальное высвобождение NO под влиянием силденафила приводит к угнетению ФДЭ5 и повышению уровня цГМФ в кавернозном теле, в результате этого происходит расслабление гладких мышц и усиление кровотока в кавернозном теле.\u003Cbr\u003EЯвляясь ингибитором ФДЭ5, силденафил увеличивает содержание цГМФ в гладкомышечных клетках легочных сосудов и вызывает их расслабление. У пациентов с легочной гипертензией прием силденафила приводит к расширению сосудов легких и, в меньшей степени, других сосудов.\u003Cbr\u003EСилденафил селективен в отношении ФДЭ5 in vitro. Его активность в отношении ФДЭ5 превосходит активность в отношении других известных изоферментов ФДЭ: ФДЭ6, участвующей в передаче светового сигнала в сетчатой оболочке глаза - в 10 раз; ФДЭ1 - в 80 раз; ФДЭ2, ФДЭ4, ФДЭ7-ФДЭ11 - более чем в 700 раз. Активность силденафила в отношении ФДЭ5 более чем в 4000 раз превосходит его активность в отношении ФДЭ3, цАМФ-специфической ФДЭ, участвующей в сокращении сердца.\u003Cbr\u003EСилденафил может вызывать легкое и преходящее нарушение различения цвета (синего/зеленого). Предполагаемым механизмом нарушения цветного зрения считается угнетение ФДЭ6, которая участвует в процессе передачи света в сетчатке. Исследования in vitro показали, что влияние силденафила на ФДЭ6 в 10 раз уступает его активности в отношении ФДЭ5."},{"name":"Фармакологическая группа","value":"эректильной дисфункции средство лечения - ФДЭ5-ингибитор"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"mochepolovaia-sistema-i-polovye-gormony","categoryId":"15756910","navnodeId":"72506","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"В сухом, защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте. Срок годности - 3 года."},{"name":"Передозировка","value":"При однократном приеме препарата в дозе до 800 мг нежелательные явления были сопоставимы с таковыми при приеме препарата в более низких дозах, но встречались чаще.\u003Cbr\u003EЛечение симптоматическое. Гемодиализ не ускоряет клиренс силденафила, так как последний активно связывается с белками плазмы и не выводится почками."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Силденафил не оказывает влияния на способность к вождению автотранспорта и управлению механизмами."},{"name":"Особые указания","value":"Перед началом приема силденафила для лечения нарушений эрекции следует провести обследование сердечно-сосудистой системы.\u003Cbr\u003EС осторожностью следует применять у пациентов с анатомической деформацией полового члена (например, ангуляция, кавернозный фиброз или болезнь Пейрони) и людей с заболеваниями, которые предрасполагают к развитию приапизма (такими как серповидно-клеточная анемия, множественная миелома или лейкемия).\u003Cbr\u003EНе следует применять у пациентов, для которых сексуальная активность нежелательна.\u003Cbr\u003EС осторожностью применять у пациентов со склонностью к кровоточивости, при язвенной болезни желудка и двенадцатиперстной кишки в фазе обострения, при наследственном пигментном ретините.\u003Cbr\u003EСилденафил не применяют у пациентов в возрасте до 18 лет."},{"name":"Взаимодействие","value":"При одновременном применении ингибиторов CYP3A4 (эритромицина, циметидина) снижается клиренс силденафила, повышается концентрация силденафила в плазме крови.\u003Cbr\u003EПри одновременном применении индинавира, саквинавира, ритонавира повышается Cmax в плазме крови и AUC силденафила, что обусловлено ингибированием изофермента CYP3A4 под влиянием индинавира, саквинавира, ритонавира.\u003Cbr\u003EМожно ожидать, что более сильные ингибиторы изофермента CYP3A4, такие как кетоконазол или итраконазол, будут повышать концентрацию силденафила в плазме крови\u003Cbr\u003EПри одновременном применении с нитратами усиливается гипотензивное действие нитратов.\u003Cbr\u003EОписан случай развития симптомов рабдомиолиза после однократного приема дозы силденафила у пациента, получающего симвастатин."},{"name":"Регистрационный номер","value":"ЛП-002313"},{"name":"Дата государственной регистрации","value":"06.05.2020"},{"name":"Владелец регистрационного удостоверения","value":"Северная Звезда","transition":{"type":"catalog","params":{"categorySlug":"mochepolovaia-sistema-i-polovye-gormony","categoryId":"15756910","navnodeId":"72506","glfilters":["34324371:35649313","7893318:16002862"]}}},{"name":"Изготовитель","value":"Северная Звезда"},{"name":"Фасовщик","value":"Северная Звезда"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Силденафил","transition":{"type":"catalog","params":{"categorySlug":"mochepolovaia-sistema-i-polovye-gormony","categoryId":"15756910","navnodeId":"72506","glfilters":["17796364:18037420"]}}},{"name":"Срок годности","value":"36 мес."}]}},"fullSpecsGrouped":{"7337882392355897456":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"половая система"},{"name":"Назначение","value":"для улучшения эректильной функции"},{"name":"Показания к применению","value":"Лечение нарушений эрекции, характеризующихся неспособностью к достижению или сохранению эрекции полового члена, достаточной для удовлетворительного полового акта.\u003Cbr\u003EЛегочная гипертензия."},{"name":"Противопоказания","value":"Одновременный прием донаторов окиси азота или нитратов в любых формах, повышенная чувствительность к силденафилу."},{"name":"Состав","value":"Действующее вещество: силденафил – 50 мг\u003Cbr\u003EВспомогательные вещества: лактозы моногидрат (сахар молочный) – 60 мг, целлюлоза микрокристаллическая – 43.86 мг, кроскармеллоза натрия – 8 мг, повидон К25 – 6 мг, магния стеарат – 1.9 мг\u003Cbr/\u003E"},{"name":"Действующее вещество","value":"Силденафил"},{"name":"Способ применения и дозы","value":"Лечение нарушений эрекции: принимают внутрь примерно за 1 ч до планируемой сексуальной активности. Разовая доза составляет 50 мг. С учетом эффективности и переносимости доза может быть увеличена до 100 мг или снижена до 25 мг. Максимальная разовая доза составляет 100 мг. Максимальная частота применения - 1 раз/сут. Для пожилых пациентов в возрасте старше 65 лет и при сопутствующих нарушениях функции почек или печени доза составляет 25 мг.\u003Cbr\u003EЛегочная гипертензия: внутрь по 20 мг 3 раза/сут с интервалом около 6-8 ч независимо от приема пищи. Максимальная суточная доза составляет 60 мг. Пациентам с нарушением функции почек коррекция дозы не требуется, однако при плохой переносимости дозу снижают до 20 мг 2 раза/сут."},{"name":"Побочные действия","value":"Со стороны ЦНС: возможны головная боль, приливы, головокружение, бессонница.\u003Cbr\u003EСо стороны пищеварительной системы: возможны диспепсия, астения, диарея, боли в животе, тошнота.\u003Cbr\u003EСо стороны костно-мышечной системы: артралгии, миалгии, повышение мышечного тонуса.\u003Cbr\u003EСо стороны дыхательной системы: заложенность носа, фарингит, ринит, синусит, инфекции дыхательных путей, нарушение дыхания.\u003Cbr\u003EСо стороны органа зрения: изменение зрения (легкое и преходящее; главным образом изменение цвета объектов, а также усиленное восприятие света и нарушение четкости зрения), конъюнктивит.\u003Cbr\u003EПрочие: возможны гриппоподобный синдром, развитие инфекционных заболеваний, симптомы вазодилатации, боли в спине, сыпь, инфекции мочевыводящих путей, нарушения функции предстательной железы; в единичных случаях - приапизм."},{"name":"Фармакологическое действие","value":"Селективный ингибитор циклогуанозинмонофосфат (цГМФ)-специфической ФДЭ5. ФДЭ5, ответственная за распад цГМФ, содержится не только в кавернозном теле полового члена, но и в сосудах легких.\u003Cbr\u003EВосстанавливает нарушенную эректильную функцию и обеспечивает естественный ответ на сексуальное возбуждение. Силденафил не оказывает прямого расслабляющего влияния на кавернозное тело, но активно усиливает расслабляющий эффект окиси азота на эту ткань. При сексуальном возбуждении локальное высвобождение NO под влиянием силденафила приводит к угнетению ФДЭ5 и повышению уровня цГМФ в кавернозном теле, в результате этого происходит расслабление гладких мышц и усиление кровотока в кавернозном теле.\u003Cbr\u003EЯвляясь ингибитором ФДЭ5, силденафил увеличивает содержание цГМФ в гладкомышечных клетках легочных сосудов и вызывает их расслабление. У пациентов с легочной гипертензией прием силденафила приводит к расширению сосудов легких и, в меньшей степени, других сосудов.\u003Cbr\u003EСилденафил селективен в отношении ФДЭ5 in vitro. Его активность в отношении ФДЭ5 превосходит активность в отношении других известных изоферментов ФДЭ: ФДЭ6, участвующей в передаче светового сигнала в сетчатой оболочке глаза - в 10 раз; ФДЭ1 - в 80 раз; ФДЭ2, ФДЭ4, ФДЭ7-ФДЭ11 - более чем в 700 раз. Активность силденафила в отношении ФДЭ5 более чем в 4000 раз превосходит его активность в отношении ФДЭ3, цАМФ-специфической ФДЭ, участвующей в сокращении сердца.\u003Cbr\u003EСилденафил может вызывать легкое и преходящее нарушение различения цвета (синего/зеленого). Предполагаемым механизмом нарушения цветного зрения считается угнетение ФДЭ6, которая участвует в процессе передачи света в сетчатке. Исследования in vitro показали, что влияние силденафила на ФДЭ6 в 10 раз уступает его активности в отношении ФДЭ5."},{"name":"Фармакологическая группа","value":"эректильной дисфункции средство лечения - ФДЭ5-ингибитор"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В сухом, защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте. Срок годности - 3 года."},{"name":"Передозировка","value":"При однократном приеме препарата в дозе до 800 мг нежелательные явления были сопоставимы с таковыми при приеме препарата в более низких дозах, но встречались чаще.\u003Cbr\u003EЛечение симптоматическое. Гемодиализ не ускоряет клиренс силденафила, так как последний активно связывается с белками плазмы и не выводится почками."},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Силденафил не оказывает влияния на способность к вождению автотранспорта и управлению механизмами."},{"name":"Особые указания","value":"Перед началом приема силденафила для лечения нарушений эрекции следует провести обследование сердечно-сосудистой системы.\u003Cbr\u003EС осторожностью следует применять у пациентов с анатомической деформацией полового члена (например, ангуляция, кавернозный фиброз или болезнь Пейрони) и людей с заболеваниями, которые предрасполагают к развитию приапизма (такими как серповидно-клеточная анемия, множественная миелома или лейкемия).\u003Cbr\u003EНе следует применять у пациентов, для которых сексуальная активность нежелательна.\u003Cbr\u003EС осторожностью применять у пациентов со склонностью к кровоточивости, при язвенной болезни желудка и двенадцатиперстной кишки в фазе обострения, при наследственном пигментном ретините.\u003Cbr\u003EСилденафил не применяют у пациентов в возрасте до 18 лет."},{"name":"Взаимодействие","value":"При одновременном применении ингибиторов CYP3A4 (эритромицина, циметидина) снижается клиренс силденафила, повышается концентрация силденафила в плазме крови.\u003Cbr\u003EПри одновременном применении индинавира, саквинавира, ритонавира повышается Cmax в плазме крови и AUC силденафила, что обусловлено ингибированием изофермента CYP3A4 под влиянием индинавира, саквинавира, ритонавира.\u003Cbr\u003EМожно ожидать, что более сильные ингибиторы изофермента CYP3A4, такие как кетоконазол или итраконазол, будут повышать концентрацию силденафила в плазме крови\u003Cbr\u003EПри одновременном применении с нитратами усиливается гипотензивное действие нитратов.\u003Cbr\u003EОписан случай развития симптомов рабдомиолиза после однократного приема дозы силденафила у пациента, получающего симвастатин."},{"name":"Регистрационный номер","value":"ЛП-002313"},{"name":"Дата государственной регистрации","value":"06.05.2020"},{"name":"Владелец регистрационного удостоверения","value":"Северная Звезда"},{"name":"Изготовитель","value":"Северная Звезда"},{"name":"Фасовщик","value":"Северная Звезда"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Силденафил"},{"name":"Срок годности","value":"36 мес."}]}],"transitionId":"tr_15536761861709549145"}}}}
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Инструкция

Показания к применению

Лечение нарушений эрекции, характеризующихся неспособностью к достижению или сохранению эрекции полового члена, достаточной для удовлетворительного полового акта.
Легочная гипертензия.

Противопоказания

Одновременный прием донаторов окиси азота или нитратов в любых формах, повышенная чувствительность к силденафилу.

Способ применения и дозы

Лечение нарушений эрекции: принимают внутрь примерно за 1 ч до планируемой сексуальной активности. Разовая доза составляет 50 мг. С учетом эффективности и переносимости доза может быть увеличена до 100 мг или снижена до 25 мг. Максимальная разовая доза составляет 100 мг. Максимальная частота применения - 1 раз/сут. Для пожилых пациентов в возрасте старше 65 лет и при сопутствующих нарушениях функции почек или печени доза составляет 25 мг.
Легочная гипертензия: внутрь по 20 мг 3 раза/сут с интервалом около 6-8 ч независимо от приема пищи. Максимальная суточная доза составляет 60 мг. Пациентам с нарушением функции почек коррекция дозы не требуется, однако при плохой переносимости дозу снижают до 20 мг 2 раза/сут.
Полная инструкция
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Силденафил таб. п/о плен.
Силденафил таб. п/о плен., 50 мг, 4 шт.
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Инструкция
Нет в продаже
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4.4
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У продавца:95 оценок·12 отзывов
У всех продавцов:258 оценок·46 отзывов
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user avatar
3 недели назад • (R) • Куплен на Маркете
Достоинства: Не достойны, только боль живота несколько дней.
Недостатки: Боль в животе несколько дней.
Комментарий: Вообще не стоит употреблять.
user avatar
2 месяца назад • Имя скрыто • Куплен на Маркете
Достоинства: Работает
Недостатки: Закладывает нос
user avatar
7 месяцев назад • Имя скрыто • Куплен на Маркете
Достоинства: работает
Недостатки: всё нормально
Комментарий: то что надо
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