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Стимуляция АТ1 рецептора ответственна за патологические эффекты ангиотензина II в почках и других органах, связанных с ангиотензином II, таких как вазоконстрикция (сужение кровеносных сосудов), задержка натрия и воды, увеличенный синтез альдостерона и протеинурия. При этом эффекты, связанные со стимуляцией АТ2 рецептора, такие как вазодилятация, натрийурез и ингибирование несоответствующего клеточного роста, не подавляются. Связывание рецептора сохраняется длительное время благодаря медленной диссоциации телмисартана из его связи с АТ1 рецептором. Телмисартан не проявляет активности агониста к АТ1 рецептору, не влияет на выведение калия при хронической болезни почек"},{"name":"Состав","value":"в 1 мл содержит в качестве действующего вещества телмисартан – 10 мг и вспомогательные вещества: пропиленгликоль, мальтитол, бензалкония хлорид, вода очищенная"},{"name":"Показания к применению","value":"для снижения уровня нефротоксической протеинурии при хронической болезни почек (ХБП) и лечения сопутствующей системной гипертензии и ХБП у кошек"},{"name":"Противопоказания","value":"• гиперчувствительность к компонентам препарата (в том числе в анамнезе) • холестаз, обструкция желчевыводящих путей • выраженная печеночная недостаточность • котята моложе 6-месячного возраста • беременные и кормящие кошки • с осторожностью при хронической сердечной и печеночной недостаточности, двустороннем стенозе почечных артерий, гиповолемии, гипонатриемии, гиперкалиемии Лекарственный препарат не предназначен для применения продуктивным животным."},{"name":"Побочные действия","value":"При применении препарата НЕФРОСПАС® в соответствии с настоящей инструкцией побочных явлений и осложнений у животных, как правило, не наблюдается. При проявлении аллергических реакций применение препарата прекращают и при необходимости назначают животному антигистаминные и симптоматические средства. В редких случаях у кошек наблюдается отрыжка, рвота, диарея или разжиженный стул, гипотония, снижение количества эритроцитов и, очень редко возможно повышение уровня печеночных ферментов. После приостановления терапии указанные показатели, как правило, нормализуются в течение нескольких дней. Особенностей действия лекарственного препарата при первом применении и при отмене не выявлено."},{"name":"Передозировка","value":"При передозировке препарата НЕФРОСПАС® у кошек может наблюдаться гипотония, тахикардия или брадикардия, острая почечная недостаточность, повышение концентрации креатинина в сыворотке крови. В этом случае проводят симптоматическое и поддерживающее лечение, в зависимости от времени прошедшего после приема препарата и выраженности симптомов. Мероприятия включают в себя: провоцирование рвоты и/или промывание желудка, прием активированного угля. Следует регулярно контролировать содержание электролитов и креатинина в плазме крови."},{"name":"Взаимодействие","value":"Не наблюдалось клинических признаков гипотензии во время сопутствующей терапии амлодипином в рекомендуемой дозе для снижения протеинурии при хронической болезни почек (ХБП). Сведения о возможных взаимодействиях у кошек с ХБП при использовании телмисартана и других лекарственных препаратов, которые влияют на ренин-ангиотензин-альдостероновую систему (РААС) (таких как блокатор рецепторов ангиотензина-П (БРА) или ангиотензинпревращающий фермент (АПФ)) отсутствуют. Сведения о несовместимости препарата с лекарственными средствами других фармакологических групп, кормами и известными кормовыми добавками отсутствуют."},{"name":"Особые указания","value":"При проведении лечебных мероприятий с использованием препарата НЕФРОСПАС следует соблюдать общие правила личной гигиены и техники безопасности, предусмотренные при работе с лекарственными препаратами."},{"name":"Применение у беременных и кормящих животных","value":"не следует применять кошкам в период беременности и вскармливания приплода, а также котятам моложе 6-месячного возраста"},{"name":"Способ применения и дозы","value":"НЕФРОСПАС® применяют кошкам перорально (внутрь) один раз в сутки, принудительно с помощью шприца-дозатора или с небольшим количеством корма, в дозе 0,1 мл/кг массы животного (соответствует 1 мг телмисартана на 1 кг массы животного). Дозу лекарственного препарата и продолжительность курса лечения определяет лечащий ветеринарный врач в зависимости от физического состояния животного и течения заболевания. Длительность курса лечения не ограничена. При пропуске одной или нескольких доз НЕФРОСПАС необходимо ввести как можно скорее в терапевтической дозе. Не следует вводить двойную дозу препарата для компенсации пропущенной. После отбора лекарственного средства необходимо плотно закрыть флакон, промыть шприц-дозатор водой и дать ему подсохнуть. Во избежание возможной контаминации используйте шприц-дозатор только для применения НЕФРОСПАС®."},{"name":"Условия отпуска","value":"без рецепта"},{"name":"Условия хранения","value":"Хранят лекарственный препарат в закрытой упаковке производителя, в защищенном от прямых солнечных лучей и недоступном для детей месте, при температуре от 2°С до 25 °С"},{"name":"Регистрационный номер","value":"№ПВР-3-27.22/03779"},{"name":"Дата государственной регистрации","value":"15.12.2022"},{"name":"Дополнительная информация","value":"шприц-дозатор в комплекте"},{"name":"Срок годности","value":"700 дн."}]}},"fullSpecsGrouped":{"14956138124466092099":{"groups":[{"name":"Общие сведения","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Действующее вещество","value":"телмисартан"},{"name":"Форма выпуска","value":"суспензия для орального применения"},{"name":"Объем","value":"25 мл"},{"name":"Назначение средства","value":"для почек и мочеполовой системы"},{"name":"Вид животного","value":"кошки, собаки"},{"name":"Возраст животного","value":"взрослые, молодые, пожилые"},{"name":"Размер животного","value":"крупный, маленький, средний"}]},{"name":"Фармакологические свойства","items":[{"name":"Описание","value":"по внешнему виду препарат представляет собой суспензию от белого до светло-жёлтого цвета"},{"name":"Фармакологическая группа","value":"антагонисты рецепторов ангиотензина II (АТ1-подтип)"},{"name":"Фармакологическое действие","value":"Телмисартан, входящий в состав лекарственного препарата - специфический антагонист рецепторов типа АТ1 ангиотензина II, который вызывает дозозависимое снижение артериального кровяного давления у млекопитающих, в том числе у кошек с хронической болезнью почек, и постепенное уменьшение протеинурии.\nТелмисартан вытесняет ангиотензин II из его связи с АТ1 рецептором, избирательно связывается с АТ1 рецептором и при этом не соединяется с другими АТ рецепторами. Стимуляция АТ1 рецептора ответственна за патологические эффекты ангиотензина II в почках и других органах, связанных с ангиотензином II, таких как вазоконстрикция (сужение кровеносных сосудов), задержка натрия и воды, увеличенный синтез альдостерона и протеинурия. При этом эффекты, связанные со стимуляцией АТ2 рецептора, такие как вазодилятация, натрийурез и ингибирование несоответствующего клеточного роста, не подавляются. Связывание рецептора сохраняется длительное время благодаря медленной диссоциации телмисартана из его связи с АТ1 рецептором. Телмисартан не проявляет активности агониста к АТ1 рецептору, не влияет на выведение калия при хронической болезни почек"},{"name":"Состав","value":"в 1 мл содержит в качестве действующего вещества телмисартан – 10 мг и вспомогательные вещества: пропиленгликоль, мальтитол, бензалкония хлорид, вода очищенная"}]},{"name":"Показания и противопоказания","items":[{"name":"Показания к применению","value":"для снижения уровня нефротоксической протеинурии при хронической болезни почек (ХБП) и лечения сопутствующей системной гипертензии и ХБП у кошек"},{"name":"Противопоказания","value":"• гиперчувствительность к компонентам препарата (в том числе в анамнезе) • холестаз, обструкция желчевыводящих путей • выраженная печеночная недостаточность • котята моложе 6-месячного возраста • беременные и кормящие кошки • с осторожностью при хронической сердечной и печеночной недостаточности, двустороннем стенозе почечных артерий, гиповолемии, гипонатриемии, гиперкалиемии Лекарственный препарат не предназначен для применения продуктивным животным."},{"name":"Побочные действия","value":"При применении препарата НЕФРОСПАС® в соответствии с настоящей инструкцией побочных явлений и осложнений у животных, как правило, не наблюдается. При проявлении аллергических реакций применение препарата прекращают и при необходимости назначают животному антигистаминные и симптоматические средства. В редких случаях у кошек наблюдается отрыжка, рвота, диарея или разжиженный стул, гипотония, снижение количества эритроцитов и, очень редко возможно повышение уровня печеночных ферментов. После приостановления терапии указанные показатели, как правило, нормализуются в течение нескольких дней. Особенностей действия лекарственного препарата при первом применении и при отмене не выявлено."},{"name":"Передозировка","value":"При передозировке препарата НЕФРОСПАС® у кошек может наблюдаться гипотония, тахикардия или брадикардия, острая почечная недостаточность, повышение концентрации креатинина в сыворотке крови. В этом случае проводят симптоматическое и поддерживающее лечение, в зависимости от времени прошедшего после приема препарата и выраженности симптомов. Мероприятия включают в себя: провоцирование рвоты и/или промывание желудка, прием активированного угля. Следует регулярно контролировать содержание электролитов и креатинина в плазме крови."},{"name":"Взаимодействие","value":"Не наблюдалось клинических признаков гипотензии во время сопутствующей терапии амлодипином в рекомендуемой дозе для снижения протеинурии при хронической болезни почек (ХБП). Сведения о возможных взаимодействиях у кошек с ХБП при использовании телмисартана и других лекарственных препаратов, которые влияют на ренин-ангиотензин-альдостероновую систему (РААС) (таких как блокатор рецепторов ангиотензина-П (БРА) или ангиотензинпревращающий фермент (АПФ)) отсутствуют. Сведения о несовместимости препарата с лекарственными средствами других фармакологических групп, кормами и известными кормовыми добавками отсутствуют."},{"name":"Особые указания","value":"При проведении лечебных мероприятий с использованием препарата НЕФРОСПАС следует соблюдать общие правила личной гигиены и техники безопасности, предусмотренные при работе с лекарственными препаратами."},{"name":"Применение у беременных и кормящих животных","value":"не следует применять кошкам в период беременности и вскармливания приплода, а также котятам моложе 6-месячного возраста"},{"name":"Способ применения и дозы","value":"НЕФРОСПАС® применяют кошкам перорально (внутрь) один раз в сутки, принудительно с помощью шприца-дозатора или с небольшим количеством корма, в дозе 0,1 мл/кг массы животного (соответствует 1 мг телмисартана на 1 кг массы животного). Дозу лекарственного препарата и продолжительность курса лечения определяет лечащий ветеринарный врач в зависимости от физического состояния животного и течения заболевания. Длительность курса лечения не ограничена. При пропуске одной или нескольких доз НЕФРОСПАС необходимо ввести как можно скорее в терапевтической дозе. Не следует вводить двойную дозу препарата для компенсации пропущенной. После отбора лекарственного средства необходимо плотно закрыть флакон, промыть шприц-дозатор водой и дать ему подсохнуть. Во избежание возможной контаминации используйте шприц-дозатор только для применения НЕФРОСПАС®."}]},{"name":"Условия отпуска и хранения","items":[{"name":"Условия отпуска","value":"без рецепта"},{"name":"Условия хранения","value":"Хранят лекарственный препарат в закрытой упаковке производителя, в защищенном от прямых солнечных лучей и недоступном для детей месте, при температуре от 2°С до 25 °С"}]},{"name":"Дополнительно","items":[{"name":"Регистрационный номер","value":"№ПВР-3-27.22/03779"},{"name":"Дата государственной регистрации","value":"15.12.2022"},{"name":"Дополнительная информация","value":"шприц-дозатор в комплекте"},{"name":"Срок годности","value":"700 дн."}]}],"transitionId":"tr_10470018852782240964"}}}}
Есть противопоказания, посоветуйтесь с врачом.
Внешний вид товаров и/или упаковки может быть изменён изготовителем и отличаться от изображенных на Яндекс Маркете.
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для снижения уровня нефротоксической протеинурии при хронической болезни почек (ХБП) и лечения сопутствующей системной гипертензии и ХБП у кошек
Противопоказания
• гиперчувствительность к компонентам препарата (в том числе в анамнезе) • холестаз, обструкция желчевыводящих путей • выраженная печеночная недостаточность • котята моложе 6-месячного возраста • беременные и кормящие кошки • с осторожностью при хронической сердечной и печеночной недостаточности, двустороннем стенозе почечных артерий, гиповолемии, гипонатриемии, гиперкалиемии Лекарственный препарат не предназначен для применения продуктивным животным.
Способ применения и дозы
НЕФРОСПАС® применяют кошкам перорально (внутрь) один раз в сутки, принудительно с помощью шприца-дозатора или с небольшим количеством корма, в дозе 0,1 мл/кг массы животного (соответствует 1 мг телмисартана на 1 кг массы животного). Дозу лекарственного препарата и продолжительность курса лечения определяет лечащий ветеринарный врач в зависимости от физического состояния животного и течения заболевания. Длительность курса лечения не ограничена. При пропуске одной или нескольких доз НЕФРОСПАС необходимо ввести как можно скорее в терапевтической дозе. Не следует вводить двойную дозу препарата для компенсации пропущенной. После отбора лекарственного средства необходимо плотно закрыть флакон, промыть шприц-дозатор водой и дать ему подсохнуть. Во избежание возможной контаминации используйте шприц-дозатор только для применения НЕФРОСПАС®.
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Неделю назад • Ольга • Куплен на Маркете
Достоинства: Наконец-то у нас стали производить достойный аналог СЕМИНТРЫ по адекватной доступной цене Недостатки: Не выявила Комментарий: Уже несколько месяцев котик с ХПН принимает этот препарат. Действие заметно: стал более активным, почти заросли залысины, которые образовались в период почечного воспаления. Теперь будем принимать его постоянно и до конца.
Неделю назад • Имя скрыто • Куплен на Маркете
Достоинства: Новая система наполнения шприца. Недостатки: нет Комментарий: Как предложение, применять на шприц более стойкую краску градуировки объема, хотя и так запоминается, со временем, объем заполнения шприца
Месяц назад • tata16rt • Куплен на Маркете
Достоинства: Бюджетная цена. По качеству не хуже импортного аналога (кот принимал и то и другое, есть с чем сравнить). Недостатки: нет Комментарий: Берём этот препарат постоянно. Коту назначено ветеринаром пожизненно. Очень довольны, что в России выпускается такой замечательный препарат. Он продлевает жизнь нашему питомцу. Чему мы безмерно рады!
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