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Ветмедин — кардиотоническое средство, способствующее повышению сердечного выброса. Окончательный инотропный эффект достигается без повышения потребления кислорода и энергии. Ветмедин способствует получению более экономичных сокращений миокарда.
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Пимобендан, входящий в состав препарата Ветмедин, обладает положительным инотропным действием и выраженным вазодилатирующим эффектом. В отличие от сердечных гликозидов положительный инотропный эффект препарата обусловлен двумя механизмами: повышением чувствительности к кальцию волокон сердечной мышцы и угнетению фосфодиэстеразы. Вазодилатирующий эффект связан с ингибированием активности фосфодиэстеразы III. Благодаря наличию положительного инотропного и вазодилатирующего действия при сердечной недостаточности препарат повышает силу сердечных сокращений и уменьшает как преднагрузку, так и постнагрузку. После перорального применения пимобендан быстро всасывается в кровь, и его биодоступность составляет 60-63%. Период полураспада пимобендана в плазме крови составляет 0,4±0,1 часа, а период полувыведения его активного метаболита составляет 2±0,3 часа. Большая часть препарата выводится из организма животных с калом. 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Доза препарата назначается ветеринарным врачом в зависимости от тяжести течения заболевания и состояния животного. Суточная доза пимобендана составляет от 0.2 мг до 0.6 мг на 1 кг массы тела животного и делится на два приема. При застойной сердечной недостаточности Ветмедин® применяют собакам пожизненно с подбором индивидуальной дозы. Особенностей действия препарата при первом приеме или отмене не выявлено. Следует избегать пропуска очередной дозы препарата, т.к. это может привести к снижению его эффективности. 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Запрещается применение Ветмедина при гипертрофической кардиомиопатии и клинических состояниях, при которых не может быть увеличен сердечный выброс крови из-за функциональных или анатомических особенностей (например, стеноз аорты). Препарат не предназначен для применения продуктивным животным."},{"name":"Побочные действия","value":"побочных явлений и осложнений при использовании Ветмедина в соответствии с настоящей инструкцией по применению, как правило, не наблюдается. В редких случаях могут возникать диарея, летаргия, анорексия. Также у некоторых животных могут наблюдаться рвота, тахикардия, которые могут быть устранены снижением дозы препарата."},{"name":"Передозировка","value":"при передозировке препарата у животного могут наблюдаться рвота, апатия, тахикардия, шумы в сердце или снижение давления. В случае передозировки следует прекратить дачу препарата и обратиться к ветеринарному врачу. При этом рекомендуется незамедлительное проведение неспецифической дезактивации препарата, включая возможное применение активированного угля и/или поддержание водно-электролитного баланса, учитывая состояние животного."},{"name":"Взаимодействие","value":"при одновременном применении препарата Ветмедин с блокатором медленных кальциевых каналов (верапамил) и бета-блокатором (пропранололом) действие пимобендана ослабляется. Препарат можно применять одновременно с сердечным гликозидом уабаином. Информация об особенностях взаимодействия с лекарственными препаратами других фармакологических групп отсутствует."},{"name":"Применение у беременных и кормящих животных","value":"Препарат назначают щенным и кормящим сукам в случае, если потенциальный риск для матери превосходит риск для плода и щенков. Препарат используется для непродуктивных животных."},{"name":"Способ применения и дозы","value":"применяют собакам перорально, за 1 ч до кормления. 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сердечная недостаточность, вызванная дилатационной кардиомиопатией, недостаточностью двустворчатого или трехстворчатого клапана, которая сопровождается характерными симптомами (кашлем, одышкой, обмороками, понижением активности, непереносимостью физических нагрузок или асцитом)
Противопоказания
противопоказанием к применению Ветмедина является повышенная чувствительность животного к его компонентам. Запрещается применение Ветмедина при гипертрофической кардиомиопатии и клинических состояниях, при которых не может быть увеличен сердечный выброс крови из-за функциональных или анатомических особенностей (например, стеноз аорты). Препарат не предназначен для применения продуктивным животным.
Способ применения и дозы
применяют собакам перорально, за 1 ч до кормления. Доза препарата назначается ветеринарным врачом в зависимости от тяжести течения заболевания и состояния животного. Суточная доза пимобендана составляет от 0.2 мг до 0.6 мг на 1 кг массы тела животного и делится на два приема. При застойной сердечной недостаточности Ветмедин® применяют собакам пожизненно с подбором индивидуальной дозы. Особенностей действия препарата при первом приеме или отмене не выявлено. Следует избегать пропуска очередной дозы препарата, т.к. это может привести к снижению его эффективности. В случае пропуска одной дозы применение препарата возобновляют в той же дозе и по той же схеме.
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17 часов назад • Алина • Куплен на Маркете
Достоинства: Оригинальное лекарство по приемлемой цене
4 дня назад • Алексей Сергеев • Куплен на Маркете
Достоинства: Собака с удовольствием есть таблетку сама. Комментарий: Берем шпицу на пожизненной основе. Собаке таблетки помогают. Кушает их сам.
4 дня назад • Евгений Винокуров • Куплен на Маркете
Недостатки: Нет Комментарий: Собака не жалуется, бегает. Не вещь и не продукты, попробовать и сказать ничего не могу
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