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Тизанидин-СЗ таб., 4 мг, 30 шт.

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Дозировка: 4 мг

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Коротко о товаре

Артикул Маркета
3123877776
Действующее вещество
Форма выпуска
таблетки
Инструкция
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Применение препарата Тизанидин-СЗ у пациентов данной популяции не рекомендовано.\u003Cbr\u003E"},{"name":"Состав","value":"1 таблетка содержит:\u003Cbr\u003Eдействующее вещество: тизанидина гидрохлорид - 2,288 мг/ 4,576 мг в пересчете на тизанидин - 2 мг/ 4 мг;\u003Cbr\u003Eвспомогательные вещества: лактозы моногидрат - 70,0 мг/140,0 мг; целлюлоза микрокристаллическая 102 - 64,912 мг/129,824 мг; кремния диоксид коллоидный (аэросил) - 1,4 мг/ 2,8 мг; магния стеарат - 1,4 мг/ 2,8 мг.\u003Cbr\u003E"},{"name":"Действующее вещество","value":"Тизанидин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-travm-boli-v-myshtsakh-i-sustavakh","categoryId":"15756903","navnodeId":"25542230","glfilters":["27144131:28708611"]}}},{"name":"Способ применения и дозы","value":"Препарат Тизанидин-СЗ обладает узким терапевтическим индексом и высокой вариабельностью концентрации тизанидина в плазме крови, поэтому необходим тщательный подбор дозы.\u003Cbr\u003EДозу и режим дозирования следует подбирать индивидуально в зависимости от потребностей пациента. Применение препарата в начальной дозе 2 мг 3 раза в день снижает риск развития побочных эффектов.\u003Cbr\u003EПрепарат принимают внутрь. Таблетки 2 мг и 4 мг могут быть разделены на две равные части.\u003Cbr\u003EПри болезненном мышечном спазме препарат Тизанидин-СЗ применяют, как правило, в дозе 2 мг или 4 мг 3 раза в сутки.\u003Cbr\u003EВ тяжелых случаях возможно дополнительное применение 2 мг или 4 мг (предпочтительно перед сном из-за возможного усиления сонливости).\u003Cbr\u003EПри спастичности скелетных мышц, обусловленной неврологическими заболеваниями, начальная суточная доза не должна превышать 6 мг, разделенных на 3 приема. Дозу можно повышать постепенно, на 2-4 мг, с интервалами от 3-4 до 7 дней. Как правило, оптимальный терапевтический эффект достигается при суточной дозе от 12 до 24 мг, разделенной на 3 или 4 приема через равные промежутки времени. Не следует превышать дозу 36 мг в сутки.\u003Cbr\u003EПрименение у пациентов старше 65 лет\u003Cbr\u003EОпыт применения препарата Тизанидин-СЗ у пациентов в возрасте старше 65 лет и старше ограничен. Рекомендуется начинать терапию с минимальной дозы с постепенным повышением до достижения оптимального соотношения переносимости и эффективности терапии.\u003Cbr\u003EПрименение у пациентов с нарушениями функции почек Лечение пациентов с почечной недостаточностью (КК менее 25 мл/мин) рекомендуется начинать с дозы 2 мг 1 раз в день. Повышение дозы проводят малыми \"шагами\" с учетом переносимости и эффективности. При необходимости достижения более выраженного эффекта, рекомендуется сначала увеличить дозу, применяемую 1 раз в сутки, после чего увеличивают кратность применения.\u003Cbr\u003EПрименение у пациентов с нарушениями функции печени\u003Cbr\u003EПрименение препарата Тизанидин-СЗ у пациентов с нарушением функции печени тяжелой степени противопоказано.\u003Cbr\u003EУ пациентов с нарушением функции печени средней степени тяжести препарат следует применять с осторожностью; рекомендовано начинать терапию с минимальной дозы, с постепенным повышением до достижения оптимального соотношения переносимости и эффективности терапии. Рекомендации по контролю показателей функции печени указаны в разделе \"Особые указания\".\u003Cbr\u003EПрерывание лечения\u003Cbr\u003EПри прекращении терапии препаратом Тизанидин-СЗ с целью уменьшения риска развития рикошетной гипертензии и тахикардии следует медленно снижать дозу до полной отмены препарата, в особенности у пациентов, получающих высокие дозы препарата в течение длительного времени.\u003Cbr\u003E"},{"name":"Побочные действия","value":"При приеме малых доз, рекомендуемых для купирования болезненного мышечного спазма, отмечались сонливость, повышенная утомляемость, головокружение, сухость во рту, снижение АД, тошнота, желудочно-кишечные расстройства, повышение активности печеночных трансаминаз. Обычно вышеописанные побочные реакции умеренно выражены и преходящи.\u003Cbr\u003EПри приеме более высоких доз, рекомендуемых для лечения спастичности, вышеперечисленные HP возникают чаще и более выражены, однако они редко требуют прекращения отмены препарата в связи с тяжестью ПР. Кроме того, могут возникать следующие явления: брадикардия, мышечная слабость, бессонница, нарушения сна, галлюцинации, гепатит.\u003Cbr\u003EНежелательные реакции (HP) сгруппированы в соответствии с классификацией органов и систем органов MedDRA, в пределах каждой группы перечислены в порядке уменьшения частоты встречаемости. Для оценки частоты развития HP использованы следующие критерии: очень часто (≥ 1/10); часто (от ≥ 1/100, \u003C 1/10); нечасто (≥ 1/1000, \u003C1/100); редко (≥ 1/10000, \u003C 1/1000); очень редко (\u003C 1/10000), включая отдельные сообщения.\u003Cbr\u003EНарушения со стороны нервной системы: очень часто - сонливость, головокружение.\u003Cbr\u003EНарушения психики: часто - бессонница, нарушения сна.\u003Cbr\u003EНарушения со стороны сердца: нечасто - брадикардия.\u003Cbr\u003EНарушения со стороны сосудов: часто - снижение АД (в отдельных случаях выраженное, вплоть до циркуляторного коллапса и потери сознания).\u003Cbr\u003EНарушения со стороны пищеварительной системы: очень часто - желудочно-кишечные расстройства, сухость во рту; часто - тошнота.\u003Cbr\u003EНарушения со стороны скелетно-мышечной и соединительной ткани: очень часто - мышечная слабость.\u003Cbr\u003EОбщие расстройства и нарушения в месте введения: очень часто - повышенная утомляемость.\u003Cbr\u003EЛабораторные и инструментальные данные: часто - повышение активности печеночных трансаминаз. При резкой отмене препарата Тизанидин-СЗ после продолжительного лечения и/или приема высоких доз препарата (а также после одновременного применения вместе с гипотензивными препаратами) отмечалось развитие тахикардии и повышения АД, способное в отдельных случаях привести к острому нарушению мозгового кровообращения, в связи с чем дозу препарата Тизанидин-СЗ следует снижать постепенно до полной отмены препарата.\u003Cbr\u003EОтдельные сообщения о HP по данным применения в клинической практике\u003Cbr\u003EПоскольку в пострегистрационном периоде сообщения о HP поступают в добровольном порядке из популяции неопределенного размера, достоверно оценить частоту их возникновения не представляется возможным (частота неизвестна).\u003Cbr\u003EНарушения со стороны иммунной системы: реакции гиперчувствительности, включая анафилактические реакции, ангионевротический отек и крапивницу.\u003Cbr\u003EНарушения психики: галлюцинации, спутанность сознания.\u003Cbr\u003EНарушения со стороны нервной системы: головокружение.\u003Cbr\u003EНарушения со стороны органа зрения: затуманивание зрения.\u003Cbr\u003EНарушения со стороны печени и желчевыводящих путей: гепатит, печеночная недостаточность.\u003Cbr\u003EНарушения со стороны кожи и подкожных тканей: кожная сыпь, эритема, кожный зуд, дерматит.\u003Cbr\u003EОбщие расстройства и нарушения вместе введения: астения, синдром отмены.\u003Cbr\u003EЕсли любые из указанных в инструкции побочных эффектов усугубляются, или Вы заметите любые другие побочные эффекты не указанные в инструкции, сообщите об этом врачу.\u003Cbr\u003E"},{"name":"Фармакологическое действие","value":"Тизанидин - миорелаксант центрального действия, Основная точка приложения его действия находится в спинном мозге. Стимулируя пресинаптические альфа2-рецепторы, он подавляет высвобождение возбуждающих аминокислот, которые стимулируют рецепторы к N-метил-В- аспартату (NMDA-рецепторы). Вследствие этого на уровне промежуточных нейронов спинного мозга происходит подавление полисинаптической передачи возбуждения. Поскольку именно этот механизм отвечает за избыточный мышечный тонус, то при его подавлении мышечный тонус снижается. В дополнение к миорелаксирующим свойствам, тизанидин оказывает также центральный умеренно выраженный анальгезирующий эффект.\u003Cbr\u003EПрепарат Тизанидин-СЗ эффективен как при остром болезненном мышечном спазме, так и при хронической спастичности спинального и церебрального генеза. Уменьшает спастичность и клонические судороги, вследствие чего снижается сопротивление пассивным движениям и увеличивается объем активных движений.\u003Cbr\u003EМиорелаксирующий аффект (измерение по шкале Ашворта и с помощью \"маятникового\" теста) и побочные действия (снижение частоты сердечных сокращений (ЧСС) и снижение артериального давления (АД)) препарата зависят от концентрации тизанидина в плазме крови.\u003Cbr\u003E"},{"name":"Фармакологическая группа","value":"миорелаксант центрального действия"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-travm-boli-v-myshtsakh-i-sustavakh","categoryId":"15756903","navnodeId":"25542230","glfilters":["35947170:36763744"]}}},{"name":"Условия хранения","value":"В защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"К настоящему времени получено несколько сообщений о передозировке препаратом Тизанидин-СЗ, включая случай, когда принятая доза составила 400 мг. Во всех случаях выздоровление прошло без особенностей.\u003Cbr\u003EСимптомы: тошнота, рвота, снижение АД, удлинение интервала QT (с), головокружение, сонливость, миоз, беспокойство, угнетение дыхания, кома.\u003Cbr\u003EЛечение. Для выведения препарата из организма рекомендуется многократное применение активированного угля. Форсированный диурез также, возможно, ускорит выведение тизанидина. В дальнейшем проводят симптоматическое лечение.\u003Cbr\u003E"},{"name":"Применение при беременности и кормлении грудью","value":"Беременность\u003Cbr\u003EПоскольку контролируемые исследования применения тизанидина у беременных женщин не проводились, его не следует применять в период беременности, за исключением тех случаев, когда потенциальная польза превышает возможный риск.\u003Cbr\u003EВ исследованиях у животных не выявлено явлений тератогенности. При применении в дозах 10 и 30 мг/кг в сутки у животных отмечено увеличение срока гестации, зарегистрированы случаи пренатальной и постнатальной потери плода, а также задержка развития плода. При применении вышеуказанных доз у самок отмечались выраженные признаки миорелаксации и седации. Исходя из площади поверхности тела, указанные дозы превышали максимальную рекомендуемую дозу для человека (0,72 мг/кг в сутки) в 2,2 и 6,7 раз.\u003Cbr\u003EГрудное вскармливание\u003Cbr\u003EВ исследованиях у животных тизанидин выделялся в небольших количествах с молоком лактирующих самок. Не следует применять препарат в период грудного вскармливания, так как нет данных о проникновении тизанидина в грудное молоко у человека.\u003Cbr\u003EТест на беременность\u003Cbr\u003EПеред началом применения препарата Тизанидин-СЗ у пациенток с сохраненным репродуктивным потенциалом рекомендовано получить результат теста на беременность.\u003Cbr\u003EВлияние на фертильность\u003Cbr\u003EВ исследованиях у животных не отмечалось неблагоприятного влияния на фертильность особей мужского и женского пола при применении тизанидина в дозе 10 мг/кг в сутки и 3 мг/кг/ сутки соответственно. Отмечалось уменьшение фертильности у особей мужского пола, получавших тизанидин в дозе, превышающей 30 мг/кг в сутки, и у особей женского пола - в дозе, превышающей 10 мг/кг сутки. Исходя из площади поверхности тела, указанные дозы превышали максимальную рекомендуемую дозу для человека (0,72 мг/кг в сутки) в 2,2 и 6,7 раз. При применении указанных доз со стороны матери отмечались поведенческие эффекты и клинические признаки, включающие выраженную седацию, уменьшение массы тела и атаксию.\u003Cbr\u003E"},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Пациентам, у которых на фоне применения препарата отмечается сонливость, головокружение или какие-либо признаки артериальной гипотензии следует рекомендовать воздержаться от видов деятельности, требующих высокой концентрации внимания и быстрой реакции, например, управления транспортными средствами и механизмами."},{"name":"Особые указания","value":"Гипотензия может возникать на фоне применения препарата Тизанидин-СЗ, а также как результат лекарственного взаимодействия с ингибиторами изофермента CYP1A2 и/или гипотензивными препаратами. Выраженное снижение АД может приводить к потере сознания и циркуляторному коллапсу.\u003Cbr\u003EСообщалось о случаях нарушений функции печени, связанных с тизанидином, однако при применении суточной дозы до 12 мг эти случаи отмечались редко. В связи с этим рекомендуется контролировать функциональные \"печеночные пробы\" 1 раз в месяц в первые 4 месяца лечения у пациентов, которые получают тизанидин в суточной дозе 12 мг и выше, а также в тех случаях, когда наблюдаются клинические признаки, позволяющие предположить нарушение функции печени, такие как необъяснимая тошнота, анорексия, чувство усталости. В случае, когда активность аланинаминотрансферазы (АЛТ) и аспартатаминотрансферазы (ACT) в сыворотке стойко превышают верхнюю границу нормы в 3 раза и более, применение препарата Тизанидин-СЗ следует прекратить.\u003Cbr\u003EКонтрацепция\u003Cbr\u003EСледует информировать пациенток с сохраненным репродуктивным потенциалом о неблагоприятном влиянии препарата на развивающийся плод, выявленном в исследованиях у животных. Во время применения препарата, а также в течение 1 суток после прекращения приема препарата пациенткам с сохраненным репродуктивным потенциалом следует использовать надежные способы контрацепции (при правильном и длительном использовании которых частота наступления беременности составляет \u003C 1 %).\u003Cbr\u003E"},{"name":"Взаимодействие","value":"При применении препарата Тизанидин-СЗ с ингибиторами изофермента CYP1A2 возможно повышение концентрации тизанидина в плазме крови. В свою очередь, повышение концентрации тизанидина в плазме крови может приводить к симптомам передозировки препаратом, в том числе удлинению интервала QT(c).\u003Cbr\u003EОдновременное применение препарата Тизанидин-СЗ с индукторами изофермента CYP1A2 может приводить к снижению концентрации тизанидина в плазме крови, что может приводить к уменьшению терапевтического эффекта препарата.\u003Cbr\u003EПротивопоказанные комбинации с тизанидином\u003Cbr\u003EОдновременное применение тизанидина с флувоксамином или ципрофлоксацином, ингибиторами изофермента CYP1А2, противопоказано. При применении тизанидина с флувоксамином или ципрофлоксацином отмечается соответственно 33-кратное и 10-кратное увеличению AUC тизанидина. Результатом одновременного применения может оказаться значимая и длительная гипотензия сопровождающаяся сонливостью, головокружением, снижением скорости психомоторных реакций (в отдельных случаях вплоть до циркуляторного коллапса и потери сознания).\u003Cbr\u003EНе рекомендуемые комбинации с тизанидином\u003Cbr\u003EНе рекомендуется применять тизанидин одновременно с другими ингибиторами изофермента CYP1A2 - антиаритмическими препаратами (амиодарон, мексилетин, пропафенон), циметидином, некоторыми фторхинолонами (эноксацин, пефлоксацин, норфлоксацин), рофекоксибом, пероральными контрацептивами, тиклопидином.\u003Cbr\u003EКомбинации с тизанидином, требующие соблюдения осторожности\u003Cbr\u003EНеобходимо соблюдать осторожность при одновременном применении препарата Тизанидин-СЗ с препаратами, удлиняющими интервал QT (например, цизаприд, амитриптилин, азитромицин).\u003Cbr\u003EГипотензивные препараты\u003Cbr\u003EОдновременное применение препарата Тизанидин-СЗ с гипотензивными препаратами, включая диуретики, иногда может вызывать выраженное снижение АД (в отдельных случаях вплоть до циркуляторного коллапса и потери сознания) и брадикардию.\u003Cbr\u003EПри резкой отмене препарата Тизанидин-СЗ после одновременного применения с гипотензивными препаратами отмечалось развитие тахикардии и повышение АД, которое в отдельных случаях может привести к острому нарушению мозгового кровообращения.\u003Cbr\u003EРифампицин\u003Cbr\u003EОдновременный прием тизанидина и рифампицина приводит к 50 % снижению концентрации тизанидина в плазме крови. Вследствие этого терапевтическое действие препарата может снижаться, что может иметь клиническую значимость для некоторых пациентов. Следует избегать длительного одновременного применения рифампицина и тизанидина при невозможности рекомендуется тщательный подбор дозы тизанидина (увеличение).\u003Cbr\u003EКурение табака\u003Cbr\u003EСистемная биодоступность тизанидина у курящих пациентов (более 10 сигарет в день) снижена примерно на 30 %. Длительная терапия препаратом у пациентов данной категории может потребовать более высоких доз тизанидина, чем средние терапевтические.\u003Cbr\u003EАлкоголь\u003Cbr\u003EВо время терапии препаратом следует избегать приема алкоголя, так как он может повысить вероятность развития нежелательных явлений (например, снижения АД и заторможенности). Тизанидин может усиливать угнетающее действие алкоголя на центральную нервную систему.\u003Cbr\u003EДругие лекарственные средства\u003Cbr\u003EСедативные, снотворные препараты (бензодиазепин, баклофен) и другие препараты, такие как антигистаминные препараты, могут также усиливать седативный эффект тизанидина. Следует избегать приема препарата с другими агонистами альфа2-адренорецепторов (например, клонидином) вследствие потенциального усиления гипотензивного эффекта.\u003Cbr\u003E"},{"name":"Регистрационный номер","value":"ЛП-005748"},{"name":"Дата государственной регистрации","value":"27.08.2019"},{"name":"Владелец регистрационного удостоверения","value":"Северная Звезда","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-travm-boli-v-myshtsakh-i-sustavakh","categoryId":"15756903","navnodeId":"25542230","glfilters":["34324371:35649313","7893318:16002862"]}}},{"name":"Изготовитель","value":"Северная Звезда"},{"name":"Фасовщик","value":"Северная Звезда"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Тизанидин","transition":{"type":"catalog","params":{"categorySlug":"sredstva-ot-travm-boli-v-myshtsakh-i-sustavakh","categoryId":"15756903","navnodeId":"25542230","glfilters":["17796364:18025487"]}}},{"name":"Срок годности","value":"1 г."}]}},"fullSpecsGrouped":{"15555781340132293736":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"костная система"},{"name":"Назначение","value":"межпозвоночная грыжа, мышечные боли и спазмы, остеоартроз, спастичность скелетных мышц"},{"name":"Показания к применению","value":"Болезненный мышечный спазм:\u003Cbr\u003Eсвязанный со статическими и функциональными заболеваниями позвоночника (шейный и поясничный синдромы);\u003Cbr\u003Eпосле хирургических вмешательств, например, по поводу грыжи межпозвонкового диска или остеоартроза тазобедренного сустава.\u003Cbr\u003EСпастичность скелетных мышц при неврологических заболеваниях, например, при рассеянном склерозе, хронической миелопатии, дегенеративных заболеваниях спинного мозга, последствиях нарушений мозгового кровообращения и детском церебральном параличе (пациенты старше 18 лет).\u003Cbr\u003E"},{"name":"Противопоказания","value":"Повышенная чувствительность к тизанидину или к любому другому компоненту препарата.\u003Cbr\u003E- Нарушение функции печени тяжелой степени.\u003Cbr\u003E- Одновременное применение с мощными ингибиторами изофермента CYP1А2, такими как флувоксамин или ципрофлоксацин.\u003Cbr\u003E- Не рекомендовано пациентам с редкими наследственными заболеваниями, такими как дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция, так как лекарственная форма содержит лактозу.\u003Cbr\u003E- Опыт применения препарата у пациентов младше 18 лет ограничен. Применение препарата Тизанидин-СЗ у пациентов данной популяции не рекомендовано.\u003Cbr\u003E"},{"name":"Состав","value":"1 таблетка содержит:\u003Cbr\u003Eдействующее вещество: тизанидина гидрохлорид - 2,288 мг/ 4,576 мг в пересчете на тизанидин - 2 мг/ 4 мг;\u003Cbr\u003Eвспомогательные вещества: лактозы моногидрат - 70,0 мг/140,0 мг; целлюлоза микрокристаллическая 102 - 64,912 мг/129,824 мг; кремния диоксид коллоидный (аэросил) - 1,4 мг/ 2,8 мг; магния стеарат - 1,4 мг/ 2,8 мг.\u003Cbr\u003E"},{"name":"Действующее вещество","value":"Тизанидин"},{"name":"Способ применения и дозы","value":"Препарат Тизанидин-СЗ обладает узким терапевтическим индексом и высокой вариабельностью концентрации тизанидина в плазме крови, поэтому необходим тщательный подбор дозы.\u003Cbr\u003EДозу и режим дозирования следует подбирать индивидуально в зависимости от потребностей пациента. Применение препарата в начальной дозе 2 мг 3 раза в день снижает риск развития побочных эффектов.\u003Cbr\u003EПрепарат принимают внутрь. Таблетки 2 мг и 4 мг могут быть разделены на две равные части.\u003Cbr\u003EПри болезненном мышечном спазме препарат Тизанидин-СЗ применяют, как правило, в дозе 2 мг или 4 мг 3 раза в сутки.\u003Cbr\u003EВ тяжелых случаях возможно дополнительное применение 2 мг или 4 мг (предпочтительно перед сном из-за возможного усиления сонливости).\u003Cbr\u003EПри спастичности скелетных мышц, обусловленной неврологическими заболеваниями, начальная суточная доза не должна превышать 6 мг, разделенных на 3 приема. Дозу можно повышать постепенно, на 2-4 мг, с интервалами от 3-4 до 7 дней. Как правило, оптимальный терапевтический эффект достигается при суточной дозе от 12 до 24 мг, разделенной на 3 или 4 приема через равные промежутки времени. Не следует превышать дозу 36 мг в сутки.\u003Cbr\u003EПрименение у пациентов старше 65 лет\u003Cbr\u003EОпыт применения препарата Тизанидин-СЗ у пациентов в возрасте старше 65 лет и старше ограничен. Рекомендуется начинать терапию с минимальной дозы с постепенным повышением до достижения оптимального соотношения переносимости и эффективности терапии.\u003Cbr\u003EПрименение у пациентов с нарушениями функции почек Лечение пациентов с почечной недостаточностью (КК менее 25 мл/мин) рекомендуется начинать с дозы 2 мг 1 раз в день. Повышение дозы проводят малыми \"шагами\" с учетом переносимости и эффективности. При необходимости достижения более выраженного эффекта, рекомендуется сначала увеличить дозу, применяемую 1 раз в сутки, после чего увеличивают кратность применения.\u003Cbr\u003EПрименение у пациентов с нарушениями функции печени\u003Cbr\u003EПрименение препарата Тизанидин-СЗ у пациентов с нарушением функции печени тяжелой степени противопоказано.\u003Cbr\u003EУ пациентов с нарушением функции печени средней степени тяжести препарат следует применять с осторожностью; рекомендовано начинать терапию с минимальной дозы, с постепенным повышением до достижения оптимального соотношения переносимости и эффективности терапии. Рекомендации по контролю показателей функции печени указаны в разделе \"Особые указания\".\u003Cbr\u003EПрерывание лечения\u003Cbr\u003EПри прекращении терапии препаратом Тизанидин-СЗ с целью уменьшения риска развития рикошетной гипертензии и тахикардии следует медленно снижать дозу до полной отмены препарата, в особенности у пациентов, получающих высокие дозы препарата в течение длительного времени.\u003Cbr\u003E"},{"name":"Побочные действия","value":"При приеме малых доз, рекомендуемых для купирования болезненного мышечного спазма, отмечались сонливость, повышенная утомляемость, головокружение, сухость во рту, снижение АД, тошнота, желудочно-кишечные расстройства, повышение активности печеночных трансаминаз. Обычно вышеописанные побочные реакции умеренно выражены и преходящи.\u003Cbr\u003EПри приеме более высоких доз, рекомендуемых для лечения спастичности, вышеперечисленные HP возникают чаще и более выражены, однако они редко требуют прекращения отмены препарата в связи с тяжестью ПР. Кроме того, могут возникать следующие явления: брадикардия, мышечная слабость, бессонница, нарушения сна, галлюцинации, гепатит.\u003Cbr\u003EНежелательные реакции (HP) сгруппированы в соответствии с классификацией органов и систем органов MedDRA, в пределах каждой группы перечислены в порядке уменьшения частоты встречаемости. Для оценки частоты развития HP использованы следующие критерии: очень часто (≥ 1/10); часто (от ≥ 1/100, \u003C 1/10); нечасто (≥ 1/1000, \u003C1/100); редко (≥ 1/10000, \u003C 1/1000); очень редко (\u003C 1/10000), включая отдельные сообщения.\u003Cbr\u003EНарушения со стороны нервной системы: очень часто - сонливость, головокружение.\u003Cbr\u003EНарушения психики: часто - бессонница, нарушения сна.\u003Cbr\u003EНарушения со стороны сердца: нечасто - брадикардия.\u003Cbr\u003EНарушения со стороны сосудов: часто - снижение АД (в отдельных случаях выраженное, вплоть до циркуляторного коллапса и потери сознания).\u003Cbr\u003EНарушения со стороны пищеварительной системы: очень часто - желудочно-кишечные расстройства, сухость во рту; часто - тошнота.\u003Cbr\u003EНарушения со стороны скелетно-мышечной и соединительной ткани: очень часто - мышечная слабость.\u003Cbr\u003EОбщие расстройства и нарушения в месте введения: очень часто - повышенная утомляемость.\u003Cbr\u003EЛабораторные и инструментальные данные: часто - повышение активности печеночных трансаминаз. При резкой отмене препарата Тизанидин-СЗ после продолжительного лечения и/или приема высоких доз препарата (а также после одновременного применения вместе с гипотензивными препаратами) отмечалось развитие тахикардии и повышения АД, способное в отдельных случаях привести к острому нарушению мозгового кровообращения, в связи с чем дозу препарата Тизанидин-СЗ следует снижать постепенно до полной отмены препарата.\u003Cbr\u003EОтдельные сообщения о HP по данным применения в клинической практике\u003Cbr\u003EПоскольку в пострегистрационном периоде сообщения о HP поступают в добровольном порядке из популяции неопределенного размера, достоверно оценить частоту их возникновения не представляется возможным (частота неизвестна).\u003Cbr\u003EНарушения со стороны иммунной системы: реакции гиперчувствительности, включая анафилактические реакции, ангионевротический отек и крапивницу.\u003Cbr\u003EНарушения психики: галлюцинации, спутанность сознания.\u003Cbr\u003EНарушения со стороны нервной системы: головокружение.\u003Cbr\u003EНарушения со стороны органа зрения: затуманивание зрения.\u003Cbr\u003EНарушения со стороны печени и желчевыводящих путей: гепатит, печеночная недостаточность.\u003Cbr\u003EНарушения со стороны кожи и подкожных тканей: кожная сыпь, эритема, кожный зуд, дерматит.\u003Cbr\u003EОбщие расстройства и нарушения вместе введения: астения, синдром отмены.\u003Cbr\u003EЕсли любые из указанных в инструкции побочных эффектов усугубляются, или Вы заметите любые другие побочные эффекты не указанные в инструкции, сообщите об этом врачу.\u003Cbr\u003E"},{"name":"Фармакологическое действие","value":"Тизанидин - миорелаксант центрального действия, Основная точка приложения его действия находится в спинном мозге. Стимулируя пресинаптические альфа2-рецепторы, он подавляет высвобождение возбуждающих аминокислот, которые стимулируют рецепторы к N-метил-В- аспартату (NMDA-рецепторы). Вследствие этого на уровне промежуточных нейронов спинного мозга происходит подавление полисинаптической передачи возбуждения. Поскольку именно этот механизм отвечает за избыточный мышечный тонус, то при его подавлении мышечный тонус снижается. В дополнение к миорелаксирующим свойствам, тизанидин оказывает также центральный умеренно выраженный анальгезирующий эффект.\u003Cbr\u003EПрепарат Тизанидин-СЗ эффективен как при остром болезненном мышечном спазме, так и при хронической спастичности спинального и церебрального генеза. Уменьшает спастичность и клонические судороги, вследствие чего снижается сопротивление пассивным движениям и увеличивается объем активных движений.\u003Cbr\u003EМиорелаксирующий аффект (измерение по шкале Ашворта и с помощью \"маятникового\" теста) и побочные действия (снижение частоты сердечных сокращений (ЧСС) и снижение артериального давления (АД)) препарата зависят от концентрации тизанидина в плазме крови.\u003Cbr\u003E"},{"name":"Фармакологическая группа","value":"миорелаксант центрального действия"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"В защищенном от света месте, при температуре не выше 25 °С. Хранить в недоступном для детей месте."},{"name":"Передозировка","value":"К настоящему времени получено несколько сообщений о передозировке препаратом Тизанидин-СЗ, включая случай, когда принятая доза составила 400 мг. Во всех случаях выздоровление прошло без особенностей.\u003Cbr\u003EСимптомы: тошнота, рвота, снижение АД, удлинение интервала QT (с), головокружение, сонливость, миоз, беспокойство, угнетение дыхания, кома.\u003Cbr\u003EЛечение. Для выведения препарата из организма рекомендуется многократное применение активированного угля. Форсированный диурез также, возможно, ускорит выведение тизанидина. В дальнейшем проводят симптоматическое лечение.\u003Cbr\u003E"},{"name":"Применение при беременности и кормлении грудью","value":"Беременность\u003Cbr\u003EПоскольку контролируемые исследования применения тизанидина у беременных женщин не проводились, его не следует применять в период беременности, за исключением тех случаев, когда потенциальная польза превышает возможный риск.\u003Cbr\u003EВ исследованиях у животных не выявлено явлений тератогенности. При применении в дозах 10 и 30 мг/кг в сутки у животных отмечено увеличение срока гестации, зарегистрированы случаи пренатальной и постнатальной потери плода, а также задержка развития плода. При применении вышеуказанных доз у самок отмечались выраженные признаки миорелаксации и седации. Исходя из площади поверхности тела, указанные дозы превышали максимальную рекомендуемую дозу для человека (0,72 мг/кг в сутки) в 2,2 и 6,7 раз.\u003Cbr\u003EГрудное вскармливание\u003Cbr\u003EВ исследованиях у животных тизанидин выделялся в небольших количествах с молоком лактирующих самок. Не следует применять препарат в период грудного вскармливания, так как нет данных о проникновении тизанидина в грудное молоко у человека.\u003Cbr\u003EТест на беременность\u003Cbr\u003EПеред началом применения препарата Тизанидин-СЗ у пациенток с сохраненным репродуктивным потенциалом рекомендовано получить результат теста на беременность.\u003Cbr\u003EВлияние на фертильность\u003Cbr\u003EВ исследованиях у животных не отмечалось неблагоприятного влияния на фертильность особей мужского и женского пола при применении тизанидина в дозе 10 мг/кг в сутки и 3 мг/кг/ сутки соответственно. Отмечалось уменьшение фертильности у особей мужского пола, получавших тизанидин в дозе, превышающей 30 мг/кг в сутки, и у особей женского пола - в дозе, превышающей 10 мг/кг сутки. Исходя из площади поверхности тела, указанные дозы превышали максимальную рекомендуемую дозу для человека (0,72 мг/кг в сутки) в 2,2 и 6,7 раз. При применении указанных доз со стороны матери отмечались поведенческие эффекты и клинические признаки, включающие выраженную седацию, уменьшение массы тела и атаксию.\u003Cbr\u003E"},{"name":"Влияние на способность управлять транспортом и механизмами","value":"Пациентам, у которых на фоне применения препарата отмечается сонливость, головокружение или какие-либо признаки артериальной гипотензии следует рекомендовать воздержаться от видов деятельности, требующих высокой концентрации внимания и быстрой реакции, например, управления транспортными средствами и механизмами."},{"name":"Особые указания","value":"Гипотензия может возникать на фоне применения препарата Тизанидин-СЗ, а также как результат лекарственного взаимодействия с ингибиторами изофермента CYP1A2 и/или гипотензивными препаратами. Выраженное снижение АД может приводить к потере сознания и циркуляторному коллапсу.\u003Cbr\u003EСообщалось о случаях нарушений функции печени, связанных с тизанидином, однако при применении суточной дозы до 12 мг эти случаи отмечались редко. В связи с этим рекомендуется контролировать функциональные \"печеночные пробы\" 1 раз в месяц в первые 4 месяца лечения у пациентов, которые получают тизанидин в суточной дозе 12 мг и выше, а также в тех случаях, когда наблюдаются клинические признаки, позволяющие предположить нарушение функции печени, такие как необъяснимая тошнота, анорексия, чувство усталости. В случае, когда активность аланинаминотрансферазы (АЛТ) и аспартатаминотрансферазы (ACT) в сыворотке стойко превышают верхнюю границу нормы в 3 раза и более, применение препарата Тизанидин-СЗ следует прекратить.\u003Cbr\u003EКонтрацепция\u003Cbr\u003EСледует информировать пациенток с сохраненным репродуктивным потенциалом о неблагоприятном влиянии препарата на развивающийся плод, выявленном в исследованиях у животных. Во время применения препарата, а также в течение 1 суток после прекращения приема препарата пациенткам с сохраненным репродуктивным потенциалом следует использовать надежные способы контрацепции (при правильном и длительном использовании которых частота наступления беременности составляет \u003C 1 %).\u003Cbr\u003E"},{"name":"Взаимодействие","value":"При применении препарата Тизанидин-СЗ с ингибиторами изофермента CYP1A2 возможно повышение концентрации тизанидина в плазме крови. В свою очередь, повышение концентрации тизанидина в плазме крови может приводить к симптомам передозировки препаратом, в том числе удлинению интервала QT(c).\u003Cbr\u003EОдновременное применение препарата Тизанидин-СЗ с индукторами изофермента CYP1A2 может приводить к снижению концентрации тизанидина в плазме крови, что может приводить к уменьшению терапевтического эффекта препарата.\u003Cbr\u003EПротивопоказанные комбинации с тизанидином\u003Cbr\u003EОдновременное применение тизанидина с флувоксамином или ципрофлоксацином, ингибиторами изофермента CYP1А2, противопоказано. При применении тизанидина с флувоксамином или ципрофлоксацином отмечается соответственно 33-кратное и 10-кратное увеличению AUC тизанидина. Результатом одновременного применения может оказаться значимая и длительная гипотензия сопровождающаяся сонливостью, головокружением, снижением скорости психомоторных реакций (в отдельных случаях вплоть до циркуляторного коллапса и потери сознания).\u003Cbr\u003EНе рекомендуемые комбинации с тизанидином\u003Cbr\u003EНе рекомендуется применять тизанидин одновременно с другими ингибиторами изофермента CYP1A2 - антиаритмическими препаратами (амиодарон, мексилетин, пропафенон), циметидином, некоторыми фторхинолонами (эноксацин, пефлоксацин, норфлоксацин), рофекоксибом, пероральными контрацептивами, тиклопидином.\u003Cbr\u003EКомбинации с тизанидином, требующие соблюдения осторожности\u003Cbr\u003EНеобходимо соблюдать осторожность при одновременном применении препарата Тизанидин-СЗ с препаратами, удлиняющими интервал QT (например, цизаприд, амитриптилин, азитромицин).\u003Cbr\u003EГипотензивные препараты\u003Cbr\u003EОдновременное применение препарата Тизанидин-СЗ с гипотензивными препаратами, включая диуретики, иногда может вызывать выраженное снижение АД (в отдельных случаях вплоть до циркуляторного коллапса и потери сознания) и брадикардию.\u003Cbr\u003EПри резкой отмене препарата Тизанидин-СЗ после одновременного применения с гипотензивными препаратами отмечалось развитие тахикардии и повышение АД, которое в отдельных случаях может привести к острому нарушению мозгового кровообращения.\u003Cbr\u003EРифампицин\u003Cbr\u003EОдновременный прием тизанидина и рифампицина приводит к 50 % снижению концентрации тизанидина в плазме крови. Вследствие этого терапевтическое действие препарата может снижаться, что может иметь клиническую значимость для некоторых пациентов. Следует избегать длительного одновременного применения рифампицина и тизанидина при невозможности рекомендуется тщательный подбор дозы тизанидина (увеличение).\u003Cbr\u003EКурение табака\u003Cbr\u003EСистемная биодоступность тизанидина у курящих пациентов (более 10 сигарет в день) снижена примерно на 30 %. Длительная терапия препаратом у пациентов данной категории может потребовать более высоких доз тизанидина, чем средние терапевтические.\u003Cbr\u003EАлкоголь\u003Cbr\u003EВо время терапии препаратом следует избегать приема алкоголя, так как он может повысить вероятность развития нежелательных явлений (например, снижения АД и заторможенности). Тизанидин может усиливать угнетающее действие алкоголя на центральную нервную систему.\u003Cbr\u003EДругие лекарственные средства\u003Cbr\u003EСедативные, снотворные препараты (бензодиазепин, баклофен) и другие препараты, такие как антигистаминные препараты, могут также усиливать седативный эффект тизанидина. Следует избегать приема препарата с другими агонистами альфа2-адренорецепторов (например, клонидином) вследствие потенциального усиления гипотензивного эффекта.\u003Cbr\u003E"},{"name":"Регистрационный номер","value":"ЛП-005748"},{"name":"Дата государственной регистрации","value":"27.08.2019"},{"name":"Владелец регистрационного удостоверения","value":"Северная Звезда"},{"name":"Изготовитель","value":"Северная Звезда"},{"name":"Фасовщик","value":"Северная Звезда"},{"name":"Страна бренда","value":"Россия"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Тизанидин"},{"name":"Срок годности","value":"1 г."}]}],"transitionId":"tr_6312905835254738495"}}}}
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Есть противопоказания, посоветуйтесь с врачом. Отпускается по рецепту врача. Приобретение лекарственных препаратов осуществляется только в торговом зале аптеки

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Где купить

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208 ₽

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  • Сегодня, самовывоз  0 ₽
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Рейтинг 5 из 5
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Инструкция

Показания к применению

Болезненный мышечный спазм:
связанный со статическими и функциональными заболеваниями позвоночника (шейный и поясничный синдромы);
после хирургических вмешательств, например, по поводу грыжи межпозвонкового диска или остеоартроза тазобедренного сустава.
Спастичность скелетных мышц при неврологических заболеваниях, например, при рассеянном склерозе, хронической миелопатии, дегенеративных заболеваниях спинного мозга, последствиях нарушений мозгового кровообращения и детском церебральном параличе (пациенты старше 18 лет).

Противопоказания

Повышенная чувствительность к тизанидину или к любому другому компоненту препарата.
- Нарушение функции печени тяжелой степени.
- Одновременное применение с мощными ингибиторами изофермента CYP1А2, такими как флувоксамин или ципрофлоксацин.
- Не рекомендовано пациентам с редкими наследственными заболеваниями, такими как дефицит лактазы, непереносимость лактозы, глюкозо-галактозная мальабсорбция, так как лекарственная форма содержит лактозу.
- Опыт применения препарата у пациентов младше 18 лет ограничен. Применение препарата Тизанидин-СЗ у пациентов данной популяции не рекомендовано.

Способ применения и дозы

Препарат Тизанидин-СЗ обладает узким терапевтическим индексом и высокой вариабельностью концентрации тизанидина в плазме крови, поэтому необходим тщательный подбор дозы.
Дозу и режим дозирования следует подбирать индивидуально в зависимости от потребностей пациента. Применение препарата в начальной дозе 2 мг 3 раза в день снижает риск развития побочных эффектов.
Препарат принимают внутрь. Таблетки 2 мг и 4 мг могут быть разделены на две равные части.
При болезненном мышечном спазме препарат Тизанидин-СЗ применяют, как правило, в дозе 2 мг или 4 мг 3 раза в сутки.
В тяжелых случаях возможно дополнительное применение 2 мг или 4 мг (предпочтительно перед сном из-за возможного усиления сонливости).
При спастичности скелетных мышц, обусловленной неврологическими заболеваниями, начальная суточная доза не должна превышать 6 мг, разделенных на 3 приема. Дозу можно повышать постепенно, на 2-4 мг, с интервалами от 3-4 до 7 дней. Как правило, оптимальный терапевтический эффект достигается при суточной дозе от 12 до 24 мг, разделенной на 3 или 4 приема через равные промежутки времени. Не следует превышать дозу 36 мг в сутки.
Применение у пациентов старше 65 лет
Опыт применения препарата Тизанидин-СЗ у пациентов в возрасте старше 65 лет и старше ограничен. Рекомендуется начинать терапию с минимальной дозы с постепенным повышением до достижения оптимального соотношения переносимости и эффективности терапии.
Применение у пациентов с нарушениями функции почек Лечение пациентов с почечной недостаточностью (КК менее 25 мл/мин) рекомендуется начинать с дозы 2 мг 1 раз в день. Повышение дозы проводят малыми "шагами" с учетом переносимости и эффективности. При необходимости достижения более выраженного эффекта, рекомендуется сначала увеличить дозу, применяемую 1 раз в сутки, после чего увеличивают кратность применения.
Применение у пациентов с нарушениями функции печени
Применение препарата Тизанидин-СЗ у пациентов с нарушением функции печени тяжелой степени противопоказано.
У пациентов с нарушением функции печени средней степени тяжести препарат следует применять с осторожностью; рекомендовано начинать терапию с минимальной дозы, с постепенным повышением до достижения оптимального соотношения переносимости и эффективности терапии. Рекомендации по контролю показателей функции печени указаны в разделе "Особые указания".
Прерывание лечения
При прекращении терапии препаратом Тизанидин-СЗ с целью уменьшения риска развития рикошетной гипертензии и тахикардии следует медленно снижать дозу до полной отмены препарата, в особенности у пациентов, получающих высокие дозы препарата в течение длительного времени.
Полная инструкция
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Тизанидин-СЗ таб.
Тизанидин-СЗ таб., 4 мг, 30 шт.
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Инструкция

208 ₽

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5.0
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У продавца:4 оценки·1 отзыв
У всех продавцов:18 оценок·10 отзывов
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4 месяца назад • Наталья • Куплен на Маркете
Комментарий: Хороший препарат
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  • Таблетница на день мини для капсул контейнер для таблеток белый
    {"widgets":{"@marketfront/SnippetConstructor/Gallery":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1915570066_3/content/content/gallery":{"title":"Таблетница на день мини для капсул контейнер для таблеток белый","images":[{"src":"https://avatars.mds.yandex.net/get-mpic/1961245/2a0000018a52b1bad4d962a614c1b1d089c4/orig","srcSet":"https://avatars.mds.yandex.net/get-mpic/1961245/2a0000018a52b1bad4d962a614c1b1d089c4/120x160 120w, https://avatars.mds.yandex.net/get-mpic/1961245/2a0000018a52b1bad4d962a614c1b1d089c4/180x240 180w, https://avatars.mds.yandex.net/get-mpic/1961245/2a0000018a52b1bad4d962a614c1b1d089c4/240x320 240w, https://avatars.mds.yandex.net/get-mpic/1961245/2a0000018a52b1bad4d962a614c1b1d089c4/300x400 300w, https://avatars.mds.yandex.net/get-mpic/1961245/2a0000018a52b1bad4d962a614c1b1d089c4/600x800 600w","sizes":"(max-width: 1456px) 15vw, 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  • Таблетница на 7 дней Органайзер для лекарств
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  • Контейнер для хранения/таблетница/кейс для таблеток
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  • Таблетница компактная /органайзер аптечка/ контейнер для таблеток БАД Panda_Home (синего цвета)
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  • Таблетница «Неделька», английские буквы, 7 секций, цвет прозрачный
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    Реклама
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  • VETTA / Таблетница-органайзер для таблеток аптечка для лекарств карманная в дорогу с разделителем на 14 секций, на неделю 7 дней, утро вечер
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  • Таблетница «Время», 3 секции, зеленая, 7,3 х 1,5 см
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  • Таблетница функциональный кейс для таблеток и капсул Iverylab
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  • Таблетница на 7 дней / органайзер / бокс / контейнер на неделю для хранения таблеток и лекарств 4 приема Clear Daswerk
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  • Таблетница на 7 дней Органайзер для лекарств
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  • Таблетница с зеркальной поверхностью, 3 секции, d 5см, цвет серебристый
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  • Таблетница пенал - органайзер ABORNS на неделю 7 ячеек 7 дней
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  • Таблетница «Неделька», английские буквы, 7 секций, цвет прозрачный
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  • Таблетница "Неделька" , английские буквы , 7 секций , цвет прозрачный
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  • {"widgets":{"@yandex-market/LazyLoader-market":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator":{"widgetName":"@marketfront/RecomLayout","widgetId":"ServerListRendererForSerp_RecommendationRoll","options":{"resolverParams":{"resources":{"garsons":[{"count":24,"limit":24,"params":{"cartProductIds":[],"snippetTypes":["product","product-block","category-block","advertisement","media-incut","promo-trigger","media-adv-banner-single","media-adv-banner-double","media-adv-carousel"],"program":"remix_desktop_model_card","hyperid":955689315},"id":"RemixData"}],"shuffle":{"mode":"exclusive"}},"limit":24},"id":"RecommendationRoll","slotOptions":{"dynamic":true},"className":"","needToProvideData":true,"wrapperProps":{},"widgetOptions":{"config":{"pictureBlock":{"maxGalleryImagesCount":5},"descriptionBlock":{"order":1,"titleRowCount":"2"},"offerBlock":{"withGreenPrice":true,"order":2,"price":{"wrap":true,"overflow":"hidden"}}},"galleryImageSize":250},"layoutOptions":{"needFallbackOnError":true,"needFallbackOnEmpty":false,"countInRows":6},"isChefRemixExp":false},"slotOptions":{"dynamic":true},"placeholder":"Invisible","infinite":true,"cspNonce":"avgFkMbqXO+r/2pe7Xcsvg==","renderStrategy":"append","renderedOnce":true}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator":{"name":"@yandex-market/LazyLoader-market"}}}
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