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Торасемид таб., 10 мг, 60 шт.

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Дозировка: 10 мг

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Количество штук в упаковке, шт.: 60

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Коротко о товаре

Артикул Маркета
3450440300
Действующее вещество
Возраст
от 18 лет
Инструкция
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артериальная гипертензия."},{"name":"Противопоказания","value":"повышенная чувствительность к торасемиду или любому из компонентов препарата; аллергия на сульфонамиды (сульфаниламидные противомикробные средства или препараты сульфонилмочевины); почечная недостаточность с анурией; печеночная кома и прекома; рефрактерная гипокалиемия; рефрактерная гипонатриемия; гиповолемия (с артериальной гипотензией или без нее) или дегидратация;\u003Cb\u003E-резко выраженные нарушения оттока мочи любой этиологии (включая одноутороннее поражение мочевыводящих путей); гликозидная интоксикация; острый гломерулонефрит; синоатриальная и атриовенокулярная блокада II-III степени; декомпенсированный артериальный и митральный стеноз; гипертрофическая обструктивная кардиомиопатия; повышение центрального венозного давления (свыше 10 мм рт.ст.); аритмия; хроническая почечная недостаточность с нарастающей азотемией; гиперурикемия; возраст до 18 лет; \nбеременность; период грудного вскармливания; одновременное применение аминогликозидов и цефалоспоринов; непереносимость лактозы, дефицит лактазы или глюкозо-галактозная мальабсобция.\u003Cb\u003EС осторожностью\u003Cb\u003Eартериальная гипотензия; стенозирующий атеросклероз церебральных артерий; гипопротеинемия; предрасположенность к гипергликемии, нарушения оттока мочи (доброкачественная гиперплазия предстательной железы, сужение мочеиспускательного канала или гидронефроз); желудочковая аритмия в анамнезе; острый инфаркт миокарда (увеличение риска развития кардиогенного шока); диарея; панкреатит; гипокалиемия; гипонатриемия; сахарный диабет (снижение толерантности к глюкозе); нарушение функции печени, цирроз печени, гепаторенальный синдром; почечная недостаточность, подагра, анемия; одновременное\tприменение сердечных\tгликозидов, кортикостероидов и адренокортикостероидного гормона (АКТГ)."},{"name":"Состав","value":"На 1 таблетку:\u003Cb\u003EДействующее вещество:\u003Cb\u003EТорасемид 5,0/10,0 мг\u003Cb\u003EВспомогательные вещества:\u003Cb\u003EЛактозы моногидрат 79,0/158,0 мг; целлюлоза микрокристаллическая (МКЦ-101) 10,0мг/20,0 мг, кросповидон 3,0 мг/6,0 мг; повидон К30 2,0 мг/4,0 мг; магния стеарат 1,0 мг/2,0 мг."},{"name":"Действующее вещество","value":"Торасемид","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["27144131:28709532"]}}},{"name":"Способ применения и дозы","value":"Внутрь, один раз в день, после завтрака, не разжевывая, запивая небольшим количеством воды.\u003Cb\u003EОтечный синдром при хронической сердечной недостаточности\u003Cb\u003EОбычная терапевтическая доза составляет 10-20 мг внутрь один раз в день. При необходимости дозу следует постепенно увеличить до 20-40 мг один раз в день, до получения требуемого эффекта.\u003Cb\u003EОтечный синдром при заболевании почек\u003Cb\u003EОбычная терапевтическая доза составляет 20 мг внутрь один раз в день. При необходимости дозу следует постепенно увеличить вдвое, до получения требуемого эффекта. С отечный синдром при заболевании печени обычная терапевтическая доза составляет 5-10 мг внутрь один раз в день. При необходимости доза может быть увеличена вдвое, до получения требуемого эффекта. Максимальная разовая доза составляет 40 мг; её превышать не рекомендуется (отсутствует опыт применения). Препарат применяют в течение длительного времени, или до получения требуемого эффекта.\u003Cb\u003EАртериальная гипертензия\u003Cb\u003EНачальная доза составляет 2,5 мг (1/2 табл. по 5 мг) один раз в день. При необходимости доза может быть увеличена до 5 мг один раз в день.\u003Cb\u003E При отсутствии адекватного снижения артериального давления при приёме препарата в дозе 5 мг один раз в день в течение 4-6 недель дозу увеличивают до 10 мг один раз в день. Если доза 10 мг не даёт требуемого результата, в лечебную схему нужно добавить гипотензивный препарат другой группы.\u003Cb\u003EПациентам пожилого возраста коррекции дозы не требуется.\u003Cb\u003EПропуск дозы: в случае пропуска очередной дозы нельзя принимать двойную дозу препарата. Следует сразу же принять бытую дозу. Следующую дозу принимают в обычное время на следующий день."},{"name":"Побочные действия","value":"Нежелательные реакции перечислены в зависимости от анатомо-физиологической классификации и встречаемости. Частота встречаемости определяется таким образом: очень часто \u003E1/10, часто -3 1/100 и 4/10, нечасто и \u003C1/100, редко и \u003C1/1000 и очень редко 4/10000.\u003Cb\u003EНарушения со стороны обмена веществ и питания: частота неизвестна гипонатриемия, гипохлоремия, гипокалиемия, гипомагниемия, гипокальциемия, метаболический алкалоз. Симптомами, указывающими на развитие нарушений водноэлектролитного состояния и кислотно-щелочного состояния, могут быть: головная боль, спутанность сознания, судороги, тетания, мышечная слабость, нарушения ритма сердца и диспепсия; гиповолемия и дегидратация (чаще у пациентов пожилого возраста), которые могут привести к гемоконцентрации с тенденцией к развитию тромбоза.\u003Cb\u003EНарушения со стороны сердца: нечасто экстрасистолия, тахикардия, аритмия.\u003Cb\u003EНарушения со стороны сосудов:астота неизвестна — чрезмерное снижение артериального давления, ортостатическая гипотензия, коллапс, снижение объёма С циркулирующей крови, тромбоз глубоких вен, тромбоэмболия.\u003Cb\u003EНарушения со стороны лабораторных и инструментальных данных: нечасто гиперхолестеринемия, гипертриглицеридемия; преходящее повышение концентрации креатинина и мочевины в крови; повышение концентрации мочевой кислоты в крови, что может вызвать или усилить проявлен подагры; снижение толерантности к глюкозе (возможна манифестация латентно протекающего сахарного диабета), повышение активности печеночных ферментов.\u003Cb\u003EНарушения со стороны почек и мочевыводящих путей: часто — увеличение частоты мочеиспускания, полиурия, никтурия; нечасто — учащенные позывы к мочеиспусканию; частота неизвестна олигурия, острая задержка мочи (например при гиперплазии предстательной железы, сужении мочеиспускательного канала, гидронефрозе); интерстициальный нефрит, гематурия, снижение потенции.\u003Cb\u003EНарушения со стороны желудочно-кишечного тракта: часто — диарея, нечасто — боль в животе, метеоризм, полидипсия; частота неизвестна — сухость во рту, тошнота, рвота, потеря аппетита, острый панкреатит.\u003Cb\u003EНарушения со стороны печени и желчевыводящих путей: внутрипеченочный холестаз. Нарушения со стороны органа слуха и лабиринтные нарушения: нечасто — нарушение слуха, обычно обратимое, и/или шум в ушах, особенно у пациентов с почечной недостаточностью или гипопротеинемией (нефротический синдром),\u003Cb\u003EНарушения со стороны нервной системы: часто — головная боль, головокружение, сонливость; нечасто — парестезия.\u003Cb\u003EНарушения со стороны кожи и подкожных тканей: нечасто — кожный зуд, крапивница, другие виды кожной сыпи или буллезное поражение кожи, полиморфная эритема, эксфолиативный дерматит, пурпура, лихорадка, васкулит, эозинофилия, фотосенсибилизация.\u003Cb\u003EНарушения со стороны общих расстройств и в месте введения: тяжелые анафилактические или анафилактоидные реакции вплоть до шока, которые до настоящего времени были описаны лишь после внутривенного введения.\u003Cb\u003EНарушения со стороны крови и лимфатической системы: частота неизвестна тромбоцитопения; лейкопения; агранулоцитоз, апластическая или гемолитическая анемия.\u003Cb\u003E"},{"name":"Фармакологическое действие","value":"Торасемид является петлевым диуретиком. Основной механизм действия препарата обусловлен обратимым связыванием торасемида с контранспортером ионов натрия/хлора/калия, расположенным в апикальной мембране толстого сегмента восходящей части петли Генле, в результате чего снижается или полностью ингибируется реабсорбция ионов натрия и уменьшается осмотическое давление внутриклеточной жидкости и реабсорбция воды. Блокирует альдостероновые рецепторы миокарда, уменьшает фиброз и улучшает диастолическую функцию миокарда.\u003Cb\u003EТорасемид в меньшей степени, чем фуросемид, вызывает гипокалиемию, при этом он проявляет большую активность, и его действие более продолжительно.\u003Cb\u003EТорасемид снижает систолическое и диастолическое артериальное давление в положении «лёжа» и «стоя».\u003Cb\u003EПрименение торасемида является наиболее обоснованным выбором для проведения длительной терапии."},{"name":"Фармакологическая группа","value":"диуретики"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["35947170:36763744"]}}},{"name":"Минимальный возраст применения","value":"от 18 лет"},{"name":"Условия хранения","value":"При температуре не выше 25 С.\u003Cb\u003EХранить в недоступном для детей месте.\u003Cb\u003E"},{"name":"Передозировка","value":"Симптомы: чрезмерно повышенный диурез, сопровождающийся снижением объёма циркулирующей крови и нарушением водно-электролитного баланса крови, с последующим выраженным снижением артериального давления, сонливостью и спутанностью сознания, коллапсом. Могут наблюдаться желудочно-кишечные расстройства.\u003Cb\u003EЛечение: специфического антидота нет. Провокация рвоты, промывание желудка, активированный уголь. Лечение симптоматическое, снижение дозы или отмена препарата и одновременное восполнение объёма циркулирующей крови и коррекция показателей водно-электролитного баланса и кислотно-основного состояния под контролем сывороточных концентраций электролитов, гематокрита.\u003Cb\u003EГемодиализ неэффективен, так как выведение торасемида и его метаболизм не ускоряется.\u003Cb\u003E"},{"name":"Применение при беременности и кормлении грудью","value":"Торасемид не обладает тератогенным эффектом и фетотоксичностью, проникает через плацентарный барьер, вызывая нарушения водно-электролитного обмена и тромбоцитопению у плода.\u003Cb\u003EНеизвестно, проникает ли торасемид в грудное молоко. При необходимости применения препарата Торасемид в период лактации необходимо прекратить грудное вскармливание.\u003Cb\u003E"},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения пациенты должны воздержаться от управления транспортными средствами и занятий другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Применять препарат Торасемид строго по назначению врача.\u003Cb\u003EПациенты с повышенной чувствительностью к сульфаниламидам и производным сульфонилмочевины могут иметь перекрестную чувствительность к торасемиду.\u003Cb\u003EПациентам, получающим высокие дозы торасемида в течение длительного периода, во избежание развития гипонатриемии, метаболического алкалоза и гипокалиемии, рекомендуется диета с достаточным содержанием поваренной соли и применение препаратов калия.\u003Cb\u003EПовышенный риск развития нарушений водно-электролитного баланса отмечается у пациентов с почечной недостаточностью. В ходе курсового лечения необходимо периодичес контролировать концентрацию электролитов плаз ы крови (в т.ч. натрия, кальция, калия, магния), кислотно-основное состояние, остаточный азот, креатинин, мочевую кислоту и проводить при необходимости соответствующую коррекционную терапию (с большей кратностью у пациентов с частой рвотой и на фоне парентерально вводимых жидкостей).\u003Cb\u003EУ пациентов с развившимися водно-электролитными нарушениями, гиповолемией или преренальноазотемией, данные лабораторных анализов могут включать: гипер- или гипонатриемю, гипер- или гипохлоремию, гипер- или гипокалиемию, нарушения кислотно-щелочного баланса и повышение концентрации мочевины в плазме крови. При возникновении этих расстройств необходимо прекратить приём препарата Торасемид до восстановления нормальных значений, а затем возобновить лечение препаратом Торасемид в меньшей дозе.\u003Cb\u003EПри появлении или усилении азотемии и олигурии у пациентов с тяжелыми прогрессирующими заболеваниями почек рекомендуется приостановить лечение.\u003Cb\u003EПодбор режима доз пациентам с асцитом на фоне цирроза печени нужно проводить в стационарных условиях (нарушения водно-электролитного баланса могут повлечь развитие печеночной комы). Данной категории пациентов показан регулярный контроль электролитов плазмы крови.\u003Cb\u003EПрименение препарата Торасемид может обусловливать обострение подагры.\u003Cb\u003EУ пациентов с сахарным диабетом или со сниженной толерантностью к глюкозе требуется периодический контроль концентрации глюкозы в крови и моче. \nУ пациентов в бессознательном состоянии, с гиперплазией предстательной железы, сужением мочеточников необходим контроль диуреза в связи с возможностью острой задержки мочи. \nУ пациентов с заболеваниями сердечно-сосудистой системы, особенно принимающих сердечные гликозиды, вызванная диуретиками гипокалиемия может стать причиной развития аритмий.\u003Cb\u003E"},{"name":"Взаимодействие","value":"При одновременном применении торасемида с минерало- и глюкокортикостероидами, фотерицином В повышается риск развития гипогликемии; с сердечными гликозидами — возрастает риск развития гликозидной интоксикации вследствие гипокалиемии (для высоко- и низкополярных сердечных гликозидов ) и удлинения периода полувыведения (для низкополярных сердечных гликозидов).\u003Cb\u003EСнижает почечный клиренс препаратов лития и повышает вероятность развития интоксикации.\u003Cb\u003EПрием торасемида повышает концентрацию и риск развития нефро- и ототоксического действия цефалоспоринов, аминогликозидов, хлорамфеникола, этакриновой кислоты, антибиотиков, салицилатов, цисплатина, препаратов платины, амфотерицина В (вследствие конкурентного почечного выведения).\nПоследовательное или одновременное применение торасемида с ингибиторами ангиотензинпревращающего фермента (АПФ) или антагонистами рецепторов ангиотензина П может привести к выраженному снижению артериального давления. Этого можно избежать, снизив дозу торасемида или временно отменив его.\nНестероидные противовоспалительные препараты, сукральфат снижают диуретический эффект вследствие ингибирования синтеза простагландина, нарушения активности ренина в плазме крови и выведения альдостерона.\nТорасемид усиливает антигипертензивное действие гипотензивных средств, нервномышечную блокаду деполяризующих миорелаксантов (суксаметоний) и ослабляет действие недеполяризующих миорелаксантов (тубокурарин).\nОдновременнный прием больших доз салицилатов на фоне терапии торасемидом увеличивает риск проявления их токсичности (вследствие конкурентного почечного выведения).\nПовышает эффективность диазоксида и теофиллина, снижает гипогликемических сред , аллопуринола.\nПрессорные амины и торасемид взаимно снижают эффективность. Лекарственные средства, блокирующие канальциевую секрецию, повышают концентрацию торасемида в сыворотке крови.\nОдновременное применение пробенецида или метотрексата может уменьшать эффективность торасемида (одинаковый путь секреции). С другой стороны, торасемид может уводить к снижению почечной элиминации этих лекарственных средств.\u003Cb\u003EПри одновременном применении циклоспорина и торасемида увеличивается риск развития подагрического артрита вследствие того, что циклоспорин может вызвать нарушение экскреции уратов почками, а торасемид — гипергликемию.\u003Cb\u003EСообщалось, что у пациентов с высоким риском развития нефропатии, принимающих торасемид внутрь, при введении рентгеноконтрастных средств нарушения функций почек наблюдались чаще, чем у пациентов с высоким риском развития нефропатии, которым перед введением рентгеноконтрастных средств проводили внутривенную гидратацию. Биодоступность и, как следствие, эффективность торасемида может быть снижена при совместной терапии с колестирамином.\u003Cb\u003E"},{"name":"Регистрационный номер","value":"ЛП-004407"},{"name":"Дата государственной регистрации","value":"19.02.2020"},{"name":"Владелец регистрационного удостоверения","value":"Hetero Labs Limited","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["34324371:35649313","7893318:17784423"]}}},{"name":"Изготовитель","value":"Макиз-Фарма"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Торасемид","transition":{"type":"catalog","params":{"categorySlug":"sredstva-dlia-serdtsa-i-sosudov","categoryId":"15756887","navnodeId":"72494","glfilters":["17796364:18003828"]}}},{"name":"Срок годности","value":"926 дн."}]}},"fullSpecsGrouped":{"14528423836758936382":{"groups":[{"name":"Общие характеристики","items":[{"name":"Тип препарата","value":"лекарственный препарат"},{"name":"Рецептурный препарат","value":"да"},{"name":"Органы и системы","value":"кровеносные сосуды, сердце"},{"name":"Назначение","value":"артериальная гипертензия, отечный синдром различного генеза"},{"name":"Показания к применению","value":"отечный синдром различного генеза, в т.ч. при хронической сердечной недостаточности, заболеваниях печени, легких и почек; артериальная гипертензия."},{"name":"Противопоказания","value":"повышенная чувствительность к торасемиду или любому из компонентов препарата; аллергия на сульфонамиды (сульфаниламидные противомикробные средства или препараты сульфонилмочевины); почечная недостаточность с анурией; печеночная кома и прекома; рефрактерная гипокалиемия; рефрактерная гипонатриемия; гиповолемия (с артериальной гипотензией или без нее) или дегидратация;\u003Cb\u003E-резко выраженные нарушения оттока мочи любой этиологии (включая одноутороннее поражение мочевыводящих путей); гликозидная интоксикация; острый гломерулонефрит; синоатриальная и атриовенокулярная блокада II-III степени; декомпенсированный артериальный и митральный стеноз; гипертрофическая обструктивная кардиомиопатия; повышение центрального венозного давления (свыше 10 мм рт.ст.); аритмия; хроническая почечная недостаточность с нарастающей азотемией; гиперурикемия; возраст до 18 лет; \nбеременность; период грудного вскармливания; одновременное применение аминогликозидов и цефалоспоринов; непереносимость лактозы, дефицит лактазы или глюкозо-галактозная мальабсобция.\u003Cb\u003EС осторожностью\u003Cb\u003Eартериальная гипотензия; стенозирующий атеросклероз церебральных артерий; гипопротеинемия; предрасположенность к гипергликемии, нарушения оттока мочи (доброкачественная гиперплазия предстательной железы, сужение мочеиспускательного канала или гидронефроз); желудочковая аритмия в анамнезе; острый инфаркт миокарда (увеличение риска развития кардиогенного шока); диарея; панкреатит; гипокалиемия; гипонатриемия; сахарный диабет (снижение толерантности к глюкозе); нарушение функции печени, цирроз печени, гепаторенальный синдром; почечная недостаточность, подагра, анемия; одновременное\tприменение сердечных\tгликозидов, кортикостероидов и адренокортикостероидного гормона (АКТГ)."},{"name":"Состав","value":"На 1 таблетку:\u003Cb\u003EДействующее вещество:\u003Cb\u003EТорасемид 5,0/10,0 мг\u003Cb\u003EВспомогательные вещества:\u003Cb\u003EЛактозы моногидрат 79,0/158,0 мг; целлюлоза микрокристаллическая (МКЦ-101) 10,0мг/20,0 мг, кросповидон 3,0 мг/6,0 мг; повидон К30 2,0 мг/4,0 мг; магния стеарат 1,0 мг/2,0 мг."},{"name":"Действующее вещество","value":"Торасемид"},{"name":"Способ применения и дозы","value":"Внутрь, один раз в день, после завтрака, не разжевывая, запивая небольшим количеством воды.\u003Cb\u003EОтечный синдром при хронической сердечной недостаточности\u003Cb\u003EОбычная терапевтическая доза составляет 10-20 мг внутрь один раз в день. При необходимости дозу следует постепенно увеличить до 20-40 мг один раз в день, до получения требуемого эффекта.\u003Cb\u003EОтечный синдром при заболевании почек\u003Cb\u003EОбычная терапевтическая доза составляет 20 мг внутрь один раз в день. При необходимости дозу следует постепенно увеличить вдвое, до получения требуемого эффекта. С отечный синдром при заболевании печени обычная терапевтическая доза составляет 5-10 мг внутрь один раз в день. При необходимости доза может быть увеличена вдвое, до получения требуемого эффекта. Максимальная разовая доза составляет 40 мг; её превышать не рекомендуется (отсутствует опыт применения). Препарат применяют в течение длительного времени, или до получения требуемого эффекта.\u003Cb\u003EАртериальная гипертензия\u003Cb\u003EНачальная доза составляет 2,5 мг (1/2 табл. по 5 мг) один раз в день. При необходимости доза может быть увеличена до 5 мг один раз в день.\u003Cb\u003E При отсутствии адекватного снижения артериального давления при приёме препарата в дозе 5 мг один раз в день в течение 4-6 недель дозу увеличивают до 10 мг один раз в день. Если доза 10 мг не даёт требуемого результата, в лечебную схему нужно добавить гипотензивный препарат другой группы.\u003Cb\u003EПациентам пожилого возраста коррекции дозы не требуется.\u003Cb\u003EПропуск дозы: в случае пропуска очередной дозы нельзя принимать двойную дозу препарата. Следует сразу же принять бытую дозу. Следующую дозу принимают в обычное время на следующий день."},{"name":"Побочные действия","value":"Нежелательные реакции перечислены в зависимости от анатомо-физиологической классификации и встречаемости. Частота встречаемости определяется таким образом: очень часто \u003E1/10, часто -3 1/100 и 4/10, нечасто и \u003C1/100, редко и \u003C1/1000 и очень редко 4/10000.\u003Cb\u003EНарушения со стороны обмена веществ и питания: частота неизвестна гипонатриемия, гипохлоремия, гипокалиемия, гипомагниемия, гипокальциемия, метаболический алкалоз. Симптомами, указывающими на развитие нарушений водноэлектролитного состояния и кислотно-щелочного состояния, могут быть: головная боль, спутанность сознания, судороги, тетания, мышечная слабость, нарушения ритма сердца и диспепсия; гиповолемия и дегидратация (чаще у пациентов пожилого возраста), которые могут привести к гемоконцентрации с тенденцией к развитию тромбоза.\u003Cb\u003EНарушения со стороны сердца: нечасто экстрасистолия, тахикардия, аритмия.\u003Cb\u003EНарушения со стороны сосудов:астота неизвестна — чрезмерное снижение артериального давления, ортостатическая гипотензия, коллапс, снижение объёма С циркулирующей крови, тромбоз глубоких вен, тромбоэмболия.\u003Cb\u003EНарушения со стороны лабораторных и инструментальных данных: нечасто гиперхолестеринемия, гипертриглицеридемия; преходящее повышение концентрации креатинина и мочевины в крови; повышение концентрации мочевой кислоты в крови, что может вызвать или усилить проявлен подагры; снижение толерантности к глюкозе (возможна манифестация латентно протекающего сахарного диабета), повышение активности печеночных ферментов.\u003Cb\u003EНарушения со стороны почек и мочевыводящих путей: часто — увеличение частоты мочеиспускания, полиурия, никтурия; нечасто — учащенные позывы к мочеиспусканию; частота неизвестна олигурия, острая задержка мочи (например при гиперплазии предстательной железы, сужении мочеиспускательного канала, гидронефрозе); интерстициальный нефрит, гематурия, снижение потенции.\u003Cb\u003EНарушения со стороны желудочно-кишечного тракта: часто — диарея, нечасто — боль в животе, метеоризм, полидипсия; частота неизвестна — сухость во рту, тошнота, рвота, потеря аппетита, острый панкреатит.\u003Cb\u003EНарушения со стороны печени и желчевыводящих путей: внутрипеченочный холестаз. Нарушения со стороны органа слуха и лабиринтные нарушения: нечасто — нарушение слуха, обычно обратимое, и/или шум в ушах, особенно у пациентов с почечной недостаточностью или гипопротеинемией (нефротический синдром),\u003Cb\u003EНарушения со стороны нервной системы: часто — головная боль, головокружение, сонливость; нечасто — парестезия.\u003Cb\u003EНарушения со стороны кожи и подкожных тканей: нечасто — кожный зуд, крапивница, другие виды кожной сыпи или буллезное поражение кожи, полиморфная эритема, эксфолиативный дерматит, пурпура, лихорадка, васкулит, эозинофилия, фотосенсибилизация.\u003Cb\u003EНарушения со стороны общих расстройств и в месте введения: тяжелые анафилактические или анафилактоидные реакции вплоть до шока, которые до настоящего времени были описаны лишь после внутривенного введения.\u003Cb\u003EНарушения со стороны крови и лимфатической системы: частота неизвестна тромбоцитопения; лейкопения; агранулоцитоз, апластическая или гемолитическая анемия.\u003Cb\u003E"},{"name":"Фармакологическое действие","value":"Торасемид является петлевым диуретиком. Основной механизм действия препарата обусловлен обратимым связыванием торасемида с контранспортером ионов натрия/хлора/калия, расположенным в апикальной мембране толстого сегмента восходящей части петли Генле, в результате чего снижается или полностью ингибируется реабсорбция ионов натрия и уменьшается осмотическое давление внутриклеточной жидкости и реабсорбция воды. Блокирует альдостероновые рецепторы миокарда, уменьшает фиброз и улучшает диастолическую функцию миокарда.\u003Cb\u003EТорасемид в меньшей степени, чем фуросемид, вызывает гипокалиемию, при этом он проявляет большую активность, и его действие более продолжительно.\u003Cb\u003EТорасемид снижает систолическое и диастолическое артериальное давление в положении «лёжа» и «стоя».\u003Cb\u003EПрименение торасемида является наиболее обоснованным выбором для проведения длительной терапии."},{"name":"Фармакологическая группа","value":"диуретики"},{"name":"Форма выпуска","value":"таблетки"},{"name":"Способ применения/введения","value":"пероральный"},{"name":"Минимальный возраст применения","value":"от 18 лет"}]},{"name":"Дополнительно","items":[{"name":"Условия хранения","value":"При температуре не выше 25 С.\u003Cb\u003EХранить в недоступном для детей месте.\u003Cb\u003E"},{"name":"Передозировка","value":"Симптомы: чрезмерно повышенный диурез, сопровождающийся снижением объёма циркулирующей крови и нарушением водно-электролитного баланса крови, с последующим выраженным снижением артериального давления, сонливостью и спутанностью сознания, коллапсом. Могут наблюдаться желудочно-кишечные расстройства.\u003Cb\u003EЛечение: специфического антидота нет. Провокация рвоты, промывание желудка, активированный уголь. Лечение симптоматическое, снижение дозы или отмена препарата и одновременное восполнение объёма циркулирующей крови и коррекция показателей водно-электролитного баланса и кислотно-основного состояния под контролем сывороточных концентраций электролитов, гематокрита.\u003Cb\u003EГемодиализ неэффективен, так как выведение торасемида и его метаболизм не ускоряется.\u003Cb\u003E"},{"name":"Применение при беременности и кормлении грудью","value":"Торасемид не обладает тератогенным эффектом и фетотоксичностью, проникает через плацентарный барьер, вызывая нарушения водно-электролитного обмена и тромбоцитопению у плода.\u003Cb\u003EНеизвестно, проникает ли торасемид в грудное молоко. При необходимости применения препарата Торасемид в период лактации необходимо прекратить грудное вскармливание.\u003Cb\u003E"},{"name":"Влияние на способность управлять транспортом и механизмами","value":"В период лечения пациенты должны воздержаться от управления транспортными средствами и занятий другими потенциально опасными видами деятельности, требующими повышенной концентрации внимания и быстроты психомоторных реакций."},{"name":"Особые указания","value":"Применять препарат Торасемид строго по назначению врача.\u003Cb\u003EПациенты с повышенной чувствительностью к сульфаниламидам и производным сульфонилмочевины могут иметь перекрестную чувствительность к торасемиду.\u003Cb\u003EПациентам, получающим высокие дозы торасемида в течение длительного периода, во избежание развития гипонатриемии, метаболического алкалоза и гипокалиемии, рекомендуется диета с достаточным содержанием поваренной соли и применение препаратов калия.\u003Cb\u003EПовышенный риск развития нарушений водно-электролитного баланса отмечается у пациентов с почечной недостаточностью. В ходе курсового лечения необходимо периодичес контролировать концентрацию электролитов плаз ы крови (в т.ч. натрия, кальция, калия, магния), кислотно-основное состояние, остаточный азот, креатинин, мочевую кислоту и проводить при необходимости соответствующую коррекционную терапию (с большей кратностью у пациентов с частой рвотой и на фоне парентерально вводимых жидкостей).\u003Cb\u003EУ пациентов с развившимися водно-электролитными нарушениями, гиповолемией или преренальноазотемией, данные лабораторных анализов могут включать: гипер- или гипонатриемю, гипер- или гипохлоремию, гипер- или гипокалиемию, нарушения кислотно-щелочного баланса и повышение концентрации мочевины в плазме крови. При возникновении этих расстройств необходимо прекратить приём препарата Торасемид до восстановления нормальных значений, а затем возобновить лечение препаратом Торасемид в меньшей дозе.\u003Cb\u003EПри появлении или усилении азотемии и олигурии у пациентов с тяжелыми прогрессирующими заболеваниями почек рекомендуется приостановить лечение.\u003Cb\u003EПодбор режима доз пациентам с асцитом на фоне цирроза печени нужно проводить в стационарных условиях (нарушения водно-электролитного баланса могут повлечь развитие печеночной комы). Данной категории пациентов показан регулярный контроль электролитов плазмы крови.\u003Cb\u003EПрименение препарата Торасемид может обусловливать обострение подагры.\u003Cb\u003EУ пациентов с сахарным диабетом или со сниженной толерантностью к глюкозе требуется периодический контроль концентрации глюкозы в крови и моче. \nУ пациентов в бессознательном состоянии, с гиперплазией предстательной железы, сужением мочеточников необходим контроль диуреза в связи с возможностью острой задержки мочи. \nУ пациентов с заболеваниями сердечно-сосудистой системы, особенно принимающих сердечные гликозиды, вызванная диуретиками гипокалиемия может стать причиной развития аритмий.\u003Cb\u003E"},{"name":"Взаимодействие","value":"При одновременном применении торасемида с минерало- и глюкокортикостероидами, фотерицином В повышается риск развития гипогликемии; с сердечными гликозидами — возрастает риск развития гликозидной интоксикации вследствие гипокалиемии (для высоко- и низкополярных сердечных гликозидов ) и удлинения периода полувыведения (для низкополярных сердечных гликозидов).\u003Cb\u003EСнижает почечный клиренс препаратов лития и повышает вероятность развития интоксикации.\u003Cb\u003EПрием торасемида повышает концентрацию и риск развития нефро- и ототоксического действия цефалоспоринов, аминогликозидов, хлорамфеникола, этакриновой кислоты, антибиотиков, салицилатов, цисплатина, препаратов платины, амфотерицина В (вследствие конкурентного почечного выведения).\nПоследовательное или одновременное применение торасемида с ингибиторами ангиотензинпревращающего фермента (АПФ) или антагонистами рецепторов ангиотензина П может привести к выраженному снижению артериального давления. Этого можно избежать, снизив дозу торасемида или временно отменив его.\nНестероидные противовоспалительные препараты, сукральфат снижают диуретический эффект вследствие ингибирования синтеза простагландина, нарушения активности ренина в плазме крови и выведения альдостерона.\nТорасемид усиливает антигипертензивное действие гипотензивных средств, нервномышечную блокаду деполяризующих миорелаксантов (суксаметоний) и ослабляет действие недеполяризующих миорелаксантов (тубокурарин).\nОдновременнный прием больших доз салицилатов на фоне терапии торасемидом увеличивает риск проявления их токсичности (вследствие конкурентного почечного выведения).\nПовышает эффективность диазоксида и теофиллина, снижает гипогликемических сред , аллопуринола.\nПрессорные амины и торасемид взаимно снижают эффективность. Лекарственные средства, блокирующие канальциевую секрецию, повышают концентрацию торасемида в сыворотке крови.\nОдновременное применение пробенецида или метотрексата может уменьшать эффективность торасемида (одинаковый путь секреции). С другой стороны, торасемид может уводить к снижению почечной элиминации этих лекарственных средств.\u003Cb\u003EПри одновременном применении циклоспорина и торасемида увеличивается риск развития подагрического артрита вследствие того, что циклоспорин может вызвать нарушение экскреции уратов почками, а торасемид — гипергликемию.\u003Cb\u003EСообщалось, что у пациентов с высоким риском развития нефропатии, принимающих торасемид внутрь, при введении рентгеноконтрастных средств нарушения функций почек наблюдались чаще, чем у пациентов с высоким риском развития нефропатии, которым перед введением рентгеноконтрастных средств проводили внутривенную гидратацию. Биодоступность и, как следствие, эффективность торасемида может быть снижена при совместной терапии с колестирамином.\u003Cb\u003E"},{"name":"Регистрационный номер","value":"ЛП-004407"},{"name":"Дата государственной регистрации","value":"19.02.2020"},{"name":"Владелец регистрационного удостоверения","value":"Hetero Labs Limited"},{"name":"Изготовитель","value":"Макиз-Фарма"},{"name":"Страна-производитель","value":"Россия"},{"name":"Название препарата","value":"Торасемид"},{"name":"Срок годности","value":"926 дн."}]}],"transitionId":"tr_6444170962765496109"}}}}
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Ещё может подойти

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Инструкция

Показания к применению

отечный синдром различного генеза, в т.ч. при хронической сердечной недостаточности, заболеваниях печени, легких и почек; артериальная гипертензия.

Противопоказания

повышенная чувствительность к торасемиду или любому из компонентов препарата; аллергия на сульфонамиды (сульфаниламидные противомикробные средства или препараты сульфонилмочевины); почечная недостаточность с анурией; печеночная кома и прекома; рефрактерная гипокалиемия; рефрактерная гипонатриемия; гиповолемия (с артериальной гипотензией или без нее) или дегидратация;-резко выраженные нарушения оттока мочи любой этиологии (включая одноутороннее поражение мочевыводящих путей); гликозидная интоксикация; острый гломерулонефрит; синоатриальная и атриовенокулярная блокада II-III степени; декомпенсированный артериальный и митральный стеноз; гипертрофическая обструктивная кардиомиопатия; повышение центрального венозного давления (свыше 10 мм рт.ст.); аритмия; хроническая почечная недостаточность с нарастающей азотемией; гиперурикемия; возраст до 18 лет; беременность; период грудного вскармливания; одновременное применение аминогликозидов и цефалоспоринов; непереносимость лактозы, дефицит лактазы или глюкозо-галактозная мальабсобция.С осторожностьюартериальная гипотензия; стенозирующий атеросклероз церебральных артерий; гипопротеинемия; предрасположенность к гипергликемии, нарушения оттока мочи (доброкачественная гиперплазия предстательной железы, сужение мочеиспускательного канала или гидронефроз); желудочковая аритмия в анамнезе; острый инфаркт миокарда (увеличение риска развития кардиогенного шока); диарея; панкреатит; гипокалиемия; гипонатриемия; сахарный диабет (снижение толерантности к глюкозе); нарушение функции печени, цирроз печени, гепаторенальный синдром; почечная недостаточность, подагра, анемия; одновременное применение сердечных гликозидов, кортикостероидов и адренокортикостероидного гормона (АКТГ).

Способ применения и дозы

Внутрь, один раз в день, после завтрака, не разжевывая, запивая небольшим количеством воды.Отечный синдром при хронической сердечной недостаточностиОбычная терапевтическая доза составляет 10-20 мг внутрь один раз в день. При необходимости дозу следует постепенно увеличить до 20-40 мг один раз в день, до получения требуемого эффекта.Отечный синдром при заболевании почекОбычная терапевтическая доза составляет 20 мг внутрь один раз в день. При необходимости дозу следует постепенно увеличить вдвое, до получения требуемого эффекта. С отечный синдром при заболевании печени обычная терапевтическая доза составляет 5-10 мг внутрь один раз в день. При необходимости доза может быть увеличена вдвое, до получения требуемого эффекта. Максимальная разовая доза составляет 40 мг; её превышать не рекомендуется (отсутствует опыт применения). Препарат применяют в течение длительного времени, или до получения требуемого эффекта.Артериальная гипертензияНачальная доза составляет 2,5 мг (1/2 табл. по 5 мг) один раз в день. При необходимости доза может быть увеличена до 5 мг один раз в день. При отсутствии адекватного снижения артериального давления при приёме препарата в дозе 5 мг один раз в день в течение 4-6 недель дозу увеличивают до 10 мг один раз в день. Если доза 10 мг не даёт требуемого результата, в лечебную схему нужно добавить гипотензивный препарат другой группы.Пациентам пожилого возраста коррекции дозы не требуется.Пропуск дозы: в случае пропуска очередной дозы нельзя принимать двойную дозу препарата. Следует сразу же принять бытую дозу. Следующую дозу принимают в обычное время на следующий день.
Полная инструкция
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Торасемид таб.
Торасемид таб., 10 мг, 60 шт.
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Инструкция

282 ₽

Скидка: 15%
–15 %
Вместо:332 ₽
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4.8
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У продавца:60 оценок·16 отзывов
У всех продавцов:84 оценки·22 отзыва
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Единственно приходится часто ходить в туалет .","commonText":"Брала для отца против отеков на стопах по рекомендации врача. Помогло !!!!!!","media":[]},"ri_305056661":{"reviewId":"305056661","author":{"nickname":"Галина++ Мачнева","avatarMediaItemId":"mi_1102520468931834716","isAnonymous":false},"rating":5,"reviewDate":"1715325312957","advantages":"Принимаю постоянно,т.к. так прописал доктор.Старый организм нуждается в медикаментозной поддержке","disadvantages":"ни разу не обнаружила, хотя принимаю м","media":[]},"ri_282017653":{"reviewId":"282017653","author":{"nickname":"Имя скрыто","avatarMediaItemId":"mi_10976536813285640517","isAnonymous":true},"rating":5,"reviewDate":"1708409237459","commonText":"лекарства, это индивидуальный подход","media":[]},"ri_251676963":{"reviewId":"251676963","author":{"nickname":"фёдоров Николай","avatarMediaItemId":"mi_4861351551922539226","isAnonymous":false},"rating":5,"reviewDate":"1699962549136","advantages":"Торасемид является мощным диуретиком . Эффективен как в составе комплексной терапии , так и самостоятельно .Петлевой диуретик торасемид характеризуется высокой биодоступностью и пролонгированным эффектом (длительность действия до 18 часов ) что обуславливает ряд благоприятных фармакодинамических свойств препарата. Показание применения , порядок и дозировку определяются ТОЛЬКО лечащим врачём .","disadvantages":"не обнаружил","commonText":"Не смотря на все превосходства над другими диуретиками недопустимо самолечение данным препаратом .","media":[]}}}}
user avatar
7 месяцев назад • фёдоров Николай • Куплен на Маркете
Достоинства: Торасемид является мощным диуретиком . Эффективен как в составе комплексной терапии , так и самостоятельно .Петлевой диуретик торасемид характеризуется высокой биодоступностью и пролонгированным эффектом (длительность действия до 18 часов ) что обуславливает ряд благоприятных фармакодинамических свойств препарата. Показание применения , порядок и дозировку определяются ТОЛЬКО лечащим врачём .
Недостатки: не обнаружил
Комментарий: Не смотря на все превосходства над другими диуретиками недопустимо самолечение данным препаратом .
user avatar
Месяц назад • Ирина Г. • Куплен на Маркете
Достоинства: Как мочегонное , хорошее средство.
Недостатки: не замечены. Единственно приходится часто ходить в туалет .
Комментарий: Брала для отца против отеков на стопах по рекомендации врача. Помогло !!!!!!
user avatar
3 месяца назад • Zoo party of Russia • Куплен на Маркете
Достоинства: Торасемид является мощным диуретиком и эффективен как в составе комплексной терапии, из-за ряда благоприятных фармакодинамических свойств препарата, мне очень помог при лечении…
Недостатки: У меня не было обнаружено
Комментарий: Рекомендую данного производителя и продавца.
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  • Омепразол капс., 20 мг, 30 шт.
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  • ЛимфоТранзит концентрат напитка фл., 100 мл
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  • Ад минус таб., 40 шт.
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    {"widgets":{"@marketfront/SnippetConstructor/ToggleWishlist":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778173791_2/content/content/toggleWishlist":{"skuId":"226177677","productId":1778173791,"offerId":"4l2lSyhPkC3V5o1As7TOkg","size":24,"color":"#BDBDBC","wishlistLink":"/my/wishlist","baobabRealTimeEventPayload":{"version":"EPV_BRT_V1","payload":"CgoQ/9Tytruxht47EhoKGHJlbWl4X2Rlc2t0b3BfbW9kZWxfY2FyZDIVCN+O888GEI3l7GsY1buhBiDX3MEH","sign":"WAf0NcWa848o07JGo6r+TJRht3ZdERvBw0O4PcEhYPQ="},"waitWishlistCollections":false,"place":{"page":"product","widget":"feed"}}}},"meta":{"/content/page/fancyPage/recommendationRoll/content/lazyGenerator/initialContent/recomLayoutItem_21#1:1778173791_2/content/content/toggleWishlist":{"name":"@marketfront/SnippetConstructor/ToggleWishlist"}}}
  • Сердечные травы таб., 300 мг, 23 г, 30 шт.
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  • Vitamin D3, 50000 МЕ, 50 мл, 50 шт.
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  • Гилан ультра комфорт увлажн. гл. р-р, 0.3%, 0.4 мл, 50 г, 10 шт.
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  • Кардиолептин таб., 0.55 г, 50 шт., 1
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  • Эвалар Чай Эвалар БИО при повышенном содержании мочевой кислоты, 20 фильтр-пакетов
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    Реклама
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  • Ад Норма капс., 56 г, 60 шт., 1
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  • БиоГая Пробиотик капли детск. фл., 5 мл, 1 уп.
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  • Вазомакс капс., 720 г, 30 шт.
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  • Пастилки California Gold Nutrition Vitamin D3 gummies со вкусом фруктов и ягод, 280 г, 90 шт.
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  • Боярышник Форте капс., 30 шт.
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  • Дигидрокверцетин капс., 30 шт., 1
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  • Дигидрокверцетин 100 мг таб., 30 шт.
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  • Бономарлот капс., 20 шт.
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  • Везуген капс., 20 шт.
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  • Кардиоген капс., 60 шт., 1
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  • Кленбутерол Софарма таб., 0.02 мг, 50 шт.
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  • IKENA Нафтифин р-р противогрибковый фл., 1%, 37 г, 10 мл, 1 шт., нейтральный, 1 уп.
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    Реклама
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  • Холисал стомат. гель, 10 г
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  • Кетоконазол шампунь лекарственный, 2%, 75 г, 75 мл
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